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Patent No. 5307162

Cloaking System Using Optoelectronically Controlled Camouflage

A Cloaking System designed to operate in the visible light spectrum, utilizes optoelectronics and/or photonic components to conceal an object within it.

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Class 514/391 - Benzene ring bonded directly to the diazole ring by nonionic bonding


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein a benzene ring is bonded directly
No. of applications: 76
Last issue date: 04/05/2012


1    
Application No.Application TitleIssue Date
20120082646Antiviral Compounds And Uses Thereof
This invention relates to: (a) compounds and salts thereof that, inter alia, inhibit HCV; (b) intermediates useful for the preparation of such compounds and salts; (c) compositions comprising such compounds and salts; (d) methods for preparing such intermediates, compou...
04/05/2012
20120083514IMIDAZOLIDINE-2,4-DIONE DERIVATIVES, AND USE THEREOF AS A CANCER DRUG
The present application relates to novel imidazolidine-2,4-dione derivatives of the general formula (I), where R1, R2, R3, R4, X, and Y are variables. Said materials have an antiproliferative activity. They are particularly us...
04/05/2012
20120083463Insecticidal and Fungicidal Active Compound Combinations
The present invention relates to active compound combinations consisting, firstly, of a known halogen-substituted derivative (component A) and, secondly, of further known pesticidally active compounds (component B), which active compound combinations are suitable for co...
04/05/2012
20120035231SPECIFIC DIARYLHYDANTOIN AND DIARYLTHIOHYDANTOIN COMPOUNDS
Compositions, such as pharmaceutical compositions, comprising specific diarylhydantoin and diarylthiohydantoin compounds, or salts or solvates thereof, are provided. Isolated and purified forms of the compounds are also described, as are unit dosage forms, compositions ...
02/09/2012
20120027879BUCCAL, POLAR AND NON-POLAR SPRAY OR CAPSULE CONTAINING DRUGS FOR TREATING METABOLIC DISORDERS
Buccal aerosol sprays or capsules using polar and non-polar solvent have now been developed which provide biologically active compounds for rapid absorption through the oral mucosa, resulting in fast onset of effect. The buccal polar compositions of the invention compri...
02/02/2012
20120015910Synergistic fungicidal active substance combinations
Novel active compound combinations comprising a carboxamide of the general formula (I) (group 1)

in which

  • A, R1, R2
01/19/2012
20110306615NOVEL IMIDAZOLIDINE DERIVATIVE AND USE THEREOF
According to the present invention, a compound represented by formula (I):

wherein Q is:

A is a hydrogen atom, a halogen atom, —ORa or a C1...

