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| Number | Title | Issue Date |
| 8049031 | Solid forms of fesoterodine fumarate New solid forms of fesoterodine fumarate are described. In particular, amorphous fesoterodine fumarate, characterized by a powder X-ray diffraction spectrum as shown in FIG. 1 and by an IR spectrum as shown in FIG. 2 is described. Also fesoterodine fum... | 11/01/2011 |
| 7763747 | Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease Bis- and tris-dihydroxyaryl compounds and their methylenedioxy analogs and pharmaceutically acceptable esters, their synthesis, pharmaceutical compositions containing them, and their use in the treatment of amyloid diseases, especially Aβ amyloidosis, such as obser... | 07/27/2010 |
| 7667069 | Ibopamine maleate, method for preparing it and pharmaceutical compositions containing it Ibopamine malcate salt (1:1), method for preparing it and pharmaceutical composition containing it. ... | 02/23/2010 |
| 7402698 | Secondary amino-and cycloamino-cycloalkanol derivatives and methods of their use The present invention is directed to secondary amino- and cycloamino-cycloalkanol derivatives, compositions containing these derivatives, and methods of their use for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia,... | 07/22/2008 |
| 7329775 | Compounds and related methods for mutant p53 reactivation Ketoamine compounds and related methods for reactivation of tumor suppressor protein p53. ... | 02/12/2008 |
| 7273952 | Substituted C-cyclohexylmethylamine derivatives Substituted C-cyclohexylmethylamine derivatives, methods for the production thereof, pharmaceuticals containing said compounds, the use of substituted C-cyclohexylmethylamine derivatives for producing pharmaceuticals, and method of pain treatment using the pharmaceu... | 09/25/2007 |
| 7253210 | Methylene-bridged selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a... | 08/07/2007 |
| RE39593 | 1-phenyl-3-dimethylaminopropane compounds with a pharmacological effects 1-phenyl-3-dimethylaminopropane compounds corresponding to the formula I a method of preparing them, and the use of these substances as analgesic active ingredients in pharmaceutical compositions. ... | 04/24/2007 |
| 7034015 | Aminobenzoephenones The invention relates to a novel class of aminobenzophenones derivatives, to pharmaceutical preparations comprising said compounds, to dosage units of such preparations, to methods of treating patients comprising administering said compounds, and to the use of said ... | 04/25/2006 |
| RE39072 | 2-aminopropane-1,3-diol compounds, medicinal use thereof, and intermediates in synthesizing the same The present invention relates to a compound of the general formula wherein R1, R2, R3 and R4 are each a hydrogen or an acyl, a pharmaceutically acceptable acid addition salt thereof or ... | 04/18/2006 |
| 7022870 | N-bridged selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a... | 04/04/2006 |
| 6858650 | Stable salts of novel derivatives of 3,3-diphenylpropylamines The present invention concerns highly pure, crystalline, stable compounds of novel derivatives of 3,3-diphenylpropylamines in the form of their salts, a method for the manufacture and highly pure, stable intermediate products. The method is in particular char... | 02/22/2005 |
| 6767923 | Benzhydryl derivatives Benzhydryl derivatives of the formula I, where the index and the variables are as defined below: X is oxygen or sulfur; R1, R3 are halogen, cyano, nitro, hydroxyl, mercapto, amino, alk... | 07/27/2004 |
| 6667341 | Delta dicarbonyl compounds and methods for using the same Amidomethyl esters, carbonylmercaptomethyl esters, keto-containing esters, amidomethyl thioesters, amidomethyl amides, and methylene dithioesters are disclosed. The novel compounds have two carbonyl groups connected by a linking moiety having an oxygen, s... | 12/23/2003 |
| 6593492 | Resolution of intermediates in the synthesis of substantially pure bicalutamide A methods of preparing a substantially pure enantiomer of an acylanilide such as Casodex.RTM. (bicalutamide) and/or its derivatives includes resolving an intermediate compound having the structure of Formula I: ##STR1## wherein R1 is alkyl or h... | 07/15/2003 |
