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| Number | Title | Issue Date |
| 7326255 | Use of latent pigments for high-remanence dyeing, composition containing the said pigments and processes using them The invention relates to the use, for dyeing keratin fibres, of at least one latent pigment, which is soluble in a medium that is suitable for dyeing, and which can be chemically, thermally or photochemically converted in the fibres into water-insoluble pigments, of... | 02/05/2008 |
| 7244756 | Benzimidazol-2-one derivatives and their use Certain 1,5-disubstituted benzimidazol-2-one compounds useful as therapeutic agents. The compounds may be of the Formula I wherein: R′ represents hydrogen or alkyl; R″ represents halogen or trihalogenmethyl; ... | 07/17/2007 |
| 7214697 | 2-Oxo-benzimidazolyl substituted ethanolamine derivatives and their use as βagonists The present invention relates to a β3 adrenergic receptor agonist of formula (I), wherein R is C3–C8 alkyl or (C3–C7 cycloalkyl)C1–C5 alk-di-yl: R1 is H, CN, halo; C1... | 05/08/2007 |
| 7196202 | 1-aryl-2-N-, S- or O-substituted benzimidazole derivatives, their use for the production of pharmaceutical agents as well as pharmaceutical preparations that contain these derivatives The invention relates to novel benzimidazole derivatives with general formula I, whereby radicals R1, R2, R3, A, B, Y and Z have the meanings that are indicated in the description and the claims, the use of these compounds for the pr... | 03/27/2007 |
| 7186745 | Indolone derivatives having vascular damaging activity This invention relates to the use of compounds of Formula (I) as vascular damaging agents: wherein X is selected from: —O—, —S—, —S(O)—, —S(O2)—, —N(R5)—, —C(O)—, —C(O)N(R5)—, —N(R5)C(O)—, â... | 03/06/2007 |
| 7176312 | Kinase inhibitor scaffolds and methods for their preparation General methods for the solution phase as well as solid phase synthesis of various substituted heteroaryls has been demonstrated. These substituted heteroaryls can be further elaborated by aromatic substitution with amines at elevated temperature or by anilines, bor... | 02/13/2007 |
| 7132547 | Preventives/remedies for urinary disturbance Preventives/remedies for voiding disturbance containing a compound having both of an acetylcholinesterase inhibitory action and an α1 antagonistic action which exhibits an excellent effect of improving the urinary function of the bladder (i.e., effects of improving... | 11/07/2006 |
| 7115644 | Heterocyclic compounds Disclosed are benzimidazolone compounds of formulas (I) & (II): wherein R1, R2, R3, R4, R5, X, L, m, n and t are defined herein. The compounds inhibit production of cytokines involved in inflammatory proc... | 10/03/2006 |
| RE39197 | Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds The present invention relates to novel cinnamide compounds that are useful for treating inflammatory and immune diseases, to pharmaceutical compositions comprising these compounds, and to methods of inhibiting inflammation or suppressing immune response in a mammal.... | 07/18/2006 |
| 7064214 | Methods of preparing sulfinamides and sulfoxides This invention encompasses novel methods of preparing sulfinamides and sulfoxides, particularly stereomerically pure sulfinamides and sulfoxides. The invention further encompasses novel compounds from which sulfinamides and sulfoxides can be prepared. ... | 06/20/2006 |
| 7009060 | 2-oxo-benzimidazolyl substituted ethanolamine derivatives and their use as βagonists The present invention relates to a β3 adrenergic receptor agonist of formula I: or a pharmaceutical salt thereof; which is capable of increasing lipolysis and energy expenditure in cells and, therefore, is u... | 03/07/2006 |
| 7002021 | Diketopyrrolopyrrole pigments Diketopyrrolopyrroles of the formula (I): wherein R1, R2, R3 and R4 independently of one another are a C1–C4 alkyl radical or a substitute... | 02/21/2006 |
| 6939887 | Benzimidazolidinone derivatives The present invention can provide novel compounds useful as orally administrable growth hormone releaser, more specifically a benzimidazolidinone derivative of formula (1) or a pharmaceutically acceptable salt thereof: (1) wherein ... | 09/06/2005 |
