Class 544/13 - Sulfamyl or substituted sulfamyl containing

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which contain a sulfamyl or substituted sulfamyl
No. of patents: 37
Last issue date: 09/01/2009

Number	Title	Issue Date
7582754	Pyrro[1,2-]pyridazinone compounds The invention is directed to pyrro[1,2-b]pyridazinone compounds and pharmaceutical compositions containing such compounds that are useful in treating infections by hepatitis C virus. ...	09/01/2009
7235548	Compounds and their use as positive AMPA receptor modulators The invention provides novel compounds represented by the general formula compound represented by the formula: wherein the bond represented by the broken line may be a single, a...	06/26/2007
7230000	Methods and compositions utilizing quinazolinones Quinazolinones of formulae 1a, 1b, 1c and 1d are disclosed. They are useful for treating cellular proliferative diseases and disorders associated with KSP kinesin activity ...	06/12/2007
7160684	Methods of selecting compounds for modulation of bladder function The present invention involves an assay system and method of selecting compounds useful in the treatment of bladder instability and related bladder conditions through the activation of KCNQ potassium channels in the bladder smooth muscle. ...	01/09/2007
7091200	Quinazolone derivatives as alpha 1A/B adrenergic receptor antagonists This invention relates to compounds which are generally alpha-1A/B adrenoceptor antagonists and which are represented by Formula I: wherein Z is —C(O)— or —S(O)2—, X is...	08/15/2006
7025816	Anthraquinone dye and inkjet recording liquid An anthraquinone dye represented by the Formula (1), (2) or (3), and an ink jet recording liquid containing a compound represented by the following Formula (1), (2) or (3): ...	04/11/2006
6656932	Benzo thiadiazine matrix metalloproteinase inhibitors Selective MMP-13 inhibitors are benzo thiadiazines of the Formula ##STR1## or a pharmaceutically acceptable salt thereof, wherein R2 is hydrogen or alkyl; R1 and R3 include hydrogen, alkyl, and aryl, with the proviso that ...	12/02/2003
5536723	S-nitroso derivatives of hydrazinoacetic acids, 1-[(acylthio and (mercapto)-1-oxoalkyl]-1,2,34-Tetrahydroquinoline-2-carboxylic acids and alanyl prolines and isoquinolines The invention relates to novel S-nitroso derivatives of ACE inhibitors and to pharmaceutical compositions comprising the S-nitrosothiol derivatives of the invention together with a pharmaceutically acceptable carrier. The invention also relates to methods for ...	07/16/1996
5281720	Pyranylphenyl hydroxyalkylnaphthoic acids as inhibitors of leukotriene biosynthesis Compounds having the formula I: ##STR1## are inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating angina, cerebral spasm, ...	01/25/1994
5025001	S-nitroso derivatives of ACE inhibitors and the use thereof The invention relates to novel S-nitroso derivatives of ACE inhibitors and to pharmaceutical compositions comprising the S-nitrosothiol derivatives of the invention together with a pharmaceutically acceptable carrier. The invention also relates to methods for ...	06/18/1991
4997833	Aryloxy-aminoalkanes, and antihypertensive use thereof Aryloxy-aminoalkanes useful as antihypertensive agents are described and disclosed....	03/05/1991
4906635	Carboxyalkyl dipeptides as antiglaucoma agents Methods and pharmaceutical compositions are disclosed for reducing intraocular pressure. The methods and compositions employ an active ingredient which comprises certain benzothiadiazinyl and quinazolinyl substituted carboxyalkyl dipeptides wherein the be...	03/06/1990
4888424	ACE-diuretics Hypotensive activity is exhibited by compounds having the formulas ##STR1##...	12/19/1989
4826816	Antihypertensive compounds Antihypertensive compounds with angiotensin-converting enzyme inhibitory activity and diuretic activity are disclosed. Such compounds are useful in the treatment of cardiovascular disorders, especially hypertension and congestive heart failure, and are us...	05/02/1989
4749698	Antihypertensive derivatives Compounds having the general structure ##STR1## and their pharmaceutically acceptable salts, wherein the substituents are defined herein, which exhibit antihypertensive activity....	06/07/1988
4746676	Carboxyalkyl dipeptide compounds Compounds having the general structure ##STR1## and their pharmaceutically acceptable salts, wherein the substituents are defined herein, which exhibit antihypertensive activity....	05/24/1988
4716161	Phenylpiperazine derivatives and their acid addition salts A phenylpiperazine derivative according to the present invention has the following general formula [I]: ##STR1## wherein R1, R2 and R3 are independently hydrogen or alkoxy group having 1 to 3 carbon atoms, or R1	12/29/1987
4713238	Water soluble complex of a poly (vinyl lactam) and chlorothiazide and process for producing same The invention relates to the novel water soluble chlorothiazide in a complexed state which is derived from the reaction between and N-Vinyl actam polymer and chlorothiazide in alkaline media and to the process for the preparation of said complex....	12/15/1987
