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| Number | Title | Issue Date |
| 7279597 | Phenyl amine carboxylic acid compounds and compositions for delivering active agents Phenyl amine carboxylic acid compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 10/09/2007 |
| 7208483 | Polymeric delivery agents and delivery agent compounds Polymeric delivery agents, delivery agent compounds and compositions comprising them which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 04/24/2007 |
| 7129274 | Phenoxy carboxylic acid compounds and compositions for delivering active agents Phenoxy carboxylic acid compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 10/31/2006 |
| 7125910 | Compounds and compositions for delivering active agents Carrier compounds and compositions therewith which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 10/24/2006 |
| 7115663 | Cyanophenoxy carboxylic acid compounds and compositions for delivering active agents Cyanophenoxy carboxylic acid compounds and compositions for the delivery of active agents are provided. Methods of administration, treatment of disease and preparation are provided as well. ... | 10/03/2006 |
| 7084279 | Oxadiazole compounds and compositions for delivering active agents Oxadiazole compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 08/01/2006 |
| 7071214 | Compounds and compositions for delivering active agents Carrier compounds and compositions therewith which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well. ... | 07/04/2006 |
| 6921747 | Basic amino acid derivatives The present invention provides a basic amino acid derivative represented by the formula (1): The present invention also provides a method of making a gelled product by employing the aforementioned compound, as well as ... | 07/26/2005 |
| 6903082 | Methods of treating inflammatory conditions of the gastrointestinal tract using 4-APAA and compositions thereof Compounds are disclosed having the structure of Formula I: where R1, R3, and R4 are independently hydrogen or C1 to C4 alkyl, and R2 is: | 06/07/2005 |
| 6696606 | Solid phase synthesis of arylretinamides A solid phase synthetic method for preparing arylretinamides is provided. The method comprises reacting hexachloroacetone with a solvent-suspended resin-bound triphenylphosphine to provide a suspension comprising an activated chlorinating reagent; reactin... | 02/24/2004 |
| 6455715 | Method of producing dicarboxylic acids suitable for synthesis of polymers or polyamides A method is described for producing saturated dicarboxylic acids with a chain length of C6 to C21 or the corresponding diamidic dicarboxylic acids from fatty acid cleavage of unsaturated fatty acids or the bis-fatty acid diamides of these unsaturated fatt... | 09/24/2002 |
| 6090958 | Compounds and compositions for delivering active agents Carrier compounds and compositions therewith which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well.... | 07/18/2000 |
| 6071510 | Modified amino acids and compositions comprising the same for delivering active agents The present invention provides modified amino acids for delivering active agents, and particularly biologically or chemically active agents. The preferred modified amino acids of the present invention include N-acylated or sulfonated amino acids. These mo... | 06/06/2000 |
| 6060513 | Compounds and compositions for delivering active agents Carrier compounds and compositions therewith which are useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well.... | 05/09/2000 |
| 5962710 | Method of preparing salicyloylamino acids A method for preparing salicyloylamino acids is provided. An oligosalicylate and an amino acid are reacted to yield the salicyloylamino acid.... | 10/05/1999 |
| 5773465 | Tartronic acids, their acetalic ethers and o-esters Tartronic acid acetalic ethers and esters of the general formula: ##STR1## are provided and are useful in treatment of bone dysmetabolism. As examples, Ra and Rb may be hydrogen, B is a C2 -C12 acyl group, R is phenyl and n is 0... | 06/30/1998 |
| 5576416 | Amide-containing self-emulsifying epoxy curing agent A new epoxy hardener composition is the product of the reaction of (A) a poly(alkylene oxide) monoamine or diamine with a molecular weight (Mn) of about 500 to 3000 and (B) a di- or polycarboxylic acid, in a ratio of moles of carboxylic acid to equivalent... | 11/19/1996 |
| 5559268 | Process for the efficient preparation of N-substituted dehydroamino acid esters A process for the preparation of N-substituted dehydroamino acid esters by contacting a ଲ-hydroxy--amino acid ester or N- or O-substituted ଲ-hydroxy--amino acid ester with an excess of acetic anhydride and a base is disclosed.... | 09/24/1996 |
| 5292915 | Compounds containing carbonate groups and carbonyl groups and the preparation and use thereof The invention relates to compounds containing carbonate groups and carbonyl groups and having the general formula ##STR1## in which R stands for a C1 -C4 -alkyl radical, an aryl radical, or a radical R1, where R1... | 03/08/1994 |
| 5266576 | N-myristoyl transferase inhibitors The invention relates to a compound of formula (I): ##STR1## which can be used as N-myristoyltransferase inhibitors, in which R1 represents hydrogen, substituted or unsubstituted (C1 -C6) alkyl, substituted or unsubst... | 11/30/1993 |
| 5252706 | Peptide derivative amphiphatic compound, intermediate thereof and liposome and film comprising peptide derivative amphiphatic compound A peptide derivative amphiphatic compound or N-terminal salt thereof represented by formula (I): ##STR1## wherein R1 and R2 each represents a straight-chain or branched alkyl or acyl group having 8 to 24 carbon atoms optionally ... | 10/12/1993 |
