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Class 548/268.2 - The triazole ring and the chalcogen are bonded directly to the same acyclic carbon


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the chalcogen and the triazole ring are
No. of patents: 111
Last issue date: 11/14/2006


1      
NumberTitleIssue Date
7135475Amide substituted xanthine derivatives
The present invention is a 1,3,8 substituted xanthine derivative of formula I or a pharmaceutically acceptable salt thereof, wherein R1, R2 and R3 are as defined in the specificat...
11/14/2006
6987112Organic compound having cyano group and insecticides/miticides
The present invention is directed to compounds represented by Formula (1); wherein A, R, X, Y and n are as defined in the description, the salts thereof, and insecticide/acaricide compositions characterized by comprisi...
01/17/2006
6649568Brassinosteroid biosynthesis inhibitor
Compounds represented by the following formula (I): ##STR1## wherein R1 represents a lower alkenyl group or a phenyl group which may be substituted, R2 and R3 independently represent a phenyl group which may be substituted...
11/18/2003
6395367Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials
The invention relates to ionic compounds in which the anionic load has been delocalized. A compound disclosed by the invention includes an anionic portion combined with at least one cationic portion Mm+ in sufficient numbers to ensure overall e...
05/28/2002
6359141Water soluble prodrugs of azole compounds
Water-soluble prodrugs of triazole antifungal compounds having a secondary or tertiary hydroxy group are provided. More particularly, new water-soluble triazole antifungal compounds are provided having the general formula ##STR1## wherein A is the no...
03/19/2002
6265584Water soluble prodrugs of azole compounds
Water-soluble prodrugs of triazole antifungal compounds having a secondary or tertiary hydroxy group are provided. More particularly, new water-soluble triazole antifungal compounds are provided having the general formula ##STR1## wherein A is the no...
07/24/2001
6159938Serine protease inhibitors comprising ଱-keto heterocycles
Provided are methods of inhibiting the activity of a serine protease using protease inhibitors that include an alpha-keto heterocycle in their structure. The methods are useful in the treatment of ischemic heart or treatment of symptoms associated with bl...
12/12/2000
60639285-lipoxygenase inhibitors
Novel compounds having the ability to inhibit 5-lipoxygenase enzyme and having the following formula I: ##STR1## and the pharmaceutically acceptable salts thereof, wherein Ar1 is a heterocyclic moiety which is selected from imidazolyl, pyr...
05/16/2000
5922867Method and compositions for the synthesis of dioxolane nucleosides with ଲ configuration
The present invention relates to methods and compositions for preparing biologically important nucleoside analogues containing 1,3-dioxolane sugar rings. In particular, this invention relates to the stereoselective synthesis of the beta (cis) isomer by gl...
07/13/1999
5874585Substituted heterocyclic compounds useful as inhibitors of (serine proteases) human neutrophil elastase
The present invention relates to certain substituted oxadiazole, thiadiazole and triazole peptoids which are useful as inhibitors of serine proteases including human neutrophil elastase, equivalently known as human leukocyte elastase....
02/23/1999
58695081,2,3-Benzothiadiazole derivatives
Novel 1,2,3-benzothiadiazole derivatives of the formula ##STR1## in which Het has the meanings set forth in the specification, and addition products thereof with an acid or metal salt are very effective for the control of undesired microorganisms. Novel i...
02/09/1999
5840894Preparation of 1,2,4-triazolium salts and 1,2,4-triazolines
A process for the preparation of 1,2,4-triazolium salts Ia ##STR1## where R1, and R2 and R3 are C-organic radicals, it being possible for R2 and R3 to be connected to give a 5- to 8-membered ring...
11/24/1998
5602196Bisphenol ester derivatives
Stabilisers of formula I ##STR1## wherein R1 and R2 may be C1 -C5 alkyl, the substituents R3 to R8 may be hydrogen, the variable n may be 1 or 2, and, when n is 1, A may be an alkoxy r...
02/11/1997
55301177-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
The disclosure is drawn to novel 7-substituted-9-(substituted amino)-6-demethyl-6-deoxytetracycline compounds. These compounds are useful to treat infections caused by a wide spectrum of bacterial organisms, including those which are resistant to tetracyc...
