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| Number | Title | Issue Date |
| 7405324 | Process for synthesising aminoadamantanes The present invention concerns a new process for synthesising aminoadamantanes of formula I in which R1 and R2 are identical or different and are H or a straight or branched alkyl group comprising from 1 to 6 carbon atoms, ... | 07/29/2008 |
| 7166744 | Retinoid derivatives and methods for producing said compounds and anti-cancer pharmaceutical composition comprising said compounds The present invention relates to a novel retinoid derivative compound represented by the formula I: wherein X, R1, R2 and R3 are as defined herein or pharmaceutically acceptalbe s... | 01/23/2007 |
| 6790992 | Scyphostatin analogues as SMase inhibitors The present invention relates to novel scyphostatin analogues, which distinguish themselves by acting as SMase inhibitors so that they are of therapeutic use for a number of diseases such as a HIV infection, neurodegenerative diseases, inflammatory diseases, apoplex... | 09/14/2004 |
| 6770784 | Use of γ-hydroxybutyric acid amides in the treatment of drug addiction and in particular of alcoholism Gamma-hydroxybutryic acid amides are used in the treatment of drug addiction and especially in the treatment of alcoholism. ... | 08/03/2004 |
| 6767925 | Sprayable analgesic composition and method of use A sprayable analgesic composition containing an analgesic which is absorbed into the bloodstream through the buccal mucosa and a pharmacologically acceptable liquid carrier. ... | 07/27/2004 |
| 6756500 | α,ω-Diene metathesis in the presence of ionic liquids A process for preparing a cyclic compound comprising subjecting a starting material in the presence of a catalyst component to metathesis reaction in the presence of an ionic liquid, wherein the starting material is a α,ω-diene bearing a α substituent NRR1 | 06/29/2004 |
| 6706765 | Aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: wherein X is O or NR9 and R1-R4, R6-R9, R11, R12, Ra | 03/16/2004 |
| 6518310 | Aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: ##STR1## wherein X is O or NR9 and R1 -R4, R6 -R9, R11, R12, Ra, Rb, R | 02/11/2003 |
| 6441232 | Selective nitrogen functionalization of organic compounds There is provided a method of selectively replacing a carbon-hydrogen bond at an unactivated saturated sp3 hybridised carbon atom in an organic compound by a carbon-nitrogen bond, the method comprising reacting the compound with a fluorinating agent in a ... | 08/27/2002 |
| 6326369 | Bicyclic quinone compounds, their production and use A compound of the formula: ##STR1## wherein R1 and R2 each represents a lower alkyl, or R1 and R2 may be bonded together to form a ring; X represents a spacer of which the number of atoms constituting the princi... | 12/04/2001 |
| 6262308 | Process for the preparation of racemic sertraline The invention relates to a process for preparing cis-N-methyl-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-naphthylamine, or racemic sertraline, corresponding to formula (I) ##STR1## in salt form, starting with 4-(3,4-dichlorophenyl)tetralone of formula (I... | 07/17/2001 |
| 6262295 | Process for the preparation of a racemic or optically active 4-(hydroxymethyl)-2-cyclopentene derivative A process for the preparation of a racemic or optically active compound of the formula ##STR1## where the group R1 is an unsubstituted or a halogen substituted C1-4 -alkyl, a C1-4 -alkoxy, an aryl, an arylalkyl, an aryloxy... | 07/17/2001 |
| 6252112 | Process for the preparation of an enantiomer of a (1R, 4S) or (1S, 4R)-1-amino-4-(hydroxymethyl)-2-cyclopentene derivative A novel process for the preparation of (1S, 4R)- or (1R, 4S)-4-(2-amino-6-chloro-9H-purin-9-yl)-2 -cyclopentene-1-methanol of the formula ##STR1## is described.... | 06/26/2001 |
