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Patent No. 6293874

User-operated amusement apparatus for kicking the user's buttocks

An apparatus including a user-operated and controlled apparatus for self-infliction of repetitive blows to the user's buttocks by a plurality of elongated arms bearing flexible extensions that rotate under the user's control.

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Class 548/301.1 - One of the two rings which form the spiro is part of a polycyclo ring system


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein one of the two rings that form the spiro
No. of patents: 124
Last issue date: 01/11/2011


1        
NumberTitleIssue Date
7868181Compounds
The present invention relates to new compounds of formula I, where R1 and R2 are independently halo or C1-3haloalkyl, X is ethenyl or ethynyl, or a salt thereof....
01/11/2011
7329759Illudin analogs useful as antitumor agents
The present invention provides illudin analogs of the general formula (I): where R1 is (CH2)n—X—Y or H; n is 0 to 4; X is O or S or N or absent; and Y...
02/12/2008
7309787Kinase inhibitors
The present invention relates to organic molecules capable of modulating tyrosine kinase signal transduction in order to regulate, modulate and/or inhibit abnormal cell proliferation. ...
12/18/2007
7288559Carboxamide spirohydantoin CGRP receptor antagonists
The present invention is directed to compounds that are antagonists of CGRP receptors and that are useful in the treatment or prevention of diseases in which the CGRP is involved, such as headache, migraine and cluster headache. The invention is also directed to pha...
10/30/2007
7220866Imidazolic compounds and use thereof as alpha-2-adrenergic receptors
The invention provides compounds having the formula (1): wherein R1 is hydrogen, fluoro or methoxyl, R1 being in position 2, 3, 4 or 5 of the aromatic carbocycle; R2 is hydrogen or methyl; R3 is hydrogen, methyl ...
05/22/2007
7202251Bicyclic anilide spirohydantoin CGRP receptor antagonists
The present invention is directed to compounds of the formula: that are antagonists of CGRP receptors and that are useful in the treatment or prevention of diseases in which the CGRP is involved, such as headache...
04/10/2007
7189722Aryl spirohydantoin CGRP receptor antagonists
The present invention is directed to compounds that are antagonists of CGRP receptors and that are useful in the treatment or prevention of diseases in which the CGRP is involved, such as headache, migraine and cluster headache. The invention is also directed to pha...
03/13/2007
7166611Pharmaceutical compositions having appetite suppressant activity
A pharmaceutical composition contains an extract obtainable from a plant of the genus Trichocaulon or Hoodia containing an appetite suppressant agent having the formula (1). A process for obtaining the extract and a process for synthesizing compound (1...
01/23/2007
7084208N-halamine vinyl compounds and their polymeric biocides
The present invention provides heterocyclic vinylic compounds that can be used to form biocidal polymers. The polymers thus generated can used alone or can be grafted onto textiles, fabrics and polymers. The polymers are readily converted to N-halamine structures on...
08/01/2006
7019148Synthesis of irbesartan
Provided are a method of making irbesartan via a Suzuki coupling reaction and a novel intermediate, 2-butyl-3-(4′-bromobenzyl)-1,3-diazaspiro[4.4]non-1-ene-4-one, for such process. The novel process includes the step of reacting such intermediate with a protected ...
03/28/2006
7014781Methods and articles for maintaining hydantoinylated polymers in a biocidally active state
A composition and the method for sustaining the biocidal activity of chlorinated polystyrene hydantoin beads. The method comprises supplying a continuous low level halogen concentration to the chlorinated polystyrene hydantoin beads in the water to be treated that f...
03/21/2006
6919364Microbiological control in animal processing
