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| Number | Title | Issue Date |
| 4874792 | Thiophenyl Alkanoic acids useful as leukotriene antagonists This invention relates to alkanoic acid compounds having phenyl and thio substituents which are useful as leukotriene antagonists and pharmaceutical compositions containing such compounds. This invention also relates to treating diseases in which leukotri... | 10/17/1989 |
| 4871756 | Leukotriene antagonists Compounds having the formula: ##STR1## are antagonists of leukotrienes of C4, D4, E4 and the slow reacting substance of anaphylaxis. As such, these compounds will be useful as anti-asthmatic, anti-allergic, anti-infla... | 10/03/1989 |
| 4859697 | Substituted acenaphthenes and their use as inhibitors of phospholipase A2 Substituted acenaphthenes and their use as inhibitors of phospholipase A2 are provided. The acenaphthenes have the formula ##STR1## wherein R1 is H or alkyl; R2 is alkyl, cycloalkyl, or aryl; and R1 and R2 | 08/22/1989 |
| 4855323 | Leukotriene antagonists, a process for the preparation thereof, and the use thereof for the treatment of diseases Leukotriene antagonists, a process for the preparation thereof, and the use thereof for the treatment of diseases ##STR1## in which R1, R2, R3, R4, R5 and X have the indicated meanings, a process... | 08/08/1989 |
| 4853403 | 3-phenylthiomethylstyrene derivative, process for preparing the same, and antiallergic agent and tyrosinekinase inhibiting agent containing the same A 3-phenylthiomethylstyrene derivative having the general formula (1): ##STR1## or salt thereof with a base, when X is hydroxyl group, R1 is hydrogen atom or R2 is hydrogen atom, a process for preparing the 3-phenylthiomethylsty... | 08/01/1989 |
| 4851440 | Leukotriene antagonists, processes for the preparation thereof, the use thereof for the treatment of diseases, and precursors Leukotriene antagonists, processes for the preparation thereof, the use thereof for the treatment of diseases, and precursors. Compounds of the formula I ##STR1## in which R1, R2, R3, R4, R5, R6 | 07/25/1989 |
| 4840969 | N-substituted benzamides An N-substituted benzamide of the formula ##STR1## in which R1 represents hydrogen or alkyl, R2 represents halogenoalkyl with more than one carbon atom, or represents cycloalkyl which is substituted by halogen or halogenoalkyl and R | 06/20/1989 |
| 4835189 | Phenolic thioalkylamides as inhibitors of 5-lipoxygenase The compounds of the present invention comprise substituted phenolic thioalkylamides that are specific inhibitors of 5-lipoxygenase and which, therefore, are useful in the treatment of local and systemic inflammation, allergy and hypersensitivity reaction... | 05/30/1989 |
| 4826876 | Chemical compounds having selective thyromimetic activity This invention relates to chemical compounds which have selective thyromimetic activity. A compound of this invention is 3,5-dibromo-3'-[6-oxo-3(1H)-pyridazinyl-methyl]-thyronine.... | 05/02/1989 |
| 4820719 | Leukotriene antagonists This invention relates to alkanoic acid compounds having phenyl and thio substituents which are useful as leukotriene antagonists and pharmaceutical compositions containing such compounds. This invention also relates to methods of treating diseases in whi... | 04/11/1989 |
| 4808628 | Amide derivatives and their use as fungicides An amide derivative of the formula (I): ##STR1## or a tautomeric form thereof, wherein R is a phenyl group substituted in the 4-position by a group of R1 XCH2--, where R1 is C1 -C4 alkyl, C3... | 02/28/1989 |
| 4808624 | Pharmacologically active substituted benzamides Novel substituted benzamides of the formula ##STR1## wherein R1, R2, R3, R4, R5 and A are as defined herein are useful in the treatment of emesis, and particularly chemotherapy-induced emesis in ... | 02/28/1989 |
| 4806570 | Therapeutic agents Compounds of formula I ##STR1## in which R1 is C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C3-7 cycloalkyl, cycloalkylalkyl or optionally substituted phenyl; R2 is H or C1-3 alk... | 02/21/1989 |