| 6933390 | Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate The invention concerns a process for the preparation of N-aryl-aza-heterocycles of the general formula I by reaction of aza-heterocycles with activated aryl halides with use of caesium carbonate without addition of fur... | 08/23/2005 |
| 6906090 | Compositions and methods for treating mycobacterial diseases The invention provides the use of certain isatin and oxindole derivatives in the preparation of a medicament for use in the treatment of mycobacterial disease. ... | 06/14/2005 |
| 6884896 | Benzo[b]thiophene derivatives and process for preparing the same The present invention is 3,4-disubstituted-benzo[b]thiophene derivatives represented by general formula (I) and processes for preparing compounds represented by general formula (V) from compounds represented by general formula (IV), preparing a mixture of compounds ... | 04/26/2005 |
| 6878700 | Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds The present invention relates to novel cinnamide compounds that are useful for treating inflammatory and immunune diseases, to pharmaceutical compositions containing these compounds, and to methods of inhibiting inflammation or suppressing immune response in a mamma... | 04/12/2005 |
| 6869913 | Pyridazin-3-one derivatives, their use and intermediates for their production Novel pyridazin-3-one derivatives of formula [1] are provided, which are useful as active ingredients of herbicides, wherein R1 is haloalkyl; R2 and R3 are hydrogen, alkyl, haloalkyl, o... | 03/22/2005 |
| 6867203 | Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds The present invention relates to novel cinnamide compounds that are useful for treating inflammatory and immune diseases and cerebral vasospasm, to pharmaceutical compositions containing these compounds, and to methods of inhibiting inflammation or suppressing immun... | 03/15/2005 |
| 6683101 | Bicyclic cyclohexylamines and their use as NMDA receptor antagonists Described are heterocycle-substituted cyclohexylamines of formula (I), and their pharmaceutically acceptable salts thereof. The compounds of the formula (I) are antagonists of NMDA receptor channel complexes useful for treating cerebral vascular disorders... | 01/27/2004 |
| 6624186 | Ion channel modulating agents comprising novel benzimidazolone derivatives The present invention relates to ion channel modulating agents. More particularly, the present invention relates to a particular class of chemical compounds that has proven useful as modulators of SKCa, IKCa and BKCa chann... | 09/23/2003 |
| 6613743 | Sulfonamide inhibitors of aspartyl protease The present invention relates to a novel class of sulfonamides of formula I which are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of HIV aspartyl protease inhibitors characterized by specific structural and phy... | 09/02/2003 |
| 6608049 | Indazoles The invention relates to new indazole derivatives, processes for their preparation, and their use in medicaments.... | 08/19/2003 |
| 6573379 | Method for preparing halomethyl heterocyclic compounds The present invention relates to a method for preparing 5- and 6-halomethyl quinoxalines. The method comprises contacting a 5- or 6-methyl quinoxaline with a halogenating agent in the presence of a radical initiator in a solvent selected from the group co... | 06/03/2003 |
| 6562972 | Method for preparing heterocyclic-carboxylic acids The present invention relates to a method for preparing quinoxaline-5- and 6-carboxylic acids. The method comprises contacting an aqueous alkaline suspension of a 5- or 6-halomethyl quinoxaline with oxygen in the presence of a transition metal catalyst, t... | 05/13/2003 |
| 6562121 | Conditioning of organic pigments Organic pigments are conditioned by introducing a liquid prepigment suspension into a miniaturized continuous reactor and thermally treating therein.... | 05/13/2003 |
