Class 544/158 - Sulfur attached directly or indirectly to morpholine ring by nonionic bonding

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein sulfur is attached directly or indirectly
No. of patents: 220
Last issue date: 04/05/2011

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Number	Title	Issue Date
7919617	Cytokine inhibitors The present invention provides low molecular weight compounds useful as cytokine inhibitors, and compositions thereof. In particular, compounds of the invention are useful as anti-inflammatory agents. There are further provided methods for the preparation of such ag...	04/05/2011
7560549	Sulfonyloxy derivatives A compound having the formula (I) wherein R1 is a substituted phenyl, R2 is a phenyl substituted with halogen atoms, R3 is a substituted phenyl, D is an oxygen or a methylene, and n is 0 or ...	07/14/2009
7393852	Piperazine derivatives and methods of use Selected compounds are effective for treatment of pain and diseases, such as inflammation mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable derivatives thereof, pharmaceutical compositions and methods for...	07/01/2008
7384941	2-(phenoxymethyl)-and 2-(phenylthiomethyl)-morpholine derivatives for use as selective norepinephrine reuptake inhibitors Compounds of formula (I): wherein A is S or O; R is H; Ar is an optionally substituted phenyl group; X is an optionally substituted phenyl group, a C1-C4 alkyl, a C3...	06/10/2008
7371747	Cyanoalkylamino derivatives as protease inhibitors The present invention is directed to novel cyanoalkylamino derivatives that are inhibitors of cysteine protease such as cathepsins K, S, B and L, in particular cathepsin K Pharmaceutical composition comprising these compounds, method of treating diseases mediated by...	05/13/2008
7341715	Method and agents on the basis of 2-mercaptopropionic acid amides for durable hair forming and a method for producing same The preparation for permanently deforming hair has a pH of 6.5 to 9.5 and contains, as keratin-reducing agent, a 2-mercaptopropion-amide of the formula (I): in which R1 and R2, independently of one ano...	03/11/2008
7294623	Benzyl morpholine derivatives A compound of formula (I) (I) wherein R is H; Ar is an aromatic group selected from phenyl; X is a phenyl group; R′ is H or C1-C4 alkyl; each R1 is independently H or C1-C4 alkyl; and pharmaceutically acceptable salts thereof	11/13/2007
7291385	Conductive film and method for preparing the same A conductive film comprising: a support; a particle-containing layer; and a metal thin film layer, in this order, wherein the particle-containing layer contains particles having a mean particle size of from 1 to 10 μm and a heat decomposed material of a metal acety...	11/06/2007
7279477	Malonyl-CoA decarboxylase inhibitors useful as metabolic modulators The present invention relates to novel compounds (I), their prodrugs, and the pharmaceutically acceptable salts as well as pharmaceutical compositions containing such compounds useful in treating certain metabolic diseases and diseases modulated by the inhibition of...	10/09/2007
7141560	Alanine 2,6-dialkoxyphenyl ester derivatives as hypnotics The present invention relates to alanine 2,6-dialkoxyphenyl ester derivatives having the general formula I The invention also relates to pharmaceutical compositions comprising said derivatives, and to the use of th...	11/28/2006
7101895	Cyclohexyl sulphone derivatives as gamma-secretase inhibitors Compounds of formula I: wherein Ar1 and Ar2 are optionally substituted aryl or heteroaryl, L is a bond, ═CH— or —(CHRa)n—, and X is SCN, SR1, S(O)R	09/05/2006
7078402	Aminothiol ester compounds, pharmaceutical and cosmetics compositions containing same and uses thereof The invention relates to novel aminothiol ester compounds having the general formula (I): and to a method for preparing them and to their use in pharmaceutical compositions intended for use in human or veterinary...	07/18/2006
