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Patent No. 5285430

Behavior Modification Wristwatch

A wristwatch including a watch band and a watch body having an octagon shaped perimeter and being red in color and having the word STOP thereon to resemble a stop sign.

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Class 514/349 - Nitrogen attached directly to the six-membered hetero ring by nonionic bonding


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein nitrogen is attached directly to
No. of patents: 299
Last issue date: 05/07/2013


            7    
NumberTitleIssue Date
4826859Fungicidal methods containing N-pyridylcarbamates
Fungicidal composition comprising a fungicidally effective amount of the N-pyridylcarbamate derivative having the formula (I) as an active ingredient: ##STR1## wherein X is 2-naphthyl, 5-indanyl, 5,6,7,8-tetrahydro-2-naphthyl, 1,4-methano-1,2,3,...
05/02/1989
4822802Method of fentanly administration for postoperative pain relief
A method of postoperative pain relief using transdermal delivery of fentanyl or its analgetically effective derivatives preceded by a dose of said material to increase the serum drug levels to steady state more quickly....
04/18/1989
4818766Novel phenoxyaliphatylphenyleneoxyalkyl esters and amides
The invention relates to novel 1,4-dihydropyridine-3-carboxylic acid phenoxyaliphatylphenyleneoxyalkyl esters of the formula ##STR1## in which Ac represents an acyl group, X represents oxy or optionally substituted imino, A represents a divalent alip...
04/04/1989
4812447Method for the treatment of nervous system degeneration
Disclosed is a method for treating nervous system deterioration associated with aging and Alzheimer's disease by administering a therapeutically-effective amount of dehydroepiandrosterone or its sulfate. Also disclosed is the co-administration of dehydroe...
03/14/1989
4798839Synergistic insecticidal compositions
Insecticidal compositions are provided which contain mixtures of certain benzoyl ureas and a synergist which is a methylenedioxyphenyl derivative. The invention also encompasses a method of controlling insects by subjecting them to an effective amount of ...
01/17/1989
4791123Insecticidal triffluormethyl alkane derivatives
There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1## in which R1, R2, R3, R4 and A have the meanings given in the description, processes for their preparation and ins...
12/13/1988
4783485Benzoylurea compounds, and insecticidal and acaricidal compositions comprising same
The invention relates to new benzoylurea compounds having insecticidal and acaricidal activity, of the general formula ##STR1## wherein R1 is a hydrogen atom or represents 1 or 2 halogen atoms; Ar is a para-phenylene group or a para-pyridylene ...
11/08/1988
4749700Novel methods of administering antihistamines, antinausea and antiemetic pharmaceutical agents and novel dosage forms containing same
Invention relates to nasal administration of physiologically active therapeutic agents and dosage forms useful for such administration....
06/07/1988
4725602Acetylene amines and their use as vasodilators and antihypertensives
Acetylenes of the following formula (I): ##STR1## wherein Y, m, R1, R2, R3, n and R4 are defined herein and R5 is hydrogen, alkyl, cycloalkyl or substituted alkyl are useful vasodilators and anti...
02/16/1988
4665073Haloalkylguanidine compounds, pharmaceutical compositions and methods processes and intermediates
The invention relates to guanidine derivatives which are histamine H-2 antagonists and which inhibit gastric acid secretion. According to the invention there is provided a guanidine derivative of the formula I: ##STR1## in which R1 and R
05/12/1987
4663334Heteroaromatic acetylenes useful as antihypertensive agents
Heterocyclic acetylenes of the formula (I): ##STR1## wherein Y is alkyl, alkoxy, alkoxyalkyl, chloro, fluoro, bromo or carboxamidoalkyl and R1 is hydrogen, alkyl, alkoxy, alkylthio, alkoxycarbonyl, chloro, fluoro or dialkylamino, m is 0-2,...
05/05/1987
4659736Benzoyl urea compounds as agents for repelling snails and slugs
