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Patent No. 5678617

Method and apparatus for making a drink hop along a bar or counter

A method for generating a drink which appears to hop from a remote spot on the bar or counter and take one or more leaps, before landing in a patron's glass.

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Class 549/268 - Polycyclo ring system having the lactone ring as one of the cyclos


Subclass of Class 549 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the lactone ring having at least seven
No. of patents: 82
Last issue date: 07/27/2010


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NumberTitleIssue Date
7763740Method for the production of mumbaistatin derivatives
The present invention relates to a process for preparing mumbaistatin derivatives (I), where the anthraquinone skeleton is constructed via a Diels-Alder reaction and the central methylene bridge via a transition metal-catalyzed reaction, and to the intermediates use...
07/27/2010
7745646Bicyclic heteroaryl inhibitors of PDE4
The present invention relates to compounds and methods which may be useful as inhibitors of phosphodiesterase 4 (PDE4) for the treatment or prevention of inflammatory diseases and other diseases involving elevated levels of cytokines and proinflammatory mediators.
06/29/2010
7374749Amino substituted hydroxyphenyl benzophenone derivatives
Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R1, and R2 independently from each other are; C1-C20alkyl; C2-C20-alken...
05/20/2008
7329654Heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators
The present invention is directed to novel heteroatom containing tetracyclic derivatives, pharmaceutical compositions containing them, their use in the treatment and/or prevention of disorders mediated by one or more estrogen receptors and processes for their prepar...
02/12/2008
7314942Methylenelactones syntheses in supercritical fluids
Alpha-methylenelactone is produced from butyrolactone and valerolactone by the addition of formaldehyde in a supercritical fluid. ...
01/01/2008
73122009-ketospinosyn derivatives
The present invention relates to derivatives of 9-keto spinosyns, which are substituted by a ═N—(O, NH or NRx)—Ry moiety in the C-9 position, to methods for their manufacture, and to their use for controlling animal pests. ...
12/25/2007
7176234Derivatives of gambogic acid and analogs as activators of caspases and inducers of apoptosis
The present invention is directed to derivatives of gambogic acid and analogs thereof. Exemplary gambogic acid derivatives of the present invention include, among others, derivatives substituted in the C10 and C28 positions of gambogic acid. The present invention al...
02/13/2007
7115651Macrocycles and uses thereof
The present invention relates to compounds having the structure (and pharmaceutically acceptable derivatives thereof) wherein R0–R4, Z, X, A—B, D—E, G—J, and...
10/03/2006
7105684Lactone compounds
An object of the present invention is to provide a novel monomer compound having a lactone structure which gives polymers having more excellent feature as resist material, etc. The present invention relates to a compound represented by the following formula [...
09/12/2006
6979721Substituted cyclohexene endcaps for polymers with thermal-oxidative stability
This invention relates to polyimides having improved thermal-oxidative stability, to the process of preparing said polyimides, and the use of polyimide prepolymers in the preparation of prepregs and composites. The polyimides are particularly useful in the preparati...
12/27/2005
6936402MONOMERS CONTAINING AN OXEPAN-2-ONE GROUP, PHOTORESIST COMPOSITIONS COMPRISING POLYMERS PREPARED FROM THE MONOMERS, METHODS FOR PREPARING THE COMPOSITIONS, AND METHODS FOR FORMING PHOTORESIST PATTERNS USING THE COMPOSITIONS
Disclosed herein is a novel norbornene, acrylate or methacrylate monomer as a photoresist monomer containing an oxepan-2-one group. Further disclosed are photoresist compositions comprising a polymer prepared from the monomer, methods for preparing the photoresist c...
08/30/2005
6919464Synthetic derivatives of 21-butenyl and related spinosyns
Macrolide compounds produced by synthetic modification of factors produced by NRRL 30141 have insecticidal and acaricidal activity and are useful intermediates for preparing additional insecticidal and acaricidal compounds ...
07/19/2005
6900339Bryostatin composition and bryostatin acquisition methodologies
Methods for obtaining bryostatins from the marine bryozoans of the Bugula neritina species complex are provided wherein the methods involve the extraction and purification of bryostatins from the larvae of Bugula neritina organisms. Further, the presen...
05/31/2005
6818667Eurotinones, and derivatives thereof, processes for preparing them, and their use
The present invention relates to novel compounds of the formula I in which R(1), R(2), R(3) and R(4) are, independently of each other, hydrogen or an alkyl radical. The compounds of the formula I are inhibitors of KDR ...
11/16/2004
6815463Laulimalide derivatives
Laulimalide compounds, intermediates thereto and methods for their preparation, and methods for their use in the treatment of diseases characterized by cellular hyperproliferation. ...
11/09/2004
6808724Artemisolide compound isolated from the aerial parts of Artemisia sylvatica, isolation method, and use thereof
The present invention relates to a novel compound isolated from Artemisia Sylvatica, expressed by the formula 1, a method of isolation, and its use thereof, and more particularly to a novel compound isolated from Artemisia Sylvatica, a method of isolat...
10/26/2004
6670389Laulimalide derivatives
Laulimalide compounds, intermediates thereto and methods for their preparation, and methods for their use in the treatment of diseases characterized by cellular hyperproliferation. ##STR1##...
12/30/2003
6670348Methods and compositions for destruction of selected proteins
