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Patent No. 5356330

Apparatus for Simulating a High Five

A self-righting hand-arm configuration which is adapted to pivot when struck by a user, thereby simulating a "high five."

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Class 514/383 - 1,2,4-triazoles (including hydrogenated)


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the five-membered hetero ring is
No. of applications: 973
Last issue date: 05/24/2012


1                      
Application No.Application TitleIssue Date
20120128750PROCESS FOR PREPARING AN AQUEOUS SUSPENSION OF AN ORGANIC PESTICIDE COMPOUND
The present invention relates to a process for preparing an aqueous suspension of an organic pesticide compound, which has a solubility in water of not more than 2 g/l at 20° C. and a melting point of not more than 110° C. and which is capable of forming at least one ...
05/24/2012
20120129901TRITERPENOID DERIVATIVES USEFUL AS ANTIPROLIFERATIVE AGENTS
Formula (I) and (II). The present invention relates to the use of a new lupane derivative of general formula (I) or (II), or a pharmaceutically acceptable salt, crystal form, complex, hydrate, or hydrolysable ester thereof, for preventing and/or inhibiting tumor growth ...
05/24/2012
20120108595PLATELET-ACTIVATING FACTOR RECEPTOR ANTAGONISTS
Cyclohexyl sulfonamide compounds which are platelet-activating factor (PAF) receptor antagonists. Said compounds may be useful, for example, for the treatment of atherosclerosis or other PAF-mediated disorders, including inflammatory, cardiovascular, and immune disorder...
05/03/2012
20120108522HDAC INHIBITORS AND HORMONE TARGETED DRUGS FOR THE TREATMENT OF CANCER
The present invention relates to the methods of treating endocrine-regulated cancers, including hormone resistant cancers, for example. More specifically, the present invention relates to a method of increasing the sensitivity of hormone resistant cancers to hormonal th...
05/03/2012
20120108570Pharmacological Treatment for Sleep Apnea
The present invention relates generally to pharmacological methods for the prevention of amelioration of sleep-related breathing disorders via administration of agents or combinations of agents that possess serotonin-related pharmacological activity....
05/03/2012
20120108635Insecticidal Arylpyrrolines
The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as an insecticide.

...

05/03/2012
20120107269THIOPHENE DERIVATIVES
Disclosed is a compound of formula (I),

wherein

    • R1
05/03/2012
20120108580Use of Fungicidal Active Substances For Controlling Mycoses on Plants of the Palm Family
The present invention relates to the use of specific fungicidal active substances, alone or in combination, for controlling mycoses in plants of the palm family and to a method for using said specific fungicidal active substances for controlling said mycoses in the fiel...
05/03/2012
20120083497Method for Combating Harmful Fungi
The present invention relates to methods, use and compositions for combating harmful fungi and bacteria in plants. More specifically, it relates to methods and compositions for controlling, preventing, or treating plant pathogens using UV filters for combating phytotoxi...
04/05/2012
20120083463Insecticidal and Fungicidal Active Compound Combinations
The present invention relates to active compound combinations consisting, firstly, of a known halogen-substituted derivative (component A) and, secondly, of further known pesticidally active compounds (component B), which active compound combinations are suitable for co...
04/05/2012
20120083494NOVEL TRIAZOLE DERIVATIVES WITH IMPROVED RECEPTOR ACTIVITY AND BIOAVAILABILITY PROPERTIES AS GHRELIN ANTAGONISTS OF GROWTH HORMONE SECRETAGOGUE RECEPTORS
The present invention provides novel triazole derivatives with improved receptor activity and bioavailability properties as ghrelin analogue ligands of growth hormone secretagogue receptors according to formula (I) that are useful in the treatment or prophylaxis of phys...
04/05/2012
20120071510Method and Composition for Treating Migraines
A method for treating migraines is disclosed. The method utilizes a rapid drug delivery system which prevents deactivation or degradation of the active agent, including small molecules and peptides being administered to a patient in need of treatment. In particular, the...
03/22/2012
20120071530AGROCHEMICAL COMPOSITION AND METHOD FOR PREPARING AND USING THE SAME
An agrochemical composition comprises an azole active ingredient and an N,N-dialkyl long chain alkylamide. The N,N-dialkyl long chain alkylamide is present in sufficient amount to prevent or inhibit the crystallization of the azole derivative during the application of t...
03/22/2012
20120053216PESTICIDAL COMPOSITIONS
Molecules having the following structure are disclosed.

