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| Number | Title | Issue Date |
| 5716993 | Anthranilic acid derivatives The present invention provides an anthranilic acid derivative having a cGMP-PDE inhibitory activity. An anthranilic acid derivative represented by the general formula (I) or a pharmacologically acceptable salt thereof: ##STR1## ›wherein R1 | 02/10/1998 |
| 5709867 | Polyaromatic amide compounds and pharmaceutical/cosmetic compositions comprised thereof Novel pharmaceutically/cosmetically-active polyaromatic amides have the structural formula (I): ##STR1## wherein Z is a radical --CO--NH-- or --NH--CO--, and are useful for the treatment of a wide variety of disease states, whether human or vete... | 01/20/1998 |
| 5705528 | Farnesyl derivatives and pharmaceutical compositions containing them Novel farnesyl derivatives which are inhibitors of the prenylated protein thyltransferase enzyme, and useful as anti-cancer drugs, have the following formula: ##STR1## wherein R1 represents farnesyl, geranyl or geranyl-geranyl; Z represent... | 01/06/1998 |
| 5696128 | Method of regulating immune function Disclosed are methods for rectifying or ameliorating abnormal responses of mammalian immune systems. Also disclosed are methods for modifying normal responses of the mammalian immune system. Further disclosed are methods for accomplishing the foregoing by... | 12/09/1997 |
| 5684049 | HIV-inhibiting benzeneacetamide derivatives A compound for use as a medicine having the formula ##STR1## a pharmaceutically acceptable acid addition salt form or a stereochemically isomeric form thereof, wherein R1 and R2 each independently are hydrogen, C1-6 a... | 11/04/1997 |
| 5677347 | Ortho-substituted phenylacetamides Ortho-substituted phenylacetamides I ##STR1## (R1 =H, alkyl, cycloalkyl, alkenyl, alkynyl, phenylalkynyl, alkoxyalkyl, alkoxycarbonyl, phenyl, phenylalkyl, phenylalkenyl or phenoxyalkyl, 5- or 6-membered heterocycle with 1-3 hetero atoms t... | 10/14/1997 |
| 5668178 | Arylthio compounds Phenylthiols and dithiobisbenzamides are potent antibacterial and antiviral agents.... | 09/16/1997 |
| 5658944 | Anti-atherosclerotic aryl compounds The present invention is concerned with compounds of formula (I) ##STR1## wherein Ar is a mono- or bicyclic aromatic group optionally containing one or two heteroatoms independently selected from nitrogen, oxygen and sulphur, said group being optiona... | 08/19/1997 |
| 5658953 | Pharmaceutical compositions of acetamidobenzamide compounds for neurodegenerative disorders A group of benzamide compounds are disclosed which are useful for treating neurodegenerative disorders. Methods for making these compounds are provided. These materials are formed into pharmaceutical compositions for oral or intravenous administration to ... | 08/19/1997 |
| 5654313 | Method for modifying or regulating the glucose metabolism of an animal or human subject A process for the long term modification and regulation of lipid and glucose metabolism--generally to reduce obesity, insulin resistance, and hyperinsulinemia or hyperglycemia, or both (these being the hallmarks of noninsulin dependent, or Type II diabete... | 08/05/1997 |
| 5652260 | Adenosine diphosphoribose polymerase binding nitroso aromatic compound useful as retroviral inactivating agents, anti-retroviral agents and anti-tumor agents The subject invention provides for novel compounds for inactivating viruses. These compounds include 6-nitroso-1,2-benzopyrone, 3-nitrosobenzamide, 5-nitroso-1(2H)-isoquinolinone, 7-nitroso-1(2H)-isoquinolinone, 8-nitroso-1(2H)-isoquinolinone. The in... | 07/29/1997 |
| 5643965 | Aminobenzamide compounds for the treatment of neurodegenerative disorders A group of benzamide compounds are disclosed which are useful for treating neurodegenerative disorders. Methods for making these compounds are provided. These materials are formed into pharmaceutical compositions for oral or intravenous administration to ... | 07/01/1997 |
| 5637613 | 15-deoxyspergualin analogs, their method of preparation and their use in therapeutics The present invention relates, by way of novel industrial products, to compounds which are structurally related to 15-deoxyspergualin and which have the formula ##STR1## in which: A is a single bond, a group --CH2 --, a group --CH2 | 06/10/1997 |
