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| Number | Title | Issue Date |
| 5955491 | Method for treating osteoporosis The present invention provides a cathepsin L inhibitor containing a compound of the formula: ##STR1## wherein R1 is a hydrogen atom or an arylalkyl, heterocyclic-alkyl or lower alkyl group which may be substituted; R2 and R... | 09/21/1999 |
| 5948792 | Fluorine-containing 1,4-disubstituted piperidine derivatives Novel fluorine-containing 1,4-disubstituted piperidine derivatives, represented by general formula I! ##STR1## such as, for example, (2R)-N-1-(6-aminopyridin-2-ylmethyl)piperidin-4-yl!-2-(1R)-3,3-difluoroc yclopentyl!-2-hydroxy-2-phenylacet... | 09/07/1999 |
| 5948551 | Use of conjugated compounds containing pyrimidine groups as electroluminescence materials The use of conjugated compounds which contain two or more pyrimidine rings as part of the conjugated system as electroluminescence materials. The conjugated compounds containing pyrimidine rings have a high thermal stability and a high photostability. The... | 09/07/1999 |
| 5948912 | Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands Disclosed are compounds encompassed by general formula (I), wherein, A represents ethenylene, or A represents --X--CH2 --; where X is carbon or oxygen, provided that when X is oxygen, the oxygen is adjacent the 6-membered ring; R1, R... | 09/07/1999 |
| 5948779 | Substituted condensation products of n-benzyl-3-indenyl acetamides with heterocyclic aldehydes Substituted condensation products of N-benzyl-3-indenylacetamides with heterocyclic aldehydes are useful for inducing or promoting apotosis and for arresting uncontrolled neoplastic cell proliferation, and are specifically useful in the arresting and trea... | 09/07/1999 |
| 5948903 | Synthesis of 3-deazapurines This invention relates to compounds based on the 3-deazapurines ring system and to methods for making such compounds. The invention also generally relates to the field of "antisense" agents, agents that are capable of specific hybridization with a nucleot... | 09/07/1999 |
| 5945572 | Method for producing aryl alkyl hydroperoxides A method for producing aryl alkyl hydroperoxides which comprises selectively oxidizing an aryl alkyl hydrocarbon having the formula: ##STR1## wherein P and Q are hydrogen or an alkyl and may be the same or different from each other; x is an integer o... | 08/31/1999 |
| 5942535 | a!-Annelated pyrrole derivatives and pharmaceutical use thereof The present invention relates to heterocyclic compounds of the formula ##STR1## in which R1 -R7, B, a and X have the meanings recited in the specification. These compounds are usable in the treatment of diseases of the rheumatoi... | 08/24/1999 |
| 5925631 | Alkylated styrenes as prodrugs to COX-2 inhibitors The invention encompasses the novel compound of Formula I useful in the treatment of cyclooxygenase-2 mediated diseases. ##STR1## The invention also encompasses certain pharmaceutical compositions for treatment of cyclooxygenase-2 mediated diseases c... | 07/20/1999 |
| 5922748 | Indole derivatives as 5-HT agonists Compounds of formula (I) ##STR1## wherein R and R1 are hydrogen, C1-4 alkyl or are linked to form a ring, A is a cycloalkyl or alkyl-cycloalkyl group, n is an integer from 0 to 3, W is an optionally substituted 5-or 6-membered hetero... | 07/13/1999 |
| 5922710 | Iminooxybenzylcrotonate esters, their preparation and their use Iminooxybenzylcrotonate esters of the formula I ##STR1## where the index and the substituents have the following meanings: n is 0, 1, 2, 3 or 4; R is nitro, cyano, halogen, unsubst. or subst. alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy o... | 07/13/1999 |
| 5922744 | Ethane-1-2-diamine derivatives and tachykinin antagonists The present invention provides a compound of formula: ##STR1## wherein R, R1, R2, R3, R4, R5, R6a and R6b are defined herein or a pharmaceutically acceptable salt thereof, a... | 07/13/1999 |
| 5919790 | Hydroxamate inhibitors of interleukin-1ଲ converting enzyme The present invention relates to compounds that are inhibitors of interleukin-1ଲ converting enzyme that have the Formula II ##STR1## This invention also relates to a method of treatment of stroke, inflammatory diseases, septic shock, reperfusio... | 07/06/1999 |