06/25/1996
5476845Use of phosphoric esters as crystallization inhibitors
A new process for preventing the crystallization of certain azole derivatives in the spray equipment upon spraying mixtures containing A) certain azole derivatives which have a tendency to crystallize and B) if appropriate one or more other active compounds and add...
12/19/1995
5369118N-alkyl-lactams as crystallization inhibitors
In the spraying of an aqueous liquor comprising at least one of 1-(4-chlorophenyl)-4,4-dimethyl-3-(1,2,4-triazol-1-yl-methyl)-pentan-3-ol and 1-(4-chlorophenoxy)-3,3-dimethyl-1-(1,2,4-triazol-1-yl)-butan-2-ol, the improvement which comprises including in ...
11/29/1994
5366984Methyl ଱-arylacrylates substituted by a heterocyclic radical and their use
Methyl ଱-arylacrylates substituted by a heterocyclic radical and having the general formula ##STR1## where R is alkyl, alkenyl, haloalkyl, cycloalkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, halogen or aryl, the aromatic ring being unsubstituted...
11/22/1994
52505551-halo-1-azolylmethane derivatives and fungicides containing these
1-Halo-1-azolylmethane derivatives of the formula ##STR1## where A and R are each alkyl, benzyl, benzoyl, acyl, biphenylyl, naphthyl, hetaryl or phenyl, it being possible for each of these radicals to be substituted; D is Cl or Br, X is CH or N, and ...
10/05/1993
5225550Process for the preparation of substituted acyclic nucleosides, and intermediates occurring therein
It is possible, by using symmetrical formaldehyde acetals of the formula ##STR1## in which the substituents R1 -R3 have the specified meanings, advantageously to introduce the substituent ##STR2## into nitrogen-containing h...
07/06/1993
5206225Alkylcarboxylic acid dimethylamides as crystallization inhibitors
Crystallization of active material in spraying an aqueous solution of one of ##STR1## and is prevented by incorporation therein of an alkylcarboxylic acid dimethylamide of the formula ##STR2## in which R represents alkyl having 5 to 19 carb...
04/27/1993
5199969Azolylethane derivatives and fungicides and growth regulators containing them
Azolylethane derivatives of the general formula I ##STR1## where A and Z are each alkyl, phenyl, biphenyl, naphthyl, benzyl, cycloalkyl or cycloalkenyl, these radicals being substituted or unsubstituted, D is alkoxy, amino, mercapto, thiophenyl, amin...
04/06/1993
5187182N-phenoxyphenoxymethyl-triazoles and a method for controlling pests
N-substituted azoles of the formula I ##STR1## where R1,R2, R3 are each hydrogen, halogen, C1 -C8 -alkyl, C1 -C8 -alkoxy, C1 -C4 -haloalkyl, C1
02/16/1993
51400361,3,5-trisubstituted-1,2,4-triazole compounds for treatment of circulatory disorders
A class of 1,3,5-trisubstituted-1,2,4-triazole compounds is described for use in treatment of circulatory disorders. Compounds of particular interest are angiotensin II antagonists of the formula ##STR1## wherein m is one; wherein R1 is se...
08/18/1992
51283571-alkoxy-1-azolylmethyloxiranes and the use thereof as crop protection agents
1-Alkoxy-1-azolylmethyloxiranes of the general ##STR1## where R1 and R2 are identical or different and each is C1 -C8 -alkyl, C3 -C8 -cycloalkyl, C5 -C8 -cycloalk...
07/07/1992
5124344Compounds containing triazole groups and use thereof as fungicides
The invention relates to compounds of formula: ##STR1## A is the group (Y)n Ph--(CH2)m where Ph is a phenyl nucleus and m=0 or 1, preferably 0, Y is a halogen atom or a cyano or nitro group or an optionally halogenated ...
06/23/1992
5101059Amino acid protecting groups
This invention relates to compounds of the formula a compound of the formula ##STR1## wherein X is O, CR7 R8, S or NR9 wherein R7 and R8 are independently hydrogen, or lower alkyl, and R9
03/31/1992
5093346Substituted 1,2,4-triazole angiotensin II antagonists
Substituted pyrroles, pyrazoles and triazoles such as ##STR1## and their pharmaceutically suitable salts are useful as antihypertensive agents and for treatment of congestive heart failure....
