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| Number | Title | Issue Date |
| 7534871 | Preparation and use of carbohydrate-based bicyclic ring structures with antimicrobial and cytostatic activity Novel carbohydrate-based compounds with an attached ring system that have antimicrobial or cytostatic activity. The compounds are administered to humans and animals for the treatment or amelioration of bacterial, fungal, viral or protozoal infections or tumors. The ... | 05/19/2009 |
| 7375213 | Methods of producing C-aryl glucoside SGLT2 inhibitors Method for the production of C-aryl glucoside SGLT2 inhibitors useful for the treatment of diabetes and related diseases. and intermediates thereof. The C-aryl glucosides may be complexed with amino acid complex forming reagents. ... | 05/20/2008 |
| 7365055 | Derivatives of morphine-6-glucuronide, pharmaceutical compositions containing them, their preparation method and their uses The invention relates to novel derivatives of morphine-6-glucuronide, the preparation method thereof and the uses of same in therapy, for example, as analgesics. ... | 04/29/2008 |
| 7244712 | Aminoglycoside antibiotics and methods of using same The present invention relates to aminoglycoside compounds having antibiotic activity. Moreover, the present invention relates to L-aminoglycoside compounds and diastereomers thereof which posses antibiotic activity and are not susceptible to development of resistant... | 07/17/2007 |
| 7220727 | Aminoglycosides as antibiotics The present invention provides aminoglycosides and pharmaceutical compositions that include the aminoglycosides. The aminogylcosides are useful to treat or prevent infectious diseases (e.g., bacterial infections) in a mammal (e.g., human). ... | 05/22/2007 |
| 7129219 | Immunoeffector compounds This invention provides compounds containing a 2-deoxy-2-amino-β-D-glucopyranose (glucosamine) glycosidically linked to a cyclic aminoalkyl (aglycon) group. The invention further provides methods for inducing an immune response using the compounds of the present in... | 10/31/2006 |
| 7060685 | Compounds and methods for inhibiting selectin-mediated function Compounds and methods are provided for modulating in vitro and in vivo processes mediated by selectin binding. More specifically, selectin modulators and their use are described, wherein the selectin modulators that modulate (e.g., inhibit or enhance) a selectin-med... | 06/13/2006 |
| 7019131 | Programmable one-pot oligosaccharide synthesis The reactivity of a number of p-methylphenyl thioglycoside (STol) donors which are either fully protected or have one hydroxyl group exposed has been quantitatively determined by HPLC in conjunction with the development of a broadly applicable approach for a facile ... | 03/28/2006 |
| 6960654 | Method of forming glycosidic bonds from thioglycosides using an N,N-dialkylsulfinamide A method of forming a glycosidic bond utilizing an activated thioglycoside is disclosed. The thioglycoside is activated by an N,N-dialkylsulfinamide and trifluoromethanesulfonic anhydride. The method allows the facile synthesis of disaccharides, oligosacchraides, an... | 11/01/2005 |
| 6911434 | Prophylactic and therapeutic treatment of infectious and other diseases with immunoeffector compounds Methods and compositions for treating or ameliorating diseases and other conditions, such as infectious diseases, autoimmune diseases and allergies are provided. The methods employ cyclic AGPs for selectively stimulating immune responses in animals and plants. ... | 06/28/2005 |
| 6887854 | Compounds as dynamic organ function monitoring agents Highly hydrophilic indole and benzoindole derivatives that absorb and fluoresce in the visible region of light are disclosed. These compounds are useful for physiological and organ function monitoring. Particularly, the molecules of the invention are useful for opti... | 05/03/2005 |
| 6875755 | Antithrombotic compound The present invention relates to compounds of the formula (I), wherein R is independently SO3− or CH3; the spacer is a flexible spacer of a length of 13-25 atoms; the charge of the pentasaccharide residue is compensated by positive... | 04/05/2005 |
| 6867194 | Enzyme activated nitric oxide donors Sugar-modified SIN-1 compositions are provided. The compositions are useful for generating NO in response to hydrolytic activity of a glycosidase specific for the O-glycosidic bond between the sugar and SIN-1 moieties. Pharmaceutical compositions containing the suga... | 03/15/2005 |
