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Class 560/49 - Nitrogen in alcohol moiety


Subclass of Class 560 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the alcohol moiety contains nitrogen covalently
No. of patents: 82
Last issue date: 05/13/2008


1      
NumberTitleIssue Date
7371831Azo dyestuffs
Compounds of formula (I) wherein all substituents have the meanings as defined in the Specification, their production and their use. ...
05/13/2008
7220749Nitrosated and/or nitrosylated cyclooxygenase-2 selective inhibitors, compositions and methods of use
The invention describes novel nitrosated and/or nitrosylated cyclooxygenase 2 (COX-2) selective inhibitors and novel compositions comprising at least one nitrosated and/or nitrosylated cyclooxygenase 2 (COX-2) selective inhibitor, and, optionally, at least one compo...
05/22/2007
7175834Sunscreen composition with enhanced SPF and water resistant properties
The present invention relates to a sunscreen formulation which exhibits superior ultraviolet protection and water resistance than prior art sunscreen compositions. The sunscreen formulation comprises (a) a dispersion comprising a sunscreen active agent and (b) a bas...
02/13/2007
7019104Diamine novel acid dianhydride and novel polyimide composition formed therefrom
An object of present invention is to provide a diamine and an acid dianhydride having photoreactivity and thermoreactivity and a polyimide composition containing the diamine and the acid dianhydride as monomer components, and specifically to synthesize a diamine and...
03/28/2006
6602869Compounds derived from benzoic acid esters, composition containing said compounds and use thereof
This invention relates to novel compounds of formula (I) wherein R1 represents a polymer, aryl or alkyl group, R2 represents a hydrogen atom, a halogen atom, a radical CN, CF3, OH, OCF3, COOH, R7, OR
08/05/2003
6576747Processes for preparing dianthranilate compounds and diazopyridone colorants
Disclosed is a process for preparing dianthranilate compounds which comprises (a) admixing reactants as follows: (1) a diol of the formula R1 (OH)2, wherein R1 is an alkylene group having at least about 20 carbon atoms, an...
06/10/2003
6262114Leukotriene B4 antagonist compounds and method for treatment
Novel amidinophenol derivatives of formula (IB) ##STR1## and processes for the preparation thereof; compositions containing a compound of formula (IB) as active ingredient useful as antagonists of leukotine B4 and inhibitors of phospholipase A
07/17/2001
6143734Nitroso esters of ଲ-oxo-amides and aryl propionic acid derivatives of non-steroidal antiinflammatory drugs
A compound comprising a non-steroidal antiinflammatory agent to which is directly or indirectly linked an NO group, a compound comprising an enolic anilide non-steroidal antiinflammatory agent to which is directly or indirectly linked an NO2 gr...
11/07/2000
6054457Benzamide derivatives and their use as vasopressin antagonists
This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkoxy, etc., R2 is lower...
04/25/2000
5985919(Het)aryloxy-, -thio- , aminocrotonates, methods of preparing them and their use as insecticides and fungicides
(Het)aryloxy-, -thio- and -aminocrotonates of the formula I ##STR1## where the substituents have the following meanings: U is oxygen, sulfur or amino; V is oxygen, sulfur, amino or alkylamino; X, Y and Z independently of one another are .dbd.N-- or .dbd.C...
11/16/1999
5948922Compounds with substituted cyclic hydrocarbon moieties linked by secondary or tertiary oxycarbonyl containing moiety providing reworkable cured thermosets
Compounds containing two cyclic hydrocarbon moieties which are substituted to provide crosslinking functionality and which are linked to each other by secondary or tertiary oxycarbonyl containing moiety are basis for compositions which are cured to provid...
09/07/1999
5861534Diaminobenzene derivatives and polyimides prepared therefrom
A diaminobenzene derivative of the formula (I): ##STR1## wherein each of P and Q which may be the same or different from each other, is a single bond, or a bivalent organic group selected from the group consisting of --O--, --COO-- and --CONH--, R
01/19/1999
5795890Sulfonamide derivatives
A sulfonamide derivatives of formula (I) ##STR1## a non-toxic salts, an acid addition salts or a solvates thereof which has an inhibitory effect on elastase....