| 4742083 | Method of relieving pain and inflammatory conditions employing substituted salicylamides A topically and systemically administered anti-inflammatory composition for human and for veterinary consumption which comprises compounds of the general formula: ##STR1## wherein R1, R2 and R3 are defined hydrocarbon... | 05/03/1988 |
| 4734435 | N-[[6-methoxy-5-(trifluoromethyl)-1-naphthalenyl]-thioxome thyl]-N-methylglycine S-oxide and the amide thereof Disclosed herein are N-[[6-methoxy-5-(trifluoromethyl)-1-naphthalenyl]-thioxomethyl]-N-methylgl ycine S-oxide (tolrestat S-oxide) and the amide thereof and methods of their preparation. The S-oxides are new aldose reductase inhibitors useful for the t... | 03/29/1988 |
| 4731359 | Prolonged action drug formulation The time during which a drug is pharmacologically active is prolonged by coating the drug with at least one chemical derivative of the drug having minor relative pharmacological activity.... | 03/15/1988 |
| 4730053 | S-[2-phenyl (alkyl) carbamoyl]-phenylselenylmercapto derivatives The present invention is related to new S-(Carbamoyl-phenylselenyl) derivatives of mercaptanes of the general formula (I) ##STR1## and to a process for the treatment of diseases caused by cell injury due to the increased formation of active oxygen me... | 03/08/1988 |
| 4727180 | Antihypertensive polyhalohydroxylisopropyl phenylalkanoic and phenylalkenoic acids, amides and esters and intermediates thereto Polyhalohydroxyisopropyl phenylalkanoic and phenylalkenoic acids, amides, and esters, such as methyl 2-methoxy-4-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]benzenepro panoate, are useful as antihypertensive agents.... | 02/23/1988 |
| 4689330 | Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines Novel substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines useful as anti-depressives, in the treatment of Parkinson's disease and in the treatment of diseases related with disturbed enterokinesia.... | 08/25/1987 |
| 4668703 | γ-allenyl-γ-aminobutyric acids This invention is for γ-allenyl-γ-aminobutyric acid derivatives which are γ-aminobutyric acid transaminase inhibitors.... | 05/26/1987 |
| 4652584 | Acetylenic phenoxypropanol derivatives and pharmaceutical compositions for the treatment of hypertension Phenoxypropanol derivatives having a 2-acetylenic moiety on the phenyl group thereof of the following formula (I): ##STR1## and their use as anti-hypertensives, e.g. in man. Also part of the invention are pharmaceutical compositions and intermediates... | 03/24/1987 |
| 4636505 | Amide derivatives Acylanilides of the formula ##STR1## wherein R1 and R2, the same or different, each is cyano, carbamoyl, nitro, halogeno, perfluoroalkyl or other defined substituents; R3 is hydrogen or halogen; R4 is hydrogen o... | 01/13/1987 |
| 4629737 | Secondary amines and use in pharmaceutical compositions A compound of formula (I): ##STR1## or a pharmaceutically acceptable salt, ester or amide thereof, in which: W is an optionally substituted phenyl group of the formula ##STR2## wherein R1 is hydrogen or fluorine, R2 is hyd... | 12/16/1986 |
| 4628062 | 1,4-naphthoquinone derivatives having anti-inflammatory action New compounds of the formula ##STR1## in which R1 is an allylamino, acetylamino or propionylamino radical, R2 is hydrogen or a 2-methoxyethoxy or ethoxy radical, R3 is hydrogen or a sulphamoyl radical, and R4 is hydr... | 12/09/1986 |
| 4621098 | Thioethers and pharmaceutical compositions containing them The present invention provides thioethers of the general formula: ##STR1## wherein Ar is a phenyl radical which is optionally substituted one, two or three times by alkyl, alkenyl, alkoxy, alkylthio, alkanoyl, hydroxyl, hydroxyalkyl, carboxyl, alkoxy... | 11/04/1986 |
| 4619944 | Antihypertensive compounds Provided are antihypertensive compounds of the formula ##STR1## wherein R1, R2, R3, R4, R5, and R6 are hydrogen, alkyl, alkenyl, alkynyl, phenyl-alkyl, or cycloalkyl, and may be the sa... | 10/28/1986 |
