Class 546/331 - Sulfur and acyclic nitrogen bonded directly to the same carbon

Subclass of Class 546 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which contain a carbon atom to which is bonded
No. of patents: 154
Last issue date: 05/08/2007

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Number	Title	Issue Date
7214701	Active substance combinations having insecticidal and acaricdal properties The invention relates to insecticidal mixtures for protecting plants against attack by pests comprising (a) compounds of the formula (I) ...	05/08/2007
6884821	Carboxylic acid derivatives and drugs containing the same Novel carboxylic acid derivatives of general formula (I), salts of the same, esters thereof, or hydrates of them, which are useful as insulin resistance improvers; and drugs containing the derivatives as the active ingredient. In said formula, R1 is hydro...	04/26/2005
6696449	Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors This invention is directed to sulfonyl aromatic hydroxamic acid compounds and salts thereof that, inter alia, inhibit matrix metalloprotease (MMP) activity and/or aggrecanase activity. In some particularly preferred embodiments, the compound corresponds i...	02/24/2004
6646009	N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof N-(Aryl)-2-arylethenesulfonamides and pharmaceutically acceptable salts and compositions thereof are useful as antiproliferative agents, including, for example, anticancer agents. They are also useful as radioprotective agents....	11/11/2003
6638950	Piperidine amides as modulators of chemokine receptor activity The present application describes modulators of CCR3 of formula (I): ##STR1## or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma and other allergic diseases....	10/28/2003
6525069	N-ureidoalkyl-piperidines as modulators of chemokine receptor activity The present application describes modulators of CCR3 of formula (I): ##STR1## or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma and other allergic diseases....	02/25/2003
6521626	Thiocarboxamide derivatives Compounds of formula (1): ##STR1## wherein R1 is a hydrogen atom or an optionally substituted cycloaliphatic, polycycloaliphatic, heterocycloaliphatic, polyheterocycloaliphatic, aromatic or heteroaromatic group; Alk1 is an optionally...	02/18/2003
6476054	Cyclic amine modulators of chemokine receptor activity The present invention is directed to cyclic amines of the formula I: ##STR1## (wherein R1, R2, R3, m and n are defined herein) which are useful as modulators of chemokine receptor activity. In particular, these compounds a...	11/05/2002
6465468	Hydroxamic and carboxylic acid derivatives The subject invention concerns methods and compounds that have utility in the treatment of a condition associated with matrix metalloproteinase, ADAM or ADAM-TS enzymes, a condition that is mediated by TNF ଱ or a condition involving a membrane-shedd...	10/15/2002
6444686	N-ureidoalkyl-piperidines as modulators of chemokine receptor activity The present application describes modulators of CCR3 of formula (I): ##STR1## or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma and other allergic diseases....	09/03/2002
6426348	Diphenyl heterocyclic thioamide derivatives It has been discovered that compounds of the formula: ##STR1## and the pharmaceutically acceptable salts and esters thereof wherein X and Y are as defined below, inhibit the binding of VCAM-1 to VLA-4 and are useful in treating inflammation associated wit...	07/30/2002
6410573	2,5-substituted benzolsulfonylureas and thioureas methods for the production thereof use thereof and pharmaceutical preparations containing the same Novel 2,5-substituted benzolsulfonyl ureas and thioureas of formula (I) as illustrated in the disclosure. The compounds are useful active ingredients for medicaments. The compounds of formula (I) act as inhibitors on ATP-sensitive potassium canals and are...	06/25/2002
6410571	Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing a substituted phenylenediamine group Compounds of the formula: ##STR1## wherein the substituents are defined herein which are useful in the treatment of diseases associated with herpes viruses including human cytomegalovirus, herpes simplex viruses, Epstein-Barr virus, varicella-zoster ...	06/25/2002
