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| Number | Title | Issue Date |
| 7576238 | Process for the preparation of substituted tetralin and substituted indane derivatives The present invention relates to novel processes for the preparation of substituted tetralin and substituted indane derivatives. The present invention is further directed to novel processes for the preparation of intermediates in the preparation of the substituted t... | 08/18/2009 |
| 7351857 | Methods of using substituted tetralins and indanes The invention features tetralin and indane compounds, compositions containing them, and methods of using them as PPAR alpha modulators to treat or inhibit the progression of, for example, diabetes. ... | 04/01/2008 |
| 6921774 | Compounds and their use as glycine transport inhibitors The invention provides novel compounds of the formula I below: wherein the meaning of each substituent is defined in the application. The compounds are useful as inhibitors of the glycine transporter and useful in the ... | 07/26/2005 |
| 6576664 | Inhibitors of aggrecanase and matrix metalloproteinases for the treatment of arthritis This invention relates to molecules which inhibit metalloproteinases, including aggrecanase, and the production of tumor necrosis factor (TNF). In particular, the compounds are inhibitors of metalloproteinases involved in tissue degradation and inhibitors... | 06/10/2003 |
| 6479646 | Metallocene compounds having indenyl ligand and catalysts for olefin polymerization containing the same A metallocene compound having an indenyl ligand substituted by a heteroaromatic group, which is useful as an olefin polymerization catalyst. The metallocene compound has the following structure ##STR1## wherein M is a transition metal atom; each Ra is a m... | 11/12/2002 |
| 6472430 | Amino thioxomethyl amino oxyacetic acid derivatives Antiatherosclerotic compounds are provided which have the following structure: ##STR1## wherein R is lower alkyl; R1 is hydroxy, amino, or lower alkoxy, R2 and R3 are each independently hydrogen, alkyl or aryl; Ar is phenyl, in... | 10/29/2002 |
| 6355836 | Process for the preparation of cis 5-fluoro-2-methyl-1[p-(methylthio)benzyliden]-inden-3-acetic acid An isomerization process of trans-5-fluoro-2-methyl-1-[p-(methylthio)benzyliden]inden-3-acetic acid for the treatment of sodium salt in methanol and in the presence of a base at 70&#b1;2° C. is described.... | 03/12/2002 |
| 6344585 | Preparation process of fluorenes A tetrahydrofluorene, which is represented by the following formula (I) ##STR1## wherein R1 to R6 each independently represent a hydrogen atom or an alkyl group having 1 to 4 carbon atoms, or R1 and R2 are combi... | 02/05/2002 |
| 6214876 | Indene-1-acetamide sPLA2 inhibitors Indene-1-acetamide compounds of the general formula (I) below; ##STR1## inhibit sPLA2 mediated release of fatty acids and are useful for treatment of conditions such as septic shock.... | 04/10/2001 |
| 6172259 | Production of enantiomer-free biarylketocarboxylic acids The invention relates to a continuous process for the preparation of enantiomerically pure biarylketocarboxylic acids, S-phenylethylamine being employed as an auxiliary base in the resolution. Biarylketocarboxylic acids, in particular substituted biaryl-4... | 01/09/2001 |
| 6172109 | 13-Thia prostaglandins for use in glaucoma therapy 13-thia prostaglandins are useful in the treatment of glaucoma and ocular hypertension. Also disclosed are ophthalmic, pharmaceutical compositions comprising said prostaglandins.... | 01/09/2001 |
| 6156750 | Bioactive bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof Novel pharmaceutically/cosmetically-active bicyclic aromatic compounds have the structural formula (I): ##STR1## and are useful for the treatment of a wide variety of disease states, whether human or veterinary, for example dermatological, rheumatic,... | 12/05/2000 |