4681886	Substituted 4-phenoxy or 4-phenylthio prolines This invention is directed to substituted 4-phenoxy and 4-phenylthio prolines of the formula ##STR1## which possess useful hypotensive activity....	07/21/1987
4634689	Phosphinylalkanoyl imino acids Phosphinylalkanoyl imino acids useful in the treatment of hypertension are disclosed....	01/06/1987
4594344	1-aryloxypropanolamines Disclosed are novel compounds having the formula ##STR1## wherein R1 is a hydrogen or halogen atom, a lower alkyl, lower alkoxy, lower alkoxy lower alkyl, lower alkenyl, lower alkenyl oxy, cyano, hydroxy, trifluoromethyl, nitro, amino, ami...	06/10/1986
4576941	Compounds for treating hypertension Compounds of the formula ##STR1## and their pharmaceutically acceptable salts, wherein the substituents are as defined herein, having antihypertensive activity....	03/18/1986
4559340	Antihypertensive agents There are disclosed benzothiadiazinyl and quinazolinyl substituted carboxylalkyl dipeptides, wherein the benzothiodiazinyl or quinazolinyl portions are joined to the dipeptide portions by an aminocarbonyl group. Compounds of this invention are useful as a...	12/17/1985
4558044	1,2,4-Benzothiadiazines Disclosed are compounds of the formula wherein R1 is guanidino or substituted guanidino, Ar is furandiyl, thiophendiyl, phenylene, pyridinediyl, pyrimidinediyl, thiazolediyl, thiadiazolediyl or imidazolediyl; a is 0, 1 or 2; b is 2, 3, 4 or 5; and ...	12/10/1985
4556655	Antihypertensive compounds having both diuretic and angiotensin converting enzyme inhibitory activity Antihypertensive compounds with angiotensin-converting enzyme inhibitory activity and diuretic activity are disclosed. Such compounds are useful in the treatment of cardiovascular disorders, especially hypertension and congestive heart failure, and are us...	12/03/1985
4536501	Substituted 4-phenoxy or 4-phenylthio prolines Compounds of the formula ##STR1## are disclosed. They possess angiotensin converting enzyme inhibition activity and diuretic activity and are therefore useful as antihypertensive agents....	08/20/1985
4468396	Antihypertensive benzothiadiazines This invention relates to benzothiadiazinyl-substituted carboxyalkyl dipeptides useful as combined antihypertensive and diuretic agents....	08/28/1984
4431645	Antihypertensive agents Compounds of the formula ##STR1## and the pharmaceutically acceptable salts thereof, wherein R1, R2, R3 and R4 are independently selected from hydrogen or lower alkyl; n is 1 or 0; A and B taken together wi...	02/14/1984
4431644	Antihypertensive agents Compounds of the formula ##STR1## and the pharmaceutically acceptable salts thereof, wherein R1, R2 and R4 are independently selected from hydrogen and lower alkyl; R3 is hydrogen, lower alkyl or amino lowe...	02/14/1984
4338435	Benzothiadiazines having diuretic activity Compounds having the formula ##STR1## wherein R1 and R2 are each independently hydrogen, halogen, trifluoromethyl, aminosulfonyl, nitro, alkyl or alkoxy; R3 is hydrogen, alkyl, or phenylmethyl; R4 is hydrogen, a...	07/06/1982
4302453	Antiarrhythmic tetrahydronaphthalene derivatives Compounds are provided having the structure ##STR1## wherein R1 and R2 may be the same or different and are hydrogen, lower alkyl, lower alkenyl, or hydroxy-lower alkyl, or R1 and R2 together with the nitro...	11/24/1981
4136033	6-Hydroxypyridone-2 compounds having a cationic group in the 3-position Compounds of the formula ##STR1## wherein K.sym. is a cationic group, preferably heterocyclic, R is hydrogen or an organic radical, preferably alkyl, phenyl or acyl, R1 is hydrogen, hydrocarbyl, substituted hydrocarbyl, heterocyclyl, ...	01/23/1979
4022774	1,2,4-Benzothiadiazines Novel 1,2,4-benzothiadiazines substituted by an oxo group in the 3-position and substituted in the 4-position with hydrogen, lower alkyl, amino-lower alkyl, mono- or di-lower alkyl amino-lower alkyl, or imino-lower alkyl, are useful as central nervous sys...	05/10/1977
3988324	3-Diazine substituted benzothiadiazines 3-Diazine(or substituted diazine)-1,2,4-benzothiadiazine-1,1-dioxide products or 3,4-dihydro derivatives thereof are described. Products are prepared by conventional methods employing the appropriate sulfamoylaniline and diazine carboxylic acid halide or ...	10/26/1976
3957769	1,2,4-Benzothiadiazines Novel 1,2,4-benzothiadiazines substituted with an amino, alkylamino, or dialkylamino group in the 3-position are useful as central nervous system depressants and as diuretics....	05/18/1976
3956335	1-Substituted-4-(2-oxo-1-imidazolidinyl) piperidines Piperidines of the formula ##SPC1## In which R1 stands for optionally substituted aryl, R2 for hydrogen, lower alkyl, lower alkenyl, acyl or ଱-aryl-lower alkyl, R3 for a free or substituted hydroxyl group, alk for lo...	05/11/1976
3951966	3-Pyrazinyl substituted-1,2,4-benzothiadiazines 3-Diazine(or substituted diazine)-1,2,4-benzothiadiazine-1,1-dioxide products or 3,4-dihydro derivatives thereof are described. Products are prepared by conventional methods employing the appropriate sulfamoylaniline and diazine carboxylic acid halide or ...	04/20/1976

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Class 544/13 - Sulfamyl or substituted sulfamyl containing