Fecal bacterial contamination in an animal is reduced by providing it with drinking water containing a microbiocidally-effective amount of halogen-based microbiocide resulting from mixing with water (A) a product formed in water from (i) bromine, chlorine, or bromin...
07/19/2005
6908636Microbiological control in poultry processing
In the processing of poultry, equipment, instruments, apparatus and/or water used in such processing, and/or carcasses and/or parts of poultry resulting from the processing of poultry, are disinfected with aqueous solutions of certain halogen-based microbiocides, es...
06/21/2005
6768009N-halamine vinyl compounds and their polymeric biocides
The present invention provides heterocyclic vinylic compounds that can be used to form biocidal polymers. The polymers thus generated can used alone or can be grafted onto textiles, fabrics and polymers. The polymers are readily converted to N-halamine structures on...
07/27/2004
6500958Carboxylic acid derivatives and process for producing the same
The present invention relates to compounds which are useful for efficient synthesis of 2-amino-4-oxobicyclo[3.1.0]hexane-2,6-dicarboxylic acids. The compounds according to the present invention comprise 2-oxobicyclo[3.1.0]hexane-6-carboxylic acid derivatives r...
12/31/2002
6316437Spirohydantoin compounds and uses thereof
Spirohydantoin compounds and their pharmaceutically acceptable salts are disclosed. The synthesis of these compounds and their use as alpha 1a adrenergic receptor antagonists is also described. One application of these compounds is in the treatment of ben...
11/13/2001
6191160Spiro-indolines as Y5 receptor antagonists
Compounds of the general structural formula I ##STR1## are selective NPY Y5 receptor antagonists. The compounds and compositions of the present invention are useful in the treatment of obesity and complications associated therewith....
02/20/2001
6172097Spiro imidazoline compounds
The invention relates to a compound of formula (I): ##STR1## wherein: A represents an optionally substituted benzene ring, B represents an imidazoline ring of formula (Ia) or (Ib): ##STR2## and medicinal products containing the same/are useful in treating or i...
01/09/2001
6124463Benzimidazoles as corticotropin release factor antagonists
The present invention describes novel benzimidazoles of formula: ##STR1## or pharmaceutically acceptable salt forms thereof, which are useful as CRF antagonists....
09/26/2000
5958960Excitatory amino acid receptor modulators
Compounds of the formula ##STR1## in which R1 and R2 are as defined in the specification, and non-toxic metabolically labile ester and amides thereof are useful as modulators of metabotropic glutamate receptor function....
09/28/1999
5670646Monomeric and polymeric cyclic amine and-halamine compounds
Cyclic amine monomers and polymers and N-halamine biocidal polymer compounds are provided. Methods of making and using the same wherein the functional groups unhalogenated or halogenated hydantoins, triazine diones, imidazolidinones, and pyrimidinones are...
09/23/1997
5648374Benzospiroalkene compounds
Compounds of formula (I): ##STR1## in which: X represents --CH2 --, --(CH2)2 --, --CH.dbd.CH--, --O--CH2 --, --S--CH2 --, --SO--CH2 -- or --SO2 --CH2 --, Y repres...
07/15/1997
5591848Spiroconjugated charge-transfer dyes for optical applications
New intramolecular charge-transfer organic dyes are described. The design of these molecules is based on the phenomenon of spiroconjugation, and it provides a modular approach to the preparation of unique materials with interesting optical properties. In ...
01/07/1997
5559233Methods for preparing n-substituted heterocyclic derivatives
The invention relates to processes for preparing N-substituted heterocyclic compounds of formula (I) ##STR1##...
09/24/1996
5534536Fused phenol derivatives
Fused phenol compounds of the formula (I): ##STR1## (wherein R1 and R2 each, independently, is H, halogen, trifluoromethyl, cyano, (substituted) alkyl, alkoxy, cycloalkyl, COOH, COOR6 (in which R6 is C1-6 a...
07/09/1996
5464859Benzospiroalkene derivatives
Compounds of formula (I): ##STR1## wherein: --X represents --CH2 --, --(CH2)2 --, --CH.dbd.CH--, --O--CH2 --, --S--CH2 --, --SO--CH2 -- or --SO2 --CH2 --, --R
