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| Number | Title | Issue Date |
| 4495104 | Quinone carboxylic acids and ester derivatives A compound of the general formula ##STR1## wherein n is an integer of 10 to 21, inclusive; R is H or lower alkyl having 1 to 4 carbon atoms has pharmaceutical activities such as hypotensive, tissue metabolism stimulating, immuno-regulatory, lysosomal... | 01/22/1985 |
| 4492704 | Quinoline quinones and anti-asthmatic use thereof This invention relates to a class of quinoline quinones, which are useful for the therapy of immediate hypersensitivity reactions, such as asthma, and in treating any condition characterized by excessive release of leukotrienes. This invention also includ... | 01/08/1985 |
| 4490373 | Method of treating asthma A new method of treating asthma is provided. The method is the administration of an effective dose of a Benzoxazole-2-carboxylic acid amide.... | 12/25/1984 |
| 4478834 | Dihydropyridines and their use in the treatment of asthma New dihydropyridines are described. These compounds are useful in the treatment of asthma.... | 10/23/1984 |
| 4478820 | Anilino-substituted isoquinoline quinones, pharmaceutical compositions and method of use thereof This invention relates to a class of isoquinoline quinones, which are useful for the therapy of immediate hypersensitivity reactions, such as asthma, and in treating any condition characterized by excessive release of leukotrienes. This invention also inc... | 10/23/1984 |
| 4477671 | 3-Acetoxy or benzyloxy-2-acetoxymethyl-6-[1-acetoxy-2-(N-tert-butylacetamido)ethyl]py ridine intermediates Processes and intermediates useful in the preparation of bronchodilator compounds of the formula ##STR1## wherein R is hydrogen, methyl or hydroxymethyl are described. Those compounds wherein R is H or CH3 have been found to have further ... | 10/16/1984 |
| 4474803 | 7-Oxabicycloheptane substituted thio prostaglandin analogs useful in treating platelet aggregation and bronchoconstriction 7-Oxabicycloheptane substituted thio prostaglandin analogs are provided having the structural formula ##STR1## wherein R is hydrogen, lower alkyl or alkali metal, R1 is lower alkyl, arylalkyl, aryl, cycloalkyl or cycloalkylalkyl. A is --CH... | 10/02/1984 |
| 4474752 | Drug delivery system utilizing thermosetting gels Present invention provides a unique drug delivery device for delivering drug by injection into a body. The drug delivery system comprises the drug and polymer which is a liquid at room temperature and a semi-solid or gel at the body temperature.... | 10/02/1984 |
| 4472586 | 6H-Dibenz[b,e][1,4]oxathiepin derivatives Novel 6H-dibenz[b,e][1,4]oxathiepin derivatives of the formulae I and IA are employed in the treatment and control of allergic conditions such as allergic asthma. ##STR1##... | 09/18/1984 |
| 4465851 | Guanidinocyclohexanecarboxylic acid derivatives A compound having the formula ##STR1## wherein R1 represents an indanyl, indolyl, quinolyl or chromonyl group, the group of the formula ##STR2## (in which R2 represents a halogen atom or a nitro group), or the group of... | 08/14/1984 |
| 4463015 | Aryl substituted 7-oxabicycloheptane compounds, useful in inhibiting platelet aggregation 7-Oxabicycloheptane and prostaglandin analogs are provided having the structural formula ##STR1## and including all stereoisomers thereof. The compounds are cardiovascular agents useful, for example, in the treatment of thrombolytic disease.... | 07/31/1984 |
| 4461769 | Nitrogen bridgehead compounds having anti-allergic effect Compounds of the formula I ##STR1## or pharmaceutically acceptable salts, hydrates, stereoisomers, optically active isomers, geometrical isomers or tautomeric forms thereof are disclosed wherein R is hydrogen or lower alkyl R1 is hydrogen,... | 07/24/1984 |
| 4451479 | Therapeutically active 3-amino-1-halogenated phenyl-2-pyrazolines and their C4 and C5 analogs A method of meliorating the inflammation and/or the progressive joint deterioration characteristic of arthritic disease, preventing the onset of asthmatic symptoms and allergic diseases, treating pain or treating bacterial and fungal infections in mammals... | 05/29/1984 |
