Yang; Lucy X. - US Patent Attorneys and Agents

Attorney: Yang; Lucy X.

Number of patents: 105
Last date: March 20, 2012

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Number	Title	Issue Date
8138177	Benzimidazolone derivatives as CB2 receptor ligands This invention relates to compounds of the formula (I): or pharmaceutically acceptable salts thereof, wherein: A, B, R1, R2 and R3 are each as described herein, and compositions containing such compounds and the use of such compounds...	03/20/2012
8133899	Pyrrolo[2,3-]pyrimidine compounds Described herein is pyrrolo{2,3-d}pyrimidine compounds, their use as Janus Kinase (JAK) inhibitors, pharmaceutical compositions containing this compounds, and methods for the preparation of these compounds. ...	03/13/2012
7902232	Substituted arylpyrazoles This invention relates to a combination product comprising a range of 1-aryl-4 -cyclopropylpyrazoles in which there is at least one fluorine attached to the cyclopropyl ring, and one o more further therapeutic agents, particularly anti-parasitic agents. ...	03/08/2011
7842791	Dispersible pharmaceutical compositions A pharmaceutical composition is provided comprising a vehicle that comprises (a) an amphipathic oil that is water dispersible and ethanol insoluble, (b) microcrystalline wax, and (c) a pharmaceutically acceptable non-aqueous carrier; and having an antibacterial subs...	11/30/2010
7829100	Pharmaceutical composition having modified carrier A composition comprising: (a) one to three bioactive agents; and (b) a modified liquid vehicle; wherein immediately after manufacture of the composition, said composition can be administered to a host such that the one to three bi...	11/09/2010
7687507	Pyrrolo[2,3-d]pyrimidine compounds A compound of the formula wherein R1, R2 and R3 are as defined above, which are inhibitors of the enzyme protein tyrosine kinases such as Janus Kinase 3 and as such are useful therapy as imm...	03/30/2010
7642350	Purine derivatives This invention relates to purine derivatives, to processes for their preparation, to compositions containing them and to their use. The present invention provides compounds of formula (I) whe...	01/05/2010
7638537	Pyrazole compounds as transforming growth factor (TGF) inhibitors Novel pyrazole compounds, including derivatives thereof, to intermediates for their preparation, to pharmaceutical compositions containing them and to their medicinal use are described. The compounds of the present invention are potent inhibitors of transforming gro...	12/29/2009
7592362	Substituted imidazoles This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides. ...	09/22/2009
7547718	Substituted imidazoles This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides. ...	06/16/2009
7544706	Substituted imidazoles This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides. ...	06/09/2009
7514464	Substituted arylpyrazoles This invention relates to a combination product comprising a compound of formula I wherein X, R1, R2, R3, R4, R5, R6, R7 and R9 are as ...	04/07/2009
7435753	Substituted arylpyrazoles This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which there is at least one fluorine attached to the cyclopropyl ring, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides. ...	10/14/2008
7411001	Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids The present invention relates to oxygenated esters of 4-iodophenylamino benzhydroxamic acid derivatives, pharmaceutical compositions and methods of use thereof. The present invention also relates to crystalline forms of oxygenated esters of 4-iodophenylamino benzhyd...	08/12/2008
7388023	Amino acids with affinity for the α2δ-protein Certain β-amino acids that bind to the alpha-2-delta (α2δ) subunit of a calcium channel are disclosed. These compounds and their pharmaceutically acceptable salts are useful in the treatment of a variety of psychiatric, pain and other disorders. Also disclosed ar...	06/17/2008
7297682	Diphosphate salt of a 4″—substituted-9-deoxo-9 A—AZA—homoerythromycin derivatives and its pharmaceutical composition This invention relates to a novel crystalline diphosphate salt of (2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-13-[[2,6-dideoxy-3-C-methyl-3-O-methyl-4-C-[(propylamino)methyl]-α-L-ribo-hexopryanosyl]oxy]-2-ethyl-3,4,10-trihydroxy-3,5,8,10,12,14-hexamethyl-11-[[3,4,6-trideo...	11/20/2007
7141588	N-aryl-2-oxazolidinone-5-carboxamides and their derivatives The present invention provides antibacterial agents having the formulae I, II, and III described herein. ...	11/28/2006
7105547	Antimicrobial 1-aryl dihydropyridone compounds The present invention provides antibacterial agents of formula I, or a pharmaceutically acceptable salt thereof. ...	09/12/2006
7101874	Antimicrobial dihydrothiazine and dihydrothiopyran oxazolidinones The present invention provides a compound of formula I or a pharmaceutically acceptable salt thereof wherein Y is —S(═O)n—, —S(═NR8)—, or —S(═NR8)(═O)—; Z is �...	09/05/2006
7087784	Process to prepare oxazolidinones The present invention relates to a one-step process to prepare pharmacologically active 2-oxo-5-oxazolidinylmethylacetamides. ...	08/08/2006
