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| Number | Title | Issue Date |
| 7157425 | Apolipoprotein A-I agonists and their use to treat dyslipidemic disorders The present invention provides peptides and peptide analogues that mimic the structural and pharmacological properties of human ApoA-I. The peptides and peptide analogues are useful to treat a variety of disorders associated with dyslipidemia. ... | 01/02/2007 |
| 7335799 | Hydroxyl compounds and compositions for cholesterol management and related uses The present invention relates to novel hydroxyl compounds, compositions comprising hydroxyl compounds, and methods useful for treating and preventing a variety of diseases and conditions such as, but not limited to aging, Alzheimer's Disease, cancer, cardiovascular ... | 02/26/2008 |
| 7192940 | Ether compounds The present invention relates to novel ether compounds, compositions comprising ether compounds, and methods useful for treating and preventing cardiovascular diseases, dyslipidemias, dysproteinemias, and glucose metabolism disorders comprising administering a compo... | 03/20/2007 |
| 7141608 | Calcium dicarboxylate ethers, methods of making same, and treatment of vascular disease and diabetes therewith Alcohol and water solvates of 6-(5-carboxy-5-methyl-hexyloxy)-2,2-dimethylhexanoic acid monocalcium salt are crystalline and have the formula wherein R1 is H or lower alkyl, and x is a number from 0 to... | 11/28/2006 |
| 7119221 | Cycloalkyl-hydroxyl compounds and compositions for cholesterol management and related uses The present invention relates to novel cycloalkyl-hydroxyl compounds, compositions comprising hydroxyl compounds, and methods useful for treating and preventing a variