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Patent No. 6049912

Mountable Printable Placard With Headband

A resilient headband in a shape for being mounted on the head of the user. The headband is equipped with a longitudinal slotted member for holding a placard.

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Class 546/169 - Acyclic nitrogen bonded directly to the -C(=X)- group


Subclass of Class 546 - Organic compounds -- part of the class 532-570 series
Definition: Compound in which acyclic nitrogen is bonded directly to
No. of applications: 183
Last issue date: 05/03/2012


1          
Application No.Application TitleIssue Date
20120108606Carboxamide, Sulfonamide and Amine Compounds and Methods for Using The Same
Disclosed are carboxamide, sulfonamide and amine compounds, as well as pharmaceutical compositions and methods of use. One embodiment is a compound having the structure

in which R1, R2, ...

05/03/2012
20120071502Novel phenoxyisobutyric acid compounds and methods for synthesis
The present invention provides a process for the synthesis of substituted phenoxymethylpropionic acid and related compounds. The compounds are useful for inhibiting the formation of AGEs (Advanced Glycation End Products)....
03/22/2012
20120053204Substituted quinoline-3-carboxamides as KCNQ2/3 modulators
The invention relates to substituted quinoline-3-carboxamides, to pharmaceutical compositions containing these compounds and also to these compounds for use in the treatment and/or prophylaxis of pain and further diseases and/or disorders....
03/01/2012
20120053148INHIBITORS OF HEPATITIS C VIRUS
The present application includes novel inhibitors of HCV, compositions containing such compounds, therapeutic methods that include the administration of such compounds....
03/01/2012
20120028938PYRAZOLE COMPOUNDS AS CRTH2 ANTAGONISTS
The present invention relates to pyrazole compounds of formula (I) and pharmaceutically acceptable salts thereof having CRTH2-activity,

wherein W, L1, L2, X, L3, Y, R1

02/02/2012
20120022057BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYGLYCEROL ACYLTRANSFERASE
The present invention relates to novel heterocyclic compounds as diacylglycerol acyltransferase (“DGAT”) inhibitors, pharmaceutical compositions comprising the heterocyclic compounds and the use of the compounds for treating or preventing a cardiovascular disease, a...
01/26/2012
20120015978THERAPEUTIC AGENTS FOR OCULAR HYPERTENSION
This invention provides well defined 6-alkyl or hydroxyalkyl-1-naphthamide or quinoline compounds for treating glaucoma or ocular hypertension....
01/19/2012
20120004227CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM
The present invention discloses novel cyclohexane derivatives having NPY Y5 receptor antagonistic activity. Specifically, the present invention discloses a compound represented by the formula (I), or a pharmaceutically acceptable salt or a solvate thereof:

01/05/2012

20110306611Transcription factor modulating compounds and methods of use thereof
Substituted benzoimidazole compounds useful as anti-infectives that decrease resistance, virulence, or growth of microbes are provided. Methods of making and using substituted benzoimidazole compounds, as well as pharmaceutical preparations thereof, in, e.g., reducing a...
12/15/2011
20110306542NOVEL GLP-1 RECEPTOR STABILIZERS AND MODULATORS
Compounds that bind the glucagon-like peptide 1 receptor (GLP-1) receptor are provided including compounds which are modulators of the GLP-1 receptors and compounds which are capable of inducing a stabilizing effect on the receptor for use in structural analyses of the ...
12/15/2011
20110294819Hepatitis C Virus Inhibitors
The present disclosure is generally directed to antiviral compounds, and more specifically directed to compounds which can inhibit the function of the NS5A protein encoded by Hepatitis C virus (HCV), compositions comprising such compounds, and methods for inhibiting the...
12/01/2011
20110286922IMAGING AND RADIOTHERAPY METHODS
The present invention relates to in vivo imaging and radiotherapeutic methods and agents which target the enzyme aldehyde dehydrogenase (ALDH) and that are suitable for the in vivo imaging of tumours and treatment of cancer....
11/24/2011
20110288117SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF
This invention provides compounds of formula (I):

