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| Number | Title | Issue Date |
| 8013164 | Insecticidal -substituted (6-halooalkylpyridin-3-yl)-alkyl sulfoximines N-Substituted (6-haloalkylpyridin-3-yl)alkyl sulfoximines are effective at controlling insects. ... | 09/06/2011 |
| 7678918 | Intermediates for imidazonaphthyridines Imidazonaphthyridine and tetrahydroimidazonaphthyridine compounds induce the biosynthesis of cytokines such as interferon and tumor necrosis factor. The compounds exhibit antiviral and antitumor properties. Methods of preparing the compounds and intermediates useful... | 03/16/2010 |
| 7511149 | Process for the oxidation of certain substituted sulfilimines to insecticidal sulfoximines Insecticidal sulfoximines are produced efficiently and in high yield by the oxidation of the corresponding sulfilimine with ruthenium tetraoxide or an alkali metal permanganate. ... | 03/31/2009 |
| 7435743 | Pyridine derivatives Pyrimidine compounds of general formula: wherein —R1 represents in which R11 is hydrogen, C1-6 alkyl, halogen, hydroxy, C1-12 alkoxy,... | 10/14/2008 |
| 7291580 | 6-(1,1-difluoroalkyl)-4-aminopicolinates and their use as herbicides 4-Aminopicolinic acids having (1,1-difluoroalkyl) substituents in the 6-position and their amine and acid derivatives are potent herbicides demonstrating a broad spectrum of weed control. ... | 11/06/2007 |
| 7173129 | Sulfonamide-substituted chalcone derivatives and their use to treat diseases The invention relates to compounds, pharmaceutical compositions and methods of using compounds of the general formula or its pharmaceutically acceptable salt or ester, wherein the substituents are defined in the ... | 02/06/2007 |
| 7125896 | Thiophene carboxamide compounds as inhibitors of enzyme IKK-2 The invention relates to thiophene carboxanmides of formula (I), wherein A, R1, R2, R3, n and X are as defined in the specification, processes and intermediates used in their preparation, pharmaceutical compositions containing them a... | 10/24/2006 |
| 7084159 | Inhibitors of c-Jun N-terminal kinases (JNK) and other protein kinases The present invention provides compounds of formula I: or a pharmaceutically acceptable derivative o thereof, wherein A, B, Ra, R1, R2, R3, and R4 are as des... | 08/01/2006 |
| 6989398 | Benzanilides as potassium channel openers Benzanilides are provided which are voltage-dependent potassium channel openers. Methods of using the benzanilides of the invention are also provided. ... | 01/24/2006 |
| 6984649 | Pyridine derivatives Pyridine compounds of general formula: wherein —R1 represents in which R11 is hydrogen, C1-6 alkyl, halogen, hydroxy, C1-12 ... | 01/10/2006 |
| 6972292 | Certain substituted polyketides, pharmaceutical compositions containing them and their use in treating tumors The present invention relates to certain substituted polyketides of formula I, wherein A, B, C, D, E, F and m are as defined herein, pharmaceutical compositions containing said compounds, and the use of said compounds ... | 12/06/2005 |
| 6951875 | Conjugated aromatic compounds with a pyridine substituent The present invention relates to compounds of formulae The compounds of the present invention are NMDA (N-methyl-D-aspartate)-receptor subtype blockers and are used in the treatment of diseases related to this receptor... | 10/04/2005 |
| 6900210 | Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers The present invention provides novel heterocyclic amides and related derivatives having the general Formula I wherein R1, R2, R3, R4, R5, R6, A, B and Z... | 05/31/2005 |
| 6887877 | Compounds and methods for the treatment or prevention of Flavivirus infections The present invention provides novel compounds represented by formula I: or pharmaceutically acceptable salts thereof useful for treating Flaviviridae viral infection. ... | 05/03/2005 |
| 6872690 | Herbicidal 2-alkynyl-pyri (mi) dines The invention relates method of combating undesired plant growth at a locus, comprising application to the locus of an effective amount of at least one compound of formula (I): wherein R1 | 03/29/2005 |
