Bizarre Patents
User-operated amusement apparatus for kicking the user's buttocks
An apparatus including a user-operated and controlled apparatus for self-infliction of repetitive blows to the user's buttocks by a plurality of elongated arms bearing flexible extensions that rotate under the user's control.
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| Number | Title | Issue Date |
| 7129345 | Keto-substituted steroid compounds Multiple novel keto-substituted intermediates are provided for the synthesis of epoxymexrenone, useful as an Aldosterone Receptor Antagonist. ... | 10/31/2006 |
| 7112669 | Processes for preparation of 9,11-epoxy steroids and intermediates useful therein Intermediates in the preparation of 9,11-epoxy steroids are disclosed. Particularly, disclosed are 11,12-epoxy steroid, 4,5-9,11-diepoxy steroid and 12-keto steroid intermediates. ... | 09/26/2006 |
| 7112670 | Crystal form The present invention involves a novel crystal form of 17β-hydroxy-7α-(5′-methyl-2′-furyl)-pregna-4,9(11)-dien-3-one-21-carboxylic acid, γ-lactone, having the formula which is an intermediate useful in pre... | 09/26/2006 |
| 6887991 | Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein Processes for the preparation of 4,5-dihydro-5,7-lactone steroid compounds are provided. ... | 05/03/2005 |
| 6335441 | 5ଲ-cyano-substituted steroid compounds Novel 5ଲ-cyano steroid compounds including compounds of Formula VII: ##STR1## wherein A--A, B--B, R3, R8 and R9 are as defined in the specification.... | 01/01/2002 |
| 5854235 | 17-spiromethylene steroids The invention relates to a steroid derivative which steroidal skeleton is bound at carbon atom 17 to a spiromethylene ring of the formula: ##STR1## wherein Ra and Rb are independently selected from the group consisting of hydrog... | 12/29/1998 |
| 5723455 | Antiandrogenic agents and related pharmaceutical compositions and methods of use Novel antiandrogenic agents are provided. An exemplary group of compounds has the structural formula (I) ##STR1## wherein R1 through R10, a and b are as defined herein. Pharmaceutical compositions and methods for using the compo... | 03/03/1998 |
| 5712264 | 17-spiromethylene steroids The invention relates to a steroid derivative which steroidal skeleton is bound at carbon atom 17 to a spiromethylene ring of the formula: ##STR1## wherein Ra and Rb are independently selected from the group consisting of hydrog... | 01/27/1998 |
| 5426179 | Steroid compounds active on the cardiovascular system Steroid compounds active on the cardiovascular system of formula ##STR1## wherein X, n, R, R1 and R2 have the meanings mentioned in the description are described.... | 06/20/1995 |
| 5372996 | Method of treatment of androgen-related diseases A method of treatment of androgen-related diseases such as prostate cancer in susceptible male animals, including humans, comprises administering novel antiandrogens and/or novel sex steroid biosynthesis inhibitors as part of a combination therapy. Sex st... | 12/13/1994 |
| 5244886 | 11ଲ-phenyl-14ଲH steroids New 11ଲ-phenyl-14ଲH-steroids of general formula (I), where Z is an oxygen atom or the hydroxyimino-grouping N~OH, and M and N are either jointly a second compound or L is a hydrogen atom and M is an -permanent hydroxy group and either A... | 09/14/1993 |
| 5026882 | Phosphinic acid substituted steroids as inhibitors of steroid 5-reductase The invention relates to 3-phosphinic acid steroidal compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5-reductase.... | 06/25/1991 |
| 5017568 | Steriod 5-alpha-reductase inhibitors Invented are substituted acrylate analogues of steroidal synthetic compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase. Also invented are intermediates used in prep... | 05/21/1991 |