| 5919930 | Process for cross-coupling aromatic boron compounds with aromatic halogen compounds or perfluoroalkylsulfonates Process for cross-coupling aromatic boron compounds with aromatic halogen compounds or perfluoroalkylsulfonates. In a process for preparing polycyclic aromatic compounds by cross-coupling aromatic boron compounds with aromatic halogen compounds or perfluo... | 07/06/1999 |
| 5919432 | Polyaminated ligands and metal complexes thereof Poly(amino acid) derivatives, which are chelating agents of paramagnetic metal ions, in which at least 3 of the donor nitrogen atoms carry identical or different substituents, of formula CH(R1)--X, in which X represents CO2 Ra,... | 07/06/1999 |
| 5912244 | Benzopyrans A compound of the formula: ##STR1## or a pharmaceutically acceptable salt thereof, wherein X is O, S or NH; R and R1 are each independently selected from H and C1 -C4 alkyl or taken together represent C2 -C... | 06/15/1999 |
| 5912350 | Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands Disclosed are compounds of the formula: ##STR1## where S and V are various organic or inorganic substituents; G and K are the same or different and represent N or CR' where R' is an organic or inorganic substituent; R is hydrogen or an alkyl group; R... | 06/15/1999 |
| 5908845 | Polyether nucleic acids A compound comprising a polyether backbone bearing a plurality of ligands that are individually bound to chiral carbon atoms located within said backbone, at least one of said ligands including a moiety selected from the group consisting of a naturally oc... | 06/01/1999 |
| 5905068 | Retroviral protease inhibiting compounds A compound of the formula: ##STR1## is disclosed as a retroviral protease inhibitor compound. Also disclosed are methods and compositions for inhibiting an HIV infection.... | 05/18/1999 |
| 5889058 | Peptidyl derivatives Methods of use for compounds of formula (I) are described wherein R represent a --CONHOH, carboxyl (--CO2 H) or esterified carboxyl group; R1 represents a hydrogen atom or an optionally substituted alkyl, alkenyl, aryl, aralkyl, hete... | 03/30/1999 |
| 5886162 | Lipophilic diakylaminomethylene prodrug derivatives for the inhibition of replication of viruses This invention provides new lipophilic dialkylaminomethylene prodrugs, particularly dialkylaminomethylene 2', 3'-dideoxynucleoside compounds and pharmaceutical compositions comprising said compounds which inhibit the replication of viruses.... | 03/23/1999 |
| 5886242 | Polymerizable, chiral compounds and their use The invention relates to chiral compounds containing at least one divalent or polyvalent chiral group, at least one polymerizable group, at least one spacer and at least one mesogenic group, and to their use as polymerizable, chiral dopes for the preparat... | 03/23/1999 |
| 5883254 | Process for making pyrimidine derivatives The present invention provides a process for the manufacture of pyrimidines of formula I: ##STR1## wherein R1, R2, R3 each independently represent hydrogen, C1-7 -alkyl, or C1-7 -alkoxy, A signif... | 03/16/1999 |
| 5869677 | 3,3-(disubstituted)cyclohexan-1-carboxylate monomers and related compounds The present invention relates to novel 3,3-(disubstituted)cyclohexan-1-carboxylate monomers and related compounds, pharmaceutical compositions containing these compounds, and their use in treating allergic and inflammatory diseases and for inhibiting... | 02/09/1999 |
| 5866576 | Epoxide-containing compounds Disclosed are enantiomers, diastereomers, salts, solvates, hydrates and mixtures thereof, of formula I: ##STR1## The core moiety is a monocyclic ring structure having five to six ring atoms and two nitrogen atoms at the 1 and 3 positions, n is an int... | 02/02/1999 |
| 5866578 | Substituted pyrimidines for control of diabetic complications This invention relates to methods of inhibiting sorbitol dehydrogenase, lowering fructose levels, and treating or preventing diabetic complications such as diabetic neuropathy, diabetic retinopathy, diabetic nephropathy, diabetic microangiopathy or diabet... | 02/02/1999 |
| 5866577 | Aromatic amidine derivatives and salts thereof An anticoagulant agent which comprises, as an active ingredient, an aromatic amidine derivative represented by the following general formula (1) or a salt thereof: ##STR1## wherein the group represented by ##STR2## is a group selected from ... | 02/02/1999 |
