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Vladimir Zworykin, television pioneer ; Talking about an invention in which he played a critical role.
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| Number | Title | Issue Date |
| 7423058 | Inhibitors of hepatitis C virus NS3 protease The present invention discloses novel compounds which have HCV protease inhibitory activity as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such compounds as well as methods of us... | 09/09/2008 |
| 7342041 | 3,4-(cyclopentyl)-fused proline compounds as inhibitors of hepatitis C virus NS3 serine protease The present invention discloses novel compounds which have HCV protease inhibitory activity as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such compounds as well as methods of us... | 03/11/2008 |
| 7314885 | Pyrrole compounds useful as kinase inhibitors The present invention relates to compounds useful of inhibitors of protein kinases. The invention also provides pharmaceutically acceptable compositions comprising said compounds, processes for making the compounds and methods of using the compositions in the treatm... | 01/01/2008 |
| 7271210 | Stabilized ester compositions and their use in film-forming compositions This invention relates to a composition comprising, consisting of or alternatively consisting essentially of a stabilized furfural or glycol ester of a vegetable oil fatty acid and an antioxidant such as butylated hydroxy toluene. This invention also relates to late... | 09/18/2007 |
| 7205330 | Inhibitors of hepatitis C virus NS3 protease The present invention discloses novel compounds which have HCV protease inhibitory activity as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such compounds as well as methods of us... | 04/17/2007 |
| 7186849 | C7 ester substituted taxanes Taxanes having an ester substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents. ... | 03/06/2007 |
| 7183300 | Inhibitors of HIV-1 capsid formation: substituted aryl aminomethyl thiazole ureas and analogues thereof Substituted aryl aminomethyl thiazole ureas and analogues thereof that act as inhibitors of viral capsid formation, including HIV capsid formation, are provided here. Generally the virus capsid formation inhibitors described herein are compounds of Formula I ... | 02/27/2007 |
| 7145025 | Structural carotenoid analogs for the inhibition and amelioration of disease A method for inhibiting and/or ameliorating the occurrence of diseases associated with reactive oxygen species, reactive nitrogen species, radicals and/or non-radicals in a subject whereby a subject is administered a carotenoid structural analog, either alone or in ... | 12/05/2006 |
| 7019024 | Pharmaceutical for treatment of neurological and neuropsychiatric disorders The invention provides a pharmaceutical for treatment of neurological and neuropsychiatric disorders comprising a compound of the formula: or a pharmaceutically acceptable salt thereof. ... | 03/28/2006 |
| 6972343 | Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity The invention concerns drug precursors with antimalarial effect, characterised in that it consists in quaternary bis-ammonium salts of general formula (I) wherein A and A′, identical or different, are respectively either a group A1 and A′1 of formula (1) wherein... | 12/06/2005 |
| 6872837 | Taxanes having a c10 Heterosubstituted acetate substituent Taxanes having a heterosubstituted acetate substituent at C(10), a hydroxy substituent at C(7), and a range of C(2), C(9), C(14), and side chain substituents. ... | 03/29/2005 |
| 6861446 | C7 heterosubstituted acetate taxane compositions Taxanes having a heterosubstituted acetate substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents. ... | 03/01/2005 |
| 6858740 | 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses The invention concerns 2-oxo-1-pyrrolidine derivatives and a process for preparing them and their uses. The invention also concerns a process for preparing α-ethyl-2-oxo-1-pyrrolidine acetamide derivatives from unsaturated 2-oxo-1-pyrrolidine derivatives. Particula... | 02/22/2005 |
| 6841571 | Compounds useful as reversible inhibitors of cysteine proteases Disclosed are cathepsin S, K, F, L and B reversible inhibitory compounds of the formulas (Ia) and (Ib) where R2, R3, R4, R6, R8 and Y are defined herein. The compounds are useful for treating autoimmune and othe... | 01/11/2005 |
| 6797712 | Substituted amino-furan-2-yl-acetic acid and amino-thien-2-yl-acetic acid derivatives and their use in the treatment of migraine and pain Compounds of formula I, or a pharmaceutically acceptable salt thereof, The compounds of the present invention are suitable for the treatment of pain and migraine. Also disclosed are method for preparing the compounds, an... | 09/28/2004 |
| 6750245 | C7 carbamate substituted taxanes Taxanes having a carbamoyloxy substituent at C(7), a hydroxy substituent at C(10, and a range of C(2), C(9), C(14), and side chain substituents. ... | 06/15/2004 |
| 6747154 | Process for preparing scopine esters A process for preparing a compound of formula 1 from a compound of formula 2 the process comprising reacting in one step the compound of formula 2 with a compound of formula ... | 06/08/2004 |
| 6673833 | C7 heterosubstituted acetate taxanes Taxanes having a heterosubstituted acetate substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents.... | 01/06/2004 |
| 6667318 | LFA-1 antagonist compounds The invention relates to novel compounds having formula (I) ##STR1## wherein Cy, X, Y, L and R1-6 are as defined herein. The compounds bind CD11/CD18 adhesion receptors such as Lymphocyte Function-associated Antigen-1 (LFA-1) and are therefore ... | 12/23/2003 |
