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"What, sir, would you make a ship sail against the wind and currents by lighting a bonfire under her deck? I pray you, excuse me, I have not the time to listen to such nonsense."
Napoleon Bonaparte ; When told of the Robert Fulton steamboat
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| Application No. | Application Title | Issue Date |
| 20120129893 | Inhibition Of Raf Kinase Using Substituted Heterocyclic Ureas Methods of treating tumors mediated by raf kinase, with substituted urea compounds, and such compounds per se.... | 05/24/2012 |
| 20120130080 | PROCESS FOR PREPARING 2-AMINO-5-CYANOBENZOIC ACID DERIVATIVES Disclosed is a method for preparing a compound of Formula 1 comprising contacting a compound of Formula 2 with a metal cyanide reagent, a copper(I) salt reagent, an iodide salt reagent and at least one compound of Formula 3 05/24/2012 | |
| 20120129844 | N-[5-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-3-YL]-4-(3,4-DIMETHYLPIPERAZIN-1-YL)BENZAMIDE AND SALTS THEREOF There is provided a compound of formula (I): or a pharmaceutically acceptable salt thereof. There are also provided processes for the manufacture of a compound of Formula 1, and the use of a compound of Formu... | 05/24/2012 |
| 20120108817 | ACETYL PYRROLIDINYL INDOLE DERIVATIVE The present invention relates to compounds, which are useful for treatment and/or prevention of diabetes mellitus, diabetes mellitus complications or obesity, since the compounds have glucokinase-activating effects, and are presented in Formula (I): wherein R1 05/03/2012 | |
| 20120110702 | Pesticidal Compositions and Processes Related Thereto This document discloses molecules having the following formula (“Formula One”): and processes related thereto.... | 05/03/2012 |
| 20120108635 | Insecticidal Arylpyrrolines The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as an insecticide. ... | 05/03/2012 |
| 20120071517 | 2-PYRIDINYLETHYLCARBOXAMIDE DERIVATIVES AND THEIR USE AS FUNGICIDES The invention discloses a compound of general formula (I) and a process for preparing this compound. The invention discloses a fungicidal composition comprising a compound of general formula (I) and a method ... | 03/22/2012 |
| 20120071325 | USE OF AMIDE COMPOUND FOR PROMOTING PLANT ROOT GROWTH The present invention relates to use of amide compounds for promoting root growth of plants.... | 03/22/2012 |
| 20120071516 | COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Described herein are compounds and pharmaceutical compositions containing such compounds, which modulate the activity of store-operated calcium (SOC) channels. Also described herein are methods of using such SOC channel modulators, alone and in combination with other co... | 03/22/2012 |
| 20120053173 | HETEROCYCLIC COMPOUND Provision of a prophylactic or therapeutic agent for diabetes, which has superior efficacy. A compound represented by the formula: wherein each symbol is as described in the spec... | 03/01/2012 |
| 20120053150 | N-PYRAZOLYL CARBOXAMIDES AS CRAC CHANNEL INIHIBITORS The present invention relates to amide compounds, processes for their preparation, pharmaceutical compositions containing these compounds and to their use in the treatment of disorders, conditions or disorders such as allergic disorders, inflammatory disorders and disor... | 03/01/2012 |
| 20120046317 | NOVEL HETEROCYCLIC COMPOUNDS The present invention relates to a new class of heterocyclic compounds and pharmaceutically acceptable salts thereof, process for preparing the same, pharmaceutical composition containing these compounds and to their use in treatment of diseases caused due to formation ... | 02/23/2012 |
| 20120046301 | Substituted Cyclic Carboxamide and Urea Derivatives as Ligands of the Vanilloid Receptor Substituted cyclic carboxamide and urea compounds, a process for their preparation, pharmaceutical compositions containing these compounds, and the use of these compounds for the treatment and/or inhibition of pain and other conditions mediated by the vanilloid receptor... | 02/23/2012 |
| 20120040950 | ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE The present invention relates to compounds useful as inhibitors of PI3K, particularly of PI3Kγ. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods of using the compositions in the treatment of various disease, con... | 02/16/2012 |
| 20120035217 | Bis Aromatic Compounds for Use as LTC4 Synthase Inhibitors There is provided compounds of formula I, wherein Y, ring A, D1, D2a, D2b, D3, L1, Y1, L2 and Y2 have meanings given in ... | 02/09/2012 |
| 20120035168 | N-((6-AMINO-PYRIDIN-3-YL)METHYL)-HETEROARYL-CARBOXAMIDES The invention relates to compound of the formula I in which the substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments ... | 02/09/2012 |
| 20120029023 | HETEROCYCLES SUBSTITUTED PYRIDINE DERIVATIVES AND ANTIFUNGAL AGENT CONTAINING THEREOF An object of the present invention is to provide an antifungal agent which has excellent antifungal effects and is superior in terms of its physical properties, safety and metabolic stability. According to the present invention, there is disclosed a compound represented... | 02/02/2012 |
| 20120028938 | PYRAZOLE COMPOUNDS AS CRTH2 ANTAGONISTS The present invention relates to pyrazole compounds of formula (I) and pharmaceutically acceptable salts thereof having CRTH2-activity, wherein W, L1, L2, X, L3, Y, R1 | |