| 6235925 | Process for synthesizing khi-substituted ring systems Using the process according to the invention, it is possible to provide, with few reaction steps, a novel route to -substituted ring systems which optionally have further substituents.... | 05/22/2001 |
| 6137007 | Enantiomer compositions of (1R,4S)-1-butyrylamino-4-(hydroxymethyl)-2-cyclopentene A novel process for the preparation of (1S,4R)- or (1R,4S)-4-(2-amino-6-chloro-9H-purin-9-yl)-2-cyclopentene-1-methanol of the formulae ##STR1## is described. This entails in the first stage (&#b1;)-2-azabicyclo[2.2.1]hept-5-en-3-one of the form... | 10/24/2000 |
| 5998653 | 1-(substituted phenyl)-2,3-disubstituted propane-1,3-diones as intermediates to 4-benzoylisoxazoles Compounds of the formula ##STR1## are useful as intermediates to new herbicidal 4-benzoylisoxazoles.... | 12/07/1999 |
| 5939554 | Diarylaminopropanediol and diarylmethyl-oxazolidinone compounds A method for preparing a diarylalanine compound is provided. The method includes reacting a diarylaminopropanediol with a reducing agent to form a diarylaminopropanol compound and/or contacting a serine ester derivative with an aryl metal reagent to form ... | 08/17/1999 |
| 5900507 | Process for the preparation of 1-amino-1-methyl-3(4)-aminomethyl cyclohexane The present invention relates to a process for the preparation of 1-amino-1-methyl-3(4)-aminomethyl cyclohexane (AMCA) by a) catalytically hydrogenating 1-formamido-1-methyl-3(4)-cyano cyclohexane (FMC) in a first reaction stage to form 1-formamido-1-meth... | 05/04/1999 |
| 5856575 | Process for the preparation of N-acetyl aminophenols This invention provides a process for the manufacture of N-acetyl amino phenol, which process comprises reacting an appropriate phenol and an amide in the presence of a heteropoly acid or its alkali metal salt catalyst.... | 01/05/1999 |
| 5852194 | N-substituted cis-n-propenyl-acetamides, and process for their preparation The present invention relates to new N-substituted cis-N-propenyl-acetamides of the general formula (I) ##STR1## in which R1 represents in each case optionally substituted alkyl, -C(alkyl)2 -alkenyl, alkynyl, cycloalkyl, cycloal... | 12/22/1998 |
| 5753652 | Antiretroviral hydrazine derivatives The invention relates to compounds of formula ##STR1## and salts, pharmaceutical compositions, intermediates and processes of preparation thereof.... | 05/19/1998 |
| 5753709 | N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics Certain N-acyl 2-aryl cyclopropylmethylamine derivatives are useful as melatonergic agents.... | 05/19/1998 |
| 5710331 | Preparation of N-alkenyl carboxamides Preparation of N-alkenyl carboxamides of the general formula I ##STR1## in which the radicals R1 to R4 independently stand for hydrogen or for aliphatic, cycloaliphatic, or aromatic radicals, which optionally carry inert substit... | 01/20/1998 |
| 5668180 | Alkoxyaryl compounds A compound selected from those of formula (I): ##STR1## in which A, R, Y, R1, R2 and R3 are as defined in the description, and a medicinal product containing the same useful for treating a disorder of the melatoninerg... | 09/16/1997 |
| 5596019 | N-acyl-cycloalkylamine derivatives as melatonergics Certain N-acyl-cycloalkylamine derivatives are useful as melatonergic agents.... | 01/21/1997 |
| 5464872 | Arylalkyl (thio) amides A compound which is selected from those of formula (I): ##STR1## in which A, R1, R2, R3, R4, R5 and R6 are as defined in the description, its optical isomers, and its addition salts th... | 11/07/1995 |
| 5463126 | Process for preparing sertraline The invention provides the substantially geometrically pure cis-stereoisomeric form of a compound of formula (I) and the substantially geometrically and optically pure cis-stereoisomeric form of a compound of formula (II): ##STR1## wherein R | 10/31/1995 |
| 5442116 | Process for preparing sertraline intermediates The invention provides the substantially geometrically and optically pure trans-stereoisomeric form of a compound of formula (I): ##STR1## wherein R1 is H or C1 -C4 alkyl, together with processes for its preparation. ... | 08/15/1995 |
