Class 548/152 - Bicyclo ring system having the thiazole ring as one of the cyclos

Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds in which the polycyclo ring system consists of
No. of patents: 251
Last issue date: 05/10/2011

«First «Previous 1 2 3 4 5 6 7 Next»Last»

Number	Title	Issue Date
6225331	Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists This invention involves compounds having the following structure: ##STR1## as described in the claims; and enantiomers, optical isomers, stereoisomers, diastereomers, tautomers, addition salts, biohydrolyzable amides and esters thereof, as well as pharmac...	05/01/2001
6224644	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophilic...	05/01/2001
6218359	Screening method using the RZR receptor family The current invention concerns the use of a receptor from the RZR/ROR receptor family or of a functional fragment thereof in a test of a compound for anti-autoimmune, anti-arthritic, anti-tumor, melatonin-like and/or melatonin-antagonistic activity and th...	04/17/2001
6204389	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 --R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophili...	03/20/2001
6197969	Process for producing substituted alkylamines or salts thereof The present invention provides a process for producing a substituted alkylamine represented by formula (3): ##STR1## or a salt thereof, which process comprises reacting a 2-aminothiophenol derivative metal salt represented by formula (1): ##STR2## wi...	03/06/2001
6197968	Decolorizable dye Described is a decolorizable dye represented by the following formula (I): ##STR1## wherein R1 represents an alkyl, aryl or heterocyclic group; R2 and R3 independently each represents a hydrogen atom or has the same meanin...	03/06/2001
6197956	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophilic...	03/06/2001
6177572	Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use Methods for preparing benzoxazoles and benzothiazoles on solid supports. Substituted benzothiazoles and benzoxazoles, libraries of the compounds, and methods of using the compounds are also disclosed....	01/23/2001
6159983	Method and composition for treatment of inflammatory bowel disease A composition in unit dosage form for the inhibition, prevention or treatment of inflammatory bowel disease comprising an effective amount of a compound having the formula: ##STR1## and a pharmaceutically acceptable carrier therefor. Also disclosed i...	12/12/2000
6156772	Antagonists of gonadotropin releasing hormone There are disclosed compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both m...	12/05/2000
6136831	Pyrazole derivatives and COX inhibitors containing them The purpose is to provide anti-inflammatory agents which have potent pharmacological actions and exert a selective inhibitory activity on COX-2, thereby being expected to reduce adverse effects such as disorders in gastric mucosa. The present invention en...	10/24/2000
6124330	N-[4-(Heteroarylmethyl)phenyl]-heteroarylamines The present invention is concerned with compounds of formula ##STR1## the N-oxides, the pharmaceutically acceptable addition salts and the stereochemically isomeric forms thereof, wherein R1 is hydrogen, hydroxy, C1-6 alkyl or a...	09/26/2000
6114350	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrop...	09/05/2000
6100405	Benzothiazole-containing two-photon chromophores exhibiting strong frequency upconversion There are provided asymmetrical two-photon chromophores of the formula: D--Ar--A wherein Ar is selected from the group consisting of ##STR1## wherein Fl is a fluorene group of the formula: ##STR2## wherein R1 and R2 are alkyl gr...	08/08/2000
6090834	Substituted oxazoles for the treatment of inflammation A class of substituted oxazolyl compounds is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula II ##STR1## wherein R is selected from halo, mercapto, hydroxyl, lower...	07/18/2000
6045696	Process for the purification of waste waters containing organic and inorganic sulphur compounds This invention relates to a process for the purification of waste waters containing organic and, should the situation arise, inorganic sulphur compounds, which waste waters contain a proportion of mercaptobenzothiazole and/or derivatives thereof and, shou...	04/04/2000
6034246	2-arylbenzazole compounds There are disclosed herein 2-phenylbenzazole compounds having a 3'-substituent and a 4'-NR2 R6 substituent in the phenyl group where R5 and R6 are each hydrogen or alkyl, or where the $'-NR5 R6	03/07/2000
6011045	Vitronectin receptor antagonists, their preparation and their use The present invention relates to compounds of the formula I A--B--D--E--F--G (I) in which A, B, D, E, F and G have the meanings given in the patent claims, to their preparation and to their use as medicaments. The compounds...	01/04/2000
6007865	Reversing the formation of advanced glycosylation endproducts The present invention relates to compositions and methods for inhibiting and reversing nonenzymatic cross-linking (protein aging). Accordingly, compositions are disclosed which comprise an agent capable of inhibiting the formation of advanced glycosylatio...	12/28/1999
6004536	Lipophilic cyanine dyes with enchanced aqueous solubilty The present invention relates to a family of cyanine dyes possessing lipophilic alkyl chains and either one or more reactive functional groups, bromo or chloro, or phenyl, sulfophenyl or polysulfophenyl substituents or combinations thereof. The dyes of th...	12/21/1999
5990145	Vitronectin receptor antagonists, their preparation and their use The present invention relates to compounds of the formula I, A--B--D--E--F--G (I) in which A, B, D, E, F and G have the meanings given in the patent claims, to their preparation and to their use as medicaments. The compound...	11/23/1999
