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| Number | Title | Issue Date |
| 7598289 | Ketones and reduced ketones as therapeutic agents for the treatment of bone conditions The present invention pertains to certain ketones and reduced ketones and derivatives thereof which, inter alia, inhibit osteoclast survival, formation, and/or activity; and/or inhibit bone resorption, and more particularly to compounds of the formulae and pharmaceu... | 10/06/2009 |
| 7572825 | Ketones and reduced ketones as therapeutic agents for the treatment of bone conditions The present invention pertains to certain ketones and reduced ketones and derivatives thereof which, inter alia, inhibit osteoclast survival, formation, and/or activity; and/or inhibit bone resorption, and more particularly to compounds of the formulae: (1) (2) wher... | 08/11/2009 |
| 7232915 | Process for the synthesis of 1,3-diols An improved process for the preparation of cis-1,3-diols is described where a beta hydroxy ketone is treated with a trialkylborane or dialkylalkoxyborane or a mixture of a trialkylborane and a dialkylalkoxyborane followed by recovery and reuse of the alkylborane spe... | 06/19/2007 |
| 7211267 | Methods of treating acne A method of treating acne in a human in need thereof comprising administering systemically to said human a tetracycline compound in an amount that is effective to treat acne but has substantially no antibiotic activity, without administering a bisphosphonate compoun... | 05/01/2007 |
| 7175860 | Enhanced wound healing method and composition A composition extracted from nut husks including a method of forming the composition, where the composition is useful in healing wounds. The method includes collecting pecan husks, pressing the pecan husks thereby expressing fluid from the husks, and collecting the ... | 02/13/2007 |
| 7115651 | Macrocycles and uses thereof The present invention relates to compounds having the structure (and pharmaceutically acceptable derivatives thereof) wherein R0–R4, Z, X, A—B, D—E, G—J, and... | 10/03/2006 |
| 7074422 | Fungicidal mixtures Fungicidal mixtures, comprising A) the compound of the formula I and B) the compound of the formula II ... | 07/11/2006 |
| 7014858 | Use methods of treating acne and telangiectasia A method of treating telangiectasia in a human in need thereof comprising administering to said human a tetracycline compound in an amount that is effective to treat telangiectasia, but has substantially no antibiotic activity. ... | 03/21/2006 |
| 7008631 | Methods of simultaneously treating ocular rosacea and acne rosacea A method for simultaneously treating ocular rosacea and acne rosacea in a human in need thereof comprising administering systemically to said human a tetracycline compound in an amount that is effective to treat ocular rosacea and acne rosacea but has substantially ... | 03/07/2006 |
| 6955820 | Coenzyme Q10 formulation and process methodology for softgel capsules manufacturing A formulation of Coenzyme Q10, beta-carotenes, Vitamin E, and medium chain triglycerides in rice bran oil and an optional thickener, such as bee's wax, is provided in a soft gel capsule so that a maximum of the Coenzyme Q10 is absorbed by the h... | 10/18/2005 |
| 6916835 | Nitrate esters and their use for neurological conditions Compounds and methods for mitigating neurodegeneration, effecting neuroprotection and/or effecting cognition enhancement in a subject are described. Neurological or cognitive conditions are treated by administering to a subject an effective amount of a therapeutic c... | 07/12/2005 |
| 6900338 | Scavenger compounds The present invention provides novel compounds having scavenging and anti-ROS properties and pharmaceutical composition comprising these compounds for treatment of conditions associated with oxidative stress or free radical injury. The compounds of the invention are... | 05/31/2005 |
| 6664287 | Antioxidants This invention comprises administering to a human or animal in need of treatment an effective amount of an antioxidant lipoic acid derivative and/or pharmaceutically acceptable salts and solvates thereof for the treatment or prevention of pathological (in... | 12/16/2003 |