| 5863926 | 4,4-(disubstituted)cyclohexan-1-carboxylate monomers and related compounds The present invention relates to novel 4,4-(disubstituted)cyclohexan-1-carboxylate monomers and related compounds, pharmaceutical compositions containing these compounds, and their use in treating allergic and inflammatory diseases and for inhibiting... | 01/26/1999 |
| 5859034 | Tri-substituted phenyl compounds which have useful pharmaceutical activity Tri-substituted phenyl derivatives having the general formula (I): ##STR1## In a preferred embodiment, Y is preferably an --XRa group, X is preferably --O--, Z is preferably an --XR5 group, Ra is preferably hydrogen o... | 01/12/1999 |
| 5856273 | Herbicidally active phenylsubstituted 5-and 6-membered heterocyclic compounds A compound of formula (I): ##STR1## where E is oxygen or sulphur; A is CR3 or N where R3 is hydrogen or hydrocarbyl; D completes a 5 or 6-membered non-aromatic heterocyclic ring which optionally contains additional heteroatoms s... | 01/05/1999 |
| 5856560 | Preparation of a-methoxyiminocarboxylic acid methylamides and intermediates therefore A process and intermediates for preparing -methoxyiminocarboxylic acid methylamides (I) by Pinner reaction of a cyanoketone (II) with an alcohol and subsequent reaction of the resulting ester (IV) with hydroxylamine to give the oxime (V), methylati... | 01/05/1999 |
| 5854232 | Acyclic anc cyclic amides as neurotransmitter release enhancers This invention relates to compounds of formula (IA), (IB), (IC) or (ID), wherein m, X, Z, R2, R3, R4, R5, R6, R14 and the dotted lines are as defined below, their pharmaceutically acceptable ... | 12/29/1998 |
| 5847035 | Substituteed tetrahydropyrimidine derivatives and their use as polymerization inhibitors for vinyl aromatic compounds The present invention is directed to substituted tetrahydropyrimidine derivatives of the general formula ##STR1## wherein R1, R2, R3, R4, R5, R6 and R7, which may be the sam... | 12/08/1998 |
| 5824682 | Vasoconstrictive dihydrobenzopyran derivatives The present invention is concerned with compounds of formula ##STR1## the pharmaceutically acceptable acid addition salts thereof, and the stereochemically isomeric forms thereof, wherein R1 is hydrogen or C1-6 alkyl; R2 | 10/20/1998 |
| 5821261 | Substituted saturated aza heterocycles as inhibitors of nitric oxide synthase Disclosed herein are compounds of Formula (I) ##STR1## and pharmaceutically acceptable salts thereof which have been found useful in the treatment of nitric oxide synthase mediated diseases and disorders, including neurodegenerative disorders, disord... | 10/13/1998 |
| 5817879 | Alicyclic peptidomimetics Compounds are provided which are crossreactive with peptides such as those bound by G-protein-linked receptors, together with preparative and therapeutic methods therefor. The compounds have the general structure: ##STR1## wherein at least one of R | 10/06/1998 |
| 5817836 | 2,4-pentadienoic acid derivatives having retinoid-like biological activity Compounds of Formula 1 ##STR1## wherein Z is selected from the group consisting of the radicals shown in Formula 2 and in Formula 3, ##STR2## Y is cycloalkyl or cycloalkenyl of 3 to 8 carbons optionally substituted with one or two R4 | 10/06/1998 |
| 5811028 | Optically active dihydropyran derivative, and liquid crystal composition, liquid crystal device, and racemic mixture comprising the derivative A 2H-5,6-optically active dihydropyran derivative represented by the general formula (I) or (I'): ##STR1## wherein Rf represents a fluoroalkyl group having 1 or 2 carbon atoms; a liquid crystal composition and a liquid crystal device comprising the ... | 09/22/1998 |
| 5811428 | Pyrimidine carboxamides and related compounds and methods for treating inflammatory conditions Compounds having utility as antinflammatory agents in general and, more specifically, for the prevention and/or treatment of immunoinflammatory and autoimmune diseases are disclosed. The compounds are pyrimidine- or pyrazine-containing compounds and, in o... | 09/22/1998 |
| 5811408 | 2'-deoxy-2'-(substituted or unsubstituted)methylidene-4'-thionucleosides The present invention relates to 2'-deoxy-2'-(substituted or unsubstituted)methylidene-4'-thionucleosides having excellent antitumor activity, represented by formula I!: ##STR1## wherein B represents a pyrimidine or purine base, R1 and R... | 09/22/1998 |
