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| Number | Title | Issue Date |
| 8173663 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound comprising: wherein M is N or CR4; Q1 and Q2 are each independen... | 05/08/2012 |
| 7960384 | Dipeptidyl peptidase inhibitors Compounds, pharmaceutical compositions, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound of the formula: wherein the substituents are as defined herein. ... | 06/14/2011 |
| 7872124 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a member selected from the group consisting of: wherein E is CH or N, Q is selected from the group consistin... | 01/18/2011 |
| 7825242 | Dipeptidyl peptidase inhibitors Compounds, pharmaceutical compositions, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound of the formula: wherein R2 is amino (C1-6)alkyl, hetero(C3... | 11/02/2010 |
| 7807689 | Dipeptidyl peptidase inhibitors The present invention provides a compound of the formula: or stereoisomers or pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof, articles of manufacture comprising the s... | 10/05/2010 |
| 7795428 | Dipeptidyl peptidase inhibitors Compounds are provided for use with DPP-IV of the formula: Also provided are pharmaceutical compositions, kits and articles of manufacture comprising such compounds; methods and intermediates useful for making the compounds... | 09/14/2010 |
| 7790736 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein. ... | 09/07/2010 |
| 7790734 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein. ... | 09/07/2010 |
| 7781584 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound comprising: wherein M is N or CR4; Q1 and Q2 are each independen... | 08/24/2010 |
| 7759339 | Hydroxysteroid dehydrogenase inhibitors Compounds, pharmaceutical compositions, kits and methods are provided for use with hydroxysteroid dehydrogenases that comprise a compound selected from the group consisting of: wherein the variables are as defined herein. | 07/20/2010 |
| 7732446 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formulae: where the substituents are as described herein. ... | 06/08/2010 |
| 7723344 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein. ... | 05/25/2010 |
| 7687625 | Dipeptidyl peptidase inhibitors Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 protease that comprise a compound comprising the formula: wherein Q is selected from the group of CO, SO, S... | 03/30/2010 |
| 7678909 | Dipeptidyl peptidase inhibitors Compounds are provided which may be used to inhibit DPP-IV comprising the formula: wherein the substituents are as described in the specification and claims. ... | 03/16/2010 |
| 7642275 | Histone deacetylase inhibitors Compounds, pharmaceutical compositions, kits and methods are provided for use with histone deacetylases (HDACs) that comprise a compound of the formulae: wherein the variables are as defined herein. ... | 01/05/2010 |
| 7642253 | Histone deacetylase inhibitors Compounds, pharmaceutical compositions, kits and methods useful for inhibiting HDAC, thereby treating a disease state for which HDAC possess activity that contributes to the pathology and/or symptomology of the disease state. The compound is selected from the group ... | 01/05/2010 |
| 7638638 | Dipeptidyl peptidase inhibitors Pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound with the formula: where the labeled substituents are as described herein. ... | 12/29/2009 |
| 7563610 | Crystalline composition of farsenyl pyrophosphate synthase (IspA) Provided are crystals relating to Farsenyl Pvrophosphate Synthase (IspA) from E. coli and its various uses. ... | 07/21/2009 |
| 7556950 | Crystallization of the catalytic domain of human phosphodiesterase 4-D3 (PDE4-D3) Provided are crystals relating to human phosphodiesterase 4-D3 (PDE4-D3), methods for forming crystals comprising PDE4-D3 and crystals comprising PDE4-D3 co-crystallized with a ligand molecule, and methods of using crystals comprising PDE4-D3. ... | 07/07/2009 |
| 7550598 | Kinase inhibitors Compounds, pharmaceutical compositions, kits and methods are provided for use with kinases that comprise a compound of the formula: wherein R1, R2, R3, Q, U, V, W, X, and Y are as defined he... | 06/23/2009 |
| 7534592 | Crystallization of carboxyltransferase domain of Acetyl-CoEnzyme A Carboxylase 2 with a ligand Provided are crystals relating to the carboxyltransferase domain of human Acetyl-Coenzyme A Carboxylase 2 and its various uses. ... | 05/19/2009 |
