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Patent No. 5307162

Cloaking System Using Optoelectronically Controlled Camouflage

A Cloaking System designed to operate in the visible light spectrum, utilizes optoelectronics and/or photonic components to conceal an object within it.

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Class 514/451 - The hetero ring is six-membered


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the hetero ring is six-membered.
No. of applications: 51
Last issue date: 05/24/2012


1    
Application No.Application TitleIssue Date
20120129833CYCLIC KETOENOLS FOR THERAPY
The invention relates to 5′-biphenyl-substituted cyclic ketoenols for therapeutic purposes, to pharmaceutical compositions and to their use in therapy, in particular for the prophylaxis and therapy of diabetes, obesity, hyperlipidaemia, fatty livers and of disorders o...
05/24/2012
20120129894Alkoxy Compounds for Disease Treatment
The present invention relates generally to compositions and methods for treating neurodegenerative diseases and disorders, particularly ophthalmic diseases and disorders. Provided herein are alkoxyl derivative compounds and pharmaceutical compositions comprising these c...
05/24/2012
20120107229NOVEL NANO-PROBES FOR MOLECULAR IMAGING AND TARGETED THERAPY OF DISEASES
The present inventions relate to compositions and methods for imaging and treating atherosclerotic diseases, pathogen infections, and tumors by administering actively targeting magnetic nanoparticles. In particular, the present inventions provide new types of targeting ...
05/03/2012
20120053208Curcumin Analogs as Dual JAK2/STAT3 Inhibitors and Methods of Making and Using the Same
Curcumin analogues and methods of making and using the same are disclosed....
03/01/2012
20120015807Trifluromethoxyphenyl-Substituted Tetramic Acid Derivatives Pesticides and/or Herbicides
The present invention relates to novel trifluoromethoxyphenyl-substituted tetramic acid derivatives of the formula (I),

in which
J, X, Y, A, B, D and G have the meanings given above,
to a number o...

01/19/2012
20110281930Use of 2-Aryl-5-heterocyclyl-cyclohexane-1,3-dione Compounds as Insecticides, Acaricides, and/ or Fungicides
The present invention relates to the use of compounds of Formula (I) wherein R1, R2, R3, R4, R5, R6, R7, R8, X and G have the meanings given above as insecticides and/or acaricides a...
11/17/2011
20110269713BRYOSTATIN ANALOGUES AND METHODS OF MAKING AND USING THEREOF
Described herein are tricyclic macrolactones. The macrolactones have a high binding affinity for PKC. The compounds described herein can be used in a number of therapeutic applications including cancer and Alzheimer's prevention and treatment. The compounds described he...
11/03/2011
20110257255COMPOSITION AND METHOD FOR INHIBITION OF NERVE TRANSMISSION
The presently claimed and disclosed invention(s) provides a therapeutically effective composition and method of inhibiting nerve cell transmission. In a preferred embodiment of the presently claimed and disclosed invention(s), the treatment of neuropathic pain utilizing...
10/20/2011
20110237592SUBSTITUTED AMIDO PHENOXYBENZAMIDES
The present invention relates to substituted amido phenoxybenzamide compounds of general formula (I):

in which A, R1, R2, R3, R4, R5, R6, R7, R8, R9 and n are as defined in the claims, to pharmaceutical compo...

09/29/2011
20110206764FORMULATIONS FOR ENHANCED BIOAVAILABILITY OF ORALLY ADMINISTERED POLAR AGENTS
A composition is described having improved oral permeability of polar agents such as neuraminidase inhibitors. The composition includes one or more polar agents and one or more permeability enhancers such that the composition increases the amount of the polar agent capa...
08/25/2011
20110144191COMPOSITIONS COMPRISING TERPENE COMPOUNDS FOR TREATING NEGATIVE SENSORY PHENOMENA
Compositions comprising terpene compounds for the treatment of negative sensory phenomena (NSP). Negative sensory phenomena is characterized by a decreased ability to sense light touch, pin prick, vibration, temperature, pain and/or reduced proprioception. The terpene c...
06/16/2011
20110086908USE OF PHOSPHATASE INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES
Provided are novel a target and drugs in the treatment of neurological disorders related to amyloid beta pathology/amyloidosis. More specifically, the use of phosphatase inhibitors for the treatment of brain impairments mediated by Aβ-oligomers is described....
04/14/2011
20110046212USE OF OLEUROPEIN AND DERIVATIVES IN THE TREATMENT OF TYPE 2 DIABETES MELLITUS AND PATHOLOGIES ASSOCIATED WITH PROTEIN AGGREGATION PHENOMENA
This invention relates to the use of oleuropein, specifically oleuropein in non-glycated form, and its derivatives in the treatment of type 2 diabetes mellitus. Furthermore, this invention relates to the use of oleuropein, specifically oleuropein in non-glycated form, a...
02/24/2011
20100261772Cycloalkylidene Compounds As Selective Estrogen Receptor Modulators
The present invention relates to compounds of formula (I) with a variety of therapeutic uses, more particularly the substituted cyclic alkylidene compounds are useful for selective estrogen receptor modulation.