6900243	Phenylheteroalkylamine derivatives There are provided novel compounds of formula (I), wherein R1, R2, X, Y, V, W and Z are as defined in the specification, and pharmaceutically acceptable salts thereof, and enantiomers and racemates thereof; together with processes for their pre...	05/31/2005
6900350	Method for the production of ω-aminoalkylsulphonic acids The invention relates to a method for the production of ω-aminoalkylsulphonic acids of general formula (I), where R1 and R2=optionally substituted alkyl groups with 1 20 C atoms and n=a whole number from 2 6, whereby an amine of formula (II), where R1 and R2 have t...	05/31/2005
6800659	Compounds for modulating cell proliferation Novel styrylacrylonitrile compounds which are useful in treating a variety of cell proliferative disorders such as cancer are disclosed. The compounds are of the Formula I: ...	10/05/2004
6730783	Process for preparing aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: wherein X is O or NR9 and R1-R4, R6-R9, R11, R12, Ra	05/04/2004
6723717	Sulfur-containing thyroxane derivatives and their use as hair growth promotors The present disclosure describes novel compounds of formula (A), wherein R1-R12, X and Y have the meanings given in the specification and compositions containing them which are particularly useful for treating hair loss in mammals, including ar...	04/20/2004
6673794	Substituted aminomethyl-phenyl-cyclohexane derivatives A substituted aminomethyl-phenyl-cyclohexane derivative of formula I or Ia, ##STR1## and their a diastereomer, enantiomer, or of a salt formed with a physiologically tolerated acid. Also disclosed are method for preparing the substituted aminomethyl-pheny...	01/06/2004
6670376	Aryl aniline 댢 adrenergic receptor agonists The invention provides novel 댢 adrenergic receptor agonist compounds of formula (I): ##STR1## wherein R1 -R13 and w have any of the values described in the specification. The invention also provides pharmaceutic...	12/30/2003
6656936	Carnitine analogues as topical, microbicidal spermicides Acylcarnitine analogues having alkyl side chains of 10 to 30 carbon atoms display excellent spermicidal and anti-HIV activity, a well as being potent inhibitors of the growth of Candida albicans....	12/02/2003
6638931	Aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: ##STR1## wherein X is O or NR9 and R1 -R4, R6 -R9, R11, R12, Ra, Rb, R	10/28/2003
6518310	Aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: ##STR1## wherein X is O or NR9 and R1 -R4, R6 -R9, R11, R12, Ra, Rb, R	02/11/2003
6511980	Substituted diamine derivatives useful as motilin antagonists The present invention relates to novel substituted diamine derivatives for the formula ##STR1## wherein R1, R2, R3, R4, X1, X2, X3, X4, A, Y and n are as described in ...	01/28/2003
6492514	Bifunctional photoinitiators suitable for photopolymerization and photopolymerizable systems containing the same The present invention relates to compounds of general formula (I) ##STR1## wherein X1 and X2 are different form each other and have the meanings reported in the following description Y is a simple bond, C1 -C12 linea...	12/10/2002
6479491	Disubstituted morpholine, oxazepine or thiazepine derivatives, their preparation and their use as dopamine d4 receptor antagonists The present invention relates to compounds of formula (I), any of it enantiomers, or any mixture thereof, or a pharmaceutically acceptable acid addition salt thereof, wherein R1, R2, R3, R4, R11, R	11/12/2002
6403830	Amidino compound and salts thereof useful as nitric oxide synthase inhibitors The present invention relates to S-[2-[(1-Iminoethyl)amino]ethyl]-2-methyl-L-cysteine, or a pharmaceutically acceptable salt thereof....	06/11/2002
