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Patent No. 5979328

Vehicular Impact Signaling Device

An apparatus for the deployment of a visible plume to alert other motorists that a proximate motor vehicle has been involved in a collision.

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Class 548/267.4 - The nitrogen is double or triple bonded to carbon


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein carbon is double or triple bonded to the
No. of patents: 166
Last issue date: 02/08/2011


1          
NumberTitleIssue Date
7884213Process for the preparation of anastrozole
A process for the preparation of anastrozole. ...
02/08/2011
7173022Bicyclic heterocycles as HIV integrase inhibitors
The invention encompasses a series cyclic bicyclic heterocyclic compounds of Formula I which are inhibitors of HIV integrase and prevent viral integration into human DNA. This action makes the compounds useful for treating HIV infection and AIDS. The invention also ...
02/06/2007
7169929Diaryl 1,2,4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor
The present invention relates to a novel diaryl 1,2,4-triazole derivative of the following formula (1) as a highly selective cyclooxygenase-2 inhibitor, wherein R1, R2, R3, R4, R5, W and A is as defined in this ...
01/30/2007
70191441,2,4-Triazole derivative, method for preparing the same, and pharmaceutical composition containing the same
A 1,2,4-Triazole derivative of formula 1 or a non-toxic salt thereof, a preparation method thereof, and a pharmaceutical composition containing the derivative or the salt as an active ingredient are provided. ...
03/28/2006
68033805-aryl-1h-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them
5-aryl-1H-triazole compounds of the formula are potent and selective COX-2 inhibitors. The invention further relates to pharmaceutical compositions containing these compounds. ...
10/12/2004
6723742Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
The use is described of 3,5-diphenyl-1,2,4-triazoles of the formula I in which R1-R5 are as defined in the description. The compounds have useful pharmaceutical properties and are particularly activ...
04/20/2004
6703411Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
Benzoylguanidines of the formula (I) ##STR1## in which R1 to R4 have the meanings given in the specification and claims are suitable as antiarrhythmic medicaments having a cardioprotective component for infarct prophylaxis and infarct treatment and for th...
03/09/2004
6503912Substituted guanidine derivatives
The present application relates to novel guanidine derivatives of the formula (I) ##STR1## in which R1 represents a five- or six-membered heterocyclic group; R2 represents hydrogen or alkyl, R3 represents the groupings --OR
01/07/2003
6465504Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
The use is described of 3,5-diphenyl-1,2,4-triazoles of the formula I ##STR1## in which R1 -R5 are as defined in the description. The compounds have useful pharmaceutical properties and are particularly active as iron chelators. They...
10/15/2002
6407100Fungicidal aromatic oximes
The invention relates to novel compounds of the formula ##STR1## in which R1 is C1-4 alkyl and (Y--X) is CH2, C1-2 alkylthio-CH.dbd. or C1-2 alkyl-ON.dbd. and Z is an aldimino or ketimino group, and t...
06/18/2002
6391903Triazole derivatives having antifungal activity
Compounds of the following formula (I) and pharmaceutically acceptable esters and salts thereof: ##STR1## Ar is a phenyl group which may optionally be substituted by from 1 to 3 substituents selected from the group consisting of halogen atoms and tri...
05/21/2002
6359141Water soluble prodrugs of azole compounds
Water-soluble prodrugs of triazole antifungal compounds having a secondary or tertiary hydroxy group are provided. More particularly, new water-soluble triazole antifungal compounds are provided having the general formula ##STR1## wherein A is the no...
03/19/2002
6337403Triazole derivatives having antifungal activity