| 20120022058 | 4,5-DIHYDRO-1H-PYRAZOLE COMPOUNDS AND THEIR PHARMACEUTICAL USES Mineralocorticoid receptor antagonists (MRa), pharmaceutical compositions containing such inhibitors and the use of such inhibitors to treat, for example, diabetic nephropathy and hypertension in mammals, including humans.... | 01/26/2012 |
| 20120015980 | ANTHRANILIC DIAMIDE DERIVATIVES The present invention relates to novel anthranilic acid derivatives of the general formula (I) in which R1, R2, R3, R4, R5, R6, A, Q and n hav... | 01/19/2012 |
| 20120010249 | Anthranilic diamide derivatives having cyclic side-chains The present invention relates to novel anthranilic diamide derivatives of the general formula (I) in which R1, R2, R3, R4, R5, R6, A, Q and n ... | 01/12/2012 |
| 20120010182 | Chemical Compounds The invention relates to sulfonamide derivatives, to their use in medicine, to compositions containing them, to processes for their preparation and to intermediates used in such processes. More particularly the invention relates to new sulf... | 01/12/2012 |
| 20120010250 | Anthranilamide derivatives as pesticides The present invention relates to novel anthranilamide derivatives of the general formula (I)
| |
| 20120004227 | CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM The present invention discloses novel cyclohexane derivatives having NPY Y5 receptor antagonistic activity. Specifically, the present invention discloses a compound represented by the formula (I), or a pharmaceutically acceptable salt or a solvate thereof: 01/05/2012 | |
| 20120004244 | Bis Aromatic Compounds for Use as LTC4 Synthase Inhibitors There is provided compounds of formula I, wherein E1, E2a, E2b, E2c, E4, D1, D2, D3, L1, Y1, L | |
| 20110319430 | FUNGICIDAL PYRAZOLES Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein
| |
| 20110312974 | HETEROARYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS Described herein are compounds that are antagonists of PGD2 receptors. Also described are pharmaceutical compositions and medicaments that include the compounds described herein, as well as methods of using such antagonists of PGD2 receptors, alone... | 12/22/2011 |
| 20110312939 | NEW CHEMICAL COMPOUNDS The present invention relates to new compounds of general formula (I), wherein the groups R1 to R3, X1, X2, X3 and L1 are defined as in claim 1, which are suitable for the treatment of diseases cha... | 12/22/2011 |
| 20110312953 | ANTHRANILIC ACID DERIVATIVES The present invention relates to novel anthranilic acid derivatives of the general formula (I) in which R1, R2, R3, R4, R5, Qx, A, Qy and n have the mean... | 12/22/2011 |
| 20110312963 | P38 MAP KINASE INHIBITORS The present disclosure relates to compounds of formula (I): which are inhibitors of p38 mitogen-activated protein kinase enzymes, particularly the alpha and gamma kinase sub-types thereof, and their use in th... | 12/22/2011 |
| 20110306645 | Novel ortho-substituted arylamide derivatives The present invention relates to novel ortho-substituted arylamide derivatives of the general formula (I) in which R1, R3, R4, R5, Qx, A, Qy, X, L and n have the me... | 12/15/2011 |
| 20110306644 | METALLOENZYME INHIBITOR COMPOUNDS The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.... | 12/15/2011 |
| 20110301034 | ISOTHIAZOLE AND PYRAZOLE DERIVATIVES FOR USE AS PLANT GROWTH REGULATORS The present invention relates to isothiazole and pyrazole compounds of formula (I) having plant growth regulating properties, to agricultural compositions comprising them, and to the use of said compounds for regulating plant growth. ... | 12/08/2011 |
| 20110301161 | BENZIMIDAZOLE INHIBITORS OF LEUKOTRIENE PRODUCTION The present invention relates to compounds of formula (I): and pharmaceutically acceptable salt thereof, wherein R1-R7 are as defined herein. The invention also relates to pharmaceutical... | 12/08/2011 |
| 20110294840 | HYDRAZIDE COMPOUND AND USE OF THE SAME IN PEST CONTROL There is provided a hydrazide compound having a controlling effect on pests represented by the formula (1): wherein, G is a 5-membered heterocyclic group, M is an oxygen atom or a sulfur atom, Q1, Q2, Q3 and Q4 is independentl... | 12/01/2011 |
| 20110294854 | SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS The present application relates to calcium channel inhibitors containing compounds of formula (I) wherein a, R1, R2, R3, and R4 are as defined in the specification.... | 12/01/2011 |
| 20110294812 | P38 MAP KINASE INHIBITORS The invention relates to compounds of formula (I): or a pharmaceutically acceptable salt thereof, including all stereoisomers, tautomers and isotopic derivatives thereof, which are inhibitors of p38 mitogen-a... | 12/01/2011 |
| 20110275676 | Triazole-substituted anthranilamides as pesticides The present invention constitutes new, triazole-substituted anthranilamides of the general formula (I), —in which R1, R2, R3, R4, R5, R6, Q,... | 11/10/2011 |
| 20110275797 | N-ACYL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF An N-acyl anthranilic acid derivative represented by general formula (1) or a salt thereof is useful for prevention or treatment of diseases associated with excessive production of collagen. (In the formula, R1 represents a carboxyl group or the like; R2... | 11/10/2011 |
| 20110275625 | Heteroaryl Diamide Compounds Useful as MMP-13 Inhibitors Disclosed are compounds and compositions of the formula (I) as described herein which are inhibitors of MMP-13. Also disclosed are methods of using and making compounds of the formula (I). ... | 11/10/2011 |