03/03/1992
5015651Treatment of hypertension with 1,2,4-angiotensin II antagonists
Substituted pyrroles, pyrazoles and traizoles such as ##STR1## and their pharmaceutically suitable salts are useful as antihypertensive agents and for treatment of congestive heart failure....
05/14/1991
5013854Process for preparing acid halides
An improved process for preparing trialkylsilyl ester and acid halide derivatives of carboxylic acids is provided along with novel trialkylsilyl ester intermediates of 2-(2-furyl)-2-methoximinoacetic acid....
05/07/1991
4970320Preparation of phenoxy-triazolyl-pinacol-ones
X represents a halogen, phenyl, phenoxy or halophenoxy moiety, and n is an integer of from 0 to 5, is produced by reacting 1,2,4-triazole with an ଱-halo-଱-phenoxy compound of the formula ##STR2## in which Y represents Br or Cl, in the presenc...
11/13/1990
4942244Diastereomeric triazolyl glycol ethers-fungicides and growth regulators
Diastereomers of the formula ##STR1## Where R1 is hydrogen, alkyl, alkenyl, alkynyl or benzyl, R2 is a alkyl or alkenyl, R3 is alkyl or benzyl, and the asymmetric centers of the molecular have (a) an RR or SS or (b) a...
07/17/1990
4931581Process and a composition for immunizing plants against diseases
A method and composition for the immunization of healthy useful plants against plant diseases containing as active ingredients compounds of formula ##STR1## in which: X is hydrogen, halogen, hydroxy, methyl, methoxy, HOOC or MOOC; Y is hydrogen, halo...
06/05/1990
4925476Azole hemiaminal derivatives and their use as nitrification inhibitors
Nitrification inhibitors contain azole hemiaminal derivatives of the formula ##STR1## where R1 and R2 are each hydrogen, alkyl, aryl or halogen, R3 is alkyl, cycloalkyl, alkoxy, alkenyl, alkynyl, styryl, aryl, he...
05/15/1990
4917720Fungicidal and plant-growth regulating azolyl ether ketones and alcohols
Azolyl ether ketones and alcohols of the formula ##STR1## in which R1 and R2 each independently represents alkyl with more than one carbon atom, or R1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlor...
04/17/1990
4895586Triazolyl glycol ethers, fungicides and bioregulators
଱-triazolyl glycol ethers of the formula I ##STR1## where R1 is alkyl, alkoxy, halogen or phenyl, R2 and R3 are each hydrogen or alkyl, R4 is alkyl or unsubstituted or substituted phenyl, Z is ##STR2## ...
01/23/1990
4878939Fungicidal and plant-growth regulating azolyl ether ketones and alcohols
Azolyl ether ketones and alcohols of the formula ##STR1## in which R1 and R2 each independently represents alkyl with more than one carbon atom, or R1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlor...
11/07/1989
4871389Heterocyclic compounds
A compound having the general formula: ##STR1## and stereoisomers thereof, wherein R1 is alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, all having up to 8 carbon atoms; or is aryl, aralkyl or heterocyclyl, any of which may be optiona...
10/03/1989
4833252Herbicidal sulfonylureas
Substituted N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'-triazinylureas of the general formula ##STR1## and the salts thereof with amines, alkali metal bases or alkaline earth metal bases, or with quaternary ammonium bases, have good ...
05/23/1989
4828603Herbicidal oxatricyclo-nonane ethers
The present invention relates to novel tricyclo ether derivative compounds, to compositions containing these ether derivative compounds, and to methods of using these compounds or compositions to control the growth of undesired vegetation....
05/09/1989
4806542Isohexide pyrimidines triazines, triazoles and imidazoles useful as cytostatic
Isohexide nucleosides of the formula I ##STR1## in which R and B have the meaning given in the description, processes for their preparation and their use as medicaments, in particular as cytostatics, virustatics and immunostimulants....
02/21/1989
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