Processes of using such molecules are disclosed....

03/01/2012
20120053217COMPOSITION FOR PREPARING EMULSION OR MICROEMULSION FORMULATIONS
Provided is a composition for preparing emulsion or microemulsion formulations that demonstrates favorable dilution properties without being affected by the solubilities of constituent components. The composition for preparing emulsion or microemulsion formulations cont...
03/01/2012
20120053165Novel Phenyl Imidazoles and Phenyl Triazoles As Gamma-Secretase Modulators
Compounds and pharmaceutically acceptable salts of the compounds are disclosed, wherein the compounds have the structure of Formula (I) as defined in the specification. Corresponding pharmaceutical compositions, methods of treatment, methods of synthesis, and intermedia...
03/01/2012
20120053181PYRROLIDINE-DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS
The present invention provides compounds of Formula (I), pharmaceutical compositions thereof, and method of using the same in the treatment or prevention of diseases mediated by the activation of β3-adrenoceptor.

...

03/01/2012
20120053139METHOD FOR IMPROVING PHARMACOKINETICS OF PROTEASE INHIBITORS AND PROTEASE INHIBITOR PRECURSORS
The present invention provides methods for improving the pharmacokinetics of protease inhibitors and protease inhibitor precursors and pharmaceutical composition comprising protease inhibitors or protease inhibitor precursors of formula I and a cytochrome P450 monooxige...
03/01/2012
20120045497PESTICIDAL COMBINATIONS
Stabilized liquid agrochemical compositions are provided which comprise flowable non-aqueous dispersion concentrates comprising a continuous substantially water-miscible liquid phase, a dispersed water-immiscible liquid phase, and a colloidal solid. In one embodiment, t...
02/23/2012
20120046324SMALL MOLECULE INHIBITORS OF KYNURENINE-3-MONOOXYGENASE
The present invention relates to compounds of Formula I below and their tautomers or pharmaceutically acceptable salts, compositions and methods of uses thereof.

...

02/23/2012
20120040985TRIAZOLE AND IMIDAZOLE DERIVATIVES FOR USE AS TGR5 AGONISTS IN THE TREATMENT OF DIABETES AND OBESITY
The present invention comprises TGR5 agonists of structural formula I,

wherein X, R1, R2, and R5 are defined herein, as well as N-oxides of them and pharmaceutically acceptabl...

02/16/2012
20120035165Use of fungicidal compound compositions for controlling certain rust fungi
The present invention relates to the use of a fungicidal composition comprising at least one carboxamide and at least one further compound selected from strobilurins or from triazoles, for controlling certain rust fungi, such as soy bean rust and coffee rust, in crop pr...
02/09/2012
20120035054PESTICIDE COMPOSITIONS OF MESO-SIZED PARTICLES WITH ENHANCED ACTIVITY
The present disclosure relates to pesticide compositions consisting of meso-sized particles in combination with certain adjuvants such as built-in adjuvants which are added directly to the formulation or to an aqueous dilution of the formulation such as tank-mix adjuvan...
02/09/2012
20120035230Compounds, Compositions, and Methods for the Treatment of Beta-Amyloid Diseases and Synucleinopathies
Dihydroxyaryl compounds and pharmaceutically acceptable esters, their synthesis, pharmaceutical compositions containing them, and their use in the treatment of synucleinopathies, such as observed in Parkinson's disease, and the manufacture of medicaments for such treatm...
02/09/2012
20120035125FULVIC ACID IN COMBINATION WITH FLUCONAZOLE OR AMPHOTERICIN B FOR THE TREATMENT OF FUNGAL INFECTIONS
A combination of fulvic acid or a salt, ester, or derivative thereof and an antifungal compound selected from fluconazole and amphotericin B for use in the treatment or prophylaxis of a disease or condition of the human or animal body is described. The fulvic acid can b...
02/09/2012
20120029032MATRIX-TYPE SUSTAINED RELEASE PREPARATION CONTAINING BASIC ADDITIVE
Disclosed is a matrix-type sustained release preparation containing a basic drug unstable against an acid as an active pharmaceutical ingredient, wherein the decomposition of the basic drug unstable against the acid can be prevented and therefore the pH-dependent releas...
02/02/2012
20120022021Mixtures of strobilurins with 1-methylcyclopropene
The present invention relates to mixtures comprising
    • a) a compound of the formula I

...
01/26/2012
20120020915Compounds and Methods for Treating Cancer and Diseases of the Central Nervous System
Disclosed are compounds of the general formula (I):

compositions comprising an effective amount of said compounds either alone or in combination with other chemotherapeutic agents, and methods useful for trea...

