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| Number | Title | Issue Date |
| 7939690 | Haloalkylsulfone substituted compounds useful for treating obesity and diabetes The present invention relates to novel compounds of formula [I], wherein R1 represents heteroaryl, at least one substituent among R5, R6 and R7 represent —SR12, —S(O)R12 or —S(O)2R | 05/10/2011 |
| 7605289 | Benzamide derivatives and uses related thereto Benzamide derivatives of formula I and II, and pharmaceutically acceptable salts, solvates, stereoisomers, and prodrugs thereof, and pharmaceutical compositions comprising the same, are described and have therapeutic utility, particularly in the treatment of diabete... | 10/20/2009 |
| 7332629 | Modulators (inhibitors/activators) of histone acetyltransferases Disclosed are compounds of the formulae: and method of using the compounds to treat cancer, AIDS, HIV infection, and asthma. ... | 02/19/2008 |
| 7188055 | Method, system, and computer program for displaying chemical data A system, method, and computer program product for visualizing and interactively analyzing data relating to chemical compounds. A user selects a plurality of compounds to map, and also selects a method for evaluating similarity/dissimilarity between the selected com... | 03/06/2007 |
| 7141385 | Microcantilever apparatus and methods for detection of enzymes, enzyme substrates, and enzyme effectors An apparatus and a method are provided for detecting an enzyme, or or for detecting a substrate of an enzyme or for detecting an enzyme effector such as an inhibitor, by measuring a change in deflection of a microcantilever having a substrate or an enzyme, respectiv... | 11/28/2006 |
| 7126027 | N-[(1-dimethylaminocycloalkyl)methyl]benzamide derivatives The present invention relates to N-[(1-dimethylaminocycloalkyl)methyl]benzamide derivatives having the general formula I wherein n is 0, 1, 2 or 3; R1 and R2 are independently H, (C1-4 | 10/24/2006 |
| 7054757 | Method, system, and computer program product for analyzing combinatorial libraries The invention provides for in silico analysis of a virtual combinatorial library. Mapping coordinates for a training subset of products in the combinatorial library, and features of their building blocks, are obtained. A supervised machine learning approach is used ... | 05/30/2006 |
| 7041702 | Pharmaceutically active compounds and methods of use The present invention relates to pharmaceutically acceptable compounds, including acylguanidine compounds, and methods of treatment and pharmaceutical compositions that utilize or comprise one or more such compounds. Compounds of the invention are particularly usefu... | 05/09/2006 |
| 7039621 | System, method, and computer program product for representing object relationships in a multidimensional space A method and computer product is presented for mapping n-dimensional input patterns into an m-dimensional space so as to preserve relationships that may exist in the n-dimensional space. A subset of the input patterns is chosen and mapped into the m-dimensional spac... | 05/02/2006 |
| 6900344 | Method of preparing alkylated salicylamides via a dicarboxylate intermediate The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for ... | 05/31/2005 |
| 6576660 | Methods and compositions for regulation of 5--reductase activity Compounds that inhibit 5-alpha-reductase are provided. The compounds are used to treat prostate cancer, breast cancer, obesity, skin disorders and baldness.... | 06/10/2003 |
| 6566394 | Salicylamide derivatives Salicylamide derivatives represented by formulae (1a) and (1b); intermediates in the production thereof; a process for producing the same; and drugs containing the same as the active ingredient. The salicylamide derivatives represented by formulae (1a) an... | 05/20/2003 |
| 6506937 | Substituted benzenesulfonylureas and -thioureas-processes for their preparation and their use as pharmaceuticals Benzenesulfonylureas and -thioureas of the formula I ##STR1## where R(1) is H or (fluoro)methyl, R(2) is H, Hal or (fluoro) (mercapto)alk(oxy)yl, E is O or S; Y is --[CR(3)2 ]n --, where R(3)=H or alkyl and n=1-4, X is H, Hal or alky... | 01/14/2003 |
