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| Number | Title | Issue Date |
| 4816451 | Antibacterial 1,8-bridged 4-quinolonecarboxylic acids Antibacterially effective 1,8-bridged 4-quinolone-3-carboxylic acids and derivatives of the formula ##STR1## in which Y represents a carboxyl group, a nitrile group, an ester group --COOR7 or an acid amide group --CONR8 R9 | 03/28/1989 |
| 4808585 | Solutions of lactic acid salts of piperazinylquinolone- and piperazinyl-azaquinolone-carboxylic acids The invention relates to solutions of piperazinylquinolone- and piperazinyl-azaquinolone-carboxylic acids, and in particular both ready-to-use injection and/or infusion solutions and dosage forms which can be converted into such injection and/or infusion ... | 02/28/1989 |
| 4762831 | Antibacterial 1,8-bridged 4-quinolone-3-carboxylic acids A process for the preparation of a 1,8-bridged 4-quinolone-3-carboxylic acid of the formula ##STR1## wherein the substituents are defined hereinbelow. Some of the compound are new. The old and new compounds are antibacterials and promote animal ... | 08/09/1988 |
| 4753953 | Pyridonecarboxylic acid derivatives and antibacterial pharmaceutical compositions thereof Pyridonecarboxylic acid derivatives of the following formula, ##STR1## wherein R is hydrogen atom or lower alkyl group, R1 is lower alkyl group, cycloalkyl group or haloalkyl group, Y is hydrogen atom or halogen atom, or Y and R1 | 06/28/1988 |
| 4735940 | Tricyclic pyridine derivatives and pharmaceutical compositions Compounds of the formula ##STR1## or a pharmaceutically acceptable acid addition salt of a compound of formula I which has one or more basic substituents, are described. The compounds of formula I possess pronounced muscle relaxant, sedative-hypnotic... | 04/05/1988 |
| 4729998 | Cyclic carbamates and fungicidal use Fungicidally active cyclic carbamates of the formula ##STR1## in which X and Y each represent oxygen or sulfur, Z represents hydrogen, halogen, alkyl or nitro, and n is 2 or 3. Some intermediates are new.... | 03/08/1988 |
| 4623647 | [1,3]oxazino[4,3-a]-isoquinoline derivatives and pharmaceutical compositions containing them The invention relates to new [1,3]oxazino[4,3-a]-isoquinoline derivatives of the formula (I) ##STR1## wherein R1 and R2 represent hydroxyl or alkoxy having from 1 to 6 carbon atoms, R3 is hydrogen, alkyl having from 1... | 11/18/1986 |
| 4623650 | Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids 1-Substituted-6-fluoro-7-aryl-(8-fluoro)-1,4-dihydroquinol-4-one 3-carboxylic acids having antibacterial activity are prepared by reacting the corresponding alkyl 1-substituted-6-fluoro-7-bromo-(8-fluoro)-1,4-dihydroquinol-4-one-3-carbox ylate with an... | 11/18/1986 |
| 4605653 | 1-(hydroxymethyl)-1,6,7,11b-tetrahydro-2H,4H-[1,3]oxazino- or -thiazino-[4,3-a]isoquinoline derivatives and pharmaceutical compositions containing them The invention relates to 1-(hydroxymethyl)-1,6,7,11b-tetrahydro-2H,4H-[1,3]oxazino- or -thiazino-[4,3-a]isoquinoline derivatives of the formula (I), ##STR1## wherein R1 and R2 are alkoxy having from 1 to 6 carbon atoms, X is oxy... | 08/12/1986 |
| 4576942 | Anti-allergic and anti-inflammatory bi- and tri- cyclo-1,4-thiazine derivatives, composition, and method of use therefor Compounds of the formulae ##STR1## wherein, A is benzo, pyrido, thieno, pyrazolo, imidazo, pyrimido, isoxazolo, thiazolo, furo or pyrrolo; X is O, S, SO or SO2 ; R1 is H, alkyl, aryl, OH, OR, aryloxy, halogen, amino, nitro, cyano, ... | 03/18/1986 |
| 4571396 | Antibacterial agents Novel naphthyridine-, quinoline- and benzoxazine-carboxylic acids as antibacterial agents are described as well as methods for their manufacture, formulation, and use in treating bacterial infections including the description of certain novel intermediate... | 02/18/1986 |
| 4564615 | Immunoactivator An immunoactivator comprising an effective amount of a thiazolobenzoxazine derivative of the formula, or its salt ##STR1## wherein R1 represents a hydrogen atom, carboxyl group or lower alkoxycarbonyl group, R2 represents a subs... | 01/14/1986 |
| 4547499 | 2,4-Dihydr o-2(omega-aminoalkyl)-1H-[1,2,4]triazolo[3,4-c]benzoxazin-1-one anti-alle rgy drug compounds, compositions and use 2,4-Dihydro-2-(omega-aminoalkyl)-1H-[1,2,4]triazolo[3,4-c][1,4]benzoxazin-1 -ones of the formula ##STR1## where n and -NRR are as defined in the specification, e.g., 2-[4-[4-(2,3-dihydro-2-oxo-1H-benzimidazol-1-yl)piperadinyl]butyl]-2,4-dih ydro-1... | 10/15/1985 |
| 4537888 | Substituted benzoxazine derivatives and fungicidal use Novel Substituted benzoxazine derivatives of the formula ##STR1## in which X is oxygen or suophur, and R1 and R2 each independently is hydrogen, alkyl, alkoxy, akylthio, halogenoalkyl, alkanoyl, aroyl, halogen, cyano, nitro, nitroso,... | 08/27/1985 |
