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| Number | Title | Issue Date |
| 5968948 | Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations Compound of general formula I ##STR1## wherein A denotes a benzo, indolo or thienyl group; B denotes the group --O--, --S-- or --CHR5 --, wherein R5 is hydrogen, (C1-6)alkyl, phenyl or benzyl; R3 denotes 2- or 3... | 10/19/1999 |
| 5945535 | Method of preparing norbenzomorphanes The present invention relates to a new process for preparing norbenzomorphan, the central intermediate step in the preparation of pharmaceutically useful benzomorphan derivatives of general formula 1 ##STR1## especially (-)-(1R,5S,2"R)-3'-hydrox... | 08/31/1999 |
| 5919807 | Benzothiazoles and benzoxazoles, drugs containing them, their use and methods of preparing them The invention relates to benzothiazoles and benzoxazoles of general formula ##STR1## wherein R1 to R3, X, Z and n are defined as in claim 1, the enantiomers, diastereomers and salts thereof, particularly the physiologically acce... | 07/06/1999 |
| 5915426 | Apparatus and process for cleaning the outside of containers An apparatus for cleaning the outside of a container to remove any adhering liquid, particularly in the region of a fill opening thereof. Adhering liquid is blown off of the container by mean of compressed air.... | 06/29/1999 |
| 5899365 | Device for assisting manual actuation of an aerosol dispenser A device for assisting the manual actuation of aerosol dispensers, especially dispensers of the sort used to dispense metered doses of phamaceuticals. Dispensers to be used with the device of the invention are of known per se design and comprise a contain... | 05/04/1999 |
| 5856497 | Asymmetric synthesis of -cycloalkylalkyl substituted methanamines This invention relates to process for asymmetrically producing enantiomerically pure -cycloalkylalkyl substitututed methanamines from -pinene. One key step of the process of this invention utilizes the oxidation product of -pinene, hy... | 01/05/1999 |
| 5852192 | Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them The invention relates to cyclic urea derivatives of general formula ##STR1## wherein Ra, Rb, X and Y are as defined herein, pharmaceutical compositions containing the derivatives and processes for preparing them.... | 12/22/1998 |
| 5847169 | Process for preparing oxiranemethanamine derivatives A process for preparing oxiranemethane derivatives which are useful as intermediates for preparing aspartyl protease inhibitors comprising the steps of activating an aminodiol, acylating the aminodiol and reacting the acylated aminodiol with a base to for... | 12/08/1998 |
| 5837712 | Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations A compound of formula I ##STR1## wherein A denotes a benzo, indolo or thieno group; R1 denotes thienyl or the group ##STR2## wherein R7, R8 and R9 independently of one another may represent methyl, eth... | 11/17/1998 |
| 5837704 | 2-heteroaryl-5,11-dihydro-6H-dipyrido3,2-B:2',3'-E!1,4!diazepines and their use in the prevention or treatment of HIV infection Novel compounds for the treatment of HIV-1 infection. These are 2-heteroary-5,11-dihydro-6H-dipyrido3,2-b:2',3'-e!1,4!diazepines of the formula ##STR1## wherein Z is oxygen, sulfur, .dbd.NCN or .dbd.NOR10 and Ar is a group of the ... | 11/17/1998 |
| 5833088 | Container with closure cap and method of filling containers without gas bubbles A closure cap for sealing containers without gas bubbles displaces some of the contents of the container when fitted onto the neck of the container and at the same time allows any trapped gas to escape through one or more vents before the closure cap enga... | 11/10/1998 |
| 5821240 | Pyrimido5,4!-dipyrimidines, pharmaceuticals containing them, their use and processes for the preparation thereof Pyrimido5,4-d!pyrimidines of the general formula ##STR1## which have an inhibitory effect on signal transduction mediated by tyrosine kinases, their use for the treatment of disorders, in particular of oncoses, and their preparation. Exemplary comp... | 10/13/1998 |
| 5817677 | 5-membered heterocycles, medicaments containing these compounds, their use and processes for their preparation 5-Membered heterocyclic compounds, of which the following compounds are exemplary: (a) 4-trans-4-(2-carboxyethyl)cyclohexyl!aminocarbonyl!-1-(4-piperidyl)imida zole, (b) 5-trans-4-(2-carboxyethyl)cyclohexyl!aminocarbonyl!-4-methyl-2-(4-piperi ... | 10/06/1998 |
| 5807875 | Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them Amino acid derivatives, suitable for the treatment of obesity. The following compound is exemplary of the class: (R,S)-N2 -(diphenylacetyl)-N-(4-hydroxyphenyl)methyl!-N5 -(1H-imidazol-2-yl)-ornithinamide.... | 09/15/1998 |
| 5807870 | Substituted pipecolinic acid derivatives as HIV protease inhibitors Disclosed herein are compounds of formula 1 ##STR1## wherein X is a terminal group, for example, an aryloxycarbonyl, an alkanoyl or an optionally mono- or disubstituted carbamoyl; B is absent or an amino acid residue, for example, Val or Asn; R1... | 09/15/1998 |
| 5770738 | Esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions The new compounds of formula A--O--CO--Z (I) (wherein A and Z are defined as explained in the specification) can be prepared by conventional methods; they are suitable as active substances for pharmaceutical compo... | 06/23/1998 |