12/15/2011
20110301108MATERIALS AND METHODS FOR SENSITIZING MULTIDRUG RESISTANT CELLS
Disclosed herein are materials and methods for sensitizing multidrug resistant cancer cells that express ABCG2 and related proteins members of a family of ATP-binding transporter superfamily that mediate drug efflux found in some types of multidrug resistant caner cells...
12/08/2011
20110288079Tannate Compositions, Methods of Making and Methods of Use
Tannate compositions containing active pharmaceutical ingredients to be used for treating nausea, vomiting, pain, convulsions, and insomnia and manufacturing processes for preparing the tannate compositions....
11/24/2011
20110281811Use Of Leukotriene Inhibitors For Treating Lung Diseases In Prematurely Born Infants
The invention relates to the use of at least one leukotriene inhibitor for preparing a pharmaceutical composition for the prophylaxis and/or treatment of lung diseases, more particularly of bronchopulmonary dysplasia, in prematurely born infants. The invention further r...
11/17/2011
20110263664Inhibitors of PIM-1 Protein Kinases, Compositions and Methods for Treating Prostate Cancer
The disclosure relates to inhibitors of Pim-1 and/or Pim-2 protein kinase, to compositions comprising one or more inhibitors of Pim-1 and/or Pim-2 protein kinase, and to methods for treating cancer....
10/27/2011
20110251165DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE BETA2 ADRENERGIC RECEPTOR
The present invention provides a compound of formula (I) wherein: R1 is a group selected from —CH2OH, —NHC(O)H and R2 is a hydrogen atom; or R1 together with R2 form the group —NH—C(O)—CH═CH— wherein t...
10/13/2011
20110251166DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE BETA2 ADRENERGIC RECEPTOR
The present invention provides a compound of formula (I) wherein: R1 is a group selected from —CH2OH, —NHC(O)H and R7 is a hydrogen atom; or R1 together with R2 form the group —NH—C(O)—CH═CH— wherein t...
10/13/2011
20110230442NA CHANNELS, DISEASE, AND RELATED ASSAYS AND COMPOSITIONS
Disclosed are molecules and their synthesis, for use in blocking gated ion channels such as voltage-gated sodium channels (VGSCs) and prostate voltage sodium channels (PVSCs). These inhibitors have superior blocking efficacy, for instance in displacing the radioligand [...
09/22/2011
201102129442-OXO-1-PYRROLIDINE DERIVATIVES
This invention relates to novel 2-oxo-1-pyrrolidines, their derivatives, and pharmaceutically acceptable salts thereof. This invention also provides compositions comprising a compound of this invention and the use of such compositions in methods of treating diseases and...
09/01/2011
20110212994Small Molecule Choline Kinase Inhibitors, Screening Assays, and Methods for Safe and Effective Treatment of Neoplastic Disorders
Small molecule choline kinase inhibitors, pharmaceutical compositions thereof, and screening methods for identifying and evaluating choline kinase inhibitors are provided. Safe and effective methods for treating subjects suffering from a disorder or disease characterize...
09/01/2011
20110207718COMPOSITIONS AND METHODS FOR TREATING PSYCHIATRIC DISORDERS
Methods of treating psychiatric disorders are provided which include administration of one or more anti-epileptic agents and, optionally, one or more a psychostimulants. Also provided are pharmaceutical compositions comprising, in combination, one or more anti-epileptic...
08/25/2011
20110178134Novel phenyl-substituted imidazolidines, process for preparation thereof, medicaments comprising said compounds and use thereof
The invention relates to compounds of formula (I) wherein the groups have stated meanings, and to their physiologically compatible salts. Said compounds are suitable, for example, as anti-obesity drugs and for treating cardiometabolic syndrome....
07/21/2011
20110177944Synergistic Fungicidal Mixtures
The present invention relates to a composition, comprising a 5-amino-3-oxo-2,3-dihydro-pyrazole of the formula I as defined in the claims and the description and at least one active compound II selected from groups A) to I) in a synergistically effective amount....
07/21/2011
20110172171TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION OF BRAIN OEDEMA
The present invention relates to taurine or taurine-like substances for the prevention of brain oedema, particularly brain intramyelinic oedema and more particularly brain intramyelinic oedema induced by an anti-convulsive drug such as vigabatrin. The invention relates ...
07/14/2011
20110130391UREIDO SUBSTITUTED BENZOIC ACID COMPOUNDS AND THEIR USE FOR NONSENSE SUPPRESSION AND THE TREATMENT OF DISEASE
The invention encompasses ureido substituted benzoic acid compounds, compositions comprising the compounds and methods for treating or preventing diseases associated with nonsense mutations of mRNA by administering these compounds or compositions....
06/02/2011
20110112097Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof
The invention relates to compounds of formula (I) wherein the groups R and R′, A, D, E, G, L, p and R1 to R10 have the stated meanings and to their physiologically compatible salts. Said compounds are suitable, for example, as anti-obesity drugs.

05/12/2011
20110098323INHIBITORS OF BACTERIAL BIOFILM FORMATION
Organic compounds are described for use in inhibiting or preventing formation of bacterial biofilms....
04/28/2011
20110077581TARGETED CELLULAR DELIVERY OF NANOPARTICLES
The various embodiments of the present disclosure relate generally to compositions and methods for the targeted cellular delivery of nanoparticles. More particularly, the various embodiments of the present invention are directed to the cellular delivery of nanoparticles...
03/31/2011
20110053947Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof
The invention relates to compounds of formula (I) wherein the groups R and R′, A, D, E, G, L, p and R1 to R10 have the stated meanings and to their physiologically compatible salts. Said compounds are suitable, for example, as anti-obesity drugs.

03/03/2011
20110046154USE OF AMINOPEPTIDASE INHIBITORS OR AZAINDOLE COMPOUNDS FOR PREVENTING OR TREATING CANCEROUS METASTASES FROM EPITHELIAL ORIGIN
The invention relates to the use of a compound selected from an aminopeptidase-inhibiting compound and an azaindole compound for producing a drug for preventing or treating cancerous metastases in humans or animals....
02/24/2011
20110046185Arylchalcogenoarylalkyl-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof
The invention relates to compounds of formula (I) wherein the groups R and R′ A, D, E, G, L, p and R1 to R10 have the stated meanings and to their physiologically compatible salts. Said compounds are suitable, for example, as anti-obesity drugs.