| 6649639 | Antipicornaviral compounds, compositions containing them, and methods for their use Picornaviral 3C protease inhibitors, obtainable by chemical synthesis, inhibit or block the biological activity of the picornaviral 3C protease. These compounds, as well as pharmaceutical compositions that contain these compounds, are suitable for treatin... | 11/18/2003 |
| 6635650 | Substituted dimeric compounds The invention relates to compounds of formula (I): wherein: A represents NR1 C(Q)R2, C(Q)NR2 R3 or NR1 C(Q)NR2 R3, B represents NR1 C(Q)R2, C(Q)NR2... | 10/21/2003 |
| 6583161 | Benzenesulfonamides and benzamides as therapeutic agents The invention provides compounds, compositions and methods relating to novel aromatic derivatives and their use as pharmacologically active agents. The compositions find particular use as pharmacological agents in the treatment of disease states, particul... | 06/24/2003 |
| 6562861 | Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors ##STR1## Compounds I-III wherein U is CH, O, or S; Z is mono- or di-substituted carbon; R is (CH2)nCO2H, (CH2)nSO3H, (CH2)nPO3H2, (CH2)nNO2, CH(SCH3)3, esters; R1 is H, hydroxyalkyl, aminoalkyl, alkoxyalkyl; RR1 is O; n is 0-4; R2, R3 is H, hydroxyalkyl, ... | 05/13/2003 |
| 6512003 | Synthetic spiroketal pyranes as potent anti-cancer agents and use Novel tubulin binding compounds (SPIKETS) having potent tubulin depolymerization activity and inhibitory activity against tubulin polymerization. The compounds are effective agents for inhibiting cellular proliferation, for example, in cancer cells. The c... | 01/28/2003 |
| 6440985 | Methods for treating viral infections Methods are provided for the treatment and prophylaxis of viral infection and disease associated with such infection.... | 08/27/2002 |
| 6407136 | 1,4-dithiin and 1,4-dithiepin-1,1,4,4, tetroxide derivatives useful as antagonists of the human galanin receptor The invention is directed to 1,4-dithiin- and 1,4-dithiepin-1,1,4,4-tetroxide derivatives useful as galanin receptor antagonists for treating disorders of the central nervous system. Pharmaceutical compositions comprising the compounds of the present ... | 06/18/2002 |
| 6358960 | Amidino derivatives and drugs containing the same as the active ingredient The novel amidino derivatives of the formula (I): ##STR1## wherein all the symbols are as in specification defined; have an inhibitory activity of a blood coagulation factor VIIa and are useful for treatment and/or prevention of several angiopathy caused by ... | 03/19/2002 |
| 6342517 | Potassium channel activators and their use Novel thienopyran compounds are disclosed, useful as anti-hypertensive agents and for asthma treatment. One group of the compounds has a heterocyclic ring spiro-connected at the 7-position of the thienopyran ring structure. Use of thienopyran compounds in... | 01/29/2002 |
| 6331554 | Antipicornaviral compounds, compositions containing them, and methods for their use Picornaviral 3C protease inhibitors of formula I, obtainable by chemical synthesis, that inhibit or block the biological activity of the picornaviral 3C protease are described. ##STR1## These compounds, as well as pharmaceutical compositions that contain ... | 12/18/2001 |
| 6288071 | 1-ethylene-2-alkylene-1,4-cyclohexadiene pesticides Pesticidally active cyclohexadienyl derivative compounds of the formula I that are esters, oximes or amides are claimed. These compounds may be used as fungicides, acaricides and insecticides in plant protection.... | 09/11/2001 |
| 6075023 | Method for combatting fish mycoses and one-celled ectoparasites Fish mycoses and single-cell ectoparasites on fish are controlled using an active compound suitable for inhibiting the mitochondrial respiratory chain at the stage of the b/c1 complex.... | 06/13/2000 |
| 6046228 | Anti-viral pharmaceutical compositions containing saturated 1,2-dithiaheterocyclic compounds and uses thereof The present invention is directed to pharmaceutical compositions including a saturated 1,2-dithiaheterocyclic compound having antiviral activity. The present invention also provides a kit containing the pharmaceutical composition and methods of treating o... | 04/04/2000 |
| 6030924 | Solid formulations The novel solid formulations obtained by low pressure extrusion of a mixture comprising at least one active ingredient; and at least one defoaming agent and/or foam breaking agent from the group consisting of perfluoroalkylphosphinic acids and/or perfluoroalkylphos... | 02/29/2000 |