| 4447603 | Substituted-6-n-propyl-8-methylimidazo[1,5-d]-as-triazin-4-(3H)-ones This disclosure describes new compounds and compositions of matter useful as anti-asthmatic agents and the method of meliorating asthma in mammals therewith, the novel active ingredients of said compositions of matter being certain 1-substituted-6-n-propy... | 05/08/1984 |
| 4443460 | 2-[4-(Diphenylmethylene)-1-piperidinyl]-acetic acids and their amides New 2-[4-(diphenylmethylene)-1-piperidinyl]-acetic acids and their amides, processes for the preparation thereof and therapeutic compositions. These compounds have the formula ##STR1## wherein Y=--OH or --NR1 R2, R1 a... | 04/17/1984 |
| 4443479 | Pharmaceutical methods and compositions using parabenzoquinone Bronchial asthma including bronchial spasms associated therewith are treated with pharmaceutical compositions containing small amounts of parabenzoquinone, for instance 2 milliliters of a one part per million solution of PBQ in sterile isotonic saline sol... | 04/17/1984 |
| 4443478 | Prostaglandin analogues Prostaglandin E1 analogues of general formula: ##STR1## [wherein R1 represents a bond or a straight- or branched-chain alkylene group containing from 1 to 5 carbon atom(s), and R2 represents a hydrogen atom, a straigh... | 04/17/1984 |
| 4442094 | (3-Aralkylamino-2-or-propoxy)heterocyclic compounds Compounds of the formula Het--O--CH2 --CHOR--CH2 --NH-aralkyl where Het is a 10 membered N-containing ring are disclosed. The compounds are useful as pharmaceuticals.... | 04/10/1984 |
| 4442099 | Leukotriene analogues A compound of the formula ##STR1## wherein n is an integer from 2 to 4; m is an integer from 3 to 5; R is OM, OR1 or NR2 R3 where M is a pharmaceutically acceptable cation; R1, R2 and R3 | 04/10/1984 |
| 4442115 | 2'Hydroxy tetrazole-5-carboxanilides and anti-allergic use thereof New tetrazole derivatives of the general formula: ##STR1## [wherein R1 represents a halogen atom, a straight- or branched-chain alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl or alkylsulphamoyl group, each such group containing f... | 04/10/1984 |
| 4440776 | Antiinflammatory 4,5-diphenyl-2-substituted-thio-imidazoles and their corresponding sulfoxides and sulfones Imidazole derivatives of the formula ##STR1## wherein Ar1 and Ar2 are each phenyl; phenyl substituted by halogen, C1-4 alkyl, C1-4 alkoxy or C2-6 dialkylamino; pyridyl; furyl; or thienyl; with th... | 04/03/1984 |
| 4439448 | Glutamine derivatives Glutamine derivatives and non-toxic salts thereof have been found to have immunomodulating activities.... | 03/27/1984 |
| 4438112 | Prostanoid compounds and pharmaceutical formulations Prostanoids are described of the formulae ##STR1## (and the salts thereof) in which: X is cis or trans --CH.dbd.CH-- or CH2 CH2 --; R1 is C1-7 alkyl terminated by --COOR10 where R10 is H, ... | 03/20/1984 |
| 4438136 | Prostaglandins Novel bicyclo [2,2,1] heptanes and hept-2-enes are substituted at the 5-position by a 6-carboxyhex-2-enyl group or a modification thereof, and at the 6-position by a grouping --C(R).dbd.N--NHCO--(NH)a --R' in which R is hydrogen, an aliphatic h... | 03/20/1984 |
| 4438111 | Prostanoid compounds and pharmaceutical formulations Prostanoids are described of the formulae ##STR1## (and the salts thereof) in which: X is cis or trans--CH.dbd.CH-- or CH2 CH2 --; R1 is C1-7 alkyl terminated by --COOR10 where R10 is H, ... | 03/20/1984 |
| 4436746 | Thromboxane synthetase inhibitory N-substituted-2-(1-imidazolyl)indoles Various 1-carboxylic acid substituted-2-(1-imidazolyl)indoles and functional derivatives thereof are highly specific thromboxane synthetase inhibitors. Synthesis of, pharmaceutical compositions thereof, and methods of treatment utilizing such compounds ar... | 03/13/1984 |
| 4435390 | Hydrocortisone derivatives, the preparation and use thereof Hydrocortisone derivatives of Formula I ##STR1## wherein is a single bond or a double bond, n is 1 or 2, R1 is hydrogen or methyl, R2 is alkyl of 1-6 carbon atoms, and R3 is hydrogen or 1-oxoalkyl (alkanoyl) of 2-6 carbon atom... | 03/06/1984 |