...

10/14/2010
20100256156HETEROCYCLIC COMPOUND
The present invention provides a heterocyclic compound represented by the following formula (I), which has a glucagon antagonistic action and is useful for the prophylaxis or treatment of diabetes and the like, a compound represented by

10/07/2010
20100226864ALKYL-SUBSTITUTED TETRAHYDROPYRANS AS FLAVORING SUBSTANCES
The present invention relates to alkyl-substituted tetrahydropyrans, mixtures containing these alkyl-substituted tetrahydropyrans, their respective use and corresponding flavored products....
09/09/2010
20100197684SUBSTITUTED HETEROCYCLIC COMPOUNDS
The present invention relates to novel heterocyclic compounds and to their use in the treatment of various disease states, including cardiovascular diseases and diabetes. In particular embodiments, the structure of the compounds is given by Formula (I):

08/05/2010

20100076068Aminoalcohol Derivatives and Their Therapeutic Use
A compound of formula (1) Including pharmaceutically acceptable salts thereof, wherein: R1 is aryl or heteroaryl optionally substituted with R8; R2 is H or alkyl or CH2 (when forming part of a ring with R3, R4 ...
03/25/2010
20100062065PHARMACEUTICAL COMPOSITION CONTAINING NAPHTHOQUINONE-BASED COMPOUND FOR INTESTINE DELIVERY SYSTEM
Provided is an oral pharmaceutical composition with improved bioavailability and pharmacokinetic properties of a drug, by increasing a bioabsorption rate and an in vivo retention time of an active ingredient via intestine-targeted formulation of a particular naphthoquin...
03/11/2010
20100048572NAPHTHALENONE COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF
Compounds of Formula I and Formula II are useful as inhibitors of HIF prolyl hydroxylases. Compounds of Formula I and Formula II have the following structures:

where the definitions of the variables are provi...

02/25/2010
20100048687USE OF PHOSPHATASE INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES
Provided are novel a target and drugs in the treatment of neurological disorders related to amyloid beta pathology/amyloidosis. More specifically, the use of phosphatase inhibitors for the treatment of brain impairments mediated by Aβ-oligomers is described....
02/25/2010
20100028460IMPROVEMENTS IN RELATION TO CANCER THERAPY
The present invention relates to an improved assay for identifying compounds that may be of use in conjunction with cancer chemotherapeutic agents and anti-proliferative agents, to improve efficacy of such agents and/or render effective compounds with relatively little ...
02/04/2010
20090269427HERBAL COMPOSITION FOR INFLAMMATORY DISORDERS
This invention relates to a novel herbal composition comprising an extract of flowering and fruiting heads of the plant, Sphaeranthus indicus. The said extract of Sphaeranthus indicus contains a compound, 3a-hydroxy-5a,9-dimethyl-3-methylene-3a,4,5,5a,6,7,...
10/29/2009
20090270494Salts of Dihydroxyanthraquinone Carboxylic Acids and Their Therapeutic Use
A compound of general formula (I): wherein Xi is H or COR1 and X2 is H or COR2 but X1 and X2 are not both H; R1 and R2 are the same or different and are each C1-4 alkyl substituted w...
10/29/2009
20090099253Internally Masked Neopentyl Sulfonyl Ester Cyclization Release Prodrugs of Acamprosate, Compositions Thereof, and Methods of Use
Internally masked neopentyl sulfonyl ester prodrugs of acamprosate, pharmaceutical compositions comprising such prodrugs, and methods of using such prodrugs and compositions thereof for treating diseases are disclosed. In particular, acamprosate prodrugs exhibiting enha...
04/16/2009
20080234258Dihydroxyanthraquinones and Their Use
A compound of formula (1)

wherein X is H or —OCR1 and Y is H or —OCR2, provided that X and Y are not both H; and R is CH2OR9, CONR11R12, C...