| 4970205 | Sulfonic acid substituted aromatic steroids as inhibitors of steroid 5--reductase Invented are sulfonic acid substituted analogues of steroidal synthetic compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase, including using these compounds to redu... | 11/13/1990 |
| 4946834 | Phosphonic acid substituted steroids as steroid 5-reductase inhibitors Invented are substituted acrylate analogues of steroidal synthetic compounds, pharmaceutical compositions containing the compounds, and methods of using these compounds to inhibit steroid 5-reductase. Also invented are intermediates used in prepari... | 08/07/1990 |
| 4937237 | Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase Invented are phosphinic acid substituted analogues of steroidal synthetic compounds, pharamaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase, including using these compounds to r... | 06/26/1990 |
| 4921846 | Novel 17-hetero substituted steroids Steroids with a 17-spiro substituent of 3,4 or 6 ring members of the formula ##STR1## wherein R1 is selected from the group consisting of carbocyclic aryl, heterocyclic aryl and aralkyl, R2 is a hydrocarbon of 1 to 18 carbon ... | 05/01/1990 |
| 4921845 | 11-arylsteroid compounds The invention relates to new 11-arylsteroid compounds, having a strong antiprogestin and a weak or nonexistent antiglucocorticoid activity, to processes for preparing said compounds and also to pharmaceutical preparations which contain these derivatives a... | 05/01/1990 |
| 4904462 | Multiply-tritiated steroidal-20,17-spirolactones and their use as tracer compounds Novel, multiple-tritiated steroid-20,17-spirolactones of general Formula I ##STR1## wherein --A--B-- is --CH2 --CH2 --, --CH.dbd.CH-- or ##STR2## and --C--D-- is ##STR3## R is hydrogen or tritium and n is 0 or 1, are ... | 02/27/1990 |
| 4882319 | Phosphonic acid substituted aromatic steroids as inhibitors of steroid 5--reductase Invented are phosphonic acid substituted analogues of steroidal synthetic compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase, including using these compounds to re... | 11/21/1989 |
| 4874754 | Novel 19-nor-steroids Novel 19-nor-steroids of the formula ##STR1## wherein the A ring is either ##STR2## Re is selected from the group consisting of hydrogen, acyl and optionally substituted alkyl of 1 to 6 carbon atoms, R is methyl or ethyl, R1 is s... | 10/17/1989 |
| 4871724 | Novel 11-aryloestrane and 11-arylpregnane derivatives The present invention is concerned with 11-aryloestrane and 11-arylpregnane derivatives, characterized in that these derivatives have the following structure: ##STR1## wherein R1 is an aryl group with an ##STR2## group as substit... | 10/03/1989 |
| 4870069 | 11ଲ-alkynyl-estrenes and -estradienes, their production and pharmaceutical preparations containing them 11ଲ-substituted steroids of the formula ##STR1## wherein A and B together represent a second bond between the 6-position and 7-position carbon atoms, or, respectively, are each H; X is O, two H atoms or hydroximino; Z is the residue of a pentagonal ... | 09/26/1989 |
| 4670551 | Epoxy steroids 7-acylthio-9,11-epoxy-20-spirox-4-ene-3,21-diones of the formula I ##STR1## in which R represents lower alkanoyl and --A--A-- represents an ethylene or cyclopropylene group, have a high aldosterone-antagonistic activity with... | 06/02/1987 |
| 4559332 | 20-Spiroxanes and analogues having an open ring E, processes for their manufacture, and pharmaceutical preparations thereof Steroid compounds of the 20-spiroxane series and their analogues having an open ring E of the formula, ##STR1## in which --A--A-- represents the group --CH2 --CH2 -- or --CH.dbd.CH--, R1 represents hydrogen, and R | 12/17/1985 |
