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| Number | Title | Issue Date |
| 8168793 | Nitrocatechol derivatives as COMT inhibitors New compounds of formula I are described. The compounds have potentially valuable pharmaceutical properties in the treatment of some central and peripheral nervous system disorders. ... | 05/01/2012 |
| 7390907 | Vanilloid receptor ligands and their use in treatments Compounds having the general structure and compositions containing them, for the treatment of acute, inflammatory and neuropathic pain, dental pain, general headache, migraine, cluster headache, mixed-vascular and non-vascu... | 06/24/2008 |
| 7390804 | N-containing five-membered ring compounds and pharmaceutical agents comprising the same as active ingredient An N-containing five-membered ring compound of formula (I) wherein all symbols are the same as described in the specification, and a non-toxic salt thereof. The compound of formula (I) has an inhibitory activity aga... | 06/24/2008 |
| 7365196 | Sulphonamido-substituted bridged bicycloalkyl derivatives A class of compounds is disclosed, comprising sulphonamido-substituted bridged bicycloalkyl structures. The compounds are inhibitors of gamma-secretase, and hence are useful in the treatment of and/or prevention of Alzheimer's disease. ... | 04/29/2008 |
| 7351724 | Oxadiazole ketone inhibitors of fatty acid amide hydrolase Certain oxadiazole ketone compounds are useful as FAAH inhibitors. Such compounds may be used in pharmaceutical compositions and methods for the treatment of disease states, disorders, and conditions mediated by fatty acid amide hydrolase (FAAH) activity. Thus, the ... | 04/01/2008 |
| 7329756 | Process for the manufacture of Isradipine The present invention relates to an improved method for the manufacture of Isradipine, 4-(4-Benzofurazanyl)-1,4-dihydro-2,6-dimethyl-3,5-pyridinedicarboxylic acid methyl 1-methylethyl ester. Which, involves reacting 2,1,3-benzoxadiazole-4-carboxaldehyde with methyl ... | 02/12/2008 |
| 7297797 | Pyrrolines The invention relates to novel Δ1-pyrrolines of the formula (I) in which R1, R2, R3, R4, A1, A2, R5, R6, R7, R | 11/20/2007 |
| 7273877 | 5-substituted-4-[(substituted phenyl) amino]-2-pyridone derivatives The present invention relates to 5-substituted-4-(substituted)phenylamino-2-pyridone derivatives, pharmaceutical compositions and methods of use thereof. ... | 09/25/2007 |
| 7196106 | Cyanothiophene derivatives, compositions containing such compounds and methods of use The present invention addresses substituted cyanothiophene derivatives of the formula I: as well as compositions containing such compounds and methods of treatment. The compounds in the present invention are gluc... | 03/27/2007 |
| 7183303 | Gamma-secretase inhibitors Compounds of formula I: inhibit gamma-secretase and hence find use in treatment of Alzheimer's disease. ... | 02/27/2007 |
| 7169929 | Diaryl 1,2,4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor The present invention relates to a novel diaryl 1,2,4-triazole derivative of the following formula (1) as a highly selective cyclooxygenase-2 inhibitor, wherein R1, R2, R3, R4, R5, W and A is as defined in this ... | 01/30/2007 |
| 7115636 | Hetrocyclic aryl sulphonamides The invention relates to novel sulfonamides of general formula (I) where the substituents R1, R2, R3, R4, A and X have the given meanings, pharmaceutical compositions c... | 10/03/2006 |
| 7105538 | 2-pyrrolidin-2-yl-[1,3,4]-oxadiazole compounds and their use as anti-depressants Substituted 2-pyrrolidin-2-yl compounds corresponding to formula I a method for their production, pharmaceutical compositions containing them, and methods of using them, especially for treating pain and/or depres... | 09/12/2006 |
| 7105556 | Conformationally constrained analogs useful as antidiabetic and antiobesity agents and method Compounds are provided which have the structure wherein Q is C or N, X1 is C or N, and R1, R2, R2a, R2b, R2c, R3, Y, A, m, n, X2 | 09/12/2006 |