| 6063807 | Cyclo-oxygenase inhibitor and amidine derivatives salts, preparation method therefor, use thereof as drugs, and pharmaceutical compositions containing said salts Cyclo-oxygenase inhibitor and amidine derivative salts, preparation methods therefor, pharmaceutical compositions containing said salts and the use thereof particularly as NO synthase and cyclo-oxygenase inhibitors, are disclosed.... | 05/16/2000 |
| 6020379 | Position 7 substituted indenyl-3-acetic acid derivatives and amides thereof for the treatment of neoplasia In position 7 substituted indenyl-3-acetic acid derivatives and pharmaceutically acceptable salts and amides thereof have anti-neoplastic activity.... | 02/01/2000 |
| 5908851 | Derivatives of succinamide and their use as metalloproteinase inhibitor Compounds of formula (I), ##STR1## wherein X is a --CO2 H or --CONHOH group; R4 is a group --CHRx Ry wherein Rx and Ry independently represent optionally substituted phenyl or monocycl... | 06/01/1999 |
| 5837807 | Tetrahydronaphthalene compounds This invention is directed to tetrahydronaphthalene compounds of the formula ##STR1## wherein R1 is hydrogen, bromine, cyano, formyl, hydroxy, lower alkyl, lower alkenyl, lower alkynyl, lower alkoxy, aryloxy, lower aralkoxy or aryl; R... | 11/17/1998 |
| 5750558 | Oxime derivatives of indole and indene compounds as inhibitors of prostaglandin biosynthesis Described herein are compounds having the formula ##STR1## or a pharmaceutically acceptable salt thereof wherein L is selected from the group consisting of ##STR2## R2 is selected from (a) ##STR3## R3 is selected ... | 05/12/1998 |
| 5719182 | Endothelin receptor anatagonists Novel indane and indene derivatives are described which are endothelin receptor antagonists.... | 02/17/1998 |
| 5712377 | Glycosides isolated from pollen, their sugar-free decomposition products and derivatives thereof What are described are new glucosides and their sugar-free decomposition products, as well as synthetically produced derivatives, which can be used as active components of pharmaceutical compositions. The novel glucosides have been isolated from aqueous e... | 01/27/1998 |
| 5578629 | Benzamide-containing inhibitors of farnesyl-protein transferase The present invention comprises peptidomimetic compounds which comprise a suitably substituted aminoalkylbenzamide moiety. The instant compounds inhibit the farnesyl protein transferase enzyme and the farnesylation of certain proteins. Furthermore, the in... | 11/26/1996 |
| 5470832 | Inhibitors of geranylgeranyl-protein transferase The compounds disclosed am analogs of the CAAX motif of proteins that can be modified by geranylgeranylation in vivo that selectively inhibit the geranylgeranylation of several proteins. The relatively poor activity of the compounds against the farnesyl p... | 11/28/1995 |
| 5459134 | (Fused) benz (thio) amides A novel (fused) benz(thio)amide of the general formula: ##STR1## or a non-toxic salt thereof, wherein R4 represents: (i) when B represents a closed ring, a group of the general formula: ##STR2## wherein U represents an oxygen atom or a sul... | 10/17/1995 |
| 5409956 | Indan derivative and thromboxane antagonist containing the same The present invention relates to indan derivatives represented by the formula (1) or pharmaceutically acceptable salts thereof: ##STR1## [wherein R1 represents C1 to C12 alkyl, benzyl, styryl, naphthyl, optionally substituted phenyl or opt... | 04/25/1995 |
| 5399748 | Derivatives of aspartic acid and glutamic acid having anticholecystokinin activity Arylsulfonamide derivatives of -amino dicarboxylic acids such as aspartic acid and glutamic acid posses anti-cholecystokinin activity. They are useful in the treatment of cholecystokinin-related disorders such as anorexia nervosa, pancreatic inflam... | 03/21/1995 |
| 5385917 | Carboxylic acid derivatives Carboxylic acid derivatives of the formula: ##STR1## are provided, which are useful for treatment of androgen dependent diseases.... | 01/31/1995 |
| 5281626 | Benzenesulfonamide derivatives A novel benzenesulfonamide derivative represented by the formula: ##STR1## has an inhibitory activity against phospholipase A2, so that it is effective in the treatment of diseases for which such an activity is efficacious.... | 01/25/1994 |
