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| Number | Title | Issue Date |
| 7435815 | Sulfonylamino-acetic acid derivatives The invention relates to novel sulfonylamino-acetic acid derivatives and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including processes for the preparation of such compounds, pharmac... | 10/14/2008 |
| 7393868 | AMPA receptor potentiators The present invention relates to AMPA receptor potentiators of Formula I: formulations comprising them, methods for their use, and intermediates useful for their preparation. ... | 07/01/2008 |
| 7279578 | Sulfonylamino-acetic acid derivatives The invention relates to novel sulfonylamino-acetic acid derivatives and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including processes for the preparation of such compounds, pharmac... | 10/09/2007 |
| 7265220 | Amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative Compound of formula (I): wherein: R1 represents aryl, heteroaryl or alkyl which is optionally substituted, or a group of formula —(CO)—CR6R7NR8R9 ... | 09/04/2007 |
| 6989398 | Benzanilides as potassium channel openers Benzanilides are provided which are voltage-dependent potassium channel openers. Methods of using the benzanilides of the invention are also provided. ... | 01/24/2006 |
| 6946474 | Nitrogen-containing compounds and their use as glycine transport inhibitors The present invention provides trichloroethyl-sulfonylurea-containing compounds that inhibit glycing transporters, pharmaceutical compositions comprising such compounds, methods for using such compounds for inhibiting glycine transporters and methods for using such ... | 09/20/2005 |
| 6911451 | Phenylalanine derivatives Phenylalanine derivatives of formula (1) are described: wherein L1 is a linker atom or group; X1 is a group selected from —N(R3)CO—, —N(R3)SO | 06/28/2005 |
| 6727265 | Phenoxyethyl-thiourea-pyridine compounds and their use for treatment of HIV-infections The invention provides compounds which inhibit reverse transcriptase (RT) and which inhibit replication of a retrovirus, such as human immunodeficiency virus-1 (HIV-1). The compound of the invention are phenoxyethyl-thiourea-pyridines. The invention additionally pro... | 04/27/2004 |
| 6645968 | Potassium channel openers Compounds of formula I: ##STR1## are useful in treating diseases prevented by or ameliorated with potassium channel openers. Also disclosed are potassium channel opening compositions and a method of opening potassium channels in a mammal.... | 11/11/2003 |
| 6586450 | Phenethyl-thiourea compounds and use Novel phenylethyl-thiourea (PHET) compounds as inhibitors of reverse transcriptase and effective agents for the treatment of HIV infection, including mutant, drug-sensitive, drug-resistant, and multi-drug resistant strains of HIV.... | 07/01/2003 |
| 6555561 | Diaminopyridine-containing thiourea inhibitors of herpes viruses This invention provides compounds of formula I having the structure ##STR1## Wherein substitutions at X, G, R1, R2, R3, R4, R5 are set forth in the specification.... | 04/29/2003 |
| 6552225 | Chemical compounds A compound of formula (I) wherein: R1, R2, R3, R4, R5, R6 and R7 are as defined within; or a pharmaceutically acceptable salt or an in vivo hydrolysable ester thereof is described. Th... | 04/22/2003 |
| 6458816 | Modified prodrug forms of AP/AMP The present invention relates to compounds according to the structure: ##STR1## Where R is H or CH3 ; R2 is phosphate which can be free acid or salt; R3 is H, F, Cl, Br, I, OCH3, OCF3 , CF3 or a C | 10/01/2002 |
| 6407246 | Phenethyl-thiourea compounds and use Novel phenylethyl-thiourea (PHET) compounds as inhibitors of reverse transcriptase and effective agents for the treatment of HIV infection, including mutant, drug-sensitive, drug-resistant, and multi-drug resistant strains of HIV.... | 06/18/2002 |