| 6472555 | Process for the production of esters from alcohols using acetic acid as acetylating and clays as catalysts The present invention relates to a process for the preparation of esters from alcohols using acetic acid as acetylating agent and clays as catalysts, which comprises the preparation of esters in a single step from the reaction of aliphatic, acyclic, cycli... | 10/29/2002 |
| 6444702 | Aminoadamantane derivatives as therapeutic agents The present invention provides novel aminoadamantane derivatives, methods of making the derivatives, compositions including the novel aminoadamantane derivatives, and methods for the treatment and prevention of neurological diseases using the derivatives ... | 09/03/2002 |
| 6414170 | Preparation of cationic surfactants containing ester group in molecules The present invention relates to a method for preparing a cationic surfactant in which physical chemical characteristics such as softness, antistatic properties, etc. as well as biodegradability are quite excellent due to having an ester group and a hydro... | 07/02/2002 |
| 6383633 | Fluorochemical composition comprising a polymer derived from a fluorochemical urethane (meth)acrylate monomer for imparting stain release properties to a substrate A fluorochemical composition is described comprising a polymer derived from a fluorochemical urethane (meth)acrylate monomer. The fluorochemical composition is useful for imparting stain release properties to a substrate.... | 05/07/2002 |
| 6359147 | Reactions catalyzed by chromium (III) carboxylates Reactions of ring systems, such as aziridines, oxetanes and oxiranes with carboxylic acids, anhydrides, imides, lactones and carbonate esters are catalyzed by C3 -C60, substituted or unsubstituted, straight or branched-chained, alkyl... | 03/19/2002 |
| 6348615 | Process for producing (2R, 3S)-3-amino-1, 2-oxirane A process for producing (2R, 3S)-3-amino-4-phenylbutane-1,2-epoxide compounds which comprises treating a (2S, 3S)-3-amino-1-halo-2-hydroxy-4-phenylbutane compound or a (2S, 3S)-3-amino-4-phenylbutane-1,2-epoxide with a carboxylic acid quaternary ammo... | 02/19/2002 |
| 6344558 | 1-phenyl-3-dimethylaminopropane compounds with a pharmacological effect 1-phenyl-3-dimethylaminopropane compounds corresponding to the formula I ##STR1## a method of preparing them, and the use of these substances as analgesic active ingredients in pharmaceutical compositions.... | 02/05/2002 |
| 6303652 | BTK inhibitors and methods for their identification and use The invention provides BTK inhibitors, methods for their identification and use, and pharmaceutical compositions comprising BTK inhibitors.... | 10/16/2001 |
| 6294575 | BTK inhibitors and methods for their identification and use The invention provides BTK inhibitors, methods for their identification and use, and pharmaceutical compositions comprising BTK inhibitors.... | 09/25/2001 |
| 6248737 | 1-phenyl-3-dimethylaminopropane compounds with a pharmacological effects 1-phenyl-3 -dimethylaminopropane compounds corresponding to the formula I ##STR1## a method of preparing them, and the use of these substances as analgesic active ingredients in pharmaceutical compositions.... | 06/19/2001 |
| 6225499 | Process for preparing aminoarylacetylenes This invention provides a process for preparing aminoarylacetylenes comprising reacting a N-arylmethylidene aminoarylhalide with a terminal acetylene in the presence of a base and a catalyst system comprising a palladium catalyst and a cuprous salt to pro... | 05/01/2001 |
| 6218536 | 1,2-bis-adducts of stable nitroxides with substituted ethylenes and stabilized compositions 1,2-Bis-adducts of stable hindered nitroxide compounds with substituted ethylenes are prepared by reacting two equivalents of nitroxyl compound with an ethylenically unsaturated compound such as styrene or an acrylate ester. These adducts are very effecti... | 04/17/2001 |