    • wherein R1a, R1,...
11/24/2011
20110263564PYRIDINE, BICYCLIC PYRIDINE AND RELATED ANALOGS AS SIRTUIN MODULATORS
Provided herein are novel sirtuin-modulating compounds and methods of use thereof. The sirtuin-modulating compounds may be used for increasing the lifespan of a cell, and treating and/or preventing a wide variety of diseases and disorders including, for example, disease...
10/27/2011
20110245226PIPERIDINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY
The present application describes substituted piperidinyl modulators of MIP-1α or CCR-1 or stereoisomers or pharmaceutically acceptable salts thereof. In addition, methods of treating and preventing inflammatory diseases such as asthma and allergic diseases, as well as...
10/06/2011
20110207737SUBSTITUTED BICYCLIC AMINES FOR THE TREATMENT OF DIABETES
Described herein are substituted bicyclic amines. In particular, described herein are substituted bicyclic amines that are effective as antagonists of SSTR5 and useful for the treatment, control or prevention of disorders responsive to antagonism of SSTR5, such as type ...
08/25/2011
20110207773NOVEL PHENYL-QUINOLINE-CARBOXYLIC ACID PYRIDINE DERIVATIVES USEFUL AS MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
This invention relates to novel phenyl-quinoline-carboxylic acid pyridine derivatives, which are found to be modulators of the nicotinic acetylcholine receptors. Due to their pharmacological profile the compounds of the invention may be useful for the treatment of disea...
08/25/2011
20110201643NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS
Compounds of a certain formula (I) wherein R1, R2, R3, X, Y, r, s, t, u and v have the meanings as defined in the specification, and the salts, solvates and hydrates thereof are novel effective HDAC 6 inhibitors.

...

08/18/2011
20110178092HIV-1 Protease Inhibitors
Described are novel protease inhibitors and methods for using said protease inhibitors in the treatment of human immunodeficiency virus (HIV) infection....
07/21/2011
20110172429STAT3 INHIBITOR CONTAINING QUINOLINECARBOXAMIDE DERIVATIVE AS ACTIVE INGREDIENT
The present invention provides a STATS inhibitor containing as an active ingredient, a quinolinecarboxamide derivative represented by the formula (I) (in the formula, W represents a bond or an alkylene chain; X represents O, S, or NR34; and R1 to R...
07/14/2011
201101246362-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS
The invention relates to novel 2-aza-bicyclo[3.1.0]hexane derivatives of Formula (I) wherein A, B, n and R1 are as described in the description, and to the use of such compounds, or of pharmaceutically acceptable salts of such compounds, as medicaments, espec...
05/26/2011
20110112058NOVEL MODULATORS OF CALCIUM RELEASE-ACTIVATED CALCIUM CHANNEL AND METHODS FOR TREATMENT OF NON-SMALL CELL LUNG CANCER
Disclosed are novel calcium release-activated calcium (CRAC) channel inhibitors, methods for preparing them, pharmaceutical compositions containing them, and methods of treatment using them. The present disclosure also relates to methods for treating non-small cell lung...
05/12/2011
20110092481QUINOLINE OR ISOQUINOLINE SUBSTITUTED P2X7 ANTAGONISTS
The present invention is related to novel compounds of formula (I) having P2X7 antagonistic properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment or prophylaxis of diseases ass...
04/21/2011
20110046177THERAPEUTIC QUINOLINE AND NAPHTHALENE DERIVATIVES
Disclosed herein is a stable compound having a structure formula (I): therapeutic methods, compositions, and medicaments related thereto are also disclosed.

...

02/24/2011
20110046110QUINOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS
Provided herein are novel sirtuin-modulating compounds and methods of use thereof. The sirtuin-modulating compounds may be used for increasing the lifespan of a cell, and treating and/or preventing a wide variety of diseases and disorders including, for example, disease...
02/24/2011
20110044899LABELLED ANALOGUES OF HALOBENZAMIDES AS MULTIMODAL RADIOPHARMACEUTICALS AND THEIR PRECURSORS
A compound of formula (I): in which R1 represents a hydrogen atom, an optionally labelled halogen, a radionuclide or a Sn[(C1-C4)alkyl]3 group, Ar represents an aryl group or a heteroaryl group, R9 represents a hydr...
02/24/2011
20110039857PIPERIDINE AND PYROOLIDINE COMPOUNDS
The invention relates to piperidine and pyrrolidine compounds of formula (I)

wherein A, B, n and X are as described in the description; to pharmaceutically acceptable salts thereof, and to the use of such com...