| 6559308 | Method for preparing heterocyclic-carboxylic acids The present invention relates to a method for preparing quinoxaline-5- and 6-carboxylic acids. The method comprises contacting an aqueous suspension of a 5- or 6-hydroxymethyl quinoxaline with oxygen in the presence of a transition metal catalyst, to form... | 05/06/2003 |
| 6552042 | Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor Xa The present application describes inhibitors of factor Xa of formula I: ##STR1## or pharmaceutically acceptable salt forms thereof, wherein W, W1, W2, and W3 may be N or C and J, Ja, and Jb combine to ... | 04/22/2003 |
| 6492517 | Method for preparing halomethyl heterocyclic compounds The present invention relates to a method for preparing 5- and 6-halomethyl quinoxalines. The method comprises contacting a 5- or 6-methyl quinoxaline with a halogenating agent in the presence of a radical initiator in a solvent selected from the group co... | 12/10/2002 |
| 6403616 | Chemical process and pharmaceutical formulation Process for the manufacturing of slightly soluble or less soluble alkaline salts of substituted sulphinyl heterocycles containing an imidazole moiety with formula I ##STR1## preferably alkaline salts of a proton pump inhibitor compound, wherein the p... | 06/11/2002 |
| 6362208 | Anilide compounds and drugs containing the same The invention relates to a novel anilide compound and a pharmaceutical composition comprising the same. The invention relates to a compound represented by the following general formula: ##STR1## represents a divalent residue of benzene with a substituent(... | 03/26/2002 |
| 6352985 | Benzimidazole compounds A benzimidazole compound represented by the formula (I): ##STR1## wherein R3 is a carboxyl group, a esterified carboxyl group, an amidated carboxyl group, an amino group, an amido group, or a sulfonyl group, or their pharmaceutically acceptable... | 03/05/2002 |
| 6316482 | Benzamide derivatives having a vasopressin antagonistic activity This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkoxy, etc., R2 is lower alkyl, et... | 11/13/2001 |
| 6316474 | 2-benzyl and 2-heteroaryl benzimidazole NMDA/NR2B antagonists Benzimidazoles, substituted in the 2-position by substituted benzyl groups or heteroaryl groups are effective as NMDA NR2B antagonists and are useful for relieving pain.... | 11/13/2001 |
| 6300325 | IL-8 receptor antagonists This invention relates to novel benzo-2-triazole substituted compounds, pharmaceutical compositions, processes for their preparation, and use thereof in treating IL-8, GRO, GROଲ, GROγ and NAP-2 mediated diseases.... | 10/09/2001 |
| 6274728 | Soluble chromophores having improved solubilizing groups Compounds of formula A(B)x (I), wherein x is an integer from 1 to 8, A is the radical of a chromophore of the quinacridone, anthraquinone, perylene, indigo, quinophthalone, indanthrone, isoindolinone, isoindoline, dioxazine, azo, phthalocyanine or ... | 08/14/2001 |
| 6268313 | Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production The dihalopropene compounds of the general formula [I] have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.... | 07/31/2001 |
| 6252104 | Naphthol derivatives and process for producing the same A naphthol derivative represented by the general formula (I), [wherein Y and Y' indicate --(CONH)n --X or --COR; X is a phenyl group, a naphthyl group, an anthraquinonyl group, a benzimidazolonyl group or a carbazolyl group; R is a hydroxyl gro... | 06/26/2001 |
| 6242445 | Benzimidazole derivative ##STR1## A novel benzimidazole derivative [specifically, for example, 2-ethoxy-1-[{4'-(2"-N,N-dimethylaminoethoxycarbonyl)phenyl}methyl]-1H-benz imidazole-6-carboxylic acid morpholide] represented by formula (I) and a salt thereof. The compound exhibits sa... | 06/05/2001 |
| 6211347 | Process for preparing fine pigment dispersions Preparation of pigment dispersions by a1) subjecting a mixture A comprising a latent pigment and a polymer to thermal, chemical or photolytic treatment and b) then adding a solvent, or a2) subjecting a mixture B comprising a latent pigment, a polymer and a sol... | 04/03/2001 |