| 5252601 | 2-mercaptomethylene-tetrahydronaphthalene and indane-2-carboxamide derivatives as enkephalinase inhibitors The present invention relates to novel 2-mercaptomethylene-tetrahydronaphthalene derivatives which are useful as enkephalinase inhibitors.... | 10/12/1993 |
| 5223529 | N-phenylamides and medicinal products containing them Compounds of formula: ##STR1## in which R1 is (a) a phenyl radical or a substituted phenyl radical, (b) a chain --CH(R8)--COOR4, (c) a chain --CH2 --CO--NR5 R6 or (d) a phenylalkyl rad... | 06/29/1993 |
| 5112868 | Hydroxamate derivatives of selected nonsteroidal antiinflammatory acyl residues having cyclooxygenase and 5-lipoxygenase inhibition The present invention is novel selected hydroxamic acid derivatives of acyl residues of selected NSAIDS, i.e. having 5-lipoxygenase and cyclooxygenase inhibiting properties, pharmaceutical compositions for treating conditions advantageously affected by th... | 05/12/1992 |
| 5081282 | Prostaglandins Bicyclo prostaglandin analogues have been prepared.... | 01/14/1992 |
| 5030653 | Antihyperlipidemic and antiatherosclerotic compounds and compositions Certain N-2,6-dialkyl- or N-2,6-dialkoxyphenyl-N'-arylalkylurea compounds are potent inhibitors of the enzyme acyl CoA:cholesterol acyltransferase (ACAT), and are thus useful agents for the treatment of hypercholesterolemia or atherosclerosis.... | 07/09/1991 |
| 5030652 | Indan derivatives and pharmaceutical preparation thereof Indan derivatives of the formula: ##STR1## wherein R1 is substituted or unsubstituted phenyl, naphthyl or sulfur-containing heterocyclic group, and R2 is hydroxy-methyl or a group of the formula: ##STR2## wherein R | 07/09/1991 |
| 4983628 | Leukotriene antagonists Compounds having the formula: ##STR1## are antagonists of leukotrienes of C4, D4 and E4, the slow reaction substance of anaphylaxis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory and c... | 01/08/1991 |
| 4980372 | Benzoylaminophenoxybutanoic acid derivatives A benzoylaminophenoxybutanoic acid derivative of general formula: ##STR1## [wherein R1 represents hydrogen atom or alkyl group of from 1 to 4 carbon atoms(s), A represents oxygen atom, sulfur atom or sulfinyl (SO) group, two R1 s ... | 12/25/1990 |
| 4975460 | Indanoxyacetic acid derivatives Novel indanoxyacetic acid derivatives of the formula: ##STR1## wherein R1 is a lower alkyl group, a substituted or unsubstituted phenyl group, naphtyl group or a sulfur-containing heterocyclic group, R2 is hydroxy group or a pro... | 12/04/1990 |
| 4963587 | Glycine derivative and pharmaceutical preparation thereof There are disclosed are glycine derivative of the formula: ##STR1## (wherein R1 represents a substituted or unsubstituted phenyl group, R2 represents a carboxyl group which may be protected, Q represents a lower alkylene group a... | 10/16/1990 |
| 4929754 | Benzenesulphonamidoindanyl compounds The invention relates to new benzenesulphonamidoindanyl compounds useful in the treatment and prophylaxis of thromboembolic diseases, arteriosclerosis and tumor metastasis.... | 05/29/1990 |
| 4868210 | Antihyperlipidemic and antiatherosclerotic compounds and compositions Certain N-2,6-dialkyl- or N-2,6-dialkoxyphenyl-N'-arylalkylurea compounds are potent inhibitors of the enzyme acyl CoA:cholesterol acyltransferase (ACAT), and are thus useful agents for the treatment of hypercholesterolemia or atherosclerosis.... | 09/19/1989 |
| 4820705 | Benzenesulphonamidoindanyl compounds, medicaments thereof, and processes of preparation The invention relates to new benzenesulphonamidoindanyl compounds having the following formula ##STR1## wherein the substituents are defined herein useful in the treatment and prophylaxis of thromboembolic diseases, arteriosclerosis and tumor me... | 04/11/1989 |
| 4783476 | 3-Phenoxy (or phenylthio)-cyclopentanecarbonylamino acid analogues This invention relates to compounds presented by the general formula: ##STR1## wherein R1 and R2 are: (i) R1, R2 and carbon atoms to which R1 and R2 are linked, together represent the group... | 11/08/1988 |