| 6403617 | Diaminopyridine-containing thiourea inhibitors of herpes viruses Compounds of the formula ##STR1## Useful in the treatment of diseases associated with herpes viruses including human cytomegalovirus, herpes simplex viruses, Epstein-Barr virus, varicella-zoster virus, humanherpesviruses-6 and -7, and Kaposi herpesvi... | 06/11/2002 |
| 6380190 | Nonnucleoside inhibitors of reverse transcriptase, composite binding pocket and methods for use thererof Novel compounds that are potent inhibitors of HIV reverse transcriptase (RT) are described in the invention. The novel compounds also inhibit replication of a retrovirus, such as human immunodeficiency virus-1 (HIV-1). The novel compounds of the invention... | 04/30/2002 |
| 6380134 | N-pyridyl herbicide compounds Compounds of the formula I ##STR1## in which A is .dbd.N-- or ##STR2## R1 is hydrogen, fluorine, chlorine, bromine or methyl; R2 is C1 -C4 alkyl, C1 -C4 haloalkyl, halogen, R6 O... | 04/30/2002 |
| 6372767 | Benzanilides as potassium channel openers Benzanilides are provided which are voltage-dependent potassium channel openers. Methods of using the benzanilides of the invention are also provided.... | 04/16/2002 |
| 6306884 | Benzamidine derivatives and their use as anti-coagulants This invention is directed to benzamidine derivatives which are useful as anti-coagulants. This invention is also directed to pharmaceutical compositions containing the compounds of the invention, and methods of using the compounds to treat disease-states... | 10/23/2001 |
| 6300351 | Beta-fluoroethyl thiourea compounds and use Novel compounds that are potent inhibitors of HIV reverse transcriptase (RT) are described in the invention. These novel compounds also inhibit replication of a retrovirus, such as human immunodeficiency virus-1 (HIV-1). The novel compounds of the inventi... | 10/09/2001 |
| 6211242 | Benzamide derivatives as vasopressin antagonists This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by the general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkyl, etc., R2 is lower alkyl,... | 04/03/2001 |
| 6207688 | Phenethyl-thiourea compounds and use Novel phenylethyl-thiourea (PHET) compounds as inhibitors of reverse transcriptase and effective agents for the treatment of HIV infection, including mutant, drug-sensitive, drug-resistant, and multi-drug resistant strains of HIV.... | 03/27/2001 |
| 6180654 | Heterocyclic nonnucleoside inhibitors of reverse transcriptase Novel compounds that are potent inhibitors of HIV reverse transcriptase (RT) are described in the invention. These novel compounds also inhibit replication of a retrovirus, such as human immunodeficiency virus-1 (HIV-1). The novel compounds of the inventi... | 01/30/2001 |
| 6172060 | Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses Disclosed are nitrosated and/or nitrosylated phosphodiesterase inhibitors having the formula NOn -PDE inhibitor where n is 1 or 2. The invention also provides compositions comprising such compounds in a pharmaceutically acceptable carrier. The ... | 01/09/2001 |
| 6008362 | Elevation of HDL cholesterol by 2-(-4-chlorol-1-aryl-butylidene)-hydrazinecarbothioamides This invention relates to the treatment of atherosclerosis via raising the level of HDL cholesterol by administration of a compound of the formula ##STR1## wherein R1, R2, and R3 are independently hydrogen, C1 ... | 12/28/1999 |
| 5919792 | Integrin antagonists This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as vitronectin receptor antagonists. The vitronectin receptor antagonist compounds of the present invention are v댣 antagonists, ... | 07/06/1999 |
| 5721259 | Method of using 2-formylpyridine thiosemicarbazone compounds A method of treatment of tumors is provided based upon a compound of the formula ##STR1## wherein one of R1 is NHR4 or NR4 R5 or R3 is NHR4, NR4 R5 or OH, and the... | 02/24/1998 |