Compounds having an ansamycin anitibiotic, or other moiety which binds to hsp90, coupled to a targeting moiety which binds specifically to a protein, receptor or marker can provide effective targeted delivery of the ansamycin antibiotic leading to the deg...
12/30/2003
6617304Method for producing macrocyclic lactone
The invention discloses a method for the production of a macrocyclic lactone represented by a formula (2), which comprises subjecting a hydroxycarboxylic acid ester represented by a formula (1) to intramolecular esterification reaction. ##STR1## In t...
09/09/2003
661073616-Halogen-epothilone derivatives, method for producing them and their pharmaceutical use
The invention relates to novel epothilone derivatives of general formula (I), wherein R8 means a halogen atom, especially a fluorine or chlorine atom, and the remaining substituents have the meanings given in the description. The novel compound...
08/26/2003
65040353-deoxy-desmycosin derivatives and process for their preparation
The present invention relates to derivatives of 3-deoxy desmycosin of the formula I, wherein, starting from triply protected desmycosin, there are performed an oxidation at C-3 in the first step and then, optionally, a hydrogenation of double bonds and an...
01/07/2003
6369099Method of locking 1 ଱-OH of vitamin D compounds in axial orientation
A method of modifying or altering the structure of a 1଱-hydroxylated vitamin D compound to increase its biological activity by altering the conformational equilibrium of the A-ring to favor a chair conformation that presents the 1଱-hydroxyl in...
04/09/2002
6307065Processes for producing epsilon caprolactones and/or hydrates and/or esters thereof
This invention relates in part to processes for producing one or more substituted or unsubstituted epsilon caprolactones and/or hydrates and/or esters thereof which comprise subjecting one or more substituted or unsubstituted penten-1-ols to carbonylation...
10/23/2001
6222048Diaryl-2-(5H)-furanones as Cox-2 inhibitors
The invention encompasses the novel compound of Formula (I) as well as a method of treating cyclooxygenase-2 mediated diseases comprising administration to a patient in need of such treatment of a non-toxic therapeutically effective amount of a compound o...
04/24/2001
6184391Processes for producing epsilon caprolactones and/or hydrates and/or esters thereof
This invention relates in part to processes for producing one or more substituted or unsubstituted epsilon caprolactones and/or hydrates and/or esters thereof which comprise subjecting one or more substituted or unsubstituted penten-1-ols to carbonylation...
02/06/2001
6100293Tetracyclic triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
08/08/2000
6090952(2R, 3S, 22R, 23R)-2,3,22,23-tetrahydroxy-24-ethyl-ଲ-homo-7-oxa-5଱-cholesta n-6-one and a process for preparing the same
The invention discloses a process for the preparation of a compound, having molecular formula C29 H50 O6 and isomeric structural formulae (2R, 3S, 22R, 23R) -2, 3, 22, 23 -tetrahydroxy-24- ethyl-ଲ-homo-7-oxa -5³...
07/18/2000
6063731Brassinosteroid analogs useful as plant growth regulators
Disclosed are compositions and methods for promoting plant growth. The compounds are cyclopropyl- and cyclobutyl-substituted brassinosteroids having high growth promoting ability. They may be used alone or in combination with other plant growth regulating...
05/16/2000
6011058Seco-cholestane derivatives and methods of making the same
The present invention is directed to novel seco-cholestane derivatives, as well as to pharmaceutical compositions thereof, and methods of making the same. More particularly, the invention relates to C5- and C8-substituted seco-cholestane derivatives. The ...
01/04/2000
6008380(2R,3S,24S)-2,3-diacetoxy-22,23-epoxy -24-ethyl-ଲ-homo-7-oxa-5଱-cholestan-6-one and a process for preparing the same
The present invention relates to a novel compound namely (2R,3S,24S)-2,3-diacetoxy-22,23-epoxy-24-ethyl-ଲ-homo-7-oxa-5଱- cholestan-6-one and a process for the preparation thereof. The said compound is represented by the structural formula ...
12/28/1999
5998408Triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
12/07/1999
5977165Radicicol derivatives
The present invention relates to radicicol derivatives represented by the following formula (I) or pharmacologically acceptable salts thereof: ##STR1## wherein R1 and R2 are the same or different and each represents hydrogen, al...
11/02/1999
5883119Triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
03/16/1999
5786492Halichondrins
Halichondrin derivatives, isolatable from a marine sponge of the Lissodendoryx Sp., have cytotoxic preparations and are of the formula: ##STR1## wherein R1 and R2 together form a spiro attached ring system selected from the grou...
07/28/1998
5763478Triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
06/09/1998
5763366Brassinosteroid derivative and plant growth regulator using the same
Brassinosteroid derivatives expressed in formula (I) and formula (II) ##STR1## and a plant growth regulator containing one type or two types of these brassinosteroid derivatives as active ingredient. The invention thereby presents novel brassinosteroid an...
06/09/1998
5741814Cyclooctadiene derivatives
Cyclooctadiene derivative of the following formula (1): ##STR1## wherein A1, A2, A3 and A4 each independently represent COOR5 (where R5 represents a hydrogen atom, a C1 -C10...
04/21/1998
5696156Triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
12/09/1997
5679705Triterpene derivatives with immunosuppressant activity
The compounds of Formula I ##STR1## are useful as immunosuppressive agents....
10/21/1997
5650430Radicicol derivatives, their preparation and their anti-tumor activity
Radicicol derivatives in which one or both hydroxy groups are acylated have valuable anti-tumor activity or may be used as chemical intermediates....
07/22/1997
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