| 5633282 | Inhibition of viral infection The use of a poly(ADP-ribose) polymerase inhibitor for the treatment of a subject against infection by a virus, in which the viral or proviral DNA integrates into the chromosome or chromosomes during its replication cycle.... | 05/27/1997 |
| 5633288 | Tri (lower alkoxy) benzene derivatives This invention relates to a tri(lower alkoxy)benzene derivative of the general formula (I), or its salt, optical isomer or solvate, ##STR1## wherein: R1, R2 and R3 : same or different and each represents a lower alkyl... | 05/27/1997 |
| 5629347 | Aromatic compounds, pharmaceutical compositions containing them and their use in therapy Compounds of formula (I), and salts and prodrugs thereof, wherein Q is R9 CR10 R11 or CH2 R9 CR10 R11 where R9 is H or OH and R10 and R11 are optional... | 05/13/1997 |
| 5622916 | Substituted 2-cylcohexen-1-yl-amine fungicidal and herbicidal agents A method of combating pests which comprises applying to such pests or to a pest habitat a pesticidally effective amount of a substituted 2-cyclohexen-1-yl-amine derivative of the formula ##STR1## and addition products thereof with acids and metal sal... | 04/22/1997 |
| 5602181 | Naphthyl ethers, their preparation, compositions containing them and their use Naphthyl ethers of the general formula I ##STR1## where the index and the substituents have the meanings defined in the specification.... | 02/11/1997 |
| 5602164 | Anti-obesity drugs Obesity is treated by the administration to a subject of a compound having the general formula (I): R4 --(CH2)n --CO--N(R1)--CH(R2)--CO(--R3), wherein R1 represents H or CH3... | 02/11/1997 |
| 5601811 | Substantive water-soluble cationic UV-absorbing compounds Substantive UV-absorbing cinnamido amine cationic quaternary salts are disclosed. Detergent and household cleaning product compositions and hair and skin personal care product compositions, as well as sunscreen and tanning lotion compositions, containing ... | 02/11/1997 |
| 5591747 | Fungicidal mixtures A fungicidal synergistic mixture containing a) a compound of the formula I ##STR1## where the substituents have the following meanings: R1 is a phenyl radical which can carry one to three of the following groups: cyano, halogen, C1 | 01/07/1997 |
| 5589479 | Fungicidal mixtures A fungicidal synergistic mixture containing a) a compound of the formula I ##STR1## where the substituents have the following meanings: R1 is a phenyl radical which can carry one to three of the following groups: cyano, halogen, C1 | 12/31/1996 |
| 5587365 | Fungicidal mixtures A fungicidal mixture containing a) the oxime ether carboxamide of the formula I ##STR1## and b) an azole derivative II selected from the group of compounds II.1 to II.16 1-[(2RS,4RS;2RS,4SR)-4-bromo-2-(2,4-dichlorophenyl)tetrahydrofuryl]-1H-1,2, 4-tri... | 12/24/1996 |
| 5587384 | Inhibitors of poly(ADP-ribose) synthetase and use thereof to treat NMDA neurotoxicity Inhibitors of poly(ADP-ribose) synthetase can be used to prevent neurotoxicity mediated through N-methyl-D-aspartate (NMDA) receptors. Poly(ADP-ribose) synthetase inhibitors can be used therapeutically in the treatment of vascular stroke and neurodegenera... | 12/24/1996 |
| 5571845 | Nitroaniline derivatives and their use as anti-tumour agents The invention provides nitroaniline derivatives represented by general formula (I) where the nitro group is substituted at any one of the available benzene positions 2-6; where R and A separately represent the groups NO2, CN, COOR1, ... | 11/05/1996 |
| 5569674 | Heteroacetic acid derivatives Disclosed are compounds of formula ##STR1## wherein R is hydroxy, esterified hydroxy or etherified hydroxy; R1 is halogen, trifluoromethyl or lower alkyl; R2 is halogen, trifluoromethyl or lower alkyl; R3 is halogen, trifluorom... | 10/29/1996 |
| 5567734 | Phenyl-substituted alkylcarboguanidides carrying perfluoroalkyl groups, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them Phenyl-substituted alkylcarboguanidides carrying perfluoroalkyl groups, of the formula I ##STR1## are described where R(A) and R(B) are H, Hal, CN, OR(6), alkyl, Or -perfluoroalkyl or NR(7)R(8); R(6) is hydrogen, (cyclo)alk(en)yl, per... | 10/22/1996 |
