U.S. patents available from 1976 to present.
U.S. patent applications available from 2005 to present.

Icon_funbox Celebrity Inventors

Mark Twain (Samuel L. Clemens) received Patent No. 121,992 for "An Improvement in Adjustable and Detachable Straps for Garments." He later received two more patents: one for a self-pasting scrapbook and one for a game to help players remember important historical dates.

Newsletter  PatentStorm News

Make the Most of Our Site

See this month's Top Inventors and Most Cited Patents.

Stay on top of the latest innovations by subscribing to an RSS feed.

Registered users: Manage your profile.

 

Class 552/644 - Unsaturation between the 5- and 10-positions


Subclass of Class 552 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which contain a double bond between the 5- and
No. of patents: 22
Last issue date: 04/22/2008


NumberTitleIssue Date
7361645Androgenic 7-substituted 11-halogen steroids
The invention relates to 11β-halogen steroids with general formula (I), whereby R11 is halogen, X—Y-Z represents a group with one of the two structures CH═C—C or CH2—C═C and the other radicals have the meaning that is indicated in th...
04/22/2008
6989378Testosterone derivative
The invention is the novel androgen (7α,17β)-7-methyl-17-[(1-oxoundecyl)oxy]estr-4en-3one (MENT undecanoate). This compound distinguishes favourably from other testosterone derivatives in that it has a good solubility in oily media. It particularly exhibits a good...
01/24/2006
6677329Non-aromatic estrogenic steroids with a hydrocarbon substituent in position 11
Disclosed are novel, selective estrogens type having a steroid skeleton with a non-aromatic A-ring and a free or capped hydroxyl group at carbon atom No. 3. The estrogens satisfy general formula (I), in which R1 is H, (C1 -C3
01/13/2004
6649779Estrenes
This invention provides a pharmaceutically acceptable salt of 3ଲ-hydroxy-5(10)-estrene-17-one 3-sulfate ester and a pharmaceutically acceptable salt of 3଱-hydroxy-5(10)-estrene-17-one 3-sulfate ester, which are useful as an estrogens....
11/18/2003
6458778Estradienes
This invention provides estra-5(10),7-dien-3ଲ-ol-17-one or a pharmaceutically acceptable salt of its 3-sulfate ester, estra-5(10),7-dien-3ଲ-ol-17-one 3-glucuronide or a pharmaceutically acceptable salt thereof, estra-5(10),7-dien-3଱-ol-1...
10/01/2002
5994568Estrenes for inducing hypothalamic effects
The invention relates to estrene steroids, which bind to neuroepithelial receptors. The steroid is preferably administered in the form of a pharmaceutical composition containing one or more pharmaceutically acceptable carriers....
11/30/1999
4923640Process for the production of 17଱-ethinyl-17ଲ-hydroxy-18-methyl-4,15-estradien-3-one and new intermediate products for this process
A process for the production of 17଱-ethinyl-17ଲ-hydroxy-18-methyl-4,15-estradien-3-one is described comprising reacting a 17-enolester of formula II ##STR1## wherein R1 represents an alkyl radical with 1-3 carbon atoms and R
05/08/1990
492184511-arylsteroid compounds
The invention relates to new 11-arylsteroid compounds, having a strong antiprogestin and a weak or nonexistent antiglucocorticoid activity, to processes for preparing said compounds and also to pharmaceutical preparations which contain these derivatives a...
05/01/1990
4871724Novel 11-aryloestrane and 11-arylpregnane derivatives
The present invention is concerned with 11-aryloestrane and 11-arylpregnane derivatives, characterized in that these derivatives have the following structure: ##STR1## wherein R1 is an aryl group with an ##STR2## group as substit...
10/03/1989
4745109Suicide inhibitors of aromatase
Thiol-substituted synthetic steriod hormones or androgens having a testosterone ring system backbone are used to inhibit aromatase's catalyzed conversion of C19 androgens having a A4,3-ketone group to estrogens in the treatment of es...