| 4492697 | 4H-Imidazo[2,3-c]pyrido[2,3-e][1,4]oxazine derivatives The invention discloses novel 4H-imidazo[2,3-c]pyrido[2,3-e][1,4]oxazine derivatives, processes for their preparation, pharmaceutical compositions thereof and methods for using the compounds. The compounds of this invention are useful in the treatment of ... | 01/08/1985 |
| 4443447 | Phenyl-substituted tricyclic antibacterial agents Antimicrobial compounds of the following formula are disclosed: ##STR1## wherein X is selected from the group consisting of --O--, --CH2 and ##STR2## m is 0 or 1; R1 is selected from the group consisting of hydrogen, nitro,... | 04/17/1984 |
| 4335129 | Thiazolo[3,2-6]isoquinolines, compositions and use thereof Nitrogen containing heterocyclic compounds shown by the formula ##STR1## wherein Y represents an oxygen atom, a sulfur atom, or a group shown by ##STR2## (wherein m is 1 or 2); n represents 0 or 1; R1 and R4, which may be t... | 06/15/1982 |
| 4307092 | 1-Oxo-5H-pyrimido[2,1-C]benzoxazine-2-carboxylic acid esters This invention discloses novel 1-oxo-5H-pyrimidol[2,1-c][1,4]benzoxa(or thia)zinc-2-carboxylic acid lower alkyl esters, derivatives thereof, process for their preparation, pharmaceutical compositions thereof and methods for using the compounds. The compou... | 12/22/1981 |
| 4291032 | Thiazolo(3,2-C)benzoxazine derivatives New thiazolo[3,2-c]-1,3-benzoxazine derivatives of the general formula (I), in which X is oxygen or sulfur, R1 and R2, which are identical or different, are hydrogen or halogen atoms or alkyl, alkoxy, alkylthio or trifluoromethyl rad... | 09/22/1981 |
| 4276292 | Triazolobenzoxazin-4-ones New triazolobenzoxazinones are described as well as the use thereof as anti-allergenic agents.... | 06/30/1981 |
| 4254121 | 3-Oxo-5H-pyrimido[2,1-c][1,4 ]benzoxazines 3-Oxo-5H-pyrimido[2,1-c][1,4]benzoxazine derivatives, optionally substituted with a hydroxymethyl, carboxy or loweer alkoxycarbonyl at position 1 and optionally substituted at positions 8 or 9, with a lowr alkyl or halo are disclosed. The derivatives are ... | 03/03/1981 |
| 4254118 | 1-Oxo-5H-pyrimido[2,1-c][1,4]benzthiazine-2-carboxylic acid esters This invention discloses novel 1-oxo-5H-pyrimido[2,1-c][1,4]benzoxa(or thia)zine-2-carboxylic acid lower alkyl esters, derivatives thereof, process for their preparation, pharmaceutical compositions thereof and methods for using the compounds. The compoun... | 03/03/1981 |
| 4224323 | Method for lowering serum uric acid A method for lowering serum uric acid is disclosed which comprises administering to a human for its uricosuric activity a pharmaceutical composition comprising 7-chloro-2-methyl-3,3a-dihydro-2H,9H-isoxazolo (3,2-b) (1,3)-benzoxazin-9-one. 7-chloro-2-methy... | 09/23/1980 |
| 4207318 | Novel imidazobenzoxazines Novel imidazobenzoxazines of the formula ##STR1## wherein X is selected from the group consisting of hydrogen, halogen and alkyl of 1 to 5 carbon atoms, R is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, and an equival... | 06/10/1980 |
| 4145419 | Novel imidazobenzoxazines Novel imidazobenzoxazines of the formula ##STR1## wherein X is selected from the group consisting of hydrogen, nitro, NH2 and a protected amino Z is selected from the group consisting of --COOR, and ##STR2## R is selected from th... | 03/20/1979 |
| 4134974 | Imidazo[5,1-c][1,4]benzoxazin-1-one Cyclic derivatives of 1,4-benzoxazine and 1,4-benzothiazine are disclosd, such as, for instance, 1H,2,3,3a,4-tetrahydro-2-carbamoylmethyl-imidazo[5,1-c][1,4]benzoxazin-1-o ne and 1H,2,3,3a,4-tetrahydro-2-carbamoylmethyl-8-chloro-imidazo[5,1-c][1,4]ben... | 01/16/1979 |
| 4035495 | Pyrrolobenzoxazines, pyrrolobenzothiazines and process therefor 4H-Pyrrolo[2,1-c][1,4]benzoxazines and 4H-pyrrolo[2,1-c]-[1,4]benzothiazines characterized by having an alkylamine substituent at position 4 are disclosed. The compounds are characterized further by having an alkyl substituent on the same carbon atom... | 07/12/1977 |
| 4012511 | Oxazinoindole derivatives useful as antidepressants Oxazinoindole derivatives characterized by having an amino(lower)alkyl radical attached to the 1 position of a 1H-1,4-oxazino[4,3-a]indole nucleus are disclosed. The amino portion of the amino(lower)alkyl radical may be further substituted with one or two... | 03/15/1977 |
| 3984548 | Substituted pyrido[1,2,3,-de]-1,4-benzoxazines as bactericides Anti-microbial agents which are 2,3-dihydro-3-substituted-7-oxo-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxy lic acids are prepared by condensation of benzoxazines with ethoxymethylene malonate esters followed by ring closure with poly phosphoric acid and ... | 10/05/1976 |