| 5760093 | Halohydrocarbon-free delayed release lacquer solution for pharmaceutical preparation The invention relates to a delayed-release lacquer solution for pharmaceutical preparations which is characterised in that it is free from halogenated hydrocarbons.... | 06/02/1998 |
| 5750135 | Stabilized feed additive and process for the preparation thereof The invention relates to a stabilized feed additive, more particularly containing zinc bacitracin, and processes for the preparation thereof.... | 05/12/1998 |
| 5747488 | 2-aryl-5,11-dihydro-6H-dipyrido3,2-B:2',3'-E!1, 4!diazepines and their use in the treatment of HIV infection Disclosed are novel 2-aryl-5,11-dihydro-6H-dipyrido3,2-b:2',3'-e!1,4!diazepines. These are useful in the of HIV infection. Exemplary compounds are: 8-Ethyl-1-methyl-10-(4-pyrazolyl)imidazo2',3':6,5!dipyrido3,2-b:2',3'-e! 1,4!diazepine; 8-c-Propyl... | 05/05/1998 |
| 5741798 | 2-benzyl-4-sulfonyl-4H-isoquinolin-1,3-diones and their use as antiinflammatory agents Antiinflammatory compounds of the formula I or IA ##STR1## wherein, R1 is hydrogen, halogen, C1-4 alkyl, or C1-4 alkoxy; R2 and R3 are the same or different and each is hydrogen, halogen, trifluo... | 04/21/1998 |
| 5726205 | O-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds and their use, as well as a method of preparing them This document describes O-acyl-4-phenyl-cycloalkanols of general formula I ##STR1## wherein n denotes the number 0 or 1, m denotes the number 1 or 2, p denotes the number 0 or 1, R1 and R2 each denote hydrogen, lower alkyl, alke... | 03/10/1998 |
| 5712273 | Amino acid derivatives, processes for the manufacture thereof and pharmaceutical compositions (II) containing these compounds The invention relates to new amino acid derivatives of general formula I R1 -R11 --A1 --B (I) and the pharmaceutically acceptable salts thereof, wherein group B is --A2 --NR2 R3 | 01/27/1998 |
| 5710155 | Arylglycinamide derivatives, processes for the manufacture thereof and pharmaceutical compositions containing these compounds The invention relates to new arylglycinamide derivatives of general formula I ##STR1## and the pharmaceutically acceptable salts thereof, wherein R1, R2, R3, R4, R5 and Ar have the meanings given... | 01/20/1998 |
| 5709305 | Dispenser for solid pharmaceutical preparations A new dispenser for solid pharmaceutical preparations consists of a flat container with a removal well 3 which can be closed or opened by the flipping round of a closure member 5 with a convexity 6 engaging in the removal well 3.... | 01/20/1998 |
| 5708006 | Neurokinin antagonists The invention relates to new compounds of general formula I ##STR1## and the pharmaceutically acceptable salts thereof, wherein A, B, Z, R1, R2, R3 and m are defined as in the specification, processes for preparing th... | 01/13/1998 |
| 5700901 | Resorbable mouldings and process for producing them The invention relates to resorbable mouldings and processes for producing them.... | 12/23/1997 |
| 5700801 | Piperazine derivatives, pharmaceutical compositions containing these compounds, their use and processes for preparing them Piperazine derivatives useful in the treatment or prevention of inflammation, bone degradation, thrombosis and tumor metastasis. Exemplary species are: (a) 4-trans-3-4-(4-Pyridyl)-piperazin-1-yl!propionyl!amino!-cyclohexanecarb oxylic acid, (b) ... | 12/23/1997 |
| 5698552 | Hetrazepinoid amides The present invention relates to thienodiazepines of formula Ib: ##STR1## wherein U, V, R5, R6 and R7 are as defined herein. This invention also relates to processes for preparing these thienodiazepines and their use ... | 12/16/1997 |
| 5688793 | Pyridazino4',5':3,4!pyrrolo-2,1-a!-isoquinolines and the use thereof for preparing pharmaceutical preparations The invention relates to new pyridazino4',5':3,4!-pyrrolo2,1-a!isoquinolines of the formula ##STR1## and the physiologically acceptable salts thereof with acids and complex-forming agents, wherein X is O, S or NHO and R1, R3... | 11/18/1997 |
| 5468758 | Crystalline forms of endo-2,3-dihydro-N-(8-methyl)-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H-benz imidazole-1-carboxamides Crystalline and pharmacologically active monohydrates of endo-2,3-dihydro-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H-benzimi dazole-1-carboxamide hydrochloride and of endo-3-ethyl-2,3-dihydro-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2-oxo-1H -be... | 11/21/1995 |
| 5463071 | 5-membered heterocyclic compounds, processes for preparing them and pharmaceutical compositions containing these compounds Compounds of the formula ##STR1## wherein X1 to X5 are as defined herein, the tautomers, the stereoisomers including the mixtures thereof and the salts thereof, particularly the physiologically acceptable salts thereof with inor... | 10/31/1995 |
| 5455266 | Enhanced chemotherapeutic compositions against microbial infections in fish, the preparation and use thereof The invention relates to enhanced chemotherapeutic compositions against microbial infections in fish, containing a benzylamine derivative of general formula ##STR1## wherein R1 to R3 are defined as in claim 1, or a physiological... | 10/03/1995 |
| 5451587 | Quinuclidines, their use as medicaments and processes for their preparation The invention relates to quinuclidines, processes for their preparation and their use as medicaments having cholinomimetic properties.... | 09/19/1995 |
| 5434242 | Catalyst-free resorbable homopolymers and copolymers The invention relates to resorbable homopolymers and copolymers which are substantially free from polymerization catalysts and processes for preparing them.... | 07/18/1995 |