| 6841536 | Prodrugs and conjugates of thiol- and selenol-containing compounds and methods of use thereof Disclosed is a prodrug of the formula: where A is a sulfur or a selenium, and R is derived from a mono- di- or oligo- saccharide. Also disclosed is a prodrug of the formula: | 01/11/2005 |
| 6828309 | Use of pentosan polysulfate to treat certain conditions of the prostate The invention relates to the field of pharmacology. More particularly, the invention relates to the treatment of prostate conditions, such as BPH. The invention provides new therapeutic compositions and methods for treating BPH, as well as chronic prostatitis, prost... | 12/07/2004 |
| 6750207 | Compositions for the regulation of cytokine activity A pharmaceutical composition for the regulation of cytokine activity in a subject. The composition features an effective amount of an oligosaccharide to inhibit the cytokine activity, preferably through inhibition of TNF-alpha activity. The oligosaccharide is more p... | 06/15/2004 |
| 6734292 | Pseudoerythromycin derivatives The present invention is to obtain novel anti-inflammatory agents having decreased antibacterial activity and increased anti-inflammatory action, and is psedoerythromycin derivatives represented by the following general formula [I], | 05/11/2004 |
| 6683056 | O-aryl glucoside SGLT2 inhibitors and method ##STR1## wherein when Y is ##STR2## or heteroaryl; A is --O(CH2)m, S, --NH(CH2)m, or (CH2)n where n is 0-3 and m is 0-2; and R1 to R6 are as defined herein... | 01/27/2004 |
| 6673907 | Methods and compositions for the manufacture of C-3' and C-4' anthracycline antibiotics The present invention discloses new and novel substituted anthracyclines with modified alkyl-aromatic ring substitutions on the C-3' of the sugar moiety or modified or unmodified alkyl-aromatic ring substitutions at the C-4' of the sugar moiety. It also d... | 01/06/2004 |
| 6656922 | Oral delivery of macromolecules Polysaccharides, which are widely used as an anticoagulation drugs, especially heparin, are clinically administered only by intravenous or subcutaneous injection because of their strong hydrophilicity and high negative charge. Amphiphilic heparin derivati... | 12/02/2003 |
| 6635622 | Glycolipid derivative The present invention is a compound of general formula (I) or a pharmaceutically acceptable salt of, ##STR1## wherein W represents carbon chain from 9 to 17 which containing double bond or hydroxy group occasionally; X represents carbon chain from 11 to 2... | 10/21/2003 |
| 6593311 | Apoptosis inducers Apoptosis inducers, anticancer drugs and carcinostatic drugs containing sulfated-fucose-containing polysaccharide(s) and/or degradation product(s) thereof, and a method for inducing apoptosis by using sulfated-fucose-containing polysaccharide(s) and/or de... | 07/15/2003 |
| 6589943 | Formulation of amphiphilic heparin derivatives for enhancing mucosal absorption Formulations for enhanced mucosal absorption of heparin are disclosed. In one embodiment, a powdered heparin composition is made by dissolving an amphiphilic heparin derivative including heparin covalently bonded to a hydrophobic agent in a water phase, d... | 07/08/2003 |
| 6534637 | Synthesis of chlorophenol red glucuronic acid This invention provides ଲ-D-Glucuronidase substrates of the formula: ##STR1## wherein R1, R2, and R7 -R12 are independently selected from the group consisting of: hydrogen, fluorine, chlorine, bromine, iodine, ... | 03/18/2003 |
| 6525028 | Immunoeffector compounds This invention provides compounds containing a 2-deoxy-2-amino-ଲ-D-glucopyranose (glucosamine) glycosidically linked to an cyclic aminoalkyl (aglycon) group. The invention further provides methods for inducing an immune response using the compounds ... | 02/25/2003 |
| 6515117 | C-aryl glucoside SGLT2 inhibitors and method An SGLT2 inhibiting compound is provided having the formula ##STR1## A method is also provided for treating diabetes and related diseases employing an SGLT2 inhibiting amount of the above compound alone or in combination with another antidiabetic agent or... | 02/04/2003 |
| 6465625 | Taxol derivatives Highly specific biocatalytic reactions have been used to create a population of taxol derivatives.... | 10/15/2002 |
