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| Number | Title | Issue Date |
| 7868205 | Inhibitors of histone deacetylase The invention relates to the inhibition of histone deacetylase. The invention provides compounds and methods for inhibiting histone deacetylase enzymatic activity. The invention also provides compositions and methods for treating cell proliferative diseases and cond... | 01/11/2011 |
| 7803970 | Multi-substitued selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a... | 09/28/2010 |
| 7772433 | SARMS and method of use thereof This invention provides SARM compounds and uses thereof in treating a variety of diseases or conditions in a subject, including, inter-alia, muscle wasting diseases and/or disorders, bone-related diseases and/or disorders, diabetes, cardiovascular disease, renal dis... | 08/10/2010 |
| 7705182 | Multi-substituted selective androgen receptor modulators and methods of use thereof This invention provides androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and anabolic act... | 04/27/2010 |
| 7576239 | Substituted amides Novel compounds of the structural formula (I) are antagonists and/or inverse agonists of the Cannabinoid-1 (CB1) receptor and are useful in the treatment, prevention and suppression of diseases mediated by the CB1 receptor. The compounds of the present invention are... | 08/18/2009 |
| 7420090 | Fungicides Fungicidal compounds of the general formula (1): wherein X, Y and Z are independently H, halogen, C1-4 alkyl, halo(C1-4)alkyl, C2-4alkenyl, halo(C2-4)alkenyl, C24 alkynyl, halo(C2-4)alkynyl, C1-4... | 09/02/2008 |
| 7358396 | Preparation of optically active amines A process for preparing optically active amines, a process for preparing racemic amines which can be resolved using optically active carboxylic acids or enzymes, and racemic and optically active amines and optically active amides are described. ... | 04/15/2008 |
| 7271289 | Biphenylcarboxylic amide derivatives as p38 kinase inhibitors Compounds of formula (I): or pharmaceutically acceptable derivatives thereof, and their use as pharmaceuticals, particularly as p38 kinase inhibitors. ... | 09/18/2007 |
| 7253318 | Benzyloxy derivatives as MAOB inhibitors The invention relates to compounds of the formula and their pharmaceutically acceptable salts wherein R1, R2, R3, R4, R5, n, m, and o are... | 08/07/2007 |
| 7105545 | N-p-propargyloxyphenethyl-thioacetic acid amides The invention relates to N-propargyloxy-phenethyl thioacetic acid amide derivatives of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R | 09/12/2006 |
| 7034015 | Aminobenzoephenones The invention relates to a novel class of aminobenzophenones derivatives, to pharmaceutical preparations comprising said compounds, to dosage units of such preparations, to methods of treating patients comprising administering said compounds, and to the use of said ... | 04/25/2006 |
| 7026500 | Halogenated selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a... | 04/11/2006 |
| 6998500 | Selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a... | 02/14/2006 |
| 6683211 | Phenyl-propargylether derivatives The invention relates to phenyl-propargylether derivatives of the general formula I ##STR1## including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R... | 01/27/2004 |
| 6083987 | Phenylenediamine derivative, radical scavenger, brain-infarction depressant, and brain-edema depressant A phenylenediamine derivative or a salt thereof in accordance with the present invention is expressed by the following formula 1: ##STR1## wherein A represents a group expressed by --CO--, --CH2 CO--, --CS--, or --SO2 --; Y repr... | 07/04/2000 |
| 5855629 | Alkoxy acetic acid derivatives This invention provides alkoxy acetic acid derivatives of general formula I: ##STR1## wherein R is the residue of an amine, an aminoalcohol or a polyol linked to the or each --CHR'--CO-- moiety via an amide or ester linkage; R' is hydrogen or a C | 01/05/1999 |
| 5728737 | N-alkoxy-amidine derivatives The present invention relates to novel N-alkoxy-arnidine derivatives of the formula (I), to a process for their preparation and to their use as pesticides. In addition, the invention also relates to novel intermediates and to a process for their preparati... | 03/17/1998 |
| 5686633 | Inks, particularly for ink jet printing Inks, particularly inks for ink jet printing, contain at least one compound of the formula I ##STR1## as a stabilizer. The symbols R1, R2, R3, R4, R3 ' and R4 ' are as defined in claim... | 11/11/1997 |
| 5663434 | Process for preparing N-(3-amino-4-chlorophenyl) acylamides The present invention provides a process for preparing N-(3-amino-4-chlorophenyl) acylamides of Formula I: ##STR1## comprising reacting, in a solvent comprising at least one polar solvent, in the presence of at least one acid acceptor, 1-chloro-2,4-d... | 09/02/1997 |
| 5430060 | Acetamide derivatives The invention concerns novel N-phenylacetyl and related acyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, ... | 07/04/1995 |
| 5393776 | Tocotrienol analogs in the treatment of hypercholesterolemia and hyperlipidemia This invention relates to structurally novel acyclic tocotrienol analogs, which are useful for cholesterol/lipid lowering in cases of hypercholesterolemia and hyperlipidemia, and for atherosclerosis. Also provided are pharmaceutical compositions and a met... | 02/28/1995 |
| 5270343 | Penta-2,4-dienamides and use as pesticides The present Application discloses pesticidally active compounds of formula (I): Q(CH2)a (O)b Q1 CR2 .dbd.CR2 .dbd.CR3 CR4 .dbd.CR5 CXNR1 Rx... | 12/14/1993 |
