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| Number | Title | Issue Date |
| 7700769 | Dihydropteridione derivatives, process for their manufacture and their use as medicament Disclosed are new dihydropteridinones of the formula (I) wherein the groups L, R1, R2, R3, R4 and R5 have the meanings provided herein, the isomers thereof, processes f... | 04/20/2010 |
| 7534880 | Clear photopolymerizable systems for the preparation of high thickness coatings The present invention relates to clear photopolymerisable systems for the preparation of high thickness coatings, to a procedure for their application and to the solid surfaces coated with them. ... | 05/19/2009 |
| 7414053 | Dihydropteridione derivatives, process for their manufacture and their use as medicament Disclosed are new dihydropteridinones of the formula (I) wherein the groups L, R1, R2, R3, R4 and R5 have the meanings provided herein, the isomers thereof, processes f... | 08/19/2008 |
| 7291654 | Storage stability of photoinitiators Compounds of formula (I), wherein R1 is hydrogen or alkyl; R2 is C1-C4alkoxy or a morpholino radical; and R3 is hydrogen or C1-C4alkoxy, are suitable for improving the solubility of specifi... | 11/06/2007 |
| 7030201 | Bottom antireflective coatings The present invention relates to bottom antireflective coating compositions and polymers useful in making such compositions. ... | 04/18/2006 |
| 6749988 | Amine compounds, resist compositions and patterning process Novel amine compounds having a nitrogen-containing cyclic structure and a hydrating group such as a hydroxy, ether, ester, carbonyl, carbonate group or lactone ring are useful for use in resist compositions for preventing a resist film from thinning and also for enh... | 06/15/2004 |
| 6689882 | Process for the synthesis of morpholinylbenzenes A new improved process for synthesizing morpholinylbenzenes of the formula I by reacting morpholine of formula II with a substituted benzene of formula III, wherein morpholine is used as a reactant and as the only one solvent. ##STR1##... | 02/10/2004 |
| 6638930 | Morpholine and thiomorpholine tachykinin receptor antagonists Substituted heterocycles of the general structural formula: ##STR1## are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, asthma and emesis, and calcium channel blockers useful in the treatment of cardiov... | 10/28/2003 |
| 6562815 | Morpholinones as light stabilizers The invention relates to new compounds containing 1-8 active groups of the type 3,3,6,6-polysubstituted 2-morpholinone and having the formula F (A'--Z)m --X (F), wherein m is a number from 1 to 8; X is an organic anchor group of valency m and in case th... | 05/13/2003 |
| 6531471 | Morpholinone and morpholine derivatives and uses thereof This invention is directed to morpholinone and morpholine derivatives which are selective antagonists for human receptors. This invention is also related to uses of these compounds for lowering intraocular pressure, inhibiting cholest... | 03/11/2003 |
| 6511980 | Substituted diamine derivatives useful as motilin antagonists The present invention relates to novel substituted diamine derivatives for the formula ##STR1## wherein R1, R2, R3, R4, X1, X2, X3, X4, A, Y and n are as described in ... | 01/28/2003 |
| 6458781 | Substituted diarylalkyl amides as calcium channel antagonists The present invention provides compounds that block calcium channels and have the Formula I: ##STR1## The present invention also provides pharmaceutical compositions containing the compounds of Formula I and methods of using them to treat stroke, cer... | 10/01/2002 |
| 6458957 | ,-dibromo--chloro-acetophenones as synthons This disclosure relates to the use of ,-dibromo--chloroacetophenone compounds as intermediates for the preparation of aromatic carbonyl compounds, especially aromatic amides. The compound 2,5-bis(2,2,2-trifluoroethoxy)-,&#... | 10/01/2002 |
| 6362182 | Morpholinone and morpholine derivatives and uses thereof This invention is directed to morpholinone and morpholine derivatives which are selective antagonists for human receptors. This invention is also related to uses of these compounds for lowering intraocular pressure, inhibiting cholest... | 03/26/2002 |