| 6831174 | Processes for preparing substituted 1, 3-oxathiolanes with antiviral properties Disclosed are processes for preparing compounds of the formula (I) and pharmaceutically acceptable salts or esters thereof: wherein R2 is a purine or pyrimidine base or an analogue or derivative thereof; and... | 12/14/2004 |
| 6825204 | N-substituted 3-hydroxy-4-pyridinones and pharmaceuticals containing thereof N-substituted 3-hydroxy-4-pyridinones and metal chelates, methods of preparing N-substituted 3-hydroxy-4-pyridinones and metal chelates, and pharmaceutical compositions containing new N-substituted 3-hydroxy-4-pyridinones and/or their metal chelates. Use of N-substi... | 11/30/2004 |
| 6624179 | Geometrical isomers of acrylonitrile compounds, mixture thereof, and process for producing these A geometrical isomer of an acrylonitrile compound represented by the formula (I) or of its salt, or a mixture thereof: ##STR1## [wherein T is phenyl or pyridyl, which is substituted by R2, Q is phenyl, thienyl, pyridyl or benzyl, which may be s... | 09/23/2003 |
| 6569860 | Alkoxycarbonylamino heteroaryl carboxylic acid derivatives as IP antagonists This invention relates to compounds which are IP receptor antagonists and which are represented by Formula (I): ##STR1## wherein G2 is a heteroaryl group containing one or two nitrogen atoms substituted with a carboxylic acid group, said hetero... | 05/27/2003 |
| 6566375 | Elevation of HDL cholesterol by 4-[(aminothioxomethyl)-hydrazono]-N-(substituted)-4-arylbutanamides Compounds of this invention increase plasma levels of high density lipoprotein or HDL, the "good" cholesterol and as such may be useful for treating diseases such as atherosclerosis. These compounds are represented by the formula ##STR1## wherein: R | 05/20/2003 |
| 6465491 | 6-phenylpyridyl-2-amine derivatives The present invention relates to certain 6-phenyl-pyridin-2-ylamine derivatives that exhibit activity as nitric oxide synthase (NOS) inhibitors, to pharmaceutical compositions containing them and to their use in the treatment and prevention of central ner... | 10/15/2002 |
| 6380214 | Heterocyclic derivatives useful as anticancer agents The present invention relates to compounds of the formula 1 ##STR1## and to pharmaceutically acceptable salts, prodrugs and solvates thereof, wherein Z, X, X1, R1, R2 and R3 are as defined herein as it relates t... | 04/30/2002 |
| 6369082 | Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment This invention encompasses the novel compounds of formula A, which are useful in the treatment of prostaglandin mediated diseases, ##STR1## or a pharmaceutically acceptable salt, hydrate or ester thereof. The invention also encompasses pharmaceutical comp... | 04/09/2002 |
| 6369084 | Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment This invention encompasses the novel compounds of formula A, which are useful in the treatment of prostaglandin mediated diseases, ##STR1## or a pharmaceutically acceptable salt, hydrate or ester thereof. The invention also encompasses certain pharmaceuti... | 04/09/2002 |
| 6331639 | Process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative A compound represented by the formula (1) which is useful as an agricultural fungicide or an intermediate thereof can be obtained by reacting a compound of the general formula (2) with a compound of the general formula (3) in the presence of an acid and r... | 12/18/2001 |
| 6331634 | Process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative A compound represented by the formula (1) which is useful as an agricultural fungicide or an intermediate thereof can be obtained by reacting a compound of the general formula (2) with a compound of the general formula (3) in the presence of an acid and r... | 12/18/2001 |
| 6329400 | Formamide compounds as therapeutic agents A family of compounds having the general structural formula ##STR1## where W is a reverse hydroxamic acid group, and R1, R2, R3, R4, R5 and R6 are as described in the specification, or a ph... | 12/11/2001 |