| 5240630 | Refrigeration compositions containing diester-amides of dialkanolamines A refrigeration lubricant suitable for use with R-134a-type refrigerants comprises at least one dialkanolamine diester-amide oil corresponding to one of the formulas: ##STR1## in which formulas R is a hydrocarbylene group containing 1-10 carbons; n ... | 08/31/1993 |
| 5147868 | Thienamycin renal peptidase inhibitors Novel chemical compounds are provided which selectively inhibit the metabolism of dipeptidase (E.C.3.4.13.11) and therefore are useful in combination with antibacterial products. These chemical compounds are z-2-acylamino-3-monosubstituted propenoates.... | 09/15/1992 |
| 5098613 | Anti-inflammatory agents This invention provides benzene derivatives, pharmaceutical formulations of those derivatives, and a method of using the derivatives for the treatment of inflammation in mammals.... | 03/24/1992 |
| 5082683 | Amide/amine ester derivatives as low calorie fat mimetics Amide/amine ester derivatives of the general formula: ##STR1## where B is an aliphatic group having 2 to 6 carbons, each R is independently, an aliphatic group having 1 to 23 carbons, Q is --N(R')-- or --O--(CH2)p --N(R')--, R' is --H, --... | 01/21/1992 |
| 5051448 | GABA esters and GABA analog esters Ester derivatives of gamma-aminobutyric acid (GABA) and GABA analogues which cross the blood-brain barrier are disclosed, as well as methods of synthesizing and using the compounds. The ester derivatives have the formula: ##STR1## where A is a radica... | 09/24/1991 |
| 5045338 | Secondary amide esters as low calorie fat mimetics Secondary amide esters of the general formula ##STR1## where A is an organic radical having 2 to 6 carbons, m=1 to 3, n=1 to 3, and each R is, independently, an aliphatic, ether or ester group having 1 or 2 to 29 carbons are edible, preferably partially d... | 09/03/1991 |
| 4978395 | Polymeric dispersing agent Polyaddition product the molecule of which is characterized by the presence of one group ##STR1## Method to prepare the above mentioned product and dispersions in polar and non polar diluents which contain the said product in addition with solid ... | 12/18/1990 |
| 4978759 | Process for the stereospecific synthesis of optically pure 4-amino-3-hydroxycarboxylic acid derivatives The process described makes it possible to obtain optically pure 4-amino-3-hydroxycarboxylic acids by means of a series of stereoselective steps. The starting material is an alpha-amino acid in the L or D configuration, with which Meldrum's acid is reacte... | 12/18/1990 |
| 4933367 | Carboxylic acid derivatives, processes for the preparation thereof, the use thereof, and pharmaceutical compositions which contain these compounds This invention relates to carboxylic acid derivatives and their use thereof. The compounds are useful in treatment of various diseases such as diabetes, prediabetic conditions, adipositas ailments or atherosclerosis.... | 06/12/1990 |
| 4892687 | Process for synthesis of amidoacids using a cobalt catalyst and a bidental phosphine ligand A process is disclosed for producing N-acetyl-aminoacid which comprises reacting a feedstock from the group consisting of simple olefins, acetamide and synthesis gas with a catalyst comprising a cobalt-containing compound promoted by a bidental-phosphine ... | 01/09/1990 |
| 4885311 | Topical transretinoids for treatment of acne and skin diseases Esters and amides of 13-trans-retinoic acid are disclosed which are used for the treatment of acne and skin diseases.... | 12/05/1989 |
| 4867915 | 16-Substituted polyunsaturated hexadecanoic fatty acids Sixteen carbon atom carboxylic acids having 16-phenoxy or 16-phenylthio substituents, and 0, 1, or 4 triple bonds, methods of preparing them, and pharmaceutical preparations containing them. These compounds are useful as lipoxygenase inhibitors.... | 09/19/1989 |
| 4847303 | Tert-butylphenyl compounds useful as anti-inflammatory agents The present invention involves compounds having the structure: ##STR1## wherein: (a) --A1 is selected from the group consisting of --OH, --H, and --O2 CR; (b) --A2 is selected from the group consisting of unsubstituted or ... | 07/11/1989 |
| 4676933 | Method for purification of amido acids A method for purification of C12 -C16 amido acids prepared from C10 -C14 amido acids is disclosed. The amido acids are purificed by dissolving the crude product in organic alcohol solvent and chloroform at a tem... | 06/30/1987 |
| 4677120 | Topical prodrugs for treatment of acne and skin diseases Esters and amides of 13-cis-retinoic acid are disclosed which are used for the treatment of acne and skin diseases.... | 06/30/1987 |
| 4628110 | Novel 9-substituted carbacyclin analogs Novel compounds of the following general formula: ##STR1##... | 12/09/1986 |
| 4570011 | Preparation of cyclobutene substituted aromatic hydrocarbons The invention is a process for the preparation of an aromatic hydrocarbon with a cyclobutene ring fused to the aromatic hydrocarbon which comprises, dissolving an ortho alkyl halomethyl aromatic hydrocarbon in an inert solvent and pyrolyzing the solution ... | 02/11/1986 |
| 4526723 | Biocidal enol esters of non-ortho substituted 2-aryl-1-3-cycloalkanedione compounds Non-ortho substituted 2-aryl-1,3-cycloalkanedione enol ester compounds exhibit outstanding acaricidal and herbicidal activity.... | 07/02/1985 |
| 4518789 | Phenyl alpha-acyloxyacetamide derivatives and their therapeutic use Therapeutic as well as preventive measures to alleviate the symptoms of dermatologic and other conditions and disorders with phenyl alpha-acyloxyacetamide derivatives is disclosed. Dermatologic and other conditions and disorders in humans in which the com... | 05/21/1985 |