| 4552871 | Steroids of the 20-spiroxane series, processes for the manufacture thereof, pharmaceutical preparations containing such compounds and the use of the latter (5)-20-spirox-1-en-3-ones (I) and 17-hydroxy-5,17-pregn-1-en-3-ones (II) of the formulae ##STR1## in which X represents O or H2, R2 represents O and R1 represents OH, OMe, OAlk, NH2, NH... | 11/12/1985 |
| 4340538 | Process for producing 6-fluoro-Ɗ1,4 -3-keto steroids Two processes are disclosed (one-pot and two-pot) for the transformation of a 6ଲ-fluoro-Ɗ1,4 -3-keto steroid (IV) to a 6-fluoro-Ɗ1,4 -3-keto steroid (VI). These processes permit the introduction of a fluorine atom at t... | 07/20/1982 |
| 4305881 | Process for 1,3ଲ-dihydroxy-Ɗ5 -steroids A process for the synthesis of 1,3ଲ-dihydroxy-Ɗ5 -steroids from steroids such as 1,2-epoxy-cholesta-4,6-dien-3-one, which is reacted with lithium in liquid ammonia in the absence of a proton donator and subseque... | 12/15/1981 |
| 4297350 | Male contraceptive steroids and methods of use The steroids of the present invention have been found to be useful as male contraceptives when administered orally. Upon cessation of administration of the male contraceptive steroids of the present invention the male promptly regains normal fertility.... | 10/27/1981 |
| 4242334 | Corticoid 17-(alkyl carbonates) and processes for their preparation What is disclosed is corticoid 17-(alkyl carbonates) of the formula ##STR1## as defined in the specification, which compounds can be used in veterinary therapy and human therapy, in the form of suspensions, ointments, creams, sprays and the like, for... | 12/30/1980 |
| 4160027 | Steroid cyanoketones and intermediates 2-Cyano-3-oxosteroids having a 4,5-epoxy group and alkylated in the 4- and/or 6-position, useful as interceptive agents, are prepared by alkaline cleavage of the corresponding steroido[2,3-d]isoxazoles.... | 07/03/1979 |
| 4119627 | Process for the manufacture of 6ଲ,7-methylene-3-oxo-4-ene steroids The invention provides a novel general process for the manufacture of 6ଲ,7-methylene-3-oxo-4-ene-steroids by successively (a) reacting a 3.xi.,5ଲ-dihydroxy-6-ene-steroid which is optionally etherified or esterified in the 3-position with a zin... | 10/10/1978 |
| 4104271 | 11ଲ,18-EPOX Y-9-HALO-17,18-DIHYDROXY-3-OXO-17-PREGN-4-ENE-21-CARBOXYLIC ACID γ-LACTONES AND CONGENERS Preparation and the diuretic utility of 11ଲ,18-epoxy-9-halo-17,18-dihydroxy-3-oxo-17-pregn-4-en e-21-carboxylic acid γ-lactones and congeners are disclosed.... | 08/01/1978 |
| 4069322 | Pro-drugs for the improved delivery of certain selected anti-inflammatory steroids Transient, pro-drug forms of conventional anti-inflammatory steroids are disclosed.... | 01/17/1978 |
| 4069219 | 7 .xi.-(Alkoxycarbonyl)-6.xi.-alkyl/halo-17-hydroxy-3-oxo-17-pregn-4 -ene-21-carboxylic acid γ-lactones and corresponding 21-carboxylic acids, their salts, and esters Various preparations and the diuretic activity of 7.xi.-(alkoxycarbonyl)-6.xi.-alkyl/halo-17-hydroxy-3-oxo-17-pregn-4 -ene-21-carboxylic acid γ-lactones and corresponding 21-carboxylic acids, their salts, and esters are disclosed.... | 01/17/1978 |
| 4031074 | Process for the preparation of 11ଲ-hydroxy-18-alkyl-estrane compounds The present invention relates to a novel process for the preparation of 11ଲ-hydroxy-18-alkyl-estrane compounds by reacting an 11ଲ-hydroxy-13-methyl-gonane compound with an excess of an acylhypoiodite to give an estrano-18,11ଲ-lactone, re... | 06/21/1977 |