| 7041685 | Substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof The present invention is directed to substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs thereof, represented by the Formula I: wherein Ar1, Ar3, A, B and D are defined herein. The present i... | 05/09/2006 |
| 6987189 | Short synthesis of pyridine-based pharmaceutical intermediates A method of making a compound of Formula VI: wherein Tr is a triphenyl group; R1, R2 and R3 are each independently selected from the group consisting of H, C1–C4 alkyl, C1–C4 alkoxy,... | 01/17/2006 |
| 6906089 | Triarylimidazole derivatives as cytokine inhibitors Compounds of formula (I) or a pharmaceutically acceptable salt thereof: wherein R1, R2 and R3 are various substituent groups; and one of X... | 06/14/2005 |
| 6855825 | Short synthesis of pyridine-based pharmaceutical intermediates A method of making a compound of Formula VI: wherein Tr is a triphenyl group; R1, R2 and R3 are each independently selected from the group consisting of H, C1-C4 alkyl, C1-C4 alkoxy, ar... | 02/15/2005 |
| 6821972 | 3-heterocyclylpropanohydroxamic acid PCP inhibitors Compounds of formula (I): and their salts, solvates, hydrates and prodrugs are useful PCP inhibitors, processes for making the same, compositions comprising the same, and methods of treating a PCP-mediated condition or... | 11/23/2004 |
| 6734143 | 2-methoxyimino-2(pyridinyloxymethyl)phenyl acetamides useful as fungicides The present invention provides 2-methoxyimino-2-(pyridinyloxymethyl) phenyl acetamides according to formula (I) as well as their use as fungicidal compounds. ... | 05/11/2004 |
| 6689779 | Oxazolidinone derivatives and a process for the preparation thereof The present invention relates to novel oxazolidinone derivatives, their pharmaceutically acceptable salts and a process for the preparation thereof. More particularly, the present invention relates to oxazolidinone derivatives having pyridine or pyrimidin... | 02/10/2004 |
| 6579880 | Isoxazoles and oxadiazoles as anti-inflammatory inhibitors of IL-8 The invention relates to isoxazole and oxadiazole compounds of Formulae I and II, ##STR1## pharmaceutical compositions containing the compounds, and methods for their production and use. These compounds are effective in inhibiting the action of IL-8 ... | 06/17/2003 |
| 6531485 | Prostaglandin agonists This invention relates to prostaglandin agonists, methods of using such prostaglandin agonists, pharmaceutical compositions containing such prostaglandin agonists and kits containing such prostaglandin agonists. The prostaglandin agonists are useful for t... | 03/11/2003 |
| 6495578 | Sulfonamide derivatives having oxadiazole rings Sulfonamide derivatives having a matrix metalloprotease inhibiting effect, which are compounds represented by general formula (I), optical isomers of the same, pharmaceutically acceptable salts of both, or solvates of them: ##STR1## wherein R1 ... | 12/17/2002 |
| 6458950 | Compounds and pharmaceutical compositions containing the same A compound shown by the formula II, wherein Het is a mono- or polycyclic heterocyclic group comprising one or more hetero atoms selected from the group consisting of N, O and S which may be the same or different from each other; R1 is hydrogen,... | 10/01/2002 |
| 6458814 | Vitronectin receptor antagonists Compounds of the formula (I) are disclosed which are vitronectin receptor antagonists and are useful in the treatment of osteoporosis: ##STR1## or a pharmaceutically acceptable salt thereof.... | 10/01/2002 |
| 6436965 | PDE IV inhibiting amides, compositions and methods of treatment Compounds represented by formula I: ##STR1## as well as pharmaceutically acceptable salts and hydrates thereof are disclosed as useful for treating or preventing diseases and conditions mediated by PDE-IV. Pharmaceutical compositions and methods of treatm... | 08/20/2002 |