| 6462234 | Process to prepare (2S)-2-(dipropylamino)-6-ethoxy-2, 3-dihydro-1H-indene-5-carboxamide The present invention is a process, including intermediates, to produce (2S)-2-dipropylamino)-6-ethoxy-2,3-dihydro-1H-indene-5-carboxamide ##STR1## which is a useful pharmaceutical agent.... | 10/08/2002 |
| 6313088 | 8-[(2-hydroxy-4-methoxy benzoyl) amino]-octanoic acid compositions for delivering active agents Carrier compounds and compositions therewith which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well.... | 11/06/2001 |
| 6288265 | Phloroglucidic acid and derivatives as antibacterial agents A series of phloroglucide derivatives are synthesized, which possess potent antibacterial activities. They include unsymmetrical phloroglucide analogs, phloroglucides attached to cephalosporins at the C-3' position, and 7-(phloroglucidamido)cephalosporins... | 09/11/2001 |
| 6153651 | Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them. Ortho-substituted benzoylguanidines of the formula I ##STR1## in which R(1) to R(4) have the meanings given in the... | 11/28/2000 |
| 6090981 | Substituted benzenesulfonylureas and -thioureas--process for their preparation and their use as pharmaceuticals Benzenesulfonylureas and -thioureas of the formula I ##STR1## where R(1) is H or (fluoro)methyl, R(2) is H, Hal or (fluoro)(mercapto)alk(ozy)yl, E is O or S; Y is --[CR(3)2 ]n --, where R(3)=H or alkyl and n=1-4, X is H, Hal or ... | 07/18/2000 |
| 6054457 | Benzamide derivatives and their use as vasopressin antagonists This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkoxy, etc., R2 is lower... | 04/25/2000 |
| 6043232 | Nitroso esters of beta-oxo-amides and aryl propionic acid derivatives of non-steroidal antiinflammatory drugs A compound comprising a non-steroidal antiinflammatory agent to which is directly or indirectly linked an NO group, a compound comprising an enolic anilide non-steroidal antiinflammatory agent to which is directly or indirectly linked an NO2 gr... | 03/28/2000 |
| 6004823 | Compounds The present invention relates to libraries of compounds based upon a N-(4-alkoxyphenyl)-N-acyl-benzylamine, N-(4-alkoxyphenylmethyl)-N-acyl-benzylamine and N-[2-(4-alkoxyphenyl)ethyl]-N-acyl-benzylamine template, to processes for the preparation of s... | 12/21/1999 |
| 5908960 | Compounds The present invention relates to libraries of compounds based upon a N-benzyl-N-alkyl-4-alkoxybenzamide, N-benzyl-N-alkyl-4-alkoxyphenylacetamide and N-benzyl-N-alkyl-3-(4-alkoxyphenyl)propionamide template to processes for the preparation of such li... | 06/01/1999 |
| 5747539 | Fluorine-containing benzoylguanidines Fluorine-containing benzoylguanidines of the formula I ##STR1## in which R1, R2 and R3 have the meanings indicated, and their physiologically acceptable salts, have antiarrhythmic properties and act as inhibitors of t... | 05/05/1998 |
| 5747541 | Substituted benzoylguanidines, a process for their preparation, their use as medicament of diagnostic agent, and medicament comprising them The present invention relates to substituted benzoylguanidines, a process for their preparation, their use as medicament or diagnostic agent, and medicament comprising them.... | 05/05/1998 |
| 5683705 | Sulfur-based amides and bis-amides useful against skin disorders Novel sulfhydryl group-containing amides and disulfide group-containing bis-amides useful for treating or preventing an abnormal biological condition or a disease, and/or improving the texture or appearance of the skin, as well as compositions containing ... | 11/04/1997 |
| 5646184 | Preparation for external application to the skin and novel benzoic acid derivatives Disclosed is a preparation for external application to the skin characterized by containing at least one of benzoic acid derivatives represented by formula (I) or pharmacologically acceptable salts thereof as an active ingredient, the preparation having s... | 07/08/1997 |