| 5714503 | Compounds and methods for inhibition of HIV and related viruses Treatment of AIDS, inhibition of the replication of HIV and related viruses thereof, and formulations using thiourea derivative compounds or salts thereof is disclosed. Also disclosed are novel thiourea derivative compounds.... | 02/03/1998 |
| 5688817 | Di(aromatic) compounds and their use in human and veterinary medicine and in cosmetics Di(aromatic) compounds corresponding to the following formula: ##STR1## in which: Ar represents either ##STR2## n=1 or 2 or: ##STR3## X represents a divalent radical, Z represents O, S or a divalent radical, and R1, R2 | 11/18/1997 |
| 5567721 | Di(aromatic) compounds and their use in human and veterinary medicine and in cosmetics Di(aromatic) compounds corresponding to the following formula: ##STR1## in which: Ar represents either ##STR2## n=1 or 2 or: ##STR3## X represents a divalent radical, Z represents O, S or a divalent radical, and R1, R2 | 10/22/1996 |
| 5519037 | N-cyanoamidine derivatives as anti-influenza agents Antiinfluenza A activity was found in compounds of the formula: ##STR1## wherein X is ##STR2## where one of R1 and R2 is H and the other is phenylamino and Z is --SCH3 or a pharmaceutically acceptable salt thereo... | 05/21/1996 |
| 5516786 | Fungicidal substituted amino acid amides Combating fungi with substituted amine acid derivatives of the formula ##STR1## in which R1 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cycloalkyl or cycloalkenyl, R2, R3, R4 | 05/14/1996 |
| 5506263 | Benzyl derivatives and pesticides containing them Benzyl derivatives of the formula I ##STR1## where A is CH2, CHCl, CH-alkyl, CH-alkoxy, CH-alkylthio or N-alkoxy, B is OH, alkylthio, alkoxy or alkylamino, U, V, W are hydrogen, halogen, alkyl or alkoxy, D is ##STR2## where R' is hydrogen ... | 04/09/1996 |
| 5416110 | Benzyl derivatives and pesticides containing them Benzyl derivatives of the formula I ##STR1## where A is CH2, CHCl, CH-alkyl, CH-alkoxy, CH-alkylthio or N-alkoxy, B is OH, alkylthio, alkoxy or alkylamino, U, V, W are hydrogen, halogen, alkyl or alkoxy, D is ##STR2## where R' is hydrogen ... | 05/16/1995 |
| 5409910 | Substituted pyridines New substituted pyridines are prepared by reducing suitably substituted pyridine derivatives. The new substituted pyridines are suitable as active compounds in pharmaceuticals, in particular for the treatment of hyperlipoproteinaemia.... | 04/25/1995 |
| 5354762 | Six-membered heterocyclic derivatives of N'-substituted N,N'-diacylhydrazines This invention relates to insecticidal compositions containing six-membered heterocyclic derivatives of N'-substituted-N,N'-diacylhydrazines, methods of using such compositions and novel six-membered heterocyclic derivatives of N'-substituted-N,N'-diacylh... | 10/11/1994 |
| 5342958 | Organic compounds derived from urea or thiourea Compounds of the formula ##STR1## wherein A is a hydrogen atoms, a halogen atom, a methyl group, or a methoxy group; B is a hydrogen atom, a halogen atom, a methyl group, or a methoxy group, with the proviso that A and B ar not both a hydrogen atom; ... | 08/30/1994 |
| 5288758 | New urea derivatives, their preparation and their application in therapy New urea derivatives corresponding to the general formula 1 ##STR1## in which: R1 represents a C1 -C4 alkyl group; R2 represents: a C5 -C7 cycloalkyl group a cycloalkylmethyl group in which the ... | 02/22/1994 |
| 5262415 | Aminopyridine compounds An aminopyridine compound represented by the formula: ##STR1## wherein n represents 0 or 1; Z represents .dbd.S, .dbd.O, .dbd.NCN or .dbd.CHNO2 ; R1 represents --CN, --NR3 R4, --CONR3 R4 | 11/16/1993 |
| 5238908 | Herbicidal glutaramic acids and derivatives This invention relates to glutaramic acids and derivatives exhibiting herbicidal activity having the structure ##STR1## wherein A is a carboxylic acid or a derivative thereof, D is CH or N, and R, R1, R2, T, X, Y, and Z are as d... | 08/24/1993 |