7049443	Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound The present invention is directed to novel amide-containing compounds which have an improved solubility and a method of improving the solubility of amide-containing compounds. The amide-containing compounds include oxazolidinone compounds and the bioavailability of ...	05/23/2006
7012088	Indolone oxazolidinones and derivatives thereof The present invention provides antibacterial agents of formula I described herein and intermediates for their preparation. ...	03/14/2006
7002020	Oxazolidinone combinatorial libraries, compositions and methods of preparation Oxazolidinones and methods for their synthesis are provided. Also provided are combinatorial libraries comprising oxazolidinones, and methods to prepare the libraries. Further provided are methods of making biologically active oxazolidinones as well as pharmaceutica...	02/21/2006
6972286	Oxazolidinones having a benzannulated 6- or 7-membered heterocycle The present invention provides oxazolidinones having a benzannelated 6- or 7-membered heterocycle as antibacterial agents. ...	12/06/2005
6927229	Difluorothioacetamides of oxazolidinones as antibacterial agents The present invention describes difluororthioacetamide oxazolidinones of formula I: R is —CH2— or —CH2CH2—; R2 and R3 are independently —H or —F; X is ...	08/09/2005
6919329	N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives The present invention provides antibacterial agents having the formulae I, II, and III described herein. ...	07/19/2005
6903097	Heterocycle carboxamides as antiviral agents The present invention provides a compound of formula I which is useful as antiviral agents, in particular, as agents against viruses of the herpes family. ...	06/07/2005
6887995	Process to prepare oxazolidinones The present invention relates to a one-step process to prepare pharmacologically active 2-oxo-5-oxazolidinylmethylacetamides. ...	05/03/2005
6884813	Antimicrobial dihydrothiazine and dihydrothiopyran oxazolidinones The present invention provides a compound of formula I or a pharmaceutically acceptable salt thereof wherein A is a structure i, ii, iii, or iv X is CR7; Y is ...	04/26/2005
6875871	Oxazolidinone photoaffinity probes Disclosed are novel compounds that are useful and effective as photoaffinity probes and methods of using oxazolidinone photoaffinity probes. ...	04/05/2005
6870070	Process to prepare 2-aminoindan derivatives The present invention relates to (2S)-enantiomers of 2-aminoindan derivatives of formula I: and a novel process for the preparation of them. ...	03/22/2005
6861433	Oxazolidinone photoaffinity probes The present invention provides compounds of the formula: compositions comprising such compounds, and methods for using the same. ...	03/01/2005
6858635	Oxazolidinone photoaffinity probes Disclosed are novel compounds that are useful and effective as photoaffinity probes and methods of using oxazolidinone photoaffinity probes. ...	02/22/2005
6828317	Antimicrobial thiadiazinone derivatives and their application for treatment of bacterial infections The present invention provides certain thiadiazinone derivatives of oxazolidinones of the following formula I: or pharmaceutically acceptable salts thereof that are antibacterial agents, pharmaceutical compositions con...	12/07/2004
6825225	Bicyclic isoxazolinones as antibacterial agents The present invention provides compounds of formula I useful as anti microbial agents wherein X, Y, R1, and n are as defined in thereof. ...	11/30/2004
6821970	Oxazinocarbazoles for the treatment of CNS diseases The present invention provides oxazinocarbazole derivatives having a ring connecting position 8 (C-8) and position 9 (N-9), and more specifically, provides compounds of formula (I) wherein R1, R2, R3 and R4 are described h...	11/23/2004
6774231	Method for the preparation of oxazolidinones The present invention relates to a process for making a compound of structure 4 which comprises reacting a compound of structure 1 with vinyl sulfone in the presence of a Lewis-acid at a temperature in a range of from 40...	08/10/2004
6730682	Heterocycle carboxamides as antiviral agents The present invention provides a compound of formula I which is useful as antiviral agents, in particular, as agents against viruses of the herpes family. ...	05/04/2004
6727248	Substituted quinolinecarboxamides as antiviral agents The present invention discloses disubstiuted 4-oxo-1,4-dihydro-3-quinolinecarboxamide derivatives. The compounds are useful as antiviral agents, in particular, as agents against viruses of the herpes family. ...	04/27/2004
6693114	4-oxo-1,4-dihydro[1,8]naphthyridine-3-carboxamides as antiviral agents A compound of formula III: ##STR1## or a pharmaceutically acceptable salt thereof wherein, the variables are as in the specification is provided. The compounds are particularly effective in the treatment or prevention of herpes viruses....	02/17/2004

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Attorney: Yang; Lucy X.