6392039	Method for preparing (R)-(+)-3 {1-[2-(4-benzoyl-2(3, 4-difluorophenyl)morpholin-2-yl)ethyl]-4-phenylpiperidin-4-yl}-1,1-dimethy lurea, its salts solvates and/or hydrates The invention relates to a process for preparing (R)-(+)-3-{1-[2-(4-benzoyl-2-(3,4-difluorophenyl)-morpholin-2-yl)ethyl]-4- phenylpiperid-4-yl}-1,1-dimethylurea and the salts, solvates and/or hydrates thereof....	05/21/2002
6281211	Substituted semicarbazides and the use thereof This invention is related to substituted semicarbazides represented by Formula (I) or a pharmaceutically acceptable salt or prodrug thereof, wherein: R1 and R2 are independently hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl, haloalky...	08/28/2001
6274632	Derivatives of 4,4-difluorobut-3-enylsulfinic acid and their use as pesticides The invention relates to compounds of the formula (I): CF2.dbd.CX--CH.sub.2 --CH2 --S(O)--R wherein X represents hydrogen, halogen or lower alkyl, and R represents a group OR1 or NR2 R3 wherein R...	08/14/2001
6235778	Aminoguanidines and alkoxyguanidines as protease inhibitors Aminoguanidine and alkoxyguanidine compounds, including compounds of the formula: ##STR1## wherein X is O or NR9 and R1 14 R4, R6 -R9, R11, R12, Ra, Rb, R	05/22/2001
6222064	Fluorination with aminosulfur trifluorides A fluorination method of oxygen and halogen sites with diaryl-, dialkoxyalkyl-, alkylalkoxyalkyl-, arylalkoxyalkyl- and cyclic aminosulfur trifluorides fluorinating reagents is disclosed....	04/24/2001
6207860	Thermally stable aminosulfur trifluorides Diaryl-, dialkoxyalkyl-, alkylalkoxyalkyl-, arylalkoxyalkyl- and cyclic aminosulfur trifluorides fluorinating agents are disclosed....	03/27/2001
6156891	Production of pyridazine herbicides Carboxylic acids of formula (1): ##STR1## wherein R2 and R3 are independently hydrogen or C1 -C3 alkyl, and Q is optionally substituted phenyl, can be easily converted by ring closing into pyridazin-3-one d...	12/05/2000
6087379	Cyclic amine derivatives A cyclic amine derivative represented by the following formula: ##STR1## wherein R1 represents a substituted or unsubstituted phenyl group, R2 represents a substituted of unsubstituted C1 -C8 aliphatic acyl...	07/11/2000
6080886	Fluorination with aminosulfur trifluorides A fluorination method of oxygen and halogen sites with diaryl-, dialkoxyalkyl-, alkylalkoxyalkyl-, arylalkoxyalkyl- and cyclic aminosulfur trifluorides fluorinating reagents is disclosed....	06/27/2000
6075146	Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals The invention relates to intermediates and processes for producing benzothiophenes employing hydroxylamines....	06/13/2000
6013649	Thiol sulfone metalloprotease inhibitors This invention is directed to proteinase (protease) inhibitors, and more particularly to thiol sulfone inhibitors for matrix metalloproteinase 13(MMP-13), compositions of proteinase inhibitors, intermediates for the syntheses of proteinase inhibitors, pro...	01/11/2000
5990105	Benzosulfone derivatives The present invention relates to novel compounds of the general formula ##STR1## wherein R1 is hydrogen; R2 is hydrogen, trifluoromethyl or lower alkyl; R3 is hydrogen or amino; or R1 and R2 or R3	11/23/1999
5965579	Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin receptors, their preparation and pharmaceutical compositions containing them The invention relates to compounds of the formula: ##STR1## Compounds of the above formula have a great affinity for the neurotensin receptors....	10/12/1999
5935585	Biaromatic amido compounds and pharmaceutical/cosmetic compositions comprised thereof Novel pharmaceutically/cosmetically-active biaromatic amido compounds have the structural formula (I): ##STR1## in which Ar is a radical selected from among those of the following formulae (a)-(e): ##STR2## and are useful for the treatment ...	08/10/1999

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Class 544/158 - Sulfur attached directly or indirectly to morpholine ring by nonionic bonding