Class 544/51 - 1,4-benzothiazines

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the sulfur and nitrogen atoms of the benzothiazine
No. of patents: 83
Last issue date: 03/25/2008

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Number	Title	Issue Date
7348426	Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents The present invention relates to novel antiobesity and hypocholesterolemic compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates...	03/25/2008
7211668	PNA monomer and precursor This application relates to monomers of the general formula (I) for the preparation of PNA (peptide nucleic acid) oligomers and provides method for the synthesis of both predefined sequence PNA oligomers and random sequence PNA oligomers:	05/01/2007
7141564	Nitrogen-containing bicyclic heterocycles for use as antibacterials Cyclohexane and cyclohexene derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly man. ...	11/28/2006
7067513	Phenylpiperazines The invention relates to a novel group of phenylpiperazines having interesting pharmacological properties such as a high affinity for the dopamine D2 receptor and/or the serotonin reuptake site, and the ability to treat conditions related to disturbances ...	06/27/2006
7049312	Benzothiazinone and benzoxazinone compounds Q is —N=or CR2 X is S, O or NOR3 Y is —O—, —S—, —SO— or —SO2— R and R1 are each...	05/23/2006
6995154	Heterocyclic topoisomerase poisons The invention provides compounds of formula I: wherein R1 to R5 have any of the values defined in the specification, as well as pharmaceutically acceptable salts of the compounds, pharmaceutical co...	02/07/2006
6974873	Modified carbocyanine dyes and their conjugates Chemically reactive carbocyanine dyes incorporating an indolium ring moiety that is substituted at the 3-position by a reactive group or by a conjugated substance, and their uses, are described. Conjugation through this position results in spectral properties that a...	12/13/2005
6919332	N-substituted-heteroaryloxy-aryloxy-pyrimidine-2,4,6-trione metalloproteinase inhibitors The present invention relates to N-substituted-heteroaryloxy-aryloxy-2,4,6-trione metalloproteinase inhibitors of the formula wherein X, A, Y, B, G, and R1 are as defined in the specification, and to pharmac...	07/19/2005
6914059	Benzoxazine and benzothiazine derivatives and the use thereof in medicaments Compounds of formula I, their tautomeric and isomeric forms and salts, as well as the process for their production and their use in pharmaceutical agents are described. ...	07/05/2005
6897305	Calcium channel drugs and uses Novel multibinding compounds are disclosed. The compounds of this invention comprise 2-10 ligands covalently connected, each of the ligands being capable of binding to a ligand binding site in a Ca++ channel , thereby modulating the biological activities ...	05/24/2005
6809095	Bicyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them A method for preventing or treating complications of diabetes by administering a compound of formula (I) its tautomeric forms, its stereoisomers, its polymorphs, its pharmaceutically acceptable salts or its pharmaceuti...	10/26/2004
6716851	Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof The present invention is directed to substituted 2-aryl-4-arylaminopyrimidine and analogs thereof, represented by the general Formula I: wherein A, Ar1, Ar2, R1 and R3 are defi...	04/06/2004
6696435	Substituted N,N-disubstituted fused-heterocyclo amino compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for treating...	02/24/2004
6667302	Heterocyclic topoisomerase poisons The invention provides compounds of formula I: ##STR1## wherein R1 to R5 have any of the values defined in the specification, as well as pharmaceutically acceptable salts of the compounds, pharmaceutical compositions comprising the c...	12/23/2003
6620809	Substituted (dihydro)benzoxazine and (dihydro)benzothiazine compounds The invention relates to compound of formula (I): ##STR1## wherein: G represents an alkylene chain containing from 1 to 4 carbon atoms, A represents ##STR2## X represents oxygen or sulphur and R2 and R1 are as defined in t...	09/16/2003
6573218	Fused-benzene derivatives useful as herbicides A compound of the formula (Ia): ##STR1## or its salts, in which the variables are as described in the disclosure; herbicidal compositions of said compounds, herbicidal processes using said compounds, defoliant processes using said compounds, and processes...	06/03/2003
6566520	Support for synthesis and purification of compounds A method for the preparation and purification of compounds using a novel support, a tetrabenzo [a, c, g, i]-fluorene group (Tbf) comprising reacting a building block (A) containing a Tbf group (Tbf-A), with a second building block (B), to afford an interm...	05/20/2003
6455519	Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity The invention relates to use of substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for t...	09/24/2002
6448241	Thiazolobenzoheterocycles, their preparation and medicaments containing them Compounds of formula (I): ##STR1## their racemates, enantiomers, diastereoisomers and inorganic acid salts and organic acid salts thereof, processes for preparing them and the medicaments containing them are discussed....	09/10/2002