02/17/2011
20110021540Bis-(Sulfonylamino) Derivatives in Therapy 066
The invention provides compounds of formula wherein R1, R3, L1, L2, G1, G2, A and m are as defined in the specification and optical isomers, racemates and tautomers thereof, and pharmaceutically acceptabl...
01/27/2011
20110021528NOVEL HYDROXAMATES AS THERAPEUTIC AGENTS
The present invention is directed to certain hydroxamate derivatives that are useful in the treatment of hepatitis C. These compounds are also inhibitors of histone deacetylase and are therefore useful in the treatment of diseases associated with histone deacetylase act...
01/27/2011
20110021514AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME
Compounds are disclosed that have a formula represented by the following: The compounds may be prepared as pharmaceutical compositions, and may be used for the prevention and treatment of a variety of conditions in mammals including humans, including by way of non-limit...
01/27/2011
20110021407USE OF METAL COMPLEX COMPOUNDS AS OXIDATION CATALYSTS
The present invention relates to the use of metal complex compounds having hydrazide ligands as oxidation catalysts. Further aspects of the invention are formulations comprising such metal complex compounds, novel metal complex compounds and novel ligands. The metal com...
01/27/2011
20100311790AMIDE COMPOUNDS AND PLANT DISEASE CONTROLLING METHOD USING SAME
The object of the present invention is to provide a compound having excellent controlling effect on plant diseases. An amide compound represented by the following formula (I) has excellent controlling effect on plant diseases:

12/09/2010

20100305154Prolyl Hydroxylase Inhibitors
The invention described herein relates to certain quinoline-8-carboxamide derivatives of formula (I)

which are antagonists of HIF prolyl hydroxylases and are useful for treating diseases benefiting from the i...

12/02/2010
20100267769Substituted Bicyclocarboxyamide Compounds
This invention provides a compound of the formula

These compounds are useful for the treatment of disease conditions caused by overactivation of the VR1 receptor such as pain, or the like in mammal. This inve...

10/21/2010
20100261675FUNGICIDAL COMPOSITION CONTAINING ACID AMIDE DERIVATIVE
Conventional many fungicidal compositions have had practical problems such that either a preventive effect or a curing effect is inadequate, the residual effect tends to be inadequate, or the controlling effect against plant diseases tends to be inadequate depending upo...
10/14/2010
20100255992Soluble Liquid Formulations of Quinclorac Ammonium Salts
The present invention relates to novel soluble liquid (SL) formulations comprising
  • A) quinclorac ammonium salts of formula I

    10/07/2010
20100233106SMALL-MOLECULE MODULATORS OF MELANIN EXPRESSION
The present invention relates to small molecule modulators of melanin expression and methods of making the small molecules. Also disclosed are methods of increasing pigmentation in a cell which involve providing compounds of the present invention and contacting a cell w...
09/16/2010
20100234424DERIVATIVES OF N-PHENYL(PIPERIDINE-2-YL) METHYL BENZAMIDE PREPARATION METHOD THEREOF AND APPLICATIONS OF SAME IN THERAPEUTICS
Compounds of formula (I) as defined herein:

are useful for treating behavioral disorders associated with dementia, psychoses, in particular schizophrenia (deficient form and productive form) and acute or chro...

09/16/2010
20100227884AMIDE COMPOUNDS AND PLANT DISEASE CONTROLLING METHOD USING SAME
The object of the present invention is to provide a compound having excellent controlling effect on plant diseases. An amide compound represented by the following formula (I) has excellent controlling effect on plant diseases:

09/09/2010

20100216803ORNITHINE DERIVATIVE
Provided is a compound which is useful as a therapeutic agent for chronic renal insufficiency and a therapeutic agent for diabetic nephropathy.

The present inventors have made extensive studies on an ornithine derivative having an antagonis...

08/26/2010
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