| 6329418 | Substituted pyrrolidine hydroxamate metalloprotease inhibitors The invention provides compounds which are potent inhibitors of metalloproteases and which are effective in treating conditions characterized by excess activity of these enzymes. In particular, the present invention relates to compounds having a structure... | 12/11/2001 |
| 6306892 | Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their use The present invention is directed to compound of the formula I: ##STR1## wherein R1, R2, R3, R4, R 5, X, Y, and ##STR2## are as defined herein. These compounds are useful for inhibiting the activity of a ... | 10/23/2001 |
| 6288091 | Antiherpes virus compounds and methods for their preparation and use This invention relates to methods for inhibiting herpes replication and for treating herpes infection in a mammal by inhibiting the herpes helicase-primase enzyme complex. This invention also relates to thiazolyphenyl derivatives that inhibit the herpes h... | 09/11/2001 |
| 6271236 | Diaminopyridine-containing thiourea inhibitors of herpes virus Compounds of the formula ##STR1## wherein R1 -R5 are independently selected from hydrogen, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl ... | 08/07/2001 |
| 6252082 | Pyridone derivatives, their preparation and their use as synthesis intermediates The invention concerns compounds of formula (I) ##STR1## in which: R is --NO2 or --NHR3, R3 being hydrogen, --COR4 (R4 selected among (C1 -C4) alkyl, aryl and aryl (C1... | 06/26/2001 |
| 6245774 | Tri-substituted phenyl or pyridine derivatives Compounds of general formula (1) are described: ##STR1## wherein .dbd.W-- is (1) .dbd.C(Y)-- where Y is a halogen atom, or an alkyl or --XRa group where X is --O--, --S(O)m -- [where m is zero or an integer of value 1 or 2], or --N(R... | 06/12/2001 |
| 6239282 | Process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative A compound represented by the formula (1) which is useful as an agricultural fungicide or an intermediate thereof can be obtained by reacting a compound of the general formula (2) with a compound of the general formula (3) in the presence of an acid and r... | 05/29/2001 |
| 6211242 | Benzamide derivatives as vasopressin antagonists This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by the general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkyl, etc., R2 is lower alkyl,... | 04/03/2001 |
| 6197795 | Preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors The present invention relates to the discovery of novel, low molecular weight, non-peptide inhibitors of matrix metalloproteinases (e.g. gelatinases, stromelysins and collagenases) and TNF- converting enzyme (TACE, tumor necrosis factor- con... | 03/06/2001 |
| 6184382 | Process for preparing N6-substituted adenosine derivatives The invention is directed to improved methods for preparing N6-substituted adenosine derivatives, to intermediates useful therefor and to methods of preparing these intermediates.... | 02/06/2001 |
| 6162814 | Preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metaloproteinase and tace inhibitors The present invention relates to the discovery of novel, low molecular weight, non-peptide inhibitors of matrix metalloproteinases (e.g. gelatinases, stromelysins and collagenases) and TNF- converting enzyme (TACE, tumor necrosis factor- con... | 12/19/2000 |
| 6143894 | Preparation of [1S-[1A,2B,3B,4A(S*)]]-4-[7-[[1-(3-chloro-2-thienyl)methyl propyl]amino] -3H-imidazo[4,5-B]pyridin-3-yl]-N-ethyl-2,3-dihydroxycyclopentanecarboxa mide This invention is directed to methods for the preparation of [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-chloro-2-thienyl) methyl]propyl]amino]-3H-imidazo[4,5-b]pyridin-3-yl]-N-ethyl-2,3-dihydroxyc yclopentanecarboxamide, methods for the preparation of intermediate... | 11/07/2000 |
| 6121202 | Thienyloxypyridines and-pyrimidines useful as herbicidal agents The present invention provides a herbicidal compound of formula I, methods for the preparation thereof and intermediates useful therefor. ##STR1## wherein X and Y are each independently O or S; Z is N or CR4.... | 09/19/2000 |