| 6355672 | Benzothiepin derivatives, process for the preparation of the same and uses thereof The invention provides compounds of the formula: ##STR1## wherein the ring A is an optionally substituted benzene ring; R1 is an optionally substituted non-aromatic heterocyclic group; R2 and R3 are independently hydrogen ... | 03/12/2002 |
| 6307087 | Ligands for metals and improved metal-catalyzed processes based thereon One aspect of the present invention relates to novel ligands for transition metals. A second aspect of the present invention relates to the use of catalysts comprising these ligands in transition metal-catalyzed carbon-heteroatom and carbon-carbon bond-fo... | 10/23/2001 |
| 6288086 | N-hydroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors Matrix metalloproteinases (MMPs) are a group of enzymes that have been implicated in the pathological destruction of connective tissue and basement membranes. These zinc containing endopeptidases consist of several subsets of enzymes including collagenase... | 09/11/2001 |
| 6218390 | Morpholinone and morpholine derivatives and uses thereof This invention is directed to morpholinone and morpholine derivatives which are selective antagonists for human receptors. This invention is also related to uses of these compounds for lowering intraocular pressure, inhibiting cholest... | 04/17/2001 |
| 6200972 | Heterocyclic esters and amides This invention relates to neurotrophic low molecular weight, small molecule heterocyclic esters and amides having an affinity for FKBP-type immunophilins, and their use as inhibitors of the enzyme activity associated with immunophilin proteins, particular... | 03/13/2001 |
| 6177564 | Process for the synthesis of N-benzyl-3-(4-fluorophenyl)-1-4-oxazin-2-one The present invention is concerned with a novel process for the preparation of N-benzyl-3-(4-fluorophenyl)-1,4-oxazin-2-one of the formula: ##STR1## This compound is useful as an intermediate in the synthesis of compounds which possess pharmacological act... | 01/23/2001 |
| 6150527 | Synthetic multimerizing agents New compounds are disclosed for multimerizing immunophilins and proteins containing immunophilin or immunophilin-related domains. The compounds are of the formula M-L-Q where M is a synthetic ligand for an FKBP protein... | 11/21/2000 |
| 6140326 | Morpholinones as light stabilizers The invention relates to new compounds containing 1-8 active groups of the type 3,3,6,6-polysubstituted 2-morpholinone and having the formula F (A'--Z)m --X (F), wherein m is a number from 1 to 8; X is an organic ... | 10/31/2000 |
| 6133456 | Synthetic multimerizing agents New compounds are disclosed for multimerizing immunophilins and proteins containing immunophilin or immunophilin-related domains. The compounds are of the formula M1 --L--M2 where M1 and M2 are independently moieties... | 10/17/2000 |
| 6107508 | Convergent synthesis of -aryl-ଲ-ketonitriles The present invention relates to processes for the production of -aryl-ଲ-ketonitriles, which serve as synthetic intermediates in the preparation of a series of biologically important molecules such as corticotropin releasing factor (CRF) rece... | 08/22/2000 |
| 6020489 | Cytoprotective fatty moiety compounds Water or lipid soluble, pharmacologically active, antioxidant, anti-phospholipase compounds that are chemically defined. The compounds protect mammalian cells by inhibiting PLA2 and preventing oxidation. In particular, each compound has at leas... | 02/01/2000 |
| 6020332 | Fluorine-containing diphenyl acrylamide antimicrobial agents Fluorine-containing diphenyl acrylamide of general formula (I) have antimicrobial properties. wherein R1 and R2 are independently selected from (C1 -C6)alkyl group, alkyl group, (C1 -C6)alk... | 02/01/2000 |
| 5935585 | Biaromatic amido compounds and pharmaceutical/cosmetic compositions comprised thereof Novel pharmaceutically/cosmetically-active biaromatic amido compounds have the structural formula (I): ##STR1## in which Ar is a radical selected from among those of the following formulae (a)-(e): ##STR2## and are useful for the treatment ... | 08/10/1999 |