08/18/1998
5783593Inhibitors of squalene synthetase and protein farnesyltransferase
The present invention provides a compound of the formula ##STR1## which inhibit squalene synthetase and cholesterol biosynthesis and are useful in the treatment of e.g., hyperlipidaemia, atherosclerosis, or fungal infections, processes for the prepar...
07/21/1998
5648513O-acyl serines
The invention relates to a method of suppressing human body malodor by utilizing a deodorant composition containing a competitive substrate for the enzymatic creation of axillary body malodor. The compound is present in a dermatologically acceptable vehic...
07/15/1997
5639746Hydroxamic acid-containing inhibitors of matrix metalloproteases
The invention provides hydroxamic acid-containing compounds which are useful as inhibitors of matrix metalloproteases and which are effective in treating conditions associated with excess activity of these enzymes. In particular, the present invention rel...
06/17/1997
5527689Enzymatic coupling of L-phenylalanine methyl ester and N-benzyloxycarbonyl-aspartic acid
The invention relates to a process for the preparation of N-benzyloxycarbonyl-଱-L-aspartyl-L-phenylalanine methyl ester by enzymatic coupling of N-benzyloxycarbonyl-L-aspartic acid and L-phenylalanine methyl ester in an aqueous medium with formation...
06/18/1996
5514794Antibody-drug conjugates
Derivatized drugs are prepared with a linker consisting of a malonate, wherein the drug is linked through a methylene to the 2-position carbon of the malonate....
05/07/1996
5453532Crystalline modification of 2-dimethylaminoethyl-n-butylaminobenzoate hydrochloride, method for production thereof and pharmaceutical preparation for anaesthesia of eyes, based thereon
A novel crystalline modification of 2-dimethylaminoethyl-n-butylaminobenzoate hydrochloride is characterized by a melting point of 148.6°&#b1;0.3° C. and has an interplanar spacing d and relative intensities defined herein, and a method for making ...
09/26/1995
5424474Fluorinated carboxylic acid esters of phosphono- and phosphinocarboxylic acids containing hydroxyl and/or mercapto groups, a method for their preparation, and their use
The present invention relates to fluorinated carboxylic acid esters of phosphono- and phosphinocarboxylic acids containing hydroxyl and/or mercapto groups, their use as waterproofing and/or oil-repellency agents, and a method for their preparation....
06/13/1995
5414102Fluorinated carboxylic acid esters of phosphono- and phosphinocarboxylic acids containing acrylate and/or methacrylate groups
The present invention relates to fluorinated carboxylic acid esters of phosphonocarboxylic acids containing acrylate and/or methacrylate groups, their use as waterproofing or oil-repellency agents, and a method for their preparation....
05/09/1995
5403951Crystalline modification of 2-dimethylaminoethyl-n-butylaminobenzoate hydrochloride, method for production thereof and pharmaceutical preparation for anaesthesia of eyes, based thereon
A novel crystalline modification of 2-dimethylaminoethyl-n-butylaminobenzoate hydrochloride and a method for production of said compound residing in that a solution of 2-dimethylaminoethyl-n-butylaminobenzoate hydrochloride of polymorphic form in wat...
04/04/1995
5395853Anti-atherosclerotic diaryl compounds
The present invention is concerned with compounds of formula (I) ##STR1## wherein m is 0 or 1; W is hydrogen, a C1-16 straight, branched, or cyclic alkyl group, or a C2-16 straight, branched, or cyclic alkenyl or alkynyl group, or Ph...
03/07/1995
5302743Preparation of N-protected .alpha.-L-aspartyl-L-phenylalanine methyl ester
Disclosed is an improved process for the preparation of an N-protected .alpha.-L-aspartyl-L-phenylalanine methyl ester from an N-protected L-aspartic anhydride and L-phenylalanine methyl ester, the improvement which comprises employing the L-phenylalanine...
04/12/1994
5298647Aromatic compounds of amide structure derived from aminobenzoic acids, hydroxy-benzoic acids, cinnamic acids, urocanic acids and benzimidazoles, absorbing UVB and/or UVA
Aromatic compounds absorbing UVB and/or UVA, substituted with an amide function, selected from the group consisting of ##STR1## whose variable substituents are as defined in the specification, e.g. ##STR2## are useful as photoprotective agents o...
03/29/1994
5290814Anti-atherosclerotic diaryl compounds
The present invention is concerned with compounds of formula (I) ##STR1## wherein m is 0 or 1; W is hydrogen, a C1-16 straight, branched, or cyclic alkyl group, or a C2-16 straight, branched, or cyclic alkenyl or alkynyl group, or ...