| 6414126 | C-aryl glucoside SGLT2 inhibitors and method SGLT2 inhibiting compounds are provided having the formula ##STR1## where R1, R2, and R2a are independently hydrogen, OH, OR5, lower alkyl, CF3, OCHF2, OCF3, SR5i or haloge... | 07/02/2002 |
| 6340746 | Prodrugs and conjugates of thiol- and selenol- containing compounds and methods of use thereof Disclosed are prodrugs as follows: (I) a prodrug of the formula ##STR1## where A is a sulfur or a selenium, and R is a mono- di- or oligo-saccharide; (II) a prodrug of the formula ##STR2## where A is sulfur or selenium, R' is a sugar, or .dbd.O, and the R... | 01/22/2002 |
| 6306837 | Heavy metal chelating agent for oral administration, its synthesis and its uses in medicine and health protection The present invention relates to a new kind of heavy metal chelating agents and a preparation process and uses thereof. The said heavy metal chelating agents are expressed in -[D(+)glucose-1-yl-amino]-댣-mercapto-(S)-propanoic acid (abbr... | 10/23/2001 |
| 6297363 | Glycoside indoles The present invention relates to a novel class of glycoside indoles. More specifically, the present invention relates to a novel class of glycoside indoles isolated from Calanthe discolor Lindl. and derivatives thereof.... | 10/02/2001 |
| 6274716 | Combinatorial library of moenomycin analogs and methods of producing same A combinatorial chemical library of compounds structurally related to the moenomycin class of antibiotics has the formula ##STR1## wherein D is a donor mono- or disaccharide, A is an acceptor monosaccharide, and P-R is a lipophosphoglycerate mimetic group... | 08/14/2001 |
| 6258784 | Acetal benzylmaltosides as inhibitors of smooth muscle cell proliferation This invention provides smooth muscle cell proliferation inhibitors of formula I having the structure ##STR1## wherein W is S, SO, SO2, NR; Y is O, S, NR, or CH2 ; R is hydrogen or alkyl of 1-6 carbon atoms, perfluoroalkyl of 1-6 carbon ... | 07/10/2001 |
| 6245753 | Amphiphilic polysaccharide derivatives Polysaccharides, which are widely used as an anticoagulation drugs, especially heparin, are clinically administered only by intravenous or subcutaneous injection because of their strong hydrophilicity and high negative charge. Amphiphilic heparin derivati... | 06/12/2001 |
| 6184366 | Substituted liposaccharides useful in the treatment and prevention of endotoxemia Novel substituted liposaccharides useful as in the prophylactic and affirmative treatment of endotoxemia including sepsis, septicemia and various forms of septic shock and methods of using these agents are provided. Also provided are methods of preparing ... | 02/06/2001 |
| 6183994 | N-containing saccharides and method for the synthesis of N-containing saccharides from amino-deoxy-disaccharides and amino-deoxy-oligosaccharides Synthesis of an amino-disaccharide, amino-oligosaccharide or a derivative thereof, characterized in that a monosaccharide, a disaccharide, an oligosaccharide, a glycoside or a derivative thereof, in the presence of a glycosidase as catalyst, is reacted wi... | 02/06/2001 |
| 6136961 | Biocatalytic methods for synthesizing and identifying biologically active compounds Highly specific biocatalytic reactions have been used to create a population of derivatives from a single starting compound. Examples demonstrate synthesis of derivatives of taxol, taxol-2'-adipate, taxol-2'-vinyl adipate, 2,3-(methylenedioxy) benzaldehyd... | 10/24/2000 |
| 6136790 | Carbohydrate mimetics having antiadhesive properties The invention relates to carbohydrate mimetics, which inhibit the binding of selectin to carbohydrate ligands, of the formula I ##STR1## excluding the compounds sialyl-Lewis-X and -A and their derivatives which, instead of an N-acetyl group, carry th... | 10/24/2000 |
| 6107284 | Water-soluble derivatives of epipodophyllotoxin, process for their preparation, their use as medicinal products and their intended use in anti-cancer treatments Water-soluble derivatives of epipodophyllotoxin, process for their preparation and their use for the treatment of rheumatoid arthritis, complaints caused by human papilloma virus and cancer.... | 08/22/2000 |
| 6087339 | Saccharide derivatives Disclosed are novel saccharide derivatives which inhibit binding of toxins, such as heat-labile enterotoxin or cholera toxin, to their receptors either in vitro or in vivo. Additionally, disclosed are compounds which inhibit binding of enterovirulent orga... | 07/11/2000 |