| 6649632 | C10 ester substituted taxanes Taxanes having an ester substituent at C(10), a hydroxy substituent at C(7), and a range of C(2), C(9), C(14), and side chain substituents.... | 11/18/2003 |
| 6620804 | Selenophene anti-tumor agents Novel selenophene compounds useful as anti-tumor agents are described. Preferred compounds include compounds of formula I: ##STR1## wherein R1 and R2 are independently selected from the group consisting of; ##STR2## H, CHO, ... | 09/16/2003 |
| 6610860 | C7 ester substituted taxanes Taxanes having an ester substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents.... | 08/26/2003 |
| 6583175 | Alkylxanthates and use of alkylxanthates in the integrated pest management This invention relates to novel alkylxanthates of formulae 1 to 3 and use of alkylxanthates of formulae 1 to 6 in the integrated pest management, more specifically alkyl xanthates are used as insect growth regulators for pest management in agricultural fi... | 06/24/2003 |
| 6552205 | C10 OXO and hydrido taxane derivatives and pharmaceutical compositions containing them Taxane derivatives having alternative C10 substituents.... | 04/22/2003 |
| 6521660 | 3'-alkyl substituted taxanes and pharmaceutical compositions containing them Taxane derivatives having an alkyl substituted C13 side chain.... | 02/18/2003 |
| 6500958 | Carboxylic acid derivatives and process for producing the same The present invention relates to compounds which are useful for efficient synthesis of 2-amino-4-oxobicyclo[3.1.0]hexane-2,6-dicarboxylic acids. The compounds according to the present invention comprise 2-oxobicyclo[3.1.0]hexane-6-carboxylic acid derivatives r... | 12/31/2002 |
| 6468444 | Chiral compounds and their use as chiral dopants for producing cholesteric liquid crystal compositions Chiral dopants of the formula I Z1 --Y1 --(A1)m --Y2 --M--Y3 --X--Y4 --(A2)n --Y5 --Z2 I in which the variables have, independently of one anot... | 10/22/2002 |
| 6462208 | C7 acyloxy and hydrido taxane derivatives and pharmaceutical compositions containing them Taxane derivatives having alternative C7 substituents.... | 10/08/2002 |
| 6410754 | Photochromic spiropyrans, and compositions and articles containing same Novel spiropyran compounds, particularly with photochromic properties, are disclosed, as well as photochromic compositions and ophthalmic articles containing said compounds. The photochromes have been designed so as to have a high colorability, a high sen... | 06/25/2002 |
| 6407268 | Substituted 4-benzoylpyrazoles 4-Benzoylpyrazoles of the formula I ##STR1## where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, C1 -C6 -alkyl, C1 -C6 -haloalkyl, C1 -C6... | 06/18/2002 |
| 6399786 | Nonacyclic nodulisporic acid derivatives The present invention relates to novel nodulosporic acid derivatives, which are acaricidal, antiparasitic, insecticidal and anthelmintic agents.... | 06/04/2002 |
| 6387908 | Epoxysuccinamide derivatives Epoxysuccinamide derivatives of the formula (1): ##STR1## wherein R1 is hydrogen, alkyl, alkenyl, alkynyl, aryl, or aralkyl; R2 is alkyl, alkenyl, alkynyl, aryl, or aralkyl; R3 is hydrogen, alkyl, alkenyl, alkynyl, aryl, a... | 05/14/2002 |
| 6359154 | C7 carbamoyloxy substituted taxanes Taxanes having a carbamoyloxy substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents.... | 03/19/2002 |
| 6331635 | Taxoids, their preparation and pharmaceutical compositions containing them New taxoids of general formula (I): ##STR1## their preparation and pharmaceutical compositions containing them. The new products of general formula (I) in which Z represents a radical of general formula (II): ##STR2## display noteworthy antitumour and ant... | 12/18/2001 |
| 6303602 | Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists A compound of the following formula: ##STR1## or a salt thereof, wherein A is hydrogen, halo, hydroxy; the broken line represents an optional double bond with proviso that if the broken line is a double bond, then A is absent; Ar1 is optionally... | 10/16/2001 |
| 6288071 | 1-ethylene-2-alkylene-1,4-cyclohexadiene pesticides Pesticidally active cyclohexadienyl derivative compounds of the formula I that are esters, oximes or amides are claimed. These compounds may be used as fungicides, acaricides and insecticides in plant protection.... | 09/11/2001 |
| 6228848 | Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities Aryl-substituted and aryl and (3-oxo-1-propenly)-substituted benzopyran, benzothiopyran, 1,2-dihydroquinoline, and 5,6-dihydronaphthalene derivatives have retinoid negative hormone and/or antagonist-like biological activities. The invented RAR antagonists... | 05/08/2001 |
| 6201140 | 7-0-ethers of taxane derivatives The present invention concerns novel 7-ethers of taxane derivatives, their use as antitumor agents and pharmaceutical compositions containing the novel compounds.... | 03/13/2001 |
| 6143780 | N-arylmethylthioanilide compounds useful for the inhibition of the replication of HIV Compounds of the formula ##STR1## wherein A and X are independently oxygen or sulphur; R6 is H, halogen, alkyl, alkoxy, alkylthio, cyano, or nitro; Y is --CH2 O--, --OCH2 --, --CH2 S--, or --CH2 SO2 | 11/07/2000 |
| 6136847 | Water-soluble trioxanes as potent and safe antimalarial agents Biologically-active, water soluble, 3-substituted trioxanes of the formula ##STR1## wherein R represents a COOH-- substituted aryl group, a substituted or unsubstituted heteroaryl group or an alkyl group, and C12 -(p-carboxy)benzyloxy trio... | 10/24/2000 |