6448246	Substituted 4H-1,4-benzothiazine-2-carboxamide: GABA brain receptor ligands Disclosed are 4H-1,4-Benzothiazine-2-carboxamides. These compounds are highly selective agonists, antagonists or inverse agonists for GABAa brain receptors or prodrugs of agonists, antagonists or inverse agonists for GABAa brain receptors. These compounds...	09/10/2002
6444615	Herbicidal imidazolidinetrione and thioxo-imidazolidinediones This invention relates to 1-substituted-phenyl-3-substituted-2-thioxo-4,5-imidazolidinediones and 2,4,5-imidazolidinetriones which have activity as herbicides, to compositions which contain these compounds and to methods of use of these compounds. In...	09/03/2002
6437141	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophilic...	08/20/2002
6432946	3-aminoalkylamino-2H-1,4-benzoxazines and 3-aminoalkylamino-2H-1,4-benzothiazines: dopamine receptor subtype specific ligands Disclosed are compounds of the formula: ##STR1## or the pharmaceutically acceptable acid addition salts thereof, wherein: Ar represents aryl or heteroaryl; R1 and R2 are the same or different and represent organic or inorganic substituent...	08/13/2002
6380235	Benzimidazolones and analogues The present invention provides compounds and pharmaceutical formulations useful as progesterone receptor agonists and antagonists and having the general formula: ##STR1## wherein: A is O, S, or NR4 ; B is a bond between A and C.dbd.Q, or the mo...	04/30/2002
6300342	Antithrombotic phenylalkyl derivatives Antithrombotic phenylalkyl derivatives of the formula ##STR1## Exemplary compounds are: (a) 1-[3-(4-amidino-phenyl)propionyl]-6-(4-fluoro-phenylsulphonamido)-1,2,3,4- tetrahydro-quinoline, (b) 1-[3-(4-amidino-phenyl)propionyl]-6-butylsulphonamido-1,2,...	10/09/2001
6265401	Bicyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them Compounds of formula (I) ##STR1## its tautomeric forms, its stereoisomers, its polymorphs, its pharmaceutically acceptable salts or its pharmaceutically acceptable solvates can be used to prevent or treat diabetes caused by insulin resistance or impa...	07/24/2001
6232310	Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use The present invention relates to fused 1,4-thiazine-2-carbonitrile derivatives, compositions thereof and methods for preparing the compounds. The compounds are useful in the treatment of diseases of the central nervous system, the cardiovascular system, the pu...	05/15/2001
6224644	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophilic...	05/01/2001
6204389	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 --R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophili...	03/20/2001
6200378	Thiazine indigo pigments, solid solutions thereof and their preparation A compound according to the formula (I) ##STR1## wherein R1 and R2 are independently the atoms necessary to complete the formation of a substituted or unsubstituted aromatic or aliphatic carbocyclic or heterocyclic ring system and R	03/13/2001
6197956	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrophilic...	03/06/2001
6191127	Substituted heterocycles and their use in medicaments Compounds of Formula I ##STR1## wherein X and R1-6, are as defined herein, tautomeric forms thereof, and isomeric forms thereof, and salts thereof, are suitable for treating diseases that are induced by the action of nitrogen monooxide at ...	02/20/2001
6114350	Cyanine dyes and synthesis methods thereof A cyanine dye having the formula ##STR1## wherein R1 -R8 are each independently selected from a group consisting of hydrogen, C1 -C6 alkyl group, and C0 -C4 alkyl group having a hydrop...	09/05/2000
6107308	Piperidine derivatives The present invention is directed to a piperidine derivative represented by the following formula (1) or a salt thereof: ##STR1## wherein R1, R2, and R3 individually represent hydrogen atoms, etc., Y represents #...	08/22/2000
6100255	3-aminoalkylamino-2H-1,4-benzoxazines and 3-aminoalkylamino-2H-1,4-benzothiazines: dopamine receptor subtype specific ligands Disclosed are compounds of the formula: ##STR1## or the pharmaceutically acceptable acid addition salts thereof, wherein: Ar represents aryl or heteroaryl; R1 and R2 are the same or different and represent organic or inorganic substi...	08/08/2000
6071860	2,4-Diamino-1, 3,5-triazines, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## where R1 to R5, A, Z, X, X', n and m are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepared analogously to known processes u...	06/06/2000
6069114	2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepa...	05/30/2000
6025355	Pharmaceutically active compounds and methods of use The present invention relates to pharmaceutically acceptable compounds, including certain substituted indolinyl and derivatives thereof, 1,2,3,4-tetrahydroquinolinyl and derivatives thereof, 1,2,3,4-tetrahydroisoquinolinyl, benz[cd]indolinyl and 5,6-...	02/15/2000
6011033	Phenylene derivatives This invention relates to a phenylene derivative represented by the following formula (1) or a salt thereof and also to a medicine containing it as an effective ingredient. ##STR1## wherein R1 represents H or halogen; A represents --CH.dbd...	01/04/2000
6011031	Azolidinediones useful for the treatment of diabetes, dyslipidemia and hypertension: process for their preparation and pharmaceutical compositions containing them Novel antidiabetic compounds, their tautomeric forms, their derivatives, their analogues, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compositio...	01/04/2000

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Class 544/51 - 1,4-benzothiazines