| 5869663 | Substituted heterocyclic compounds The invention relates to compounds of the formula ##STR1## in which: A is a divalent radical selected from: A1) --O--CO-- A2) --CH2 --O--CO-- A3) --O--CH2 --CO-- A4) --O--CH2 --CH | 02/09/1999 |
| 5840745 | Hydrosoluble 3-arylidene-2-oxindole derivatives as tyrosine kinase inhibitors Novel hydrosoluble 3-arylidene-2-oxindole derivatives, having tyrosine kinase inhibitor activity, encompassed by general formula (I), wherein m is zero, 1 or 2; A is a bicyclic ring chosen from tetralin, naphthalene, quinoline and indole; R1 is... | 11/24/1998 |
| 5795891 | Acylphenylglycine derivative and preventive and remedy for diseases caused by increased collagenase activity containing said compound as active ingredient An acylphenylglycine derivative represented by general formula (I) or a pharmaceutically acceptable salt thereof, and a preventive and remedy for diseases caused by an increased collagenase activity containing the same as the active ingredient, wherein R | 08/18/1998 |
| 5753707 | Amide derivatives and their use in cosmetic composition An amide derivative represented by the following formula (1): ##STR1## wherein R1 represents a C1-40 hydrocarbon; R2 represents a C1-6 alkylene; R3 represents H, OH or alkoxyl; R4 repr... | 05/19/1998 |
| 5700761 | Herbicidal tricyclic heterocycles Compounds of Formula I having herbicidal utility are disclosed: ##STR1## wherein Q, R1, R2, V, m and p are defined in the text, including compositions containing such compounds, and a method for controlling weeds employing such ... | 12/23/1997 |
| 5464836 | Benzophenones having an antifungal activity A description follows of benzophenones having an antifungal activity and responding to the general formula (I): ##STR1## wherein: R1 and R2, the same or different, represent C1 -C6 alkyl groups, C7 | 11/07/1995 |
| 5436335 | Preparation of 2,6-dimethylmorpholine from N-(2-hydroxypropyl)-2,6-dimethylmorpholine A process for the preparation of 2,6-dimethylmorpholine from N-(2-hydroxypropyl)-2,6-dimethylmorpholine, in which N-(2-hydroxypropyl)-2,6-dimethylmorpholine, in which a) N-(2-hydroxypropyl)-2,6-dimethylmorpholine is caused to react in the presence of a ca... | 07/25/1995 |
| 5153322 | Perfluoro (cycloaliphatic methyleneoxyalkylene) carbonyl fluorides and derivatives thereof Perfluoro (cycloaliphatic methyleneoxyalkylene) compositions are provided. These compositions comprise perfluoro(cycloaliphatic methyleneoxyalkylene) carbonyl fluoride compounds having (a) a perfluorocycloaliphatic moiety which can have up to two perfluor... | 10/06/1992 |
| 5077402 | Novel alpha-aminoacetophenones as photoinitiators Compounds of the formula I, II, III and IIIa ##STR1## in which Ar1 is an unsubstituted or substituted aromatic radical and at least one of the radicals R1 and R2 is an alkenyl, cycloalkenyl or arylmethyl group, are ef... | 12/31/1991 |
| 5068393 | Aromatic derivatives of butyric acid, a process for their preparation and their use in cosmetics and in human and veterinary medicine An aromatic deviative of butyric acid has the formula ##STR1## wherein R1, R2, R3 and R4, each independently, represent hydrogen or alkyl, with at least two of R1 -R4 being other than ... | 11/26/1991 |
| 5041639 | Polysubstituted derivatives of naphtalene, their process of preparation and their application in the cosmetic and pharmaceutical fields New polysubstituted derivatives of naphthalene. These derivatives correspond to the following formula: ##STR1## in which: R1 to R4 is H or CH3 R5 is ##STR2## or (iv) the radical: 2-oxazolinyl m is 0 or... | 08/20/1991 |
| 5001156 | Lipophilic quaternary ammonium salicylates, their use in cosmetics and in dermopharmacy Lipophilic quaternary ammonium salicylate, characterized in that it corresponds to the formula: ##STR1## in which: (i) R1, R2, R3 and R4, which may be identical or different, denote an alkyl or alkylcycloal... | 03/19/1991 |
| 4992547 | Aminoaryl ketone photoinitiators The photopolymerizable mixture described contains (A) at least one ethylenically unsaturated photopolymerisable compound, (B) a photoinitiator of the formula I ##STR1## and (C) a photosensitiser from the group of aromatic carbonyl compounds having a tripl... | 02/12/1991 |