| 6214873 | 2-aminopropane-1,3-diol compounds, medicinal use thereof, and intermediates in synthesizing the same The present invention relates to a compound of the general formula ##STR1## wherein R1, R2, R3 and R4 are each a hydrogen or an acyl, a pharmaceutically acceptable acid addition salt thereof or a hydrate thereof... | 04/10/2001 |
| 6160010 | BTK inhibitors and methods for their identification and use The invention provides BTK inhibitors, methods for their identification and use, and pharmaceutical compositions comprising BTK inhibitors.... | 12/12/2000 |
| 6124270 | Use of a cationic amphipathic compound as a transfection agent, vaccine additive or drug A cationic amphipathic compound of formula (I), ##STR1## wherein A is a single bond, an NH--R' grouping or (a), wherein --R'-- is a straight or branched, optionally substituted, saturated or unsaturated C1-22 aliphatic chain optionally int... | 09/26/2000 |
| 6100425 | Process for the preparation of an intermediate useful in the synthesis of iodinated contrast media A process for the preparation of the compound L-5-(2-acetoxypropionylamino)-2,4,6-triiodoisophthaloyl dichloride by reacting 5-amino-2,4,6-triiodoisophthaloyl dichloride with L-2-acetoxypropionyl chloride in N,N-dimethylacetamide as a solvent, charac... | 08/08/2000 |
| 6069247 | Process for preparing substituted acrylamides by reaction of propiolamides and aromatic rings The present invention relates to a process for preparing acrylamides; wherein, a propiolamide is reacted with an activated aromatic ring to yield a wide variety of acrylamides.... | 05/30/2000 |
| 5929272 | Aliphatic epoxide-amine adducts with substantial side-chain, branching process for their preparation, and their use Epoxide-amine adducts having a proportion by mass of at least 20% of aliphatic epoxide or amine units which comprise at least one tertiary or quaternary carbon atom are disclosed. The adducts are employed as binders for coatings of relatively high environ... | 07/27/1999 |
| 5917038 | Process of preparing substituted acrylamides The present invention relates to a process for preparing acrylamides; wherein, a propiolamide is reacted with an activated aromatic ring to yield a wide variety of acrylamides.... | 06/29/1999 |
| 5892061 | Process for preparing isoimides A preparation process of isoimide comprising reacting a compound having one or more carboxyl group and one or more amide bond in the same molecule in the presence of a haloiminium salt and basic substance, and a preparation process of isoimide comprising ... | 04/06/1999 |
| 5753707 | Amide derivatives and their use in cosmetic composition An amide derivative represented by the following formula (1): ##STR1## wherein R1 represents a C1-40 hydrocarbon; R2 represents a C1-6 alkylene; R3 represents H, OH or alkoxyl; R4 repr... | 05/19/1998 |
| 5710279 | N-acyloxyalkyl-carboxamides and process for their preparation The invention provides novel N-acyloxyalkyl-carboxamides of the general formula (I): ##STR1## in which R1 is alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, arylalkyl or heteroarylalkyl, each of which is optionally substituted, R | 01/20/1998 |
| 5705680 | Process for the preparation of O-acylglycolanilides The present invention relates to a process for the preparation of O-acylglycolanilides of the formula (1) ##STR1## in which R1 and R2 are identical or different and are hydrogen, halogen, a nitro group, a cyano group, a straight... | 01/06/1998 |
| 5698523 | Acylated enol derivatives as prodrugs of elastase inhibitors This invention relates to acylated enol derivatives of known elastase inhibitors. These compounds are useful in the treatment of various inflammatory diseases, including cystic fibrosis and emphysema or as prodrugs of compounds which are useful in the tre... | 12/16/1997 |
| 5693852 | Process for the preparation of o-acyloxycarboxanilides The present invention relates to a process for the preparation of O-acyloxycarboxanilides of the formula (I) ##STR1## in which R is a radical having 1 to 6 carbon atoms, n is an integer from 1 to 10, R1 is hydrogen or an alkyl radical havi... | 12/02/1997 |