01/26/2012
20120022083SMALL MOLECULE MODULATORS OF CELL ADHESION
Compounds, particularly compounds having activity as modulators of cadherin-mediated cell adhesion having the following structure:

or a pharmaceutically acceptable salt, stereoisomer or prodrug thereof,

    01/26/2012
    20120022090NOVEL SUBSTITUTED BENZOXAZOLE, BENZIMIDAZOLE, OXAZOLOPYRIDINE AND IMIDAZOPYRIDINE DERIVATIVES AS GAMMA SECRETASE MODULATORS
    The present invention is concerned with novel substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives of Formula (I)

    wherein R1, R2, R3, R...

    01/26/2012
    20120015919THERAPIES FOR TREATING CANCER USING COMBINATIONS OF COX-2 INHIBITORS AND AROMATASE INHIBITORS OR COMBINATIONS OF COX-2 INHIBITORS AND ESTROGEN RECEPTOR ANTAGONISTS
    Described herein are compositions and methods for using these compositions in the treatment of cancer, tumors, and tumor-related disorders in a subject....
    01/19/2012
    20120015988Sulfone Compounds Which Modulate The CB2 Receptor
    Compounds which modulate the CB2 receptor are disclosed. Compounds according to the invention bind to and are agonists of the CB2 receptor, and are useful for treating inflammation. Those compounds which are agonists are additionally useful for treating pain.

    01/19/2012
    20120015993Novel Pharmaceutical Forms, and Methods of Making and Using the Same
    Crystalline salts, polymorphs, solvates, and hydrates of bicalutamide, 5-fluorouracil, donepezil, anastrozole, nelfinavir, mirtazapine, lansoprazole, and tamsulosin, or derivatives thereof are provided by the subject invention. Methods of making and using the same are a...
    01/19/2012
    20120015910Synergistic fungicidal active substance combinations
    Novel active compound combinations comprising a carboxamide of the general formula (I) (group 1)

    in which

    • A, R1, R2
    01/19/2012
    20120014962METHOD OF INHIBITING FIBROGENESIS AND TREATING FIBROTIC DISEASE
    The present invention relates to the discovery of an epigenetic relay pathway that controls hepatic stellate cell activation and the wound-healing response in fibrogenesis, including fibrogenesis of the injured liver. Methods of inhibiting fibrogenesis, including liver ...
    01/19/2012
    20120015807Trifluromethoxyphenyl-Substituted Tetramic Acid Derivatives Pesticides and/or Herbicides
    The present invention relates to novel trifluoromethoxyphenyl-substituted tetramic acid derivatives of the formula (I),

    in which
    J, X, Y, A, B, D and G have the meanings given above,
    to a number o...

    01/19/2012
    20120015981Active compound combinations
    The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) the compound 3-(difluoromethyl)-1-methyl-N-(3′,4′,5′-trifluorobiphenyl-2-yl)-1H-pyrazole-4-carboxamide of formula (I) and/or the compou...
    01/19/2012
    20120010072DIMETHOMORPH AS SAFENER FOR PESTICIDES WITH PHYTOTOXIC EFFECTS
    The present invention relates to a method for reducing or preventing damage caused by pesticides to plants treated therewith and/or to plant propagation material treated therewith and/or to plants growing from this plant propagation material and/or to plants which grow ...
    01/12/2012
    20120010184Therapeutic Uses of Compounds Which Selectively Modulate The CB2 Receptor
    Compounds of formula (I)

    are disclosed. Compounds according to the invention bind to and are agonists, antagonists or inverse agonists of the CB2 receptor, and are useful for treating inflammation. Those comp...

    01/12/2012
    20120009238METHOD FOR TREATMENT OF CROP WITH AN ENCAPSULATED PESTICIDE
    The present invention is related to a method for the pesticidal treatment of crops which have a final growth height of at least 140 cm, comprising the treatment with an encapsulated pesticide at a growth height of the crop of up to 120 cm. The invention further relates ...
    01/12/2012
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