11/07/1995
5447946Hydantoin derivatives for treating complications of diabetes
Hydantoin derivatives and salts thereof, intermediates therefor, process for the preparation thereof, and medicines containing the derivative, wherein said derivatives have the formula ##STR1## wherein one of V and W is hydrogen and the other is a ha...
09/05/1995
5436261Benzospiroalkene heterocyclic compounds
Compounds of formula (I): ##STR1## in which: X represents --CH2 --, --(CH2)2 --, --CH.dbd.CH--, --O--CH2 --, --S--CH2 --, --SO--CH2 -- or --SO2 --CH2 --, Y repres...
07/25/1995
5430048Spirocyclic benzopyran imidazolines
Spiro- [4H- 1 -benzopyran-4,4'-5'H-imidazol]-5'-ones of the Formula 1: ##STR1## wherein R1 is H, R2 F, Cl, Br, CF3, CF3 O, CN, NO2, R2 SO2, R2 NHSO2, R...
07/04/1995
5329006Chromogenic lactam compounds, their preparation and their use
Chromogenic lactam compounds of the formula ##STR1## in which the ring A is an aromatic or heteroaromatic radical which has 6 ring atoms and may contain a fused aromatic ring, it being possible for both the ring A and the fused ring to be substituted...
07/12/1994
5274104N-substituted heterocyclic derivatives useful in the treatment of cardiovascular disorders
The present invention relates to N-substituted heterocyclic derivatives of formula: ##STR1## processes for their preparation, and pharmaceutical compositions which contain them. The compounds according to the invention are non-peptide compounds ...
12/28/1993
5270317N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present
The invention relates to N-substituted heterocyclic derivatives and its salts. These derivatives have the formula ##STR1## in which the substituents are as defined in the specification. Application: Angiotensin II antagonists...
12/14/1993
5212186Cardioactive pyrrolobenzimidazoles
Compounds for the treatment of cardiac insufficiency, an arterial thrombo embolism, an arterial occlusive disease, psoriasis, neurodermatitis, asthma, platelet aggregation and hypertension, of the formula ##STR1## in which R1 is hydrogen, ...
05/18/1993
5211736Azole derivatives of spiroheterocycles
A compound having the structural formula ##STR1## where R is C2 -C8 alkylene having 2 to 4 carbon atoms linking X and Y; R1 is C1 -C8 linear or branched alkylene, C1 -C6 oxyalkylene, ...
05/18/1993
5182289Heterobicyclic compounds having antiinflammatory activity
Heterobicyclic and heterocyclic intermediate compounds and their use in treating inflammation, hyperproliferative skin conditions such as psoriasis and allergy are disclosed....
01/26/1993
5180825Mitomycin derivatives
Disclosed in a mitomycin derivative represented by the formula (I): ##STR1## wherein W is a heterocyclic group....
01/19/1993
5180419Herbicidal 2-(2-imidazolin-2-yl)-benzo-(5-membered)-heterocycles and the use thereof
There are provided o-carboxy-(5-oxo-2-imidazolin-2-yl)benzo-(5-membered)-heterocyclic compounds and derivatives thereof and a method for the use therewith to control monocotyledenous and dicotyledenous plant species....
01/19/1993
5164391Hydantoin derivatives for treating complications of diabetes and circulatory diseases
The invention relates to a hydantoin derivative, salt thereof, process for the preparation thereof, and medicine containing the derivative. The derivative is represented by the formula ##STR1## wherein M is --CONH--NHR1 group, --CONH--OR
11/17/1992
5140031Pyranyl cyanoguanidine derivatives
Novel compounds having the formula ##STR1## wherein ##STR2## are disclosed. These compounds have potassium channel activating activity and are useful, for example, as cardiovascular agents, especially as antiischemic agents....
08/18/1992
5108485Herbicidal 2-(2-imidazolin-2-yl)-benzazoles
There are provided o-carboxy-(5-oxo-2-imidazolin-2-yl)benzoheterocyclic compounds wherein the fused heterocyclic ring system is a 5-membered ring containing one, two or three nitrogen atoms, derivatives of said benzoheterocyclic compounds and a method for...
04/28/1992
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