6407248	଱-unsaturated amines, their production and use ଱-Unsaturated amines of the formula: ##STR1## wherein X1 and X2 are such that one is an electron-attracting group with the other being a hydrogen atom or an electron-attracting group; R1 is a group attached through a...	06/18/2002
6395737	Malonic acid derivatives, processes for their preparation, for their use and pharmaceutical compositions containing them New compounds for the inhibition of blood clotting proteins, and more particularly, to malonic acid derivatives of the formula I, ##STR1## wherein R(1), R(2), R(3), R(4), R(5), and R(6) have the meanings indicated in the claims. The compounds of formula I...	05/28/2002
6391881	Thiourea derivatives of dihydropyridine NPY antagonists A series of antagonists of NPY have been synthesized and are comprised of thiourea linked piperazine and piperidine derivatives of 4-phenyl-1,4-dihydropyridines of Formula 1. ##STR1## where Z is NR7 R8 or ##STR2## and X is CH or...	05/21/2002
6342633	O-benzyl oxime ether derivatives and their use as pesticides Compounds of the formula I ##STR1## in which Y is hydrogen, C1 -C4 alkyl, C1 -C4 alkoxy, OH, CN, NO2, Si(CH3)3, CF3 or halogen, Z is a group a) ##STR2## R1 ...	01/29/2002
6294549	Method for eliciting an ଱v댥 or dual ଱v댣/଱v댥 antagonizing effect A method for eliciting an ଱vଲ.sub.5 or dual ଱vଲ.sub.3 /଱vଲ.sub.5 antagonizing effect in a mammal which comprises administering to the mammal a therapeutically effective amount of a compo...	09/25/2001
6211240	O-benzyl oxime ether derivatives and their use as pesticides Compounds of the formula I ##STR1## in which Y is hydrogen, C1 -C4 alkyl, C1 -C4 alkoxy, OH, CN, NO2, Si(CH3)3, CF3 or halogen, Z is a group a) ##STR2## R1 ...	04/03/2001
6166214	Process for preparing pyridylmethyl isothiocyanates The present invention relates to a novel process for preparing pyridylmethyl isothiocyanates of the formula (I) ##STR1## in which R1 represents halogen or C1 -C4 -alkyl, characterized in that in a first step, amines o...	12/26/2000
6090824	Therapeutic neurokinin receptor antagonist compounds Compounds of formula I ##STR1## wherein Q1, Q2, Q3, and Q4 have any of the meanings given in the specification, their N-oxides, and their pharmaceutically acceptable salts are nonpeptide antagonists Substan...	07/18/2000
6063798	Substituted N-methylenethioureas as pesticides The present invention relates to new substituted N-methylenethioureas of the general formula (I) ##STR1## in which n, Het, R1 and R2 have the meanings given in the description, to a process for their preparation, and to their us...	05/16/2000
6015573	Nucleoside phosphate therapy for viral infection Compositions for topical use in herpes virus infections comprising anti-herpes nucleoside analogue phosphate esters, such as acyclovir monophosphate and acyclovir diphosphate, which show increased activity against native strains of herpes virus as well as...	01/18/2000
6008362	Elevation of HDL cholesterol by 2-(-4-chlorol-1-aryl-butylidene)-hydrazinecarbothioamides This invention relates to the treatment of atherosclerosis via raising the level of HDL cholesterol by administration of a compound of the formula ##STR1## wherein R1, R2, and R3 are independently hydrogen, C1 ...	12/28/1999
5952306	Integrin receptor antagonists Fibrinogen receptor antagonists having the formula ##STR1## for example ##STR2## which are useful for inhibiting the binding of fibrinogen to blood platelets and for inhibiting the aggregation of blood platelets....	09/14/1999
5945436	Pyridylmethyl nitriles, amides and thioamides useful as fungicides Compounds of of the formula ##STR1## wherein R is a C6 -C10 aryl group, optionally substituted with one or more halogen atoms, phenoxy, or, linear or branched, C1 -C6 alkyl, C1 -C6 alk...	08/31/1999
5936093	Process for preparing pyridylmethyl isothiocyanates Process for preparing pyridylmethyl isothiocyanates of the formula (I) ##STR1## comprising reacting amines of the formula (II): ##STR2## with xanthogenates of the formula (III): R2 O--CS--S.crclbar. M.sym. ...	08/10/1999
