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| Number | Title | Issue Date |
| 7994338 | Small molecule inhibitors of kynurenine-3-monooxygenase The present invention relates to compounds of formula Ia or Ib below and their tautomers and/or pharmaceutically acceptable salts and compositions and methods of uses thereof. ... | 08/09/2011 |
| 7256205 | Nitrosated and nitrosylated Hreceptor antagonist compounds, compositions and methods of use The invention describes novel nitrosated and/or nitrosylated H2 receptor antagonist compounds, and novel compositions comprising at least one H2 receptor antagonist compound that is optionally substituted with at least one NO and/or NO2 | 08/14/2007 |
| 7189750 | Thiazole-based nitric oxide donors having at least two thiazole moieties and uses thereof Disclosed are novel NO-donating compounds, designed such that when NO is released from the compound a residue which is a naturally occurring metabolite is formed, and thus a development of tolerance to the compounds upon repetitive administration is prevented or dec... | 03/13/2007 |
| 7132436 | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which act... | 11/07/2006 |
| 7125900 | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which act... | 10/24/2006 |
| 6620767 | Pesticidal n-heteroaryl alpha-alkoximino-carboxamides The invention relates to compounds of the general formula ##STR1## wherein R1 is hydrogen, halogen, C1 -C6 -alkyl, C1 -C6 -alkoxy, C1 -C6 -haloalkyl or unsubstituted or mono- to ... | 09/16/2003 |
| 6617341 | Insecticidal 2-iminothiazole derivatives A novel 2-iminothiazole derivatives and the use as an insecticide and acaricide of the compounds of formula (1): ##STR1## wherein R1 is CN or fluoroalkyl (especially C1 -C4 fluoroalkyl), R2 is H, halogen or CN, ... | 09/09/2003 |
| 6448286 | Imino pyrrolidine derivatives useful as nitric oxide synthase inhibitors The current invention discloses useful pharmaceutical compositions containing amidino derivative useful as nitric oxide synthase inhibitors.... | 09/10/2002 |
| 6218408 | Selective NPY (Y5) antagonists (bicyclics) This invention is directed to bicyclic compounds which are selective antagonists for NPY (Y5) receptors. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of the compound of the invention and a pharmaceutica... | 04/17/2001 |
| 6214853 | Selective NPY (Y5) antagonists (bicyclics) This invention is directed to bicyclic compounds which are selective antagonists for NPY (Y5) receptors. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of the compound of the invention and a pharmaceutica... | 04/10/2001 |
| 6166215 | Process for producing guanidine derivatives, intermediates therefor and their production A process for producing the compound [I] or a salt thereof having excellent pesticidal activity as shown in the following schema. ##STR1##... | 12/26/2000 |
| 6140505 | Synthesis of benzo fused heterocyclic sulfonyl chlorides A process for preparing a benzo fused heterocyclic sulfonyl halide comprising reacting a benzo fused heterocyclic compound with an SO3 complex in the presence of a water immiscible, non-reactive solvent, at a temperature of from about 0° C. to... | 10/31/2000 |
| 6057349 | 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxphenyl, and aminophenyl alkylsulfonamides and ureas and their use The present invention concerns novel compounds represented by the Formula: ##STR1## wherein: A is R1q (R3 R60 N)m (Z)(NR2)n ; m and q are each 0 or 1, with the proviso that when ... | 05/02/2000 |
| 5965601 | Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors Selected amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, rela... | 10/12/1999 |
| 5925651 | Inhibitors of farnesyl-protein transferase The present invention is directed to compounds which inhibit farnesyl-protein transferase (FTase) and the farnesylation of the oncogene protein Ras. The invention is further directed to chemotherapeutic compositions containing the compounds of this invent... | 07/20/1999 |