03/01/1994
5283258Procaine double salt complexes
A procaine acid addition salt, wherein the acid is attached to the diethylamino nitrogen, is complexed with a biologically active organic acid such as a vitamin acid, essential unsaturated fatty acid, C4 to C6 hydroxycarboxylic acid ...
02/01/1994
5218137Light activated acyl-enzymes
Light activated acyl-enzymes of the formula: ##STR1## are disclosed. In the compounds of Formula (III), ENZ is an enzyme, X is O or S, Y is --NR3 R4, --OR5, or --SR5, and Z is a nucleophile. m is 0 to 3 and...
06/08/1993
51029114-Substituted HMG-CoA reductase inhibitors
HMG-CoA reductase inhibitors of formulae (I) and (II) are disclosed. ##STR1##...
04/07/1992
5087726Carbamate ACAT inhibitors
This invention relates to novel compounds which are ACAT inhibitors rendering them useful in lowering blood cholesterol levels. The compounds are carbamates represented by the general formula ##STR1## wherein Ar and Ar' represent phenyl or naphthyl e...
02/11/1992
5073641Prodrug derivatives of carboxylic acid drugs
Novel ester derivatives of carboxylic acid medicaments of formula (I), wherein R--COO--represents the acyloxy residue of a carboxylic acid drug or medicament, n is an integrer from 1 to 3, and R1 and R2 are the same or different and ...
12/17/1991
5001148Mevinic acid derivatives
Antihypercholesterolemic activity, due to competitive inhibition of HMG CoA reductase, has been found in compounds of the formula ##STR1## wherein: R1, R2 and R3 are independently selected from: (1) alkyl, (2) substituted ...
03/19/1991
5001156Lipophilic quaternary ammonium salicylates, their use in cosmetics and in dermopharmacy
Lipophilic quaternary ammonium salicylate, characterized in that it corresponds to the formula: ##STR1## in which: (i) R1, R2, R3 and R4, which may be identical or different, denote an alkyl or alkylcycloal...
03/19/1991
4999186Novel sunscreen agents, sunscreen compositions and methods for preventing sunburn
The present invention relates to novel sunscreen agents which have the ability to absorb both UVA and UVB wavelength radiation. The sunscreen agents comprise a specific type of UVA-absorbing chromophore covalently bonded to a specific type of UVB-absorbin...
03/12/1991
4992575Process for the preparation of N,N'-dimethyl aromatic diamines, intermediates and products
N,N'-dimethyl aromatic diamines are prepared from the corresponding diprimary amines via a two step synthesis forming first the corresponding di-succinylimidomethylamine and then reductively cleaving the succinylimido group. The products are useful, e.g.,...
02/12/1991
4940813Resolution of a carboxylic acid
A process is described for the preparation of an optically active carboxylic acid or ester derivative thereof from a ketene and an optically active ଱-hydroxyester or an ଱-hydroxy amide....
07/10/1990
4937370Novel chromophores, sunscreen compositions and methods for preventing sunburn
The present invention relates to novel chromophore-containing compounds useful as sunscreen agents which have the ability to absorb both UVA and UVB wavelength radiation. These compounds comprise a specific type of UVA-absorbing chromophore covalently bon...
06/26/1990
4914223Acrylamidoacylated oligomers
A composition of matter comprising an acrylamido-acyl or methacrylamido-acyl oligomer derived from at least one nucleophilic oligomer having at least one amino-, hydroxyl-, or thio-substituted polyoxyalkylene, polyalkyleneimine, polyester, polyolefin, pol...
04/03/1990
4894181Carbocyclic compounds
Carbocyclic compounds of the formula I ##STR1## wherein Q is a benzene or cyclohexane ring or a naphthalene system, X is in each case --CH2 --(CH2)p -- where it is also possible for one or two non-adjacent CH2
01/16/1990
4851562Aromatic amide groups-containing diamines and polymers in which these diamines are incorporated
There is provided a new class of diamines of the formula ##STR1## wherein X=NH or O, and R represents a divalent, substituted or unsubstituted organic group having at the most 20 carbon atoms. The diamines, wherein X has the meaning of an O-atom, may be c...
07/25/1989
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