| 4598087 | Substituted trans-1,2-diaminocyclohexyl amide compounds Substituted trans-1,2-diaminocyclohexyl amide compounds demonstrating selective opioid receptor binding possess utility as analgesic, diuretic, and psychotherapeutic agents. A method of preparing the compounds, pharmaceutical compositions employing the co... | 07/01/1986 |
| 4528286 | Method of using certain aryl-mercapto-lower-alkanamides as antiseborrheic agents Aryl-mercapto-lower-alkanamides having the following formula ##STR1## wherein R1 is selected from the group consisting of phenyl, C1-4 -alkylphenyl, halophenyl, hydroxyphenyl, C1-4 -alkoxyphenyl, aminophenyl, acetamid... | 07/09/1985 |
| 4513009 | Aminoacid derivatives and their therapeutic applications This invention relates to aminoacid derivatives, and compositions containing the same and having enkephalinase-inhibiting, antalgic, antidiarrhea and hypotensive activities, of the formula ##STR1## whose variables are as set forth herein, for example... | 04/23/1985 |
| 4485115 | Method for treating depressive syndrome by administering N-(diethylaminoethyl)-2-methoxy-5-methylsufonyl benzamide The depressive syndrome associated with alcoholic withdrawal is treated by administering N-(diethylaminoethyl)-2-methoxy-5-methylsulfonyl benzamide.... | 11/27/1984 |
| 4460600 | Adjacently substituted ketal derivatives of cycloalkane-amide analgesics Cis- and trans-N-[2-amino(adjacenty substituted bis(alkyloxy), bis(alkylthio), alkylthio or mercapto group substituted)-cycloaliphatic]benzeneacetamide and -benzamide compounds, e.g., (&#b1;)-(1,2ଲ)-4-bromo-N-[3,3-dimethoxy-2-(1-pyrrolid... | 07/17/1984 |
| 4425357 | Acyl anilines exerting a fungicidal action Acyl anilines are disclosed having the formula ##STR1## wherein R and R1 (like or unlike each other)=H; CH3 ; C2 H5 ; n.C3 H7 ; --CH2 --CH.dbd.CH2 ; --CH.dbd.CH--... | 01/10/1984 |
| 4425360 | Pharmacologically active novel O-substituted pyruvic acid oximes The present invention provides pyruvic acid oximes of the general formula: ##STR1## wherein R is a hydrogen atom, a C3 -C8 cycloalkyl, C1 -C6 alkoxy, cinnamyloxy, phenylamino, phenyl-N-alkylamino or phenylt... | 01/10/1984 |
| 4416889 | Combating fungi with N-allenyl-acetanilides N-allenyl-acetanilides of the formula ##STR1## in which R1 represents hydrogen, alkyl or halogen, R2 represents hydrogen or alkyl, R3 represents hydrogen or alkyl, R4 represents hydrogen or alkyl, R5 repre... | 11/22/1983 |
| 4407816 | 3-Substituted-2-propenimidamides and method of manufacturing the same New derivatives of 3-furyl-, 3-thienyl- and 3-phenyl-2-propenimidamides are disclosed, which are useful as anti-ulcer agents. These new compounds are synthesized by reacting an imino ether derived from a corresponding 3-substituted-2-propenenitrile with a... | 10/04/1983 |
| 4386080 | Anti-androgenic amide derivative Novel 3,4-disubstituted-N-acylanilines of the formula: ##STR1## wherein R1, R2 and ring A are defined in claim 1; wherein R3 is hydrogen or alkyl of up to 4 carbon atoms, or is joined to R5 as stated below;... | 05/31/1983 |
| 4340603 | Novel inotropic prodrugs Novel, transient inotropic prodrug forms of the N-(2-phenylethyl)-ω-phenylalkylamines, notably of dobutamine, have (i) the structural formula (I): ##STR1## with the proviso that at least one R1, R2 or OR1, when ... | 07/20/1982 |
| 4329363 | Substituted mercapto acid amides and their use The present application discloses a method of correcting an imbalance of immune homeostasis caused by cytostatic treatment or radiotherapy by administering to a patient in need of such treatment an effective amount of a novel substituted mercapto acid ami... | 05/11/1982 |
| 4312862 | Therapeutically active derivatives of benzamide Novel therapeutically active derivatives of benzamide, having the general formula ##STR1## in which R1 and R2, independently of each other, are hydrogen or a lower alkyl group, R3 is a phenyl or lower alkyl or lower a... | 01/26/1982 |
| 4310545 | Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino) phenyl compounds This disclosure describes novel 4-(polyfluoroalkylamino)phenyl compounds useful as hypolipidemic and antiatherosclerotic agents.... | 01/12/1982 |