| 5877193 | Use of N-(4-aryl-thiazol-2-yl)-sulfonamides The invention is concerned with the use of sulfonamide derivatives of the general formula ##STR1## wherein R signifies lower-alkyl, phenyl, benzyl, naphthyl, pyridyl or thienyl, optionally substituted by one or more lower-alkyl, lower-alkoxy, lo... | 03/02/1999 |
| 5846990 | Substituted biphenyl isoxazole sulfonamides Compounds of the formula ##STR1## inhibit the activity of endothelin. The symbols are defined as follows: R1, R2, R3 and R4 are each directly bonded to a ring carbon and are each independently (a) hydrogen;... | 12/08/1998 |
| 5612483 | Process for the preparation of nitro-substituted arylamines Nitro-substituted aromatics can be directly aminated with amines in the presence of simple bases and oxygen.... | 03/18/1997 |
| 5506262 | Cholesterol lowering compounds Disclosed herein are compounds of structural formula (I) ##STR1## which are useful as cholesterol lowering agents. These compounds are also useful as inhibitors of squalene synthetase, inhibitors of fungal growth, inhibitors of farnesyl-protein trans... | 04/09/1996 |
| 5449783 | Diphenylthiazole derivative A novel diphenythiazole derivative represented by the following general formula (I): ##STR1## wherein m and n are each 1 or 2; R1 and R2 represent each a hydrogen atom, a lower alkyl group, a lower alkoxy group, a lower alk... | 09/12/1995 |
| 5411975 | Thiazolidinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension Compounds characterized generally as thiazolidinyl-terminated alkylamino ethynyl alanine amino diol derivatives are useful as renin inhibitors for the treatment of hypertension. Compounds of particular interest are those of Formula I ##STR1## wh... | 05/02/1995 |
| 5376677 | Benzo[b]thiophene derivatives The invention relates to novel compounds of the formula ##STR1## in which R is as defined in the description, to their preparation, to fungicidal compositions which contain such compounds as active substances, and to the use of the active substances ... | 12/27/1994 |
| 5350736 | Iminothiazolines, their production and use as herbicides, and intermediates for their production There is disclosed an iminothiazoline compound of the formula: ##STR1## wherein R1 is halogen, halo(lower)alkyl, halo(lower)alkoxy or halo(lower)alkylthio; R2 is lower alkyl, chlorine; bromine or iodine; R3 is (lower ... | 09/27/1994 |
| 5334614 | Hydroxylamine derivatives The invention concerns hydroxylamine derivatives of the formula I ##STR1## wherein R4 is hydrogen, carbamoyl, (1-4C)alkyl, cyclopentyl, cyclohexyl, tetrahydrofuran-3-yl, tetrahydropyran-4-yl, piperidin-4-yl, N-(1-4C)alkylpiperidin-4-yl, (2... | 08/02/1994 |
| 5326783 | Cholesterol lowering compounds This invention is directed to compounds of formula (I) which are novel C3- or C5-acyl sulfonamide, carboxamic acid or tetrazolyl analogs of the Zaragozic acids. These compounds inhibit the enzyme squalene synthase and are useful as cholesterol lowering ag... | 07/05/1994 |
| 5314891 | Benzenesulphonamide derivatives The invention concerns benzenesulphonamide derivatives of the formula I ##STR1## wherein R1 is (1-4C)alkyl, (3-4C)alkenyl or (3-4C)alkynyl; R2 and R3 together form --A2 --X2 --A3 -- which d... | 05/24/1994 |
| 5308857 | Furylthiazole derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same The invention relates to compounds of the formula: ##STR1## wherein R1, R2, R3, R4, A and Q are as described, useful in the treatment of ulcers.... | 05/03/1994 |
| 5290802 | 3-substituted-2-oxindole derivatives This invention relates to novel 3-substituted-2-oxindole derivatives which are inhibitors of prostaglandin H2 synthase, 5-lipoxygenase and interleukin-1 biosynthesis. The compounds of the invention are useful as inhibitors of prostaglandin H | 03/01/1994 |