5919792	Integrin antagonists This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as vitronectin receptor antagonists. The vitronectin receptor antagonist compounds of the present invention are ଱v댣 antagonists, ଱...	07/06/1999
5808082	Method of preparing phosphodiesterase IV inhibitors A process for the preparation of Phosphodiesterase IV inhibitors is described. The process consists of eight chemical steps involving five isolations to prepare the title compound from readily available isovanillin in 35% overall yield (Scheme 1). The pro...	09/15/1998
5789422	Substituted arylalkylamines as neurokinin antagonists Compounds represented by the structural formula ##STR1## or a pharmaceutically acceptable salt thereof are disclosed, wherein: A1 is --CH2 R6, --OR6, --N(R6)(R7), --S(O)e R	08/04/1998
5756116	Nucleoside phosphate therapy for viral infection Compositions for topical use in herpes virus infections comprising anti-herpes nucleoside analogue phosphate esters, such as acyclovir monophosphate and acyclovir diphosphate, which show increased activity against native strains of herpes virus as well as...	05/26/1998
5741796	Pyridyl and naphthyridyl compounds for inhibiting osteoclast-mediated bone resorption Compounds of the following general structure X-Y-Z-Aryl-A-B, for example, ##STR1## which inhibit osteoclast mediated bone resorption. Specifically, the compounds are useful for treating mammals suffering from a bone condition caused or mediated by in...	04/21/1998
5728588	Coating of hydrophobic surfaces to render them protein resistant while permitting covalent attachment of specific ligands A surface of specific reactivity is formed by adsorbing a modified block polymeric surfactant of the Pluronic-type, i.e., containing pendant poly(ethylene oxide) blocks attached at an end to poly(propylene oxide) center blocks and with specifically reacti...	03/17/1998
5726314	Pyridinium compounds Novel quaternary pyridinium compounds useful in inhibiting acetylcholinesterase in mammals of the general structure: ##STR1## or pharmaceutically acceptable salts thereof, where R5 is pentafluorophenyl, phenyl monosubstituted with K, pheny...	03/10/1998
5705513	Fungicides for the control of take-all disease of plants A compound, composition, and method for controlling Take-all disease of plants by applying to the seed prior to planting, a fungicide of the formula: ##STR1## wherein Z1 and Z2 are C and are part of an aromatic ring which i...	01/06/1998
5670528	Thioamides and their use as crop protection agents Thioamides of the formula I ##STR1## where A, B, R' are hydrogen, cyano, alkyl, alkoxy or halogen, X is .dbd.CHCH3 or .dbd.N--OCH3, R1, R2 - are hydrogen or alkyl, Y is a group ##STR2## --O--CH2,...	09/23/1997
5580571	Nucleoside analogues Compositions for topical use in herpes virus infections comprising anti-herpes nucleoside analogue phosphate esters, such as acyclovir monophosphate and acyclovir diphosphate, which show increased activity against native strains of herpes virus as well as...	12/03/1996
5552418	Trisubstituted Naphthylalkylamides The invention relates to a compound selected from those of formula (I): ##STR1## in which R, R1, R2 and R3 are as defined in the specification, and a medicinal product containing said compound for treating a disorder of ...	09/03/1996
5470855	Certain heterocyclic thiazole derivatives and their therapeutic use The invention relates to compounds of formula: ##STR1## in which: A is selected from O or S; B is selected from C or N; Z1 is selected from C1 -C4 alkylene or phenylene; Z2 is C1 -C4 alkylene; W...	11/28/1995
5464847	Branched alkylamino derivatives of thiazole, processes for preparing them and pharmaceutical compositions containing them The invention relates to the derivatives of formula I: ##STR1## in which R1 represents a phenyl or naphthyl radical (optionally substituted), R2 represents a hydrogen or halogen atom or an alkyl, hydroxymethyl or formyl radical,...	11/07/1995

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Class 546/331 - Sulfur and acyclic nitrogen bonded directly to the same carbon