| 7510690 | System for performing crystallization trials A crystallization system is provided comprising a trial generation station configured to generate crystallization trials in trial zones of a crystallization plate; an imaging station configured to take images of crystallization trials in the crystallization plate; a... | 03/31/2009 |
| 7507552 | Crystallization of histone deacetylase 2 Provided are crystals relating to histone deacetylase 2 (HDAC-2) and its various uses. ... | 03/24/2009 |
| 7452419 | Method for performing crystallization trials A method is provided for operating a crystallization system comprising identifying a screen storage plate from among the plurality of screen storage plates stored in a screen storage station, each screen storage plate having a plurality of wells that contain a scree... | 11/18/2008 |
| 7444273 | Crystallization of aurora/LPL1P-related kinase Provided are crystals relating to Aurora/LPL1P-related kinase and its various uses. ... | 10/28/2008 |
| 7435397 | System for performing crystallization trials A crystallization system is provided comprising a screen generation station; a screen storage station; including a housing configured to store a plurality of screen storage plates and mechanics for retrieving a selected screen storage plate from among the plurality ... | 10/14/2008 |
| 7435379 | System for performing crystallization trials A trial generation station is provided comprising: a deck configured to receive a crystallization plate from a transport mechanism, the crystallization plate including a plurality of trial zones where crystallization trials are generated; and a head configured to be... | 10/14/2008 |
| 7431768 | System for performing crystallization trials A crystallization system is provided comprising: a screen replicator configured to transfer screen solutions from wells of a screen storage plate into well regions of multiple crystallization plates; a trial generation station configured to generate crystallization ... | 10/07/2008 |
| 7416710 | Method and system for performing crystallization trials A crystallization system is provided that comprises a screen replicator having a transfer mechanism configured to transfer portions of different screen solutions contained in a screen storage plate to well regions of a crystallization plate; a screen storage station... | 08/26/2008 |
| 7344852 | Crystallization of dipeptidyl peptidase IV (DPPIV) Provided are crystals relating to DPPIV and its various uses. ... | 03/18/2008 |
| 7326552 | Wild-type kinase domain of human Ephrin receptor A2 (EPHA2) and crystallization thereof Provided are crystals relating to human Ephrin Receptor A2 and its various uses. ... | 02/05/2008 |
| 7319016 | Crystallization of cathepsin S Provided are crystals relating to Cathepsin S and its various uses. ... | 01/15/2008 |
| 7309594 | Crystallization of protein kinase Bα/AKT1 Provided are crystals relating to Protein kinase Bα/AKT1 and its various uses. ... | 12/18/2007 |
| 7303892 | Crystallization of AKT3 Provided are crystals relating to AKT3 and its various uses. ... | 12/04/2007 |
| 7303893 | Crystallization of c-KIT tyrosine kinase leading to autoinhibited crystal structure Provided are crystals relating to the autoinhibited structure of c-KIT tyrosine kinase (c-KIT) and its various uses. ... | 12/04/2007 |
| 7297508 | Crystallization of fibroblast activation protein alpha (FAPα) Provided are crystals relating to FAPα and its various uses. ... | 11/20/2007 |
| 7294309 | Small volume liquid handling apparatus and method A fluid dispensing system comprising: a fluid container; a dispensing head in fluid communication with the fluid container; a displacement mechanism which delivers fluid from the fluid container to the dispensing head such that an aliquot of liquid is delivered to a... | 11/13/2007 |
| 7270987 | Crystallization of FMS-like tyrosine kinase 3 Provided are crystals and structure coordinates relating to FMS-like tyrosine kinase 3 and its various uses. ... | 09/18/2007 |
| 7250514 | Histone deacetylase inhibitors Histone deacetylase inhibitors and uses thereof are provided that have the general formula: wherein R1, R2, R3, R4, R5, R6, R7, R8... | 07/31/2007 |
| 7241868 | Crystallization of Glucocorticoid Receptor Provided are crystals relating to human Glucocorticoid Receptor and its various uses. ... | 07/10/2007 |