| 5565454 | Method for preventing intervention-associated stenosis and other symptoms associated with stenosis of blood vessels following non-bypass, invasive interventions The present invention relates to methods for reducing stenosis after non-bypass invasive intervention and for ameloriating symptomatic chest pains following non-bypass invasive intervention comprising administering a daily amount of a dopamine-potentiatin... | 10/15/1996 |
| 5559140 | Difluoro statone analogs This invention relates to novel difluoro statone analogs, to the processes and intermediates useful for their preparation and to their use as anti-viral agents.... | 09/24/1996 |
| 5556884 | Substituted oxime ethers, their preparation and their use for controlling pests and fungi Substituted oxime ethers of the general formula I ##STR1## where R1 is alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxyalkyl, cycloalkyl, cycloalkylalkyl, cyanoalkyl, alkoxycarbonylalkyl, arylalkyl, heteroarylalkyl, arylalkenyl or a... | 09/17/1996 |
| 5554616 | Fungicidal mixtures A fungicidal mixture containing a) the oxime ether carboxamide of the formula I ##STR1## and either b.1 the oxime ether carboxylic acid ester of the formula II ##STR2## or b.2 the methoxyacrylic acid ester of the formula III ##STR3## in a s... | 09/10/1996 |
| 5554653 | Inhibitors of HIV protease useful for the treatment of AIDS The present invention provides novel HIV protease inhibitors, pharmaceutical formulations containing those compounds and methods of treating and/or preventing HIV infection and/or AIDS.... | 09/10/1996 |
| 5552444 | Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes The present invention provides novel ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes, including their corresponding sulfoxides and sulfones, which ring-substituted compounds exhibit agonist activity at t... | 09/03/1996 |
| 5532260 | Fungicidal mixtures A fungicidal mixture containing a) the oxime ether carboxamide of the formula I ##STR1## and b) an azole derivative II selected from the group of compounds II.1 to II.16 1-[(2RS,4RS;2RS,4SR)-4-bromo-2-(2,4-dichlorophenyl)tetrahydrofuryl]-1H-1,2, 4-tri... | 07/02/1996 |
| 5532259 | Isoxazole-4-carboxamides and hydroxyalkylidenecyanoacetamides, pharmaceuticals containing these compounds and their use Isoxazole-4-carboxamides and hydroxyalkylidenecyanoacetamides, pharmaceuticals containing these compounds and their use Isoxazole-4-carboxamide derivatives and hydroxyalkylidene-cyanoacetamide derivatives are suitable for the treatment of carcinoses. These com... | 07/02/1996 |
| 5516804 | Ortho-substituted phenylacetamides Ortho-substituted phenylacetamides I ##STR1## (R1 =H, alkyl, cycloalkyl, alkenyl, alkynyl, phenylalkynyl, alkoxyalkyl, alkoxycarbonyl, phenyl, phenylalkyl, phenylalkenyl or phenoxyalkyl, 5- or 6-membered heterocycle with 1-3 hetero atoms t... | 05/14/1996 |
| 5514683 | Bicyclo 2,2,2!octane derivatives The compounds of the formula I ##STR1## and their pharmaceutical acceptable salts, which are defined herein, are ligands for cholecystokinin and/or gastrin receptors.... | 05/07/1996 |
| 5512582 | Fungicidal mixtures A fungicidal mixture containing a) the oxime ether carboxamide of the formula I ##STR1## and b) a morpholine or piperidine derivative II selected from the group of compounds IIa, IIb and IIc ##STR2## (n=10,11,12 (60-70%) or 13) in a synergisti... | 04/30/1996 |
| 5512596 | Aromatic compounds A composition comprising a compound of the formula: ##STR1## wherein: X is H or OH; Y is a group capable of hydrogen bonding to amino, guanidino, or imidazole function, or a group comprising an acidic hydrogen atom, a protected acidic group, or an an... | 04/30/1996 |
| 5510348 | Fungicidal mixtures A fungicidal mixture containing a) the oxime ether carboxamide of the formula I ##STR1## and b) a morpholine or piperidine derivative II selected from the group of compounds IIa, IIb and IIc ##STR2## in a synergistically active amount is descr... | 04/23/1996 |