A method of combating slugs and snails comprising applying to a plant or to an area from which it is desired to exclude such slugs and snails a repellent amount of at least one benzoyl urea of the formula ##STR1## in which R, R1 and R...
04/21/1987
4657908Carbonyl derivatives
The invention relates to carbonyl derivatives which are histamine H-2 antagonists and which inhibit gastric acid secretion. According to the invention where is provided a guanidine derivative of the formula I: ##STR1## in which R1 and R
04/14/1987
46525722-(furanyl alkylamino or thienyl alkylamino or phenylalkylamino)-3-carboxy (or hydroxy)-pyridines
This invention relates to 2-amino-3-hydroxy, and 3-carboxy pyridine derivatives, in which the amino group is substituted by a methylthioethyl, butyl or oxypropyl group bearing a terminal heterocyclic group. The compounds have histamine H2 -anta...
03/24/1987
4647569Antiarthritic pyridylaminoethene disulfonyl compounds and use
Pyridylaminoethene derivatives of the formula: ##STR1## wherein R1 is pyridyl, unsubstituted or substituted by one or more substituents R4 selected from halogen, amino, carboxy, cyano nitro, hydroxy, formyl, trifluoromethyl, ary...
03/03/1987
4624962Substituted derivatives of 2-azabicyclo-[3.3.0]octanes
Compounds of the formula I ##STR1## in which n denotes 0-3, R1 and R1' are the same or different and denote hydrogen, alkyl or alkenyl, phenyl or benzyl, each substituted as desired; R2 denotes hydrogen, alkyl or alkenyl; ...
11/25/1986
4555517Pyridone esters as inotropic agents
Described are compounds of the formula ##STR1## wherein R is hydrogen, lower alkyl, halo, cyano, hydroxy, amino, lower alkylamino, --CH2 NH2, CH2 OH or COOR"; R' is hydrogen, lower cycloalkyl or lower alkyl; R" is low...
11/26/1985
4540578Pesticidal phenoxypyridyl benzoyl ureas
Novel phenoxyphenyl and phenoxypyridyl benzoyl ureas and a process for their preparation are provided. The novel ureas are useful as the active toxicant in pesticidal compositions....
09/10/1985
4518603[2-[(Nitropyridinyl)amino]phenyl]arylmethanones in a process for preparing pyrido[1,4]benzodiazepines
[2-[(Nitropyridinyl)amino]phenyl]arylmethanones as chemical intermediates and/or having antidepressant activity having the formula: ##STR1## wherein; B is carbonyl, thioxomethyl, ketal or thioketal, R is hydrogen or --alk1 -Q, Q is hydrogen, --...
05/21/1985
45157973-Amino-5-(hydroxy- and/or aminophenyl)-6-(lower-alkyl)-2(1H)-pyridinones and cardiotonic use thereof
1-R1 -3-amino-5-(3-R'-4-R"-phenyl)-6-R-2(1H)-pyridinones or salts thereof, which are useful as cardiotonics, where R1 is hydrogen, lower-alkyl, or lower-hydroxyalkyl, R is hydrogen or lower-alkyl, and, R' and R" are each hydrogen, hy...
05/07/1985
4515803Substituted derivatives of octahydroindole-2-carboxylic acids
Compounds of the formula I ##STR1## in which n denotes 0-3, R1 and R1' are the same or different and denote hydrogen, alkyl or alkenyl, phenyl or benzyl, each substituted as desired; R2 denotes hydrogen, alkyl or alkenyl;...
05/07/1985
4439427Method and composition for treating pediculosis
A method of treating lice infestations in patients in need of such treatment and composition useful therefor is disclosed and includes topically applying to the lice-infected area an effective amount of one or more of the pediculocide agents selected from...
03/27/1984
4438136Prostaglandins
Novel bicyclo [2,2,1] heptanes and hept-2-enes are substituted at the 5-position by a 6-carboxyhex-2-enyl group or a modification thereof, and at the 6-position by a grouping --C(R).dbd.N--NHCO--(NH)a --R' in which R is hydrogen, an aliphatic h...
03/20/1984
4426385Insecticidal bicyclooxyphenyl ureas
Novel bicyclooxyphenyl ureas, such as 1-(bicyclooxyphenyl)-benzoyl ureas, are provided which exhibit pesticidal activity. The compositions are conveniently prepared by reacting an isocyanate with either an amide or a bicyclooxyaniline....
01/17/1984
4414218Cyano-(substituted and unsubstituted pyridinyl) methyl and aryl esters of carbonic acid
The novel compounds of this invention are pyridinyl cyano carbonates corresponding to the formula ##STR1## wherein: R is alkyl or aryl of up to 20 carbons; X is hydrogen, halo, cyano, nitro, R or OR; and n is 1, 2, 3 or 4....
11/08/1983
44055521-Benzoyl-3-(arylphyridyl)urea compounds
