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| Number | Title | Issue Date |
| 7361654 | Substituted heteroaryl amide modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof The present invention relates to new class of non-steroidal compounds which are useful in treating diseases associated with modulation of the glucocorticoid receptor, AP-1, and/or NF-κB activity including obesity, diabetes, inflammatory- and immune-associated disea... | 04/22/2008 |
| 7326728 | Modulators of glucocorticoid receptor, AP-1, and/or NF-κβ activity and use thereof Novel non-steroidal compounds are provided which are useful in treating diseases associated with modulation of the glucocorticoid receptor, AP-1, and/or NF-κB activity including obesity, diabetes, inflammatory and immune diseases, and have the structure of formula ... | 02/05/2008 |
| 7214701 | Active substance combinations having insecticidal and acaricdal properties The invention relates to insecticidal mixtures for protecting plants against attack by pests comprising (a) compounds of the formula (I) ... | 05/08/2007 |
| 6995181 | Modulators of the glucocorticoid receptor and method Novel non-steroidal compounds are provided which are glucocorticoid receptor modulators which are useful in treating diseases requiring glucocorticoid receptor agonist or antagonist therapy such as obesity, diabetes, inflammatory and immune disorders, and have the s... | 02/07/2006 |
| 6919357 | α adrenergic agents Aspects of the present invention are directed towards compounds of Formula I for the treatment of human erectile disorders including erectile dysfunction in men. wherein: R1 is hydrogen, halo, h... | 07/19/2005 |
| 6916924 | Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents This invention relates to novel processes for preparing heteroaryl-substituted urea compounds of formula (I): which are useful for treating diseases and pathological conditions involving inflammation such as chronic in... | 07/12/2005 |
| 6911595 | Charge transfer material, and photoelectric conversion device and photoelectric cell using same, and pyridine compound A charge transfer material comprising a basic compound having negative charge and represented by the following general formula (I): (A1-L)n1-A2·M (I), wherein A1 represents a group having negativ... | 06/28/2005 |
| 6762190 | Thienylalanine derivatives as inhibitors of cell adhesion The present invention relates to compounds of formula (I), in which A, B, X, Y, R1, R2, R3 and n have the meanings indicated in the claims. The compounds of formula (I) are valuable pharmacologically active compounds. They are vitron... | 07/13/2004 |
| 6465650 | Substituted N-ethylglycine derivatives for preparing PNA and PNA/DNA hybrids The invention provides a processes for the preparation of a compound of Formula I, or a salt thereof ##STR1## wherein PG is a urethane- or trityl-type protective group; X is NH, O, or S; Y is CH2, O, or NH; and B' is a base customary in nucleot... | 10/15/2002 |
| 6448286 | Imino pyrrolidine derivatives useful as nitric oxide synthase inhibitors The current invention discloses useful pharmaceutical compositions containing amidino derivative useful as nitric oxide synthase inhibitors.... | 09/10/2002 |
| 6410542 | Aminotetrazole derivatives useful as nitric oxide synthase inhibitors The current invention discloses aminotetrazole derivatives useful as nitric oxide synthase inhibitors.... | 06/25/2002 |
| 6277845 | Hydrazono-benzazulene derivatives, pharmaceutical compositions and intermediates Compounds of the formula ##STR1## wherein the substituents are as defined in the application and their pharmaceutically acceptable acid and base salts thereof which are useful for preventing loss of bone matrix.... | 08/21/2001 |
| 6169089 | Aminotetrazole derivatives useful as nitric oxide synthase inhibitors The current invention discloses aminotetrazole derivatives useful as nitric oxide synthase inhibitors.... | 01/02/2001 |