| 6432960 | Squarate derivatives of dihydropyridine NPY antagonists A series of antagonists of NPY have been synthesized and are comprised of squarate derivatives of 4-phenyl-1,4-dihydropyridines of Formula (I). ##STR1## As antagonists of NPY-induced behavior, these compounds are expected to act as effective anorexiant ag... | 08/13/2002 |
| 6369226 | Substituted benzamide inhibitors of rhinovirus 3C protease Nonpeptide benzamide-containing inhibitors of human rhinovirus (HRV) 3C protease are described.... | 04/09/2002 |
| 6306873 | Substituted ଲ-thiocarboxylic acids This invention relates to compounds of general formula (I): ##STR1## in which Ar is a group selected from: ##STR2## A1, A2, B, C, D, E, Q1-Q3, R1-R9, Z1 and Z2 are as defined in the disclosure, and Y represents carboxy or an acid bioisostere. These c... | 10/23/2001 |
| 6303600 | Substituted azabicyclic compounds This invention is directed to certain physiologically active compounds of formula (I) ##STR1## wherein ##STR2## represents a bicyclic ring system, of about 10 to about 13 ring members, in which the ring ##STR3## is an azaheterocycle, and the rin... | 10/16/2001 |
| 6288236 | Benzimidazole compounds containing a benzoxazole or benzothiazole ring, and compositions and methods of use containing the same Benzimidazole compounds represented by the formula set out below and analogs thereof, wherein Y represents a single bond or sulfur atom; Z represents oxygen atom, sulfur atom, or N--R4 ; R1 and R2 independently represent h... | 09/11/2001 |
| 6133294 | 2-methoxyimino-2-(pyridinyloxymethyl) phenyl acetamides with 5 membered heterocyclic rings on the pyridine ring The present invention provides novel 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamide compounds with 5 membered heterocyclic rings on the pyridine ring, their use as fungicidal compounds, and their use in fungicidal compositions comprising at least ... | 10/17/2000 |
| 6107314 | Pesticides Compounds of formula (I) or pesticidally acceptable salts thereof, compositions containing them and methods of use. ##STR1##... | 08/22/2000 |
| 6083957 | Heterocyclic compounds and their preparation and use The present invention relates to therapeutically active quaternary azacyclic or azabicyclic compounds with formula I: ##STR1## wherein X is oxygen or sulfur and wherein G is selected from the group of azacyclic or azabicyclic ring systems consisting ... | 07/04/2000 |
| 5998446 | 2-[2-(Hetaryl oxymethylene)phenyl] crotonates used as pesticides and fungicides There are described compounds of the general formula I ##STR1## where the index and the substituents have the following meanings: R is cyano, halogen, alkyl or alkoxy; n is 0, 1 or 2, it being possible for the substituents R to differ from each other... | 12/07/1999 |
| 5998456 | Benzimidazole compounds containing 1,2,4-triazole ring, and compositions and methods of use containing the same Benzimidazole compounds represented by the formula set out below and analogs thereof, wherein Y represents a single bond or sulfur atom; Z represents oxygen atom, sulfur atom, or N--R4 ; R1 and R2 independently represent h... | 12/07/1999 |
| 5985904 | 1,2,4-oxadiazole derivatives and their use as parasiticides for animals The invention relates to 1,2,4-oxadiazole derivatives of the formula (I) ##STR1## in which R1, R2, R3, R4, R5, R6, X, Y, m and n have the meanings given in the description, to a plurality o... | 11/16/1999 |
| 5962656 | Indazole containing coupler A photographic element comprising a support having situated thereon at least one silver halide emulsion layer, the layer containing a photographic coupler represented by the formula COUP--T1 --T2 --(T3)b --PUG wherei... | 10/05/1999 |
| 5922724 | Benzimidazole compounds and their use as modulators of the GABA a receptor complex The present patent application discloses compounds having the formula ##STR1## or a pharmaceutically acceptable salt thereof or an oxide thereof wherein R3 is ##STR2## wherein A, B and D each is CH, or one or two of A, B and D is N an... | 07/13/1999 |