05/17/1988
433392816 ଱-Alkyl steroids, their preparation, and pharmaceutical preparations thereof
16 ଱-Alkyl steroids of the formula ##STR1## wherein R1 is hydrogen or methyl, R2 is hydrogen, alkyl, acyl, or glycosyl R3 is hydrogen or a substituted or unsubstituted, saturated or unsaturated lower hydrocarbon resi...
06/08/1982
4212864Branched chain and cycloaliphatic esters of the androstane and oestrane series and pharmaceutical compositions containing same
There are disclosed branched chain and cycloaliphatic esters of steroids having the formula: ##STR1## or the 5଱H analog thereof, where R is H or CH3 ; R1 is H or CH3 ; R2 is H or CH3 ; R3
07/15/1980
4150126Novel enol esters of steroids, compositions containing such compounds, processes for their preparation and methods of treatment therewith
This invention relates to novel enol esters of steroids having an antitumor activity and to the preparation thereof. The invention is also concerned with pharmaceutical compositions containing the said compounds and methods of treatment therewith....
04/17/1979
405242113-Ethinyl-steroids and processes for their manufacture
A new class of 13-ethinyl-steroids is prepared by a novel process comprising Wittig reaction of a 13-formyl steroid with a chloro- or bromomethylenephosphorane and dehydrohalogenation of the intermediate 13-(2-halogenovinyl)steroid with an extremely stron...
10/04/1977
4036695Process for the preparation of estrene-3,17-dione derivatives
Estrene-3,17-diones of the formula ##STR1## wherein X is oxo, or ketalized oxo, preferably alkylenedioxy of 2-6 carbon atoms or o-phenylenedioxy; Ɗ is a carbon atom linked to the adjacent carbon atoms by a double bond and two single bonds; R1
07/19/1977
4002746Synthesis of gon-4-enes
1. A therapeutic composition having progestational activity comprising as active ingredient a 17-aliphatic carboxylic acid ester of 17଱-ethynyl-18-methyl-19-nortestosterone and a pharmaceutical carrier for said compound....
01/11/1977
39975749-଱-methyl-steroids
The compounds are 13-(lower)alkyl-9଱-methyl-17଱-propadienylgona-4-en-17ଲ-ol -3-ones and derivatives thereof, e.g. 9଱-methyl-17଱-propadienylestra-17ଲ-ol-3-one, and are useful as progestational agents....
12/14/1976
3983144Novel 11ଲ-alkyl steroids of the estrane series
The present invention relates to novel steroids of the estrane series having the general formula I: ##SPC1## wherein R1 and R2 = an alkyl group having 1-4 carbon atoms, R3 = oxygen or (଱P)(ଲQ), wherein P = hydrogen ...
09/28/1976
3972906Novel - 11-substituted steroids of the estrane series
The present invention relates to novel 11-substituted steroids of the estrane series having the general formula ##SPC1## In which R1 = a free, esterified or etherified hydroxyl group or halogen; R2 = an alkyl group with 1-4 C-atoms; R
08/03/1976
3963707Novel N-nitroso compounds, compositions containing such compounds, processes for their preparation and methods of treatment therewith, and novel intermediates
This invention relates to novel N-halogenoalkyl-N-nitroso carbamates and N4 halogenalkyl-N4 -nitroso allophanates of steroid compounds, having an anti-tumor activity, and to the preparation thereof. The invention is also concerned wi...
06/15/1976
3962291Total synthesis of 11-alkyl steroids
A novel total synthesis of 11-alkyl steroids, utilizing readily available and inexpensive raw materials, is described. The resulting products are useful and novel pharmacological agents possessing, for example, selective hormonal properties....
06/08/1976
3944576Novel steroids of the oestrane series substituted in 7-position
The invention relates to novel 7-substituted-steroids of the oestrane series of the general formula: ##SPC1## In which Ring A including carbon atom 6 is ##SPC2## R1 = an alkyl group with 1-4 C-atoms, R2 = oxygen or (଱Y)(ଲ...
03/16/1976
 
Sign InRegister
Username  
Password   
forgot password?