| 6147097 | Imidazole derivatives as anti-HIV agents An imidazole derivative represented by general formula (I) or a salt thereof, having the effect of specifically inhibiting the growth of HIV as a pathogenic virus and being reduced in toxicity. In said formula R1 represents hydrogen, C1 | 11/14/2000 |
| 6075143 | Substituted N-ethylglycine derivatives for preparing PNA and PNA/DNA hybrids There are described N-ethylglycine derivatives of the formula I ##STR1## in which PG is a urethane-type or trityl-type amino protective group which is labile to weak acids, X is NH, O or S, Y is CH2, NH or O, and B' are bases customary in ... | 06/13/2000 |
| 6005117 | Imino compounds, process for their preparation and their use as victronectin antagonists There are described imino derivatives of formula (I) R1 --Y--A--B--D--E--F--G (I) their preparation and their use as medicaments. The compounds according to the invention may be used as vitronectin receptor antagonists and as... | 12/21/1999 |
| 5919787 | Aminotetrazole derivatives useful as nitric oxide synthase inhibitors The current invention discloses aminotetrazole derivatives useful as nitric oxide synthase inhibitors.... | 07/06/1999 |
| 5919792 | Integrin antagonists This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as vitronectin receptor antagonists. The vitronectin receptor antagonist compounds of the present invention are v댣 antagonists, ... | 07/06/1999 |
| 5886190 | Rapid synthesis and use of 18F-fluoromisonidazole and analogs The present invention involves a rapid synthesis of 18 F-FMISO and analogs thereof. New precursors such as 1-(2'-nitro-1'-imidazolyl)-2-0-acetyl-3-0-tosylpropanol, glycerol-1,3-ditosylate-2-0-acetylate, 1-(2'-nitro-1'-imidazolyl)-2,3-0-dia... | 03/23/1999 |
| 5854251 | Aminotetrazole derivatives useful as nitric oxide synthase inhibitors Aminotetrazole derivatives of the formula (I) wherein the variables are as defined in the disclosure are useful as nitric oxide synthase inhibitors. ##STR1##... | 12/29/1998 |
| 5840911 | Imidazole derivatives, their preparation and their use as S-adenosylmethionine decarboxylase (=SAMDC) inhibitors Described are compounds of formula I ##STR1## wherein R1 is hydrogen or hydroxy; R2, R2 ' and R2 " are each independently of the others hydrogen or a substituent other than hydrogen; either R3 is hydr... | 11/24/1998 |
| 5733934 | Antiarrythmic and cardioprotective substituted indenoylguanidines Indenoylguanidines of formula I and formula II, the process for their preparation, their use as medicaments, medicaments containing them, their use as diagnostic agents and medicaments containing them are described. Compounds I are useful for treating car... | 03/31/1998 |
| 5733882 | Retroviral protease inhibitors The present invention provides compounds, more particularly dipeptide analogs, which bind to retroviral proteases. These compounds are inhibitors of retroviral proteases and are useful for treating diseases related to infection by retroviruses.... | 03/31/1998 |
| 5684008 | Aminotetrazole derivatives useful as nitric oxide synthase inhibitors The current invention discloses aminotetrazole derivatives useful as nitric oxide synthase inhibitors.... | 11/04/1997 |
| 5554633 | Substituted amines as tachykinin receptor antagonists Compounds of formula (I), and salts and prodrugs thereof, wherein Q is optionally substituted phenyl or benzhydryl; X and Y are each H or together form a group=O; Z is O, S or NR9, where R9 is H or C1-6 alkyl; R1 | 09/10/1996 |
| 5552427 | Glutaminase inhibitory compounds, compositions, and methods of use There is disclosed a pharmaceutical composition for inhibiting glutaminase which comprises a imidazole derivative or a salt thereof. This compound selectively inhibits the proliferation of tumor cells, and the composition is useful as an anti-cancer agent... | 09/03/1996 |
| 5543433 | Azine-substituted phenylacetic acid derivatives and fungicides containing these Compounds of the formula I ##STR1## where X is hydrogen, halogen, alkyl, alkoxy, trifluoromethyl, cyano or nitro, Y is an amino, methylamino or dimethylamino group, Z is a group CHCH3, CHOCH3 or NOCH3, R is hydrogen or alk... | 08/06/1996 |
