Celebrity Inventors
Superstar singer Michael Jackson co-patented a "Method and means for creating anti-gravity illusion" in 1993.
PatentStorm News
Make the Most of Our Site
See this month's Top Inventors and Most Cited Patents.
Stay on top of the latest innovations by subscribing to an RSS feed.
Registered users: Manage your profile.
| Number | Title | Issue Date |
| 7468453 | Production process of gamma-cyhalothrin A process for the preparation of gamma-cyahlothrin comprising a) chlorinating 1R cis-Z 3-(2-chloro-3,3,3-trifluoro-1-propenyl)-2,2-dimethyl cyclopropanecarboxylic acid to give 1R cis-Z 3-(2-chloro-3,3,3-trifluoro-1-propenyl)-2,2-dimethyl cyclopropanecarboxylic acid ... | 12/23/2008 |
| 7407959 | Cathepsin cysteine protease inhibitors This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, s... | 08/05/2008 |
| 7375134 | Cathepsin cysteine protease inhibitors This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, s... | 05/20/2008 |
| 6703379 | Benzene derivatives and pharmaceutical use thereof The present invention provides an AP-1 activation inhibitor, NF-kappa B activation inhibitor, inflammatory cytokine production inhibitor, matrix metalloprotease production inhibitor, inflammatory cell adhesion molecule expression inhibitor, anti-inflammat... | 03/09/2004 |
| 6699904 | PPAR agonists PPAR alpha activators, pharmaceutical compositions containing such compounds and the use of such compounds to elevate certain plasma lipid levels, including high density lipoprotein-cholesterol and to lower certain other plasma lipid levels, such as LDL-c... | 03/02/2004 |
| 6596878 | Methods and compositions for inhibiting cell proliferative disorders The present invention concerns compounds and their use to inhibit the activity of a receptor tyrosine kinase. The invention is preferably used to treat cell proliferative disorders such as cancers characterized by over-activity or inappropriate activity H... | 07/22/2003 |
| 6465657 | Method of preparing refined organic compound for use in photography with improved liquid-liquid extraction from organic reaction mixture There is disclosed a method of preparing a refined organic compound, comprising the steps of adding water to an organic reaction mixture and mixing them, and then subjecting the mixture to filtration processing using a filter, to separate an organic phase... | 10/15/2002 |
| 6294573 | Reverse hydroxamate inhibitors of matrix metalloproteinases Compounds having the formula ##STR1## are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.... | 09/25/2001 |
| 6288261 | Inhibitors of matrix metalloproteinases Compounds having the formula ##STR1## and pharmaceutically acceptable salts and prodrugs thereof are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloprot... | 09/11/2001 |
| 6194463 | N-sulphonyl and N-sulphinyl amino acid amides as microbicides -Amino acid amides of formula (I) wherein the substituents are defined as follows: n is a number zero or one; R1 to R7 are as defined herein; R8 is C1 -C6 alkyl, C3 -C6 al... | 02/27/2001 |
| 6083986 | Potassium channel inhibitors Compounds useful as potassium channel inhibitors and especially useful for the treatment of cardiac arrhythmias and cell proliferative disorders are described.... | 07/04/2000 |
| 5968977 | Ketonitrile derivatives and antibacterial agent and drugs containing the same The present invention is directed to a ketonitrile derivative represented by the following formula (1): ##STR1## (wherein R1 is a hydrogen atom or a lower alkyl group; each of R2, R3, R4, and R5,... | 10/19/1999 |
| 5932766 | Process for the preparation of substituted keto-enamines The present invention discloses a process for the preparation of a compound having formula 4: ##STR1## The process comprises the step of reacting an enolate having the formula: ##STR2## with a Grignard reagent. The enolate salt is formed in situ... | 08/03/1999 |