| 5434190 | N-aryl and N-cycloalkyl neoalkanamide insect repellents N-monosubstituted neoalkanamides of 11 to 14 carbon atoms wherein the substituent on the amide nitrogen is cyclic (aromatic or cycloaliphatic, such as aryl or cycloalkyl) and of at least five carbon atoms, have been discovered to be insect repellent, prov... | 07/18/1995 |
| 5414017 | Trifluoromethyl mercaptan and mercaptoacyl derivatives and method of using same Compounds of the formula ##STR1## wherein m is zero or 1; n is zero, 1 or 2; p is zero or 1 to 6 provided that m and p are not both zero; R3 is hydrogen, acyl, or benzyl; and R1 is hydrogen, alkyl, phenyl, substituted phenyl, ph... | 05/09/1995 |
| 5411989 | Nitric acid esters of cyclohexanol derivatives The invention concerns nitric acid esters of cyclohexanol of formula I ##STR1## in which A signifies a valency bond or a C1 -C6 -alkylene chain and B the group --NR1 --CO--Z, --NR1 --SO2 --Z or -... | 05/02/1995 |
| 5403853 | Substituted N-aryl-1,2-diaminocyclobutene-3,4-diones The compounds of the formula: ##STR1## wherein R1 and R2 are, independently, hydrogen, straight or branched chain alkyl or mono- or bi-cyclic alkyl; A is a substituted phenyl group containing one or two substituents selected fro... | 04/04/1995 |
| 5338884 | Method for the preparation of arylalkanolamineacylates Acylamides or amine acylate salts of arylalkanolamines are prepared by reacting an arylisonitrosoalkanone with hydrogen and a carboxylic acid, carboxylic acid anhydride or carboxylic acid ester or mixture thereof in the presence of a transition metal cata... | 08/16/1994 |
| 5292952 | Process for producing 2-fluoro-4-(trifluoromethyl) acetanilide Disclosed is a process for producing 2-fluoro-4-(trifluoromethyl) acetanilide which comprises reacting 3,4-difluorobenzotrifluoride with acetamide in the presence of a base in an aprotic polar solvent or in a mixture of an aprotic polar solvent and an apr... | 03/08/1994 |
| 5292938 | Synthesis of 4-substituted-trans-1, 2-diaminocyclohexyl polyaminocarboxylate metal chelating agents for the preparation of stable radiometal antibody immunoconjugates for therapy and spect and pet imaging Cyclo agents useful in forming antibody-metal conjugates useful for diagnostic and therapeutic purposes. New compounds and processes of forming these compounds are disclosed including 4-haloacetamido-trans-1,2-diaminocyclohexyl polyaminocarboxylate and ... | 03/08/1994 |
| 5254732 | N-fluorosulfonimides and their application as fluorinating agents The invention describes N-fluorosulfonimides which are useful as fluorinating agents. The N-fluorosulfonimides are stable, easily synthesized, and allow the introduction of fluorine into organic compounds under mild conditions.... | 10/19/1993 |
| 5243080 | Method of fluorinating by using N-fluoropyridinium pyridine heptafluorodiborate The present invention provides a novel compound represented as ##STR1## The present novel compound is prepared by reacting fluorine with pyridine-boron trifluoride and is useful as a fluorinating agent in the fluorination of organic compounds.... | 09/07/1993 |
| 5221769 | Production of p-acetylaminophenol from p-aminophenyl acetate p-Aminophenyl acetate is isomerized to p-acetylaminophenol in the presence of an acid such as acetic acid or phosphoric acid.... | 06/22/1993 |
| 5107022 | Process for the preparation of aromatic amines The invention relates to a process for the preparation of compounds of formula ##STR1## wherein R is unsubstituted or substituted C1 -C4 alkyl or unsubstituted or substituted phenyl, X is hydrogen or unsubstituted or substi... | 04/21/1992 |
| 5086060 | Compound and method for treating skin for acne or psoriasis The effects of acne and psoriasis are relived by applying either topically or by oral adminstration, a compound having the structure: ##STR1## wherein R1, R2, R3, R4 and R5 are independently sele... | 02/04/1992 |