| 5244863 | Iminothiazolines, their production and use as herbicides, and intermediates for their production An iminothiazoline compound of the formula: ##STR1## which is useful as a herbicide.... | 09/14/1993 |
| 5225548 | Indophenol dyes and thermal transfer thereof Indophenol dyes of the formula ##STR1## where X is nitrogen or the radical CH, Q is a five-membered heterocyclic radical, and K is a radical of an aniline, aminonaphthalene, aminoquinoline or aminothiazole derivative, and the radical A can be benzofused, ... | 07/06/1993 |
| 5128477 | Process for the preparation of morphologically homogeneous forms of thiazole derivatives The invention relates to two morphologically homogeneous forms of Famotidine [chemical name: N-sulfamoyl-3-(2-guanidino-thiazole-4-yl-methylthio)-propionamidine]. Said forms are prepared by selective crystallization or precipitation.... | 07/07/1992 |
| 5120850 | Process for the preparation of morphologically homogeneous forms of thiazole derivatives The invention relates to two morphologically homogeneous forms of Famotidine [chemical name: N-sulfamoyl-3-(2-guanidino-thiazole-4-yl-methylthio)-propionamidine]. Said forms are prepared by selective crystallization or precipitation.... | 06/09/1992 |
| 5081142 | Derivatives of 1-hydroxy-1,2,4-triazole and fungicides and growth regulators containing them Compounds of the formula I ##STR1## where Ar is unsubstituted or substituted phenyl, pyridyl, thienyl or napthyl, R1 is hydrogen or CN, R2 is unsubstituted or substituted aryl, hetaryl, alkyl or cycloalkyl, or is unsubstituted o... | 01/14/1992 |
| 5043443 | Aminomethyloxooxazolidinyl arylbenzene derivatives Novel aminomethyloxooxazolidinyl arylbenzene derivatives, wherein the aryl includes the phenyl, substituted phenyl, pyridyl, and substituted pyridyl groups, such as (l)-N-{3-[4- (4'-pyridyl)phenyl]-2-oxooxazolidin-5-ylmethyl}acetamide, possess useful ... | 08/27/1991 |
| 5034417 | New alkanesulfonanilide derivatives, processes for preparation thereof and pharmaceutical composition comprising the same This invention relates to new alkanesulfonanilide derivatives and pharmaceutically acceptable salts thereof which have inflammatory activities and analgesic activities, to pharmaceutical compositions containing the same and to a method for the treatment o... | 07/23/1991 |
| 5021582 | Famotidine polymorphic forms and their preparation process It is described the preparation of the famotidine polymorphs with low melting point and relative high or low apparent densities. They differ from the polymorph of high melting point and high density, in the physical-chemical and biological properties, of ... | 06/04/1991 |
| 5006660 | Process for producing alkoxybenzene compound and aryloxybenzene compound The present invention relates to a process for producing an alkoxybenzene compound or an aryloxybenzene compound by reacting a halogenobenzene compound with an alcohol or a phenol compound in the presence of copper or a copper compound, an amine, and a ba... | 04/09/1991 |
| 5001138 | Novel heterocyclic compounds Novel insecticides of the formula ##STR1## in which n is 0 or 1, X is S, O, ##STR2## Y is N or ##STR3## Z is a 5- or 6-membered nitrogen-containing heterocyclic ring, and R to R9 variously represent hydrogen or specified org... | 03/19/1991 |
| 4913722 | Iminophenylthiazolidines, process of preparation and method of use A 2-iminophenyl thiazolidine having the formula ##STR1## wherein R is hydrogen or methyl; R1 is halo, nitro, cyano, C1 -C4 alkyl, C1 -C4 alkoxy, perhalomethyl, difluoromethyl, pentafluoroethyl, t... | 04/03/1990 |
| 4914112 | Aminoazole derivatives and their production and use A compound of the formula: ##STR1## wherein A is the group of the formula: Ar1 --D--Ar2 -- wherein Ar1 is a phenyl or thienyl group which may be optionally substituted with at least one of the same or different halogen ato... | 04/03/1990 |
