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Class 548/365.1 - Plural 1,2-diazoles (including hydrogenated)


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the additional hetero ring is a five membered
No. of patents: 120
Last issue date: 08/09/2011


1      
NumberTitleIssue Date
7994341Process for the production of amides
The present invention relates to a process for the preparation of compounds of formula (I) wherein R1 and R2 are each independently of the other hydrogen or C1-C5alkyl and R3 is CF3 or CF2H...
08/09/2011
7288572Active substance combinations having insecticidal and acaricidal properties
The present invention relates to novel insecticidally and acaricidally active compound combinations of N2-[1,1-dimethyl-2-(methylsulphonyl)ethyl]-3-iodo-N1-{2-methyl-4-[1,2,2,2-tetrafluoro-1-(trifluoromethyl)ethyl]phenyl}phthalamide of the form...
10/30/2007
7285569Tricycles, their manufacture and use as pharmaceutical agents
The present invention relates to compounds of formula I their pharmaceutically acceptable salts, enantiomeric forms, diastereoisomers and racemates, the preparation of the above-mentioned compounds, medicaments c...
10/23/2007
7253169Aza compounds, pharmaceutical compositions and methods of use
The present invention relates to N-substituted cyclic aza compounds, pharmaceutical compositions comprising such compounds, and methods of their use for effecting neuronal activities. ...
08/07/2007
7176321Method for producing 3-amino-4-substituted-5-pyrazolones
The invention provides a method for producing a compound represented by the following formula (II), comprising executing alkali hydrolysis of a compound represented by the following formula (I) with an alkali metal hydroxide in the presence of a barium compound to f...
02/13/2007
7135499Active substance combinations having insecticidal and acaricidal properties
The present invention relates to novel insecticidally and acaricidally active compound combinations of N2-[1,1-dimethyl-2-(methylsulphonyl)ethyl]-3-iodo-N1-{2-methyl-4-[1,2,2,2-tetrafluoro-1-(trifluoromethyl)ethyl]phenyl}phthalamide of the form...
11/14/2006
7125997Differential tumor cytotoxicity compounds and compositions
The invention is directed to novel biaryl derivatives, to the uses of these compounds in various medicinal applications, including the treatment, prevention and control of proliferative diseases such as tumors, and to pharmaceutical compositions comprising these com...
10/24/2006
7101533Agent for inducing receptor potential
Disclosed is an agent for inducing receptor potential, which comprises an organic dye compound capable of inducing/evoking receptor potential in response to photostimulation in the optic nerve, wherein the organic dye compound is a polymethine organic dye compound. ...
09/05/2006
7084138Active ingredient combinations with insecticidal and acaricidal properties
The invention relates to novel active compound combinations having very good insecticidal and acaricidal properties and containing (a) cyclic ketoenols having the formula in which the gro...
08/01/2006
6919090Active substance combinations with insecticidal and acaricidal properties
The invention relates to novel active combinations of certain cyclic ketoenols and certain active compounds that together have unexpectedly good insecticidal and acaricidal properties. ...
07/19/2005
6916798Inhibitors of GSK-3 and uses thereof
The present invention relates to compounds of formula I that are useful as GSK-3 inhibitors. The invention also relates to methods of using compounds of formula I or pharmaceutical compositions comprising compounds of formula I to inhibit GSK-3 activity. The inventi...
07/12/2005
6906199Process for preparing distamycin derivatives
It is described a process for preparing, in high yields and purity and without the need of carrying out several steps and/or isolating many intermediates which could lead to undesired by-products, a distamycin derivative of formula
06/14/2005
68310393-(heterocyclyl)-substituted benzolpyrazols
The invention relates to 3-(heterocyclyl)-substituted benzoylpyrazois of formula (I), wherein the variables have the following meanings: X is O, NH or N-alkyl; R1 is alkyl; R2, R3, R4, R5 are hydrogen, alkyl or ...
12/14/2004
6831163Bichromophoric molecules
Disclosed is a molecule containing a first chromophore that exhibits a first absorption maximum above 700 nm and a second chromophore that exhibits a second absorption maximum different from the first absorption maximum, wherein the absorption of the first and secon...
12/14/2004
6831075Heterocyclic substituted pyrazolones
The present invention is directed to novel heterocyclic substituted pyrazolones, including pharmaceutical compositions, diagnostic kits, assay standards or reagents containing the same, and methods of using the same as therapeutics. The invention is also directed to...
12/14/2004
6774229Coupling condensation synthesis of heterocycles
The invention relates to a process for the preparation of heterocycles, characterised in that the following components: i) a propargyl derivative of the general structural formula I  a wherein Het is an optional...
08/10/2004
6753316Acryloyl derivatives analogous to distamycin, process for preparing them, and their use as antitumor agents
Compounds which are acryloyl substituted distamycin derivatives of formula (I) wherein: n is 2, 3 or 4; m is 1 or 2; X and Y are the same or different and are selected, independently for each heterocyclic ring of the polyetherocyclic chain, from N and CH; R1
06/22/2004
6746989Substituted benzoylpyrazoles as herbicides
The invention relates to novel substituted benzoylpyrazoles of the general formula (I), in which n represents the numbers 0, 1, 2 or 3, A represents a single bond or represents alkanediyl(alkylene), ...
06/08/2004
6716257Bridged diaminopyrazole compounds and dye compositions containing same
The new diaminopyrazole compounds are bridged 4,5-diaminopyrazole compounds or salts thereof. These diaminopyrazole compounds have the formula (I): wherein R1 represents hydrogen, a C1- to C6-alkyl,...