Compounds of the following formula (I) and pharmaceutically acceptable esters and salts thereof: ##STR1## Ar is a phenyl group which may optionally be substituted by from 1 to 3 substituents selected from the group consisting of halogen atoms and tri...
01/08/2002
6316459O-benzyloxime ethers and crop protection agents containing these compounds
O-Benzyloxime ethers of the formula I ##STR1## where X is substituted or unsubstituted CH2, NOalkyl Y is O, S, NR5 R1, R2, R5 are H, alkyl Z1, Z2 are H, halogen, methyl, methoxy, cyano R
11/13/2001
6316505Pharmaceutical compositions comprising fluorinated co-polymers
Block copolymers containing a fluorinated hydrocarbon unit, a hydrocarbon unit, and a poly(oxyethylene) unit are useful in fluid formulations of pharmaceutical agents. A typical embodiment is: C11 H23 --CONHC2 H4 NHC...
11/13/2001
62880711-ethylene-2-alkylene-1,4-cyclohexadiene pesticides
Pesticidally active cyclohexadienyl derivative compounds of the formula I that are esters, oximes or amides are claimed. These compounds may be used as fungicides, acaricides and insecticides in plant protection....
09/11/2001
62620993-(substituted phenyl)-5-(substituted cyclopropyl)-1,2,4-triazole compounds
3-(Substituted phenyl)-5-(substituted cyclopropyl)-1,2,4-triazole compounds are useful as insecticides and acaricides. New synthetic procedures and intermediates for preparing the compounds, pesticide compositions containing the compounds, and methods of ...
07/17/2001
5977152Triazole antifungal agent
A triazole compound having the formula: ##STR1## wherein Ar1 represents an optionally substituted phenyl, Ar2 represents an optionally substituted phenyl, R0 represents a hydrogen atom or a lower alkyl; R1 ...
11/02/1999
5912355Chiral synthesis of tertiary alcohols with a hydrolase
Method of preparing an optically active compound of formula, wherein R and R1 are independently alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, cycloalkyl, aryl, aralkyl, a heterocyclic group or a C1 -C4 alkyl-heterocycle, e...
06/15/1999
5905087Iminooxybenzyl compounds and their use as pesticides and fungicides
Iminooxybenzyl compounds of the formula I ##STR1## where R1 is C(CO2 Ra).dbd.CHRb, C(CO2 Ra).dbd.CHORb, C(CO2 Ra).dbd.NORb or C(CONRa ...
05/18/1999
5888941Carbozamides with antifungal activity
Compounds of general formula I and their salts and solvates are antifungal agents and as such are useful in the treatment of various fungal infections. Pharmaceutical compositions including these compounds and processes for their preparation are also prov...
03/30/1999
5846907Herbicidally active pyrazol-4-ylbenzoyl compounds
Pyrazol-4-ylbenzoyl compounds of the formula I ##STR1## where Z is a 5- or 6-membered heterocyclic saturated or unsaturated radical, Q is a pyrazole ring and L and M are as defined in the specification, their use as herbicidal compounds and to proces...
12/08/1998
5846906Herbicidally active phenyldiketone compounds
Herbicidally active phenyldiketone compounds of the formula I ##STR1## in which the substituents have the following meanings: L and M are hydrogen, C1 -C6 -alkyl, C2 -C6 -alkenyl, C2 -C6
12/08/1998
57671513,3-(disubstituted) cyclohexan-1-ylidine acetate dimers and related compounds
The present invention relates to novel 3,3-(disubstituted)-cyclohexan-1-ylidene acetate dimers of Formula (I): ##STR1## and related compounds, pharmaceutical compositions containing these compounds, and their use in treating allergic and inflammateor...
06/16/1998
5763640Fungicide intermediates
Compounds having the formula (I): ##STR1## and stereoisomers thereof, wherein A is hydrogen, halo, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4...
06/09/1998
5760067Halogen alkenyl azolyl microbicides
Novel halogenoalkenyl-azolyl derivatives of the formula ##STR1## in which R1 represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl, optionally substituted aryl or represents optionally ...
06/02/1998
5723473Propenoic acid derivatives useful as fungicides
A fungicidal compound of formula (I): ##STR1## wherein A is hydrogen, halogen, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4 alkoxycarbony...
03/03/1998
