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| Number | Title | Issue Date |
| 7462725 | Chloromethylation of thiophene The process according to the invention relates to the preparation of 2-chloromethyl-thiophene of the formula (I). During this process thiophene is chloromethylated in the presence of one or more compounds containing keto group and optionally it is transformed into t... | 12/09/2008 |
| 7442708 | 1,2,3-substituted indolizine derivatives, inhibitors of fgfs, method for making same and pharmaceutical compositions containing same Compounds of formula I or salts thereof: in which R1 represents —OH, (C1-C5)alkoxy, carboxyl, (C2-C6)alkoxycarbonyl, —NR5R6, —N... | 10/28/2008 |
| 7326720 | Phenyl- and pyridylpiperidines with TNF activity The present invention relates to compounds of formula (I): in which X represents N or CH; R1 represents a hydrogen or halogen atom or a CF3 group; R2 and R3 independent... | 02/05/2008 |
| 7326723 | Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same The present invention relates to compounds of formula (I): in which X represents N or CH; R1 represents a hydrogen or halogen atom or a CF3 group; n is an ... | 02/05/2008 |
| 7186720 | Tetrahydropyridyl-alkyl-heterocycles, method for preparing the same and pharmaceutical compositions containing the same The present invention relates to compounds of formula (I): in which X represents N or CH; R1 represents a hydrogen or halogen atom or a CF3 group; R2 and R3 independent... | 03/06/2007 |
| 7153969 | Hydroxyacetic ester derivatives, preparation method and use as synthesis intermediates Methyl (R)-2-(R1OSO2)-2-(2-chlorophenyl)acetates useful as intermediates in the preparation of methyl (S)-2(2-chlorophenyl)-2-(4,5,6,7-tetrahydrothieno[3,2-c]-5-pyridyl)acetate. ... | 12/26/2006 |
| 6951940 | Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them The invention relates to the compounds of formula: as well as to the salts thereof with inorganic or organic acids, to solvates thereof and/or to hydrates thereof, which have strong affinity and high selectivity for th... | 10/04/2005 |
| 6894186 | Hydroxyacetic ester derivatives, preparation method and use as synthesis intermediates Methyl (R)-2-(R1OSO2)-2-(2-chlorophenyl)acetates useful as intermediates in the preparation of methyl (S)-2(2-chlorophenyl)-2-(4,5,6,7-tetrahydrothieno[3,2-c]-5-pyridyl)acetate. ... | 05/17/2005 |
| 6864277 | 1,3-dihydro-2H-indol-2-one derivatives, method for preparing same and pharmaceutical compositions containing them The invention relates to compounds of formula: and to solvates and/or hydrates thereof, with affinity for and selectivity towards the Vreceptors or both the V1b and V1a receptors of arginine-vasop... | 03/08/2005 |
| 6861072 | Pharmaceutical composition with gastric residence and controlled release The invention concerns a pharmaceutical composition with gastric residence and controlled release, characterized in that it comprises two or three layers and contains (a) an active principle associated with a excipient modifying its release; (b) a system generating ... | 03/01/2005 |
| 6846936 | 2-butyl-3-(4-[3(dibutylamino)propoxy]benzoyl)-5-nitro-benzofuran hydrochloride and preparation thereof The invention relates to 2-butyl-3-(4-[3-(dibutylamino)propoxy]benzoyl-5-nitrobenzofuran hydrochloride, to its preparation and to its use as synthetic intermediate, in particular in preparing 2-butyl-3-(4-[3-(dibutylamino)propoxy]benzoyl)-5-nitrobenzofuran, itself a... | 01/25/2005 |
| 6844329 | Polysaccharides with antithrombotic activity comprising at least a covalent bond with biotin or a biotin derivative The present invention relates to novel synthetic polysaccharides with antithrombotic activity exhibiting at least one covalent bond with biotin or a biotin derivative and to a process employing avidin or streptavidin which makes it possible to neutralize these polys... | 01/18/2005 |
| 6844335 | 2-amino-3-(alkyl)-pyrimidone derivatives as GSK3.β.inhibitors A pyrimidone derivative represented by formula (I) or a salt thereof: Wherein: R1 represents a hydrogen atom or a C1-6 alkyl group which may be substituted by a C | 01/18/2005 |