| 5503776 | N-acylcarnosines and their use as antioxidants An N-acylamino acid compound represented by the general formula (1): R--CO--(NH--X--CO)n --OR1 (1) wherein (NH--X--CO) is an amino acid residue, X in (NX--X--CO) is variable with the kind of amino acid to be used, R--CO ... | 04/02/1996 |
| 5403930 | Substituted salicylic acids A compound of the formula Het--NR--SO2 --Ph2 --A--Ph1 (COOH)(OH) and tautomic form, salts, solvates, C1-6 alkyl esters and pharmaceutical compositions of the compound. Ph1 and Ph2 are benze... | 04/04/1995 |
| 5352831 | Oligomeric cyanoguanidines Oligomeric cyanoguanidines of formula I ##STR1## wherein, for example, R1 and R2 are each phenyl, R is 1,4-phenylene and n is an integer from 1 to 20, are suitable latent hardeners for epoxy resins. They are readily soluble in s... | 10/04/1994 |
| 5317021 | 3-mercapto-glutamic acid derivatives Amino acid compounds of the formula: ##STR1## wherein the various symbols are as hereinafter described, which have inhibiting effect on enkephalinase.... | 05/31/1994 |
| 5302718 | Compounds containing an amino salicylic acid moiety linked to a sulphapyridine moiety via stable bridge A compound of the formula Het--NR--SO2 --Ph2 --A--Ph1 (COOH)(OH) and tautomeric form, salts, solvates, C1-6 alkyl esters and pharmaceutical compositions of the compound. Ph1 and Ph2 are ben... | 04/12/1994 |
| 5264584 | Dialkoxymethylimidazolidine derivatives Novel dialkoxymethylimidazolidine derivatives of the formula (1) ##STR1## are described. Also, a preparation process of the derivatives and insecticidal compositions comprising the same are set forth. In addition, novel intermediate compounds of the ... | 11/23/1993 |
| 5258381 | 2-substituted-2-imidazolines The present invention relates to compositions and methods for inhibiting nonenzymatic cross-linking (protein aging) which contain novel 2-substituted-2-imidazolines. Accordingly, a composition is disclosed which comprises an agent capable of inhibiting th... | 11/02/1993 |
| 5234946 | Substituted alkylamine derivatives The substituted alkylamine derivatives represented by formula (I) ##STR1## wherein R1 represents (a) substituted or unsubstituted C2-6 alkenyl group, (b) substituted or unsubstituted C3-6 cycloalkenyl group, (c) subst... | 08/10/1993 |
| 5229404 | Azacyclic carboxylic acid derivatives and their preparation and use Novel O-alkylated oximes of the general formula I ##STR1## wherein R1 and R2 are optionally substituted aromatic or heteroaromatic rings, R3 is hydrogen or lower alkyl, R4 is a nitrogen containing, substitu... | 07/20/1993 |
| 5223525 | Pesticidal 1-arylimidazoles The invention describes novel 1-arylimidazoles of formula (I) ##STR1## wherein typically preferred substituents are: X is S(O)n R1, in which R1 is an alkyl group, preferably a methyl group, which is fully substituted ... | 06/29/1993 |
| 5192778 | Dialkoxymethylimidazolidine derivatives, preparation thereof, insecticides containing same as an effective ingredient and intermediates therefor Novel dialkoxymethylimidazolidine derivatives of the formula (1) ##STR1## are described. Also, a preparation process of the derivatives and insecticidal compositions comprising the same are set forth. In addition, novel intermediate compounds of the ... | 03/09/1993 |
| 5086184 | N-heterocyclic benzamides N-Aryl benzamides wherein the aryl group is a nitrogen containing heterocycle are useful as selective herbicidal agents. Compositions containing the novel benzamides and a herbicidal method of selective weed control are disclosed.... | 02/04/1992 |
| 5068365 | Hexahydrophthalic anilide derivatives Disclosed is novel hexahydrophthalic anilide derivatives and herbicide compositions comprising the derivatives. The hexahydrophthalic anilide derivatives of this invention are represented by the formula [I], [II] or [III]. ##STR1## (wherein R | 11/26/1991 |