| 6022895 | Substituted amino compounds and their use as substances having an analgesic effect Substituted amino compounds of general formula (I) ##STR1## are described, as are a method of preparing them and their use as drugs, especially as analgesics.... | 02/08/2000 |
| 6020371 | Antipicornaviral compounds compositions containing them and methods for their use Picornaviral 3C protease inhibitors, obtainable by chemical synthesis, inhibit or block the biological activity of the picornaviral 3C protease. These compounds, as well as pharmaceutical compositions that contain these compounds, are suitable for treatin... | 02/01/2000 |
| 5914351 | Anti-viral aromatic hydrazones Compounds of the formula ##STR1## wherein Q is a hydrazone derivative; R1 is hydrogen, halogen, alkyl or alkoxy; R2 is hydrogen, halogen, alkyl, alkoxy, alkenoxy, alkynyloxy, halomethyl, trifluoromethoxy, alkylthio, nitro or cyano; a... | 06/22/1999 |
| 5747542 | Oxo-substituted tetrahydronaphthalene derivatives having retinold and/or retinoid antagonist-like biological activity Compounds of the formula ##STR1## where the symbols have the meaning described in the application, have retinoid-like or retinoid antagonist-like biological activity.... | 05/05/1998 |
| 5705501 | Certain substituted 1-aryl-3-morpholinopropanones to treat Alzheimer's Disease Disclosed are compounds of formula I: ##STR1## wherein X is selected from oxygen, sulfur and NR; wherein R is selected from hydrogen, loweralkyl and CH2 CH2 COAr1 ; and Z is hydrogen; straight or branched chain alkyl havin... | 01/06/1998 |
| 5698580 | Antiviral agent containing benzodithiin derivative as active ingredient Antiviral agents comprising, as an active ingredient, a 1,4-dihydro-2,3-benzodithiin derivative of the formula ##STR1## wherein each symbol is as defined in the Specification, or a pharmacologically acceptable salt thereof. The antiviral agents of th... | 12/16/1997 |
| 5668168 | 1,2-dithiin antiinfective agents This invention pertains to a novel group of 1,2-dithiin compounds useful as antiinfective agents, and a novel synthetic process to produce the same. The compounds are particularly effective in treating fungal infections, especially those caused by Candida... | 09/16/1997 |
| 5648354 | 1,2-dithiins having antifungal activity Novel 1,2-dithiin compounds useful as antifungal or anti-infective agents, as well as methods for their use as such, are described. The 1,2-dithiin compounds are particularly effective in treating infections, especially those caused by Candida albicans, C... | 07/15/1997 |
| 5580897 | 1,2-dithiins having antifungal activity Novel 1,2-dithiin compounds useful as antifungal or anti-infective agents, as well as methods for their use as such, are described. The 1,2-dithiin compounds are particularly effective in treating infections, especially those caused by Candida albicans, C... | 12/03/1996 |
| 5556875 | 1,2-dithiin antiinfective agents This invention pertains to a novel group of 1,2-dithiin compounds useful as antiinfective agents, and a novel synthetic process to produce the same. The compounds are particularly effective in treating fungal infections, especially those caused by Candida... | 09/17/1996 |
| 5543433 | Azine-substituted phenylacetic acid derivatives and fungicides containing these Compounds of the formula I ##STR1## where X is hydrogen, halogen, alkyl, alkoxy, trifluoromethyl, cyano or nitro, Y is an amino, methylamino or dimethylamino group, Z is a group CHCH3, CHOCH3 or NOCH3, R is hydrogen or alk... | 08/06/1996 |
| 5508275 | Lipid-selective antioxidants and their preparation and use Lipid-selective antioxidants of the formula I (A)a (L)(X)a, (I), in which A=an antioxidative component, L=a bridging member, X=a lipophilic component a and a'=independently of one another the numbers 1 or 2. The c... | 04/16/1996 |
| 5502073 | Heterocyclic pesticidal compounds Compounds of the formula (I) ##STR1## which contain between 10 and 27 carbon atoms, and wherein m and n are independently selected from 0, 1 and 2; R2a is hydrogen, methyl, or ethyl; R2b is acetylene or contains between 3 and 18... | 03/26/1996 |