| 6828448 | Methanesulphonamido-benzofuran, preparation method and use thereof as synthesis intermediate The invention relates to 2-butyl-5-(methanesulfonamido)benzofuran, its preparation and its use. This compound is a synthesis intermediate, in particular for the preparation of dronedarone. ... | 12/07/2004 |
| 6828321 | 1,2,4-Benzotriazine oxides as radiosensitizers and selective cytotoxic agents A method of using 1,2,4-benzotriazine oxides, some of which are novel compounds, as radiosensitizers and selective cytotoxic agents is disclosed. These compounds are shown to specifically radiosensitize hypoxic tumor cells. Some are additionally disclosed to be usef... | 12/07/2004 |
| 6806282 | Branched substituted amino derivatives of 3-amino-1-phenyl-1h-[1,2,4]triazol, methods for producing them and pharmaceutical compositions containing them The present invention relates to novel branched substituted amino derivatives of 3-amino-1-phenyl-1H-[1,2,4]triazole, processes for their preparation and pharmaceutical compositions comprising them. ... | 10/19/2004 |
| 6800761 | Form of irbesartan, methods for obtaining said form and pharmaceutical compositions containing same The invention relates to a novel crystalline form of irbesartan, to pharmaceutical compositions containing it, to processes for preparing it, and to a method for treating cardiovascular diseases utilizing it. ... | 10/05/2004 |
| 6794382 | Benzimidazole derivatives, preparation and therapeutic use thereof The invention relates to benzimidazole derivatives of general formula in which X represents a nitrogen atom or a carbon atom; and when X represents a nitrogen atom: R3 represents a hydrogen atom or a... | 09/21/2004 |
| 6767533 | Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress A composition containing a peripheral benzodiazepine receptor ligand for topical use in the treatment of cutaneous stress. ... | 07/27/2004 |
| 6761879 | Titanium derived compounds, preparation and use thereof The invention relates to a titanium-derived compounds, and to processes for preparing the same. ... | 07/13/2004 |
| 6730695 | 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for V1b and V1a arginine-vasopressin receptors The invention relates to compounds of formula: as well as the possible salts thereof with mineral or organic acids, and the solvates and/or hydrates thereof, which have affinity for and selectivity towards the V1b | 05/04/2004 |
| 6713053 | Use of IL-7 for treating auto-immune diseases and insulin-dependent diabetes mellitus in particular The use of interleukin 7 or T cells pre-incubated in the presence of IL-7 for preparing a drug or pharmaceutical composition for treating an auto-immune disease, particularly an auto-immune disease induced by a defect in CD4+ T cell immunoregulation, is disclosed. | 03/30/2004 |
| 6710042 | Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them Compounds of formula (I) are useful as human NK3 receptor antagonists. ... | 03/23/2004 |
| 6673790 | Indolin-2-one derivatives, preparation and their use as ocytocin receptor ligands The present invention relates to novel indolin-2-one derivatives of formula: ##STR1## to the preparation and to the pharmaceutical compositions comprising them. These compounds have an affinity for oxytocin receptors.... | 01/06/2004 |
| 6610882 | N-(arylsulphonyl) amino acid derivatives The invention relates to compounds of formula ##STR1## in which R1 to R9, R16 and R17 are as defined in claim 1. These compounds are pharmacologically active.... | 08/26/2003 |
| 5665763 | Therapeutic phenoxyalkylpyridazines and intermediates therefor Compounds of the formula ##STR1## wherein: R1, R2, R3 and R4 are as defined in the specification, Y is alkylene of 3 to 9 carbon atoms, R5 is alkoxycarbonyl, alkyltetrazolyl, phenyl or a heterocycle c... | 09/09/1997 |
| 5661020 | Low diol polyalkylene oxide biologically active proteinaceous substances Disclosed are pharmaceutical compositions containing low diol polyethylene glycol, covalently attached to superoxide and dismutase process of making the compositions. Also disclosed is a method of treatment of disease processes associated with the adverse... | 08/26/1997 |