09/25/2008
20080226716AMINO ACID CONJUGATES PROVIDING FOR SUSTAINED SYSTEMIC CONCENTRATION OF GABA ANALOGUES
Compounds that provide for sustained systemic concentrations of GABA analogs following oral administration to animals are disclosed. Pharmaceutical compositions including, and methods using, such compounds are also disclosed....
09/18/2008
20080194673Environment-Friendly Pollution-Proof Agent
The present invention relates to an environmental friendly antifouling agent, and more particularly, to a novel Sargassum-derived antifouling agent which is harmless to environment, has antifouling activity against a broad spectrum of fouling organisms, can be ex...
08/14/2008
20080188548Cyclic ether vitamin D3 compounds, 1alpha(OH)3-epi-vitamin D3 compounds and uses thereof
Novel cyclic ether vitamin D3 compounds having a cyclic ether side chain are disclosed. These compounds were first identified as metabolites of 3-epi vitamin D3 produced via a tissue-specific metabolic pathway which catalyzes the formation of a cyclic ether structure. A...
08/07/2008
20080138297Pyran derivatives, process of preparation and use thereof in perfumery and flavouring
Pyran derivatives of general formula (I)

wherein

    • Y is a 5...
06/12/2008
20080085893MATRIX METALLOPROTEASE INHIBITORS
The present invention relates to compounds of Formula I, wherein R1, R2, R3, R4, R5, R6, and R7 are defined in the specification. In addition, the present invention relates to methods treating disorders related to matrix metalloproteases. More particularly, the comp...
04/10/2008
20080039506Aminoalcohol Derivatives
The present invention relates to a compound of the formula [I]: wherein (a), in which —Y—, R4, R5 and R6 are4 R5 each as defined in the description, etc., R1 is hydrogen, halogen, lower alkyl, hydroxy...
02/14/2008
20080027096Novel Pharmaceutical Compositions
The invention provides compounds of formula (I) or a pharmaceutically acceptable ester, amide, solvate or salt thereof, including a salt of such an ester or amide, and a solvate of such an ester, amide or salt, for use in the treatment or prophylaxis of condition mediat...
01/31/2008
20070287745Laulimalide Analogs and Uses Thereof
The present invention provides compounds having formula I:
    • and pharmaceutically acceptable derivatives thereof, whe...
12/13/2007
20070270452Novobiocin analogues as neuroprotective agents and in the treatment of autoimmune disorders
Novobiocin analogues and pharmaceutical composition containing such compounds useful for the treatment and/or prevention of neurodegenerative disorders and autoimmune disorders. ...
11/22/2007
20070249565Class of Gamma Delta T Cells Activators and Use Thereof
The present invention relates to a new class of compounds having γδ T cells activating properties of Formula (I), a composition comprising these compounds and methods for regulating an immune response in a subject comprising the step of administering these compoun...
10/25/2007
20070244187Intermediates for the Preparation of Halichondrin B
The present invention provides macrocyclic compounds, synthesis of the same and intermediates thereto. Such compounds, and compositions thereof, are useful for treating or preventing proliferative disorders Formula (F-4). ...
10/18/2007
20070238769Bone Densifying Agent Characterized By Use Of Cathepsin K Inhibitor With Pth
The present invention relates to an agent for increasing BMD characterized by use of a cathepsin K inhibitor as a bone resorption inhibitor in combination with a type of PTH as a bone formation stimulator. This agent for increasing BMD is useful for the treatment of os...
10/11/2007
20070232686Cyanoamidine P2X7 Antagonists for the Treatment of Pain
Novel cyanoamidines compounds of formula (I) and (II)

and their derivatives wherein R1-R12 are as defined in the specification act as antagonists of the P2X7 receptor. These compounds are particularly u...

10/04/2007
20070225357Formulation for Stimulating Hair Growth
The present invention is directed to a topical formulation comprising the Compound 6-[[(3S,4R)-3,4-dihydro-3-hydroxy-6-[(3-hydroxyphenyl)sulfonyl)-2,2,3-trimethyl-2H-1-benzopyran-4-yl]oxy]-2-methyl-3(2H)-pyridazinone in a formulation comprising at least one pharmaceutic...
09/27/2007
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