| 4435420 | Anti-inflammatory agents and antiasthmatic agents N-(1,3-dithiolan-2-ylidene)-4-alkylanilines are useful as anti-inflammatory agents, as analgesic agents and as antiasthmatic agents. The compounds involved can be prepared by the reaction of an appropriate 4-alkylaniline with a methyl(1,3-dithiolan-2-ylid... | 03/06/1984 |
| 4435404 | Carbostyril derivatives Novel carbostyril derivative and its salt represented by the general formula (1), ##STR1## wherein R1 is a hydrogen atom, a lower alkyl group, a lower alkenyl group or a phenyl-lower alkyl group; R2 is a hydrogen atom, a lower ... | 03/06/1984 |
| 4432986 | Tetrazoles bonded to certain polycyclic aromatic systems and anti-allergic use thereof Amides obtained by reaction of aminotetrazole and certain optionally substituted polycyclic aromatic acids are potent anti-allergic agents.... | 02/21/1984 |
| 4432976 | Cyclocarbonate esters of 16,17, dihydroxy anti-inflammatory steroids Corticoids of Formula I ##STR1## wherein is a single bond or a double bond, X is hydrogen, fluorine, or chlorine, Y represents two hydrogen atoms or an oxygen atom, and Z is hydrogen or acyloxy of 2-6 carbon atoms, are pharmacologically active compounds... | 02/21/1984 |
| 4432991 | Therapeutically active 3-amino-1-phenyl(and substituted phenyl)-2-pyrazolines This disclosure describes certain 3-amino-1-phenyl-2-pyrazolines and 3-amino-1-substituted phenyl-2-pyrazolines and their C4 and C5 analogs useful for meliorating the inflammation and/or the progressive joint deterioration characteristic of arthritic dise... | 02/21/1984 |
| 4430345 | Prostaglandins Novel bicyclo [2,2,1] heptanes and hept-2Z-enes are substituted at the 5-position by a 6-carboxyhex-2-enyl group or a modification thereof, and at the 6-position by an aldoxime or ketoxime group which is O-substituted by an aliphatic hydrocarbon residue, ... | 02/07/1984 |
| 4427671 | Steroids esterified in position 17 and thioesterified in position 21, a process for preparing them and their use as medicaments Compounds of formula: ##STR1## wherein A and B each represent, independently of each other, a straight-chained or branched alkyl group having from 1 to 6 carbon atoms or a phenyl group optionally mono- or polysubstituted by alkyl radicals having... | 01/24/1984 |
| 4427682 | Pyridine alkyl benzoic and thenoic acid compounds and their pharmaceutical compositions The pyridine derivatives of the general formula: ##STR1## [wherein A represents an alkylene group containing from 1 to 5 carbon atoms unsubstituted or substituted by a hydroxy group, B represents a single bond, or an oxygen or sulphur atom, or an alk... | 01/24/1984 |
| 4427680 | 1,2-Dihydroquinolines connected via an oxyalkyl group with a piperidine ring and having anti-allergic action The present invention provides aryl ether derivatives of the general formula: ##STR1## wherein A is an oxygen atom or the group >N--R1, R1 being a hydrogen atom or a lower alkyl radical, R2 and R3, which ca... | 01/24/1984 |
| 4427686 | Pharmacologically active benzopyranotriazole compounds A compound of the formula (I): ##STR1## wherein R1 is hydrogen or C1-6 alkyl; R2, R3 and R4 are the same or different and are chosen from hydrogen, hydroxyl, halogen, C1-4 alkyl, C1-4 | 01/24/1984 |
| 4426383 | Theophylline and theobromine derivatives A novel compound has the following formula: ##STR1## in which R1 and R2 are methyl or a group having the formula: ##STR2## provided that one of R1 and R2 is methyl and the other is said group, wherein ... | 01/17/1984 |
| 4425349 | Sulfur-containing isoquinoline derivatives in pharmaceutical compositions and methods of use The invention concerns new sulfur-containing isoquinoline derivatives. More particularly, the invention relates to isoquinoline derivatives of the general formula (I) ##STR1## wherein R independently represents hydrogen, hydroxyl or alkoxy having 1 ... | 01/10/1984 |
| 4424231 | Compounds There are described compounds of formula I, ##STR1## in which Ra, Rb, Rc, Rd, Re, Rf and Rg, which may be the same or different, each represent hydrogen, amino, hydroxy, alkoxy, alkenyloxy, halogen, acyl, alkenyl, alkyl, or alkoxy substituted by phen... | 01/03/1984 |