02/24/2011
20110021573ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS
Described herein are compounds that are antagonists of PGD2 receptors. Also described are pharmaceutical compositions and medicaments that include the antagonists of PGD2 receptors described herein, as well as methods of using such antagonists of P...
01/27/2011
20100330032HETEROCYCLIC ANTIVIRAL COMPOUNDS
Compounds having the formula I wherein R1, R2, R3, R4, and R5 are as defined herein are Hepatitis C virus NS5b polymerase inhibitors. Also disclosed are compositions and methods for treating an HCV infection and inh...
12/30/2010
20100311701Pharmaceutical Co-Crystal Compositions
A pharmaceutical composition comprising a co-crystal of an API and a co-crystal former; wherein the API has at least one functional group selected from ether, thioether, alcohol, thiol, aldehyde, ketone, thioketone, nitrate ester, phosphate ester, thiophosphate ester, e...
12/09/2010
20100292187METHODS FOR TREATING HEPATITIS C
The present invention provides compounds, pharmaceutical compositions, and methods of using such compounds or compositions for treating infection by a virus, or for affecting viral IRES activity....
11/18/2010
20100279991TETRAHYDRO-CYCLOPENTYL PYRAZOLE CANNABINOID MODULATORS
This invention is directed to a tetrahydro-cyclopentyl pyrazole cannabinoid modulator compound of formula (I):

and a method for use in treating, ameliorating or preventing a cannabinoid receptor mediated synd...

11/04/2010
20100255116FUNGICIDAL COMPOSITION AND METHOD FOR CONTROLLING NOXIOUS FUNGI
A fungicidal composition is provided. A fungicidal composition comprising synergistically effective amounts of (a) a carboxylic acid amide derivative of the formula (I) or its salt: wherein B is a heterocyclic group which may be substituted; each of R1 and R<...
10/07/2010
20100247583NOVEL N-PHENYLACETAMIDE INHIBITORS OF THE ENZYME SOAT-1 AND PHARMACEUTICAL/COSMETIC COMPOSITIONS COMPRISED THEREOF
Novel N-phenylacetamide compounds of formula (I):

and cosmetic and pharmaceutical compositions containing same are useful for treating disorders of the sebaceous gland, e.g., acne, or have cosmetic applicatio...

09/30/2010
20100239668SEGMENTED PHARMACEUTICAL DOSAGE FORMS
Described is a layered or segmented controlled release pharmaceutical tablet adapted for separating one segment from another by breaking through a segment....
09/23/2010
20100234331HEXAHYDRO-CYCLOOCTYL PYRAZOLE CANNABINOID MODULATORS
This invention is directed to a hexahydro-cyclooctyl pyrazole cannabinoid modulator compound of formula (I):

and a method for use in treating, ameliorating or preventing a cannabinoid receptor mediated syndro...

09/16/2010
20100222298SPILL RESISTANT FORMULATIONS CONTAINING CLAYS
The invention relates to novel spill resistant formulations comprising either a weak base or a weak acid as the pharmaceutical ingredient, a liquid base, a clay and a water soluble cellulose ether. The clay and cellulose ether allow for a broader pH range into which the...
09/02/2010
20100222311SOLID FORMULATIONS OF CRYSTALLINE COMPOUNDS
Described herein are formulations of active pharmaceutical ingredients, where the active pharmaceutical ingredients or drugs are included in a solid suspension with one or more solid additives. The formulations described herein are useful for formulating any drug or act...
09/02/2010
20100210699IMIDAZOLIDINE DERIVATIVES, USES THEREFOR, PREPARATION THEREOF AND COMPOSITIONS COMPRISING SUCH
Compounds of formula (I):

wherein

  • X is O or S,
  • R1 is acyl, aldehyde, cycloalkyl, an o...
08/19/2010
20100210665DIARYLHYDANTOIN COMPOUNDS
The present invention relates to diarylhydantoin compounds, including diarylthiohydantoins, and methods for synthesizing them and using them in the treatment of hormone refractory prostate cancer....
08/19/2010
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