| 5270342 | Acetamide derivatives The invention concerns novel N-phenylacetyl and related acyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, ... | 12/14/1993 |
| 5250570 | Amidobenzene derivatives, compositions and use The invention concerns novel phenoxy- and phenylthio-acetyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, i... | 10/05/1993 |
| 5235092 | Phenoxyacetic acid derivatives and plant growth regulating agents containing them as active ingredients A phenoxycetic acid derivative of the formula: ##STR1## wherein R is a hydroxyl group, an alkoxy group, a group of the formula OM wherein M is an alkali metal ion, an alkaline earth metal ion, a transition metal ion, an ammonium ion or an organic amm... | 08/10/1993 |
| 5155271 | Process for the alkylation of aromatic amines The invention relates to a process for the preparation of compounds of the formula ##STR1## in which Q is substituted or unsubstituted C1 -C6 alkyl, A is a direct bond or a bridging member, s is the number 1 or 2, Z is a radical... | 10/13/1992 |
| 5098613 | Anti-inflammatory agents This invention provides benzene derivatives, pharmaceutical formulations of those derivatives, and a method of using the derivatives for the treatment of inflammation in mammals.... | 03/24/1992 |
| 5064861 | Acylated amine compounds which are useful fungicigal agents A compound selected from the group consisting of a compound of the formula ##STR1## wherein R1 is selected from the group consisting of Ar-O- and aryl, polyaryl and condensed polyaryl unsubstituted or substituted and heterocycle unsubstitu... | 11/12/1991 |
| 5041653 | Substituted benzamide radiosensitizers A method for sensitizing hypoxic tumor cells to radiation using derivatives of benzamide are disclosed. Some of the compounds useful in the method of the invention are novel.... | 08/20/1991 |
| 4948812 | 1-phenoxy-3-amino-2-propanols use thereof Compounds of formula ##STR1## (the substituents R1, R2, R3, R4 and R5 are explained in the specification) may be prepared by conventional methods. Owing to their favorable activity profile the compoun... | 08/14/1990 |
| 4929273 | N-benzyl-2-(4-fluoro-3-trifluoromethylphenoxy)butanoic amide and herbicidal composition containing the same There are disclosed N-benzyl-2-(4-fluoro-3-trifluoromethylphenoxy)butanoic amide represented by the formula: ##STR1## and a herbidical composition containing the same as an active ingredient.... | 05/29/1990 |
| 4882357 | Novel N-(substituted-phenyl)-5-(substituted-2,5-dimethylphenoxy)-2,2-dimethylp entanamides Novel N-(substituted-phenyl)-5-(substituted-2,5-dimethylphenoxy)-2,2-dimethylpen tan amides which are useful in preventing the intestinal absorption of cholesterol and also increasing high-density lipoprotein (HDL) cholesterol, as well as novel pharma... | 11/21/1989 |
| 4845264 | Phenoxycarboxylic acid and herbicide comprising it as active ingredient A novel phenoxycarboxylic acid of formula (I) is disclosed. The compound is effective as herbicide for eradicating broad-leaved weeds. A combination of the phenoxycarboxylic acid and a N-phosphonomethylglycine or a glufosinate which is known as a herbicid... | 07/04/1989 |
| 4753674 | Herbicidal composition containing a phenoxyalkylamide derivative and method for controlling weeds by the use of the same There are disclosed a herbicidal composition containing, as an active ingredient, a phenoxyalkylamide derivative represented by the formula ##STR1## wherein X, n, Y, Z, R1, R2 and R3 have the same meanings as defined ... | 06/28/1988 |
| 4677122 | Substituted trans-1,2-diaminocyclohexyl amide compounds Substituted trans-1,2-diaminocyclohexyl amide compounds demonstrating selective opioid receptor binding possess utility as analgesic, diuretic, and psychotherapeutic agents. A method of preparing the compounds, pharmaceutical compositions employing the co... | 06/30/1987 |
| 4554282 | Substituted 2,2-dimethyl-5-phenoxypentanoic acid benzamides as anti-arteriosclerotic agents and method New substituted 2,2-dimethyl-5-phenoxypentanoic acid benzamides which are useful as anti-arteriosclerotic agents are disclosed. These compounds elevate the high density lipoprotein fraction of cholesterol, and also lower the low density lipoprotein fracti... | 11/19/1985 |
| 4531969 | Herbicidal esters of D-1-(phenoxy-4-phenoxy)propionic acid Optically active enantiomers of the formula I ##STR1## where R is a group of the formulae ##STR2## R1 and R2, among others, are halogen or CF3 and Z is a carboxyl, carboxylate, carboxylic acid ester, thioester, c... | 07/30/1985 |
| 4487953 | 9-Bromoprostaglandins, their preparation, and their use as medicaments Compounds of Formula (I) ##STR1## wherein the 9-bromine atom can be in the - or ଲ-position, R1 is CH2 OH or C(O)OR2, wherein R2 is hydrogen, alkyl, cycloalkyl, aryl, or a heterocyclic residue; or R | 12/11/1984 |
| 4465507 | Herbicidal acetanilides A tri- or tetra-substituted phenoxy alkylene- or alkenylene-anilide compound represented by the following formula ##STR1## wherein R, R1, R2, X, Y, l, m and n are as defined in claim 1; a process for producing the aforesaid anil... | 08/14/1984 |
| 4454339 | 9-Fluoroprostaglandin derivatives, and use as medicinal agents 9-Fluoroprostane derivatives of Formula I ##STR1## wherein R1 is CH2 OH or ##STR2## wherein R2 is hydrogen, alkyl, cycloalkyl, aryl, or a heterocyclic residue; or R1 is the residue ##STR3## ... | 06/12/1984 |