| 5637121 | Poly(oxyalkylene) aromatic amides and fuel compositions containing the same Poly(oxyalkylene) aromatic amides having the formula: ##STR1## or a fuel-soluble salt thereof; wherein a is hydroxy, nitro, amino, N-alkylamino wherein the alkyl group contains 1 to 6 carbon atoms, or N,N-dialkylamino wherein each alkyl group indepen... | 06/10/1997 |
| 5591776 | Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV Rolipram-based PDE IV inhibitors containing phenyl- or benzyl-substituted moieties of the formula: ##STR1## wherein X1 and X2 may be the same or different and each is O or S; R1 is selected from the group consisting o... | 01/07/1997 |
| 5543572 | Monocarboxamides of polyamines Monocarboxamides of formula I ##STR1## wherein R is a radical of formula ##STR2## C9 -C19 alkyl, C9 -C19 alkenyl or C9 -C19 alkdienyl, wherein each R2 independently of... | 08/06/1996 |
| 5426224 | Mammalian DNA topoisomerase II inhibitor and method A novel antiproliferative drug and methods are disclosed. The drug has the general structural formula: ##STR1## where R1=OR1 ', SR1 ', or N(R1 'R1 ")2, where R1 ' and R1 " a... | 06/20/1995 |
| 5416118 | Bicyclic amides as inhibitors of acyl-coenzyme A: cholesterol acyl transferase Novel bicyclic amides of the formula ##STR1## wherein Ar1 and Ar2 are phenyl, R2 -substituted phenyl, heteroaryl or R2 -substituted heteroaryl, wherein R2 is 1 to 3 substituents independently sel... | 05/16/1995 |
| 5393776 | Tocotrienol analogs in the treatment of hypercholesterolemia and hyperlipidemia This invention relates to structurally novel acyclic tocotrienol analogs, which are useful for cholesterol/lipid lowering in cases of hypercholesterolemia and hyperlipidemia, and for atherosclerosis. Also provided are pharmaceutical compositions and a met... | 02/28/1995 |
| 5326898 | Substituted phenylethenyl compounds having retinoid-like biological activity Compounds of the formula ##STR1## wherein R1, R2, R3 and R4 independently are hydrogen, lower alkyl of 1 to 6 carbons, halogen or lower alkoxy of 1 to 6 carbons; R5 and R5 ' independen... | 07/05/1994 |
| 5283359 | Process for preparing albuterol, acetal, hemi-acetal, and hydrates of arylglyoxal intermediates thereof The preparation of arylethanolamines, and in particular albuterol (salbutamol), together with their novel boron, acetal and hemi-acetal intermediates is described.... | 02/01/1994 |
| 5233082 | Method of making 3-hydroxy-2,4,5-trifluorobenzoic acid Disclosed is a method of making 3-hydroxy-2,4,5-trifluorobenzoic acid. A aqueous solution is prepared of an alkali metal base and a tetrafluorophthalimide. The solution is heated to produce a mixture of a salt of a 4-hydroxy-3,5,6-trifluorophthalamic acid... | 08/03/1993 |
| 5223645 | Unsaturated phenone derivatives and their use as contact adhesives Unsaturated phenone derivatives of the general formula I ##STR1## where R1 is C1 -C4 -alkyl, cyclopropyl, cyclopentyl, cyclohexyl, indanonyl, tetralonyl, phenyl or phenyl in which some or all of the hydrogen atoms have bee... | 06/29/1993 |
| 5183828 | Polyhydroxybenzoic acid derivatives Polyhydroxy-substituted benz, phenylacet and mandelamidines, amidates, amidoximes and hydroxyamidoximes--ribonucleotide reductase inhibitors, and free radical scavengers.... | 02/02/1993 |
| 5155271 | Process for the alkylation of aromatic amines The invention relates to a process for the preparation of compounds of the formula ##STR1## in which Q is substituted or unsubstituted C1 -C6 alkyl, A is a direct bond or a bridging member, s is the number 1 or 2, Z is a radical... | 10/13/1992 |
| 5155106 | Cysteamine derivatives and antirheumatic agents containing cysteamine derivatives A cysteamine derivative represented by general formula (I): ##STR1## wherein R1 represents a straight-chain or a branched alkyl radical having 1 to 6 carbon atoms, R2 represents hydrogen atom or n-propyl radical, and X represent... | 10/13/1992 |
| 5089158 | Additives for lubricating oils and processes for producing them The invention provides oil-soluble multivalent metal ion salts of a compound of the formula XNR1 R2, in which R1 and R2 are the same or different and each are selected from hydrogen and hydrocarbon based radical... | 02/18/1992 |