5980779	Liquid crystalline compound and use thereof A process for producing a liquid crystalline compound represented by the following general formula (A): ##STR1##...	11/09/1999
5981559	Azole derivative with leukotriene (LTs) antagonizing activity and thromboxane (TX) A₂ antagonizing activity An azole derivative represented by general formula (I) or a pharmaceutically acceptable salt thereof, having both of a leukotriene antagonistic effect and a thromboxane A2 antagonistic effect and being useful in preventing or treating allergic diseases, i...	11/09/1999
5955458	Penicillin glycolate New solvates of penicillin, in particular amoxycillin glycolate has been provided for together with a simple one-step process to prepare the same....	09/21/1999
5952354	Tris carbamic acid esters: inhibitors of cholesterol absorption Inhibition of the enzymes cholesterol ester hydrolase (CEH) and/or acyl coenzyme A: cholesterol acyltransferase (ACAT) results in the inhibition of the esterification of cholesterol and are therefore implicated in the inhibition of absorption of cholester...	09/14/1999
5942535	a!-Annelated pyrrole derivatives and pharmaceutical use thereof The present invention relates to heterocyclic compounds of the formula ##STR1## in which R1 -R7, B, a and X have the meanings recited in the specification. These compounds are usable in the treatment of diseases of the rheumatoi...	08/24/1999
5939415	A!-annellated pyrrole derivatives and their use in pharmacology The present invention relates to heterocyclic compounds with the formula ##STR1## in which R1 to R7, B, a, and X have the meanings indicated in the specification. These compounds can be used for the treatment of diseases of the ...	08/17/1999
5932740	Thioheterocyclic near-infrared dyes Disclosed is a novel near-infrared absorbing dye of formula: ##STR1## wherein X1, X2 independently represents --CR8 R9 --, --S--, --Se--, --NR10 --, --CH.dbd.CH-- or --O--; n is an integer of 2 or 3; ...	08/03/1999
5889022	Indole, indoline and quinoline derivatives with 5HT_1D (anti-depressive) activity Novel indole, indoline and quinoline derivatives of formula (I) processes for their preparation, pharmaceutical compositions containing them, and their use in medicine is disclosed. A structurally distinct class of compounds have now been discovered and h...	03/30/1999
5874431	Benzazole compounds There are disclosed herein benzazole compounds, exemplified by 2-(4-aminophenyl)benzothiazole and analogues or salts thereof, which exhibit very significant selective cytotoxic activity in respect of tumor cells, especially breast cancer cells, and which ...	02/23/1999
5853703	Preventing and reversing the formation of advanced glycosylation endproducts The present invention relates to compositions and methods for inhibiting and reversing nonenzymatic cross-linking (protein aging). Accordingly, compositions are disclosed which comprise an agent capable of inhibiting the formation of advanced glycosylatio...	12/29/1998
5843972	Heterocyclic ଲ-adrenergic agonists The present invention relates to certain compounds of the formula (I) the racemic-enantiomeric mixtures and optical isomers of said compounds and the pharmaceutically acceptable salts or prodrugs thereof, depicted below, which are ଲ-adrenergic recep...	12/01/1998
5840721	Imidazole derivatives as MDR modulators The present invention relates to polysubsituted imidazole having formula 1 ##STR1## These compounds are useful for restoring the sensitivity of multidrug resistant cells to cancer chemotherapeutic agents....	11/24/1998
5821362	Method of desilylating silylether compounds Method of desilylating a silylether compound by reacting a silylether compound of the general formula (I): ##STR1## or a salt thereof with an amine hydrogen fluoride salt or a pyridine hydrogen fluoride salt in an organic solvent to produce a compoun...	10/13/1998
5801246	Substituted heteroarylphenyloxazolidinones The present invention discloses novel substituted aryl- and heteroarylphenyloxazolidinones which are useful as anti-bacterial agents. More specifically, the substituted aryl- and heteroarylphenyloxazolidinones of the invention are characterized by ox...	09/01/1998
5766510	Liquid crystalline compound and use thereof A process for producing a liquid crystalline compound represented by the following general formula (A): ##STR1##...	06/16/1998
5733648	Organic compounds suitable as reactive diluents, and binder precursor compositions including same Organic compounds having at least one ethylenically-unsaturated group are described, the organic compounds being suitable for use in coatable compositions as reactive diluents; compounds of the invention preferably have a divalent organic linking moiety d...	03/31/1998
5714479	Endothelin antagonistic heteroaromatic ring-fused cyclopentene derivatives A heteroaromatic ring-fused cyclopentene derivative of the formula: ##STR1## wherein the variables are as defined in the specification; or a pharmaceutically acceptable salt thereof....	02/03/1998
5698574	5-membered heteroaryl-oxazolidinones The present invention relates to 5-membered heteroaryl-oxazolidinones, to processes for their preparation and to their use as medicaments, in particular as antibacterial medicaments....	12/16/1997
5684152	Preparation of carboxyalkyl derivatives as inhibitors of matrix metalloproteinases Carboxy-peptidyl compounds of Formula I are found to be useful inhibitors of matrix metalloendoproteinase-mediated diseases including osteoarthritis, rheumatoid arthritis, septic arthritis, tumor invasion in certain cancers, periodontal disease, corneal u...	11/04/1997

«First «Previous 1 2 3 4 5 6 7 Next»Last»

PatentStorm

Bizarre Patents

PatentStorm News

Class 548/152 - Bicyclo ring system having the thiazole ring as one of the cyclos