04/06/2004
6677341(R)-Chiral halogenated substituted heteroaryl benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
The invention relates to substituted aryl and heteroaryl (R)-Chiral Halogenated 1-Substitutedamino-(n+1)-Alkanol compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and m...
01/13/2004
6638624Squarylium dye and filter for display device
A filter for a display device, which comprises a dipyrazolylsquarylium dye represented by formula: ##STR1## wherein A and B each independently represent a substituted or unsubstituted pyrazolyl group. The filter is excellent in resistance to heat and ligh...
10/28/2003
6583182Compounds with chelation affinity and selectivity for first transition series elements: use in medical therapy and diagnosis
This invention involves synthesis and use of a class of compounds with chelation affinity and selectivity for first transition series elements. Administration of the free or conjugated compound, or physiological salts of the free or conjugated compound, r...
06/24/2003
6552051Energetic nitramine-linked azoles and related compounds as oxidizers, initiators and gas generators
Novel compounds are provided having the structural formula R[--N(NO2)--L--R1 ]n wherein R, L, R1 and n are defined herein. The compounds are useful in a variety of contexts, but are primarily to be used as high ...
04/22/2003
65067083-(heterocyclyl)-benzoylpyrazole-derivatives
3-(Heterocyclyl)benzoylpyrazole derivatives of the formula I ##STR1## where: X is O, NH or N-alkyl; R1 is nitro, halogen, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfonyl or haloalkylsulfonyl; R2,R3,R4,R
01/14/2003
6465658Process for the preparation of N,N'-carbonyldiazoles and azolide salts
This invention relates to the preparation of N,N'-carbonyldiazoles in a particularly advantageous manner by reacting corresponding azolide salts with phosgene in an aromatic compound or an ether as solvent. The azolide salts are preferably prepared by a n...
10/15/2002
6452017Complexes having tris(pyrazolyl)methanate ligands
Methods of forming a film on a substrate using chemical vapor deposition techniques and pyrazolyl complexes. The complexes and methods are particularly suitable for the preparation of semiconductor structures....
09/17/2002
6444696Pyrazole derivatives P38 MAP kinase inhibitors
The present invention relates to certain pyrazole derivatives of Formula (I): ##STR1## that are p-38 MAP kinase inhibitors, pharmaceutical compositions containing them, methods for their use, and methods for preparing these compounds....
09/03/2002
6380393Ligands, transition metal complexes and methods of using same
Compositions including at least one organic ligand including a first hetero atom and a second hetero atom directly bonded to the first hetero atom or located one carbon atom away from the first hetero atom, with at least one of the hetero atoms being nitr...
04/30/2002
6358631Mixed vapor deposited films for electroluminescent devices
A light emitting device (LED) structure and devices containing the same in which the LED structure contains a plurality of at least a first and a second light emitting organic device (LED) stacked one upon the other, to form a layered structure, with each...
03/19/2002
6335357Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient
A 1-aryl-3-cyano-5-(het)arylalkylaminopyrazole derivative represented by the general formula (1): ##STR1## process of making, intermediate thereof and pesticide therewith....
01/01/2002
6271237Nitrogen containing heteromatics with ortho-substituted P1s as factor Xa inhabitors
The present application describes nitrogen containing heteroaromatics with ortho-substituted P1's and derivatives thereof of formula I: ##STR1## or pharmaceutically acceptable salt or prodrug forms thereof, wherein J is N or NH and D is substituted ortho ...
08/07/2001
6271179Benzylidene pyrazolones, production and use thereof
Benzylidenepyrazolones of the formula I, ##STR1## Useful as herbicides....
08/07/2001
6265351Phenylpyrazoles with a herbicidal activity
The invention relates to phenylpyrazoles having general formula (I): ##STR1## The compounds having formula (I) have a high herbicidal activity and are used for controlling weeds in the agronomic field....
07/24/2001
6207618Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
Substituted 4-benzoylpyrazole of the formula I ##STR1## where: Q is a pyrazole of the formula II ##STR2## X1 is a straight-chain or branched C1 -C6 -alkylene, a C2 -C6 -alkenylene or a C2 -...
03/27/2001
6201003Pesticidal 1-arylpyrazoles
1-Arylpyrazoles of the formula: ##STR1## wherein R31, R32, R33, R4, R5, R12, R13, R14, R15 and Z are as defined in the specification, are useful as pesticid...
03/13/2001
61659444-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
4-(3-Heterocyclyl-1-benzoyl)pyrazoles of the formula I ##STR1## where: R1 and R3 are each hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsu...
12/26/2000
6159673Oxonol compound, light-sensitive material and process for the synthesis of oxonol compound
An oxonol compound is represented by the following formula (I): ##STR1## in which Z is an atomic group that forms a cyclic amide ring; each of W1 and W2 independently is an atomic group that forms an acidic nucleus ring; and M i...
12/12/2000
6156702Substituted 4-benzoylpyrazoles
4-Benzoylpyrazoles of the formula I ##STR1## useful for controlling harmful plants, are disclosed....
12/05/2000
6143696Substituted 4-(3-alkenylbenzoyl)pyrazoles
4-(3-Alkenylbenzoyl)pyrazoles of the formula I ##STR1## and agriculturally useful salts thereof; processes for preparing the compounds of the formula I; compositions comprising them; and the use of these derivatives or of compositions comprising them...
11/07/2000
6020357Nitrogen containing heteroaromatics as factor Xa inhibitors
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I: ##STR1## or pharmaceutically acceptable salt or prodrug forms thereof, wherein J is N or NH and D may be C(.dbd.NH)NH2, which are u...
02/01/2000
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