| 5925676 | Ester compounds pesticidal compositions containing the same and itermediates for synthesis thereof An ester compound represented by the formula ##STR1## wherein R1 and R2 may be the same or different and each represent a C1 -C6 alkyl group, or other specified groups, which may be optionally substituted w... | 07/20/1999 |
| 5888481 | Cinnamamides and their use as stabilizers The invention relates to novel cinnamamides, a process for their manufacture and their use as UV absorbers. The cinnamamides of the invention may be used as UV absorbers in a variety of engineered resins such as polyamides (especially nylon 6 and 6,6), po... | 03/30/1999 |
| 5859279 | Compound and process A process for the preparation of a compound of formula (VI), optionally in enantiomerically-enriched form (R or S), comprises chemoselective reduction of a novel compound of formula (V), wherein Ar1 and Ar2 are independently selected... | 01/12/1999 |
| 5847147 | 3-Amino-2-mercaptobenzoic acid derivatives and processes for their preparation Compounds of the formula I ##STR1## and disulfides thereof and salts thereof are important intermediate products for the preparation of compounds having a microbicidal and plant-immunizing action, of the formula III ##STR2## In the compound... | 12/08/1998 |
| 5750726 | Process for the manufacture of 2-aryl-5-perfluoroalkylpyrrole derivatives and intermediates useful therefor There is provided a single step procedure to prepare 2-aryl-5-perfluoroalkylpyrrole derivatives directly from the perfluoroacetylated Strecker reaction product. Said pyrrole derivatives are insecticidal and also useful as precursors to other insecticidal ... | 05/12/1998 |
| 5696161 | Substituted phenoxymethylphenyl derivatives, their preparation and their use for controlling pests and fungi Substituted phenoxymethylphenyl derivatives I ##STR1## X is .dbd.CH--OCH3, .dbd.CH--CH3 or .dbd.N--OCH3 ; R1 is, inter alia, R2 and R3 are, inter alia, H, halogen, CN, NO2, C | 12/09/1997 |
| 5650511 | Process for the preparation of 9-deazaguanine derivatives Derivatives of 9-deazaguanine are prepared by reacting an aldehyde or ketone with a dialkylaminomalonate to form the corresponding enamine. The enamine is then reacted with a base to form a cyclic pyrrole. The cyclic pyrrole is reacted with an urea compou... | 07/22/1997 |
| 5637770 | Hexa-cyclic compound A novel hexa-cyclic compound, a derivative of camptothecin, of the general formula: ##STR1## The compound is prepared from an aminoketone compound and a pyranoindolizine compound by the condensation-ring closing reaction. It is abundantly water-... | 06/10/1997 |
| 5563278 | Angiotensin II antagonists This invention provides novel phenyl and heterocyclic derivatives, their pharmaceutical formulations and their use for antagonizing angiotensin II receptors in mammals.... | 10/08/1996 |
| 5545664 | Substituted phenoxymethylphenyl derivatives, their preparation and their use for controlling pests and fungi Substituted phenoxymethylphenyl derivatives I ##STR1## X is .dbd.CH--OCH3, .dbd.C--CH3 or .dbd.N--OCH3 ; R1 is, inter alia, R2 and R3 are, inter alia, H, halogen, CN, NO2, C... | 08/13/1996 |
| 5530014 | Cyclohexadiene derivatives The cyclohexadiene derivatives are prepared by reaction of cyclohexanones with amines and subsequent dehydration. The compounds are suitable as active compounds in medicaments on account of their property of being selective modulators of calcium channel-d... | 06/25/1996 |
| 5446194 | Pharmacologically active catechol derivatives A compound according to formula 1 ##STR1## wherein R1 and R2 independently represent hydrogen, carbamoyl which is substituted by an alkyl of 1 to 4 carbon atoms, alkylcarbonyl of 2 to 5 carbon atoms or phenyl carbonyl, X represe... | 08/29/1995 |
| 5430060 | Acetamide derivatives The invention concerns novel N-phenylacetyl and related acyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, ... | 07/04/1995 |
| 5405987 | Process for preparing pyridine and quinoline derivatives The present invention pertains to a method of preparing substituted and unsubstituted N-hydroxy-2-aminobutane diacid derivatives which can be dehydrated to 2-aminobut-2-ene dioic acid derivatives, which can be subsequently converted to pyridine and quinol... | 04/11/1995 |