The present invention is directed to 1-benzoyl-3-(arylpyridyl)urea compounds useful as insecticides....
09/20/1983
4331670Pyridylanilines
A novel compound for combatting insect, mite, fungus or bacterium is a pyridylaniline represented by the following formula (I) ##STR1## wherein X is a trifluoromethyl group, a halogen atom, a lower alkyl group or a lower alkoxy group; n is an integer...
05/25/1982
4305946Propargyl thio-nitro-pyridines
Novel propargylthio-nitropyridines of the formula ##STR1## wherein X is hydrogen or halogen, processes for producing these compounds, as well as compositions containing them, for use in combating pests, particularly for use as ovicides for combating ...
12/15/1981
4297357N-Phenethylacetamide compounds and process for preparation thereof
N-phenethylacetamide compounds of the formula: ##STR1## wherein X1 represents a lower alkoxy group, X2 represents a hydrogen atom or a lower alkoxy group and R represents a phenyl group, a pyridyl group, a pyrimidinyl group or a...
10/27/1981
4285952Pyridyl, thiazolyl and isothiazolyl alkyl bisamidines
Bisamidines carrying one unsaturated nitrogen heterocycle-containing substituent, representative of which is 1-[N'-(2-(5-methyl-4-imidazolyl)methylthio)ethyl)guanidino]-8-[N'-methylgu anidino]octane, are histamine H2 -antagonists....
08/25/1981
4252813Oxamides, pharmaceutical compositions thereof and method of use
Compounds of the formula ##STR1## are useful as anti-allergy agents....
02/24/1981
4252804Therapeutically useful 3,4,5-trimethoxybenzene derivatives
Compounds of the formula I ##STR1## wherein m and n are 0, 1 or 2, X represents oxygen, imino, benzylimino, or morpholinoethylimino, Y represents CO, CONH, COO or SO2, and NR1 R2 represents a dimethylamino, diethylami...
02/24/1981
42410682-(Pyridyl-amino)-benzoic acids and salts thereof
Compounds of the formula ##STR1## wherein A is .dbd.CH-- or .dbd.N--; R1 is (a) hydrogen, lower alkyl, lower alkoxy or a fused benzene ring, or (b) --CO--R4, tetrazol-5-yl or cyano in the 4- or 5-position; R2 is --CO--R
12/23/1980
4226871Heterocyclic carbamates
Heterocyclic carbamates are disclosed which have potent gastric secretion inhibitory properties. The heterocyclic substituent is a pyridyl group or a 6-membered heterocycle with two nitrogen heteroatoms, which may be optionally substituted. Further substi...
10/07/1980
4215126Alkoxy pyridine compounds
The compounds are alkoxypyridine compounds which are histamine H2 -antagonists. Two specific compounds of the present invention are N-cyano-N'-methyl-N"-[2-((3-methoxy-2-pyridyl)methylthio)ethyl]guanidine and 1-methylamino-1-[2-((3-methoxy...
07/29/1980
4205073Anti-diarrheal anilino nicotinic acids and method of using same
This invention relates to compositions of matter useful as anti-diarrheal agents and to the method of controlling and treating diarrhea in warm blooded animals. The active anti-diarrheal agents are substituted anilino nicotinic acids, and salts thereof an...
05/27/1980
41950902-(3-Amino-2-hydroxy-propoxy)pyridine derivatives and pharmaceutical compositions therewith
Heterocyclic compounds of the formula ##STR1## wherein Het denotes optionally substituted pyridazinyl, pyrimidinyl, pyrazinyl or substituted pyridyl, R1 is hydrogen or methyl and R2 is lower alkyl, optionally substituted phenyl-...
03/25/1980
4189488Amidinoformic and amidinosulphinic acids
Amidinoformic acids and amidinosulphinic acids which are histamine H2 -antagonists. Two specific compounds of the present invention are N-[2-(5-methyl-4-imidazolylmethylthio)ethyl]amidinoformic acid and N-methyl-N'-[2-(5-methyl-4-imidazolylmeth...
02/19/1980
4173637N-Benzoyl-N'-pyridyloxy phenyl urea and insecticidal compositions thereof
N-benzoyl N'-pyridyloxy phenyl urea having the formula ##STR1## wherein X1 represents a halogen atom or methyl group; X2 represents hydrogen or halogen atom; X3 and X4 respectively represent hydrogen or hal...
11/06/1979
41736391-Benzoyl-3-(alkoxy- or alkylthiopyridinyl)ureas
The present invention is directed to 1-benzoyl-3-(alkoxy- or alkylthiopyridinyl)urea compounds useful as insecticides....
11/06/1979
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