| 5652254 | 2-saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof 4-R4 -R5 -2-Saccharinylmethyl heterocyclic carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R4 -R5 -2-halomethylsaccharin with either a heterocyclic carboxylic acid in... | 07/29/1997 |
| 5650419 | Thiadiazoles and their use as antipicornaviral agents Described herein are compounds of the formula; ##STR1## wherein: Thi is a unsubstituted or substituted thiadiazolyl; Y is an alkylene bridge of 3-9 carbon atoms; R1 and R2 are each independently chosen from hydrogen, halo, alkyl, alk... | 07/22/1997 |
| 5643929 | 1,2,4-oxidiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents Compounds of the formula ##STR1## wherein: R1 is alkyl, alkoxy, hydroxy, cycloalkyl, hydroxyalkyl, alkoxyalkyl, hydroxyalkoxy, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alk... | 07/01/1997 |
| 5624922 | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents Aryl-fused- and hetaryl-fused-2,4-diazepines of formula XXXVI, benzodiazocines of formula XXX, benzodiazepines of formula II ##STR1## δ-aminoamides of formula III and aryldimethanamines of formula XXXVII ##STR2## wherein A is an aryl or he... | 04/29/1997 |
| 5614530 | Substituted N-arylmethyl and heterocyclmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines and compositions and methods of use thereof Substituted N-arylmethyl and heterocyclylmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines, pharmaceutical compositions containing them and methods for a) effecting c-GMP-phosphodiesterase inhibition, b) treating heart failure and/or hypertension, c) revers... | 03/25/1997 |
| 5597841 | 2-saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof 4-R4 -R5 -2-Saccharinylmethyl aryl carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R4 -R5 -2-halomethylsaccharin with an arylcarboxylic acid in the presence of an aci... | 01/28/1997 |
| 5578623 | Saccharin derivative proteolytic enzyme inhibitors Compounds having the structural formula ##STR1## wherein L is O; L-R1 is a leaving group, H-L-R1 is the conjugate acid thereof and H-L-R1 has a pKa value less than or equal to to 8; R2 is primary or s... | 11/26/1996 |
| 5563163 | 2-saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof 4-R4 -R5 -2-Saccharinylmethyl heterocyclic carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R4 -R5 -2-halomethylsaccharin with either a heterocyclic carboxylic acid in... | 10/08/1996 |
| 5494925 | 2-heterocyclyloxymethyl and 2-heterocyclylthiomethyl-1,2,5-thiadiazolidin-3-one 1,1-dioxides and compositions and method of use thereof 2-Heterocyclyloxymethyl and 2-heterocyclylthiomethyL-1,2,5-thiadiazolidin-3-one 1,1-dioxides, pharmaceutical compositions containing them and methods for the treatment of degenerative diseases utilizing them.... | 02/27/1996 |
| 5488055 | Substituted N-cycloalkylmethyl-1H-pyrazolo(3,4-b)quinolin-4 amines and compositions and methods of use thereof Substituted N-cycloalkylmethyl-1H-pyrazolo[3,4-b]quinolin-4-amines, pharmaceutical compositions containing them and methods for a) effecting c-GMP-phosphodiesterase inhibition, b) treating heart failure and/or hypertension, c) reversing or reducing nitrat... | 01/30/1996 |
| 5242924 | Tetrazolyl-(phenoxy and phenoxyalkyl)-piperidinylpyridazines as antiviral agents Compounds of the formula ##STR1## wherein: Y is a bond, or C1 -C6 alkylene; R1 is hydrogen or C1 -C3 lower-alkyl; R2 and R3 are each independently hydrogen, C1 -C3 | 09/07/1993 |
| 5239110 | Phenylcyclohexanol derivatives as agents for treating CNS disorders Compounds of the formula ##STR1## wherein R1 is lower-alkanoyl or hydrogen; R2 and R3 are the same or different lower-alkyl; or pharmaceutically acceptable acid-addition salts thereof are useful in the treatment of di... | 08/24/1993 |
| 5206231 | 2,5-benzodiazocine antiarrhythmic agents Novel 2,5-benzodiazocines of formulas II and IV, pharmaceutical compositions containing them, processes for preparing them and methods of treating cardiac arrhythmias in mammals utilizing them. ##STR1##... | 04/27/1993 |