| 5403953 | 1-phenylbicyclo[2.2.2]octane compounds Compound of formula (I): ##STR1## in which: R1 represents halogen, or hydroxy, alkyl, alkoxy, cyano, amino, mercapto, alkylthio or phenoxy, R2 and R'2 represent two hydrogen when the ring is unsaturated, or alternativ... | 04/04/1995 |
| 5380755 | Alkyl and alkylbenzyl ethers of substituted hydroquinones The present invention provides alkyl and alkylbenzyl ethers of substituted hydroquinones and pharmaceutical compositions containing them. The present invention further provides methods of using these compounds and compositions to inhibit monoamine oxidase... | 01/10/1995 |
| 5358968 | Substituted oxime ethers, their preparation and their use for controlling pests and fungi Substituted oxime ethers of the general formula I ##STR1## where R1 is alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxyalkyl, cycloalkyl, cycloalkylalkyl, cyanoalkyl, alkoxycarbonylalkyl, arylalkyl, heteroarylalkyl, arylalkenyl or a... | 10/25/1994 |
| 5296454 | Acetanilide herbicides The invention relates to novel acetanilides of the formula (I) ##STR1## wherein Ar represents phenyl, furyl or thienyl, R1 represents hydrogen, C1-5 -alkyl, C3-6 -cycloalkyl, C3-6 -cycloalkyl-methyl, C3-5 | 03/22/1994 |
| 5270342 | Acetamide derivatives The invention concerns novel N-phenylacetyl and related acyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, ... | 12/14/1993 |
| 5247119 | Phenylacetonitrilehydroxyalkylaminoalkyl-ortho-substituted aryl compounds as immunosuppressives A class of substituted phenylacetonitrilehydroxyalkylaminoalkyl-ortho-substituted aryl compounds having immunosuppressive properties is described. Compounds of this class would be useful in reducing recipient rejection of transplanted organs and for ... | 09/21/1993 |
| 5223536 | 1,4-diaryl-1-cyclopropyl-4-substituted butanes as insecticides and acaricides The 1,4-diaryl-1-cyclopropyl-4-substituted butane pesticides of the following formula are effective as insecticides and acaricides: ##STR1## in which X and Y are independently hydrogen, halogen, alkyl, alkoxy, cycloalkylalkoxy, alkylcarbonyl, alkoxyc... | 06/29/1993 |
| 5196147 | Organic nonlinear optical substance An organic nonlinear optical substance having the formula (I): ##STR1## wherein R1 represents --H or --CH3 ; n is 0, 1, or 2; A represents Z1 --Ar, ##STR2## wherein Ar represents a 6-14 membered aromatic group includ... | 03/23/1993 |
| 5196562 | Substituted 1,3,5-triazinetriones, for use against parasitic protozoa Protecting against parasitic protozoa with substituted 1,3,5-triazinetriones of the formula ##STR1## in which R1 represents aromatic or heteroaromatic radicals, each of which is optionally substituted, R2 represents H, alkyl, al... | 03/23/1993 |
| 5190999 | -carbonylphenylacetonitrile derivatives as stabilizers for organic materials Compositions comprising an organic material liable to oxidative, thermal and/or actinic degradation and at least one compound of the formula I ##STR1## are described in which n is 1-6, R, R1, R2, R3 and R4 ... | 03/02/1993 |
| 5189039 | 7-disubstituted-methyl-4-oxo-3H,5H-pyrrolo[3,2d]pyrimidine and pharmaceutical uses and compositions containing the same Disclosed is a compound of the formula ##STR1## wherein R1 is H, NH2, or OCH3, R2 is an optionally substituted cyclic group optionally containing one or more heteroatoms, R3 and R4 are... | 02/23/1993 |
| 5182303 | Substituted semicarbazone arthropodicides Certain substituted semicarbazones, including all geometric and stereoisomers thereof, agricultural compositions containing them and their use as arthropodicides.... | 01/26/1993 |
| 5175170 | ଲ-amino acid derivatives Non-peptidyl compounds characterized generally as cycloalkyl/cycloalkylkyl-N-terminal amino hydroxy ଲ-amino acid derivatives are useful as renin inhibitors for treatment of hypertension. Compounds of particular interest of the formula ##STR1## ... | 12/29/1992 |