5703109Selective aromatase inhibiting compounds
New compounds of formula (I) wherein R1 is H, CH3, OCH3, NO2, NH2, CN, CF3, CHF2, CH2 F or halogen, R2 is a heterocyclyl radical selected from 1-imidazolyl, tria...
12/30/1997
5700824Triazole derivatives, insecticide, acaricide and methods thereof
The invention provides a triazole derivative represented by a general formula ##STR1## (wherein R1 is an alkyl group, X is a hydrogen atom, a halogen atom or an alkyl group, n is an integer of 1-5, Y is a halogen atom, a nitro group o...
12/23/1997
5677465Benzaldehyde oxime derivatives, production and use thereof
The present invention relates to novel benzaldehyde derivatives, specifically ଱-azolyl-2-substituted benzaldehyde oxime derivatives, their production, and fungicidal, herbicidal and growth regulating compositions containing them....
10/14/1997
5665739Substituted benzoylguanidines, process and their preparation, their use as pharmaceutical or diagnostic, and pharmaceutical containing them
Benzoylguanidines of the formula I are described ##STR1## in which R(1)=hydrogen, Hal, --NO2, --C.tbd.N, --CF3, R(4)--SOm or R(5)R(6)N--SO2 --, R(4) and R(5) are alk(en)yl or CF3, R(5) also havin...
09/09/1997
5637605଱-fluoro-଱-1-(1,2,4-triazolyl)-phenylmethyl derivatives useful as aromatase inhibitors
Compounds of formula I ##STR1## wherein Z, R, R1, R2 and X are as defined in the description, have valuable pharmaceutical properties and are effective especially against tumours. They are prepared in a manner known per se....
06/10/1997
5605921Triazole derivatives and salts thereof, and antifungal agent containing the same
The present invention relates to a compound represented by the general formula (1) or its salt, a process for producing the same, and an antifungal agent comprising the same as an effective component: ##STR1## wherein R1 represents a subst...
02/25/1997
5587392Azolyl methyl phenyl derivatives having aromatase inhibitory activity
Compounds exerting excellent aromatase inhibitory activity in vivo and in vitro with higher specificity and greater safety are provided together with the salts thereof. Using the same, there are also provided, prophylactic agents and/or therapeutical agen...
12/24/1996
5543433Azine-substituted phenylacetic acid derivatives and fungicides containing these
Compounds of the formula I ##STR1## where X is hydrogen, halogen, alkyl, alkoxy, trifluoromethyl, cyano or nitro, Y is an amino, methylamino or dimethylamino group, Z is a group CHCH3, CHOCH3 or NOCH3, R is hydrogen or alk...
08/06/1996
5527816Fungicidal 2-aryl-2-cyano-2-(aryloxyalkyl)ethyl-1,2-4-triazoles
2-aryl-2-cyano-2-(aryloxyalkyl)ethyl-1,2,4-triazoles of the formula ##STR1## wherein Ar1 and Ar2 are optionally substituted aryl groups which may or may not be different, R is hydrogen or alkyl, n is an integer of at least one, ...
06/18/1996
5510493Process for alkylation with triazoles
The present invention provides an improved process for the production of triazoles of the formula: ##STR1## wherein Z is an optionally substituted (C6 -C10)aryl group; R is a hydrogen atom, a (C1 -C12)alkyl...
04/23/1996
5489603Guanidine derivatives, their production and insecticides
An insecticidal composition containing a guanidine derivative of the formula: ##STR1## wherein R1 is an optionally substituted homocyclic or heterocyclic group, n is 0 or 1, R2 is a hydrogen atom or an optionally substitute...
02/06/1996
5476845Use of phosphoric esters as crystallization inhibitors
A new process for preventing the crystallization of certain azole derivatives in the spray equipment upon spraying mixtures containing A) certain azole derivatives which have a tendency to crystallize and B) if appropriate one or more other active compounds and add...
12/19/1995
5470863Oximic derivatives with a fungicide activity
A description follows of oximic derivatives with a fungicide activity, for agricultural use, having the formula (I): ##STR1## wherein: A, B, D, are N, or .dbd.C--G; G is H, halogen, NO2, CN, --COOR4, C1 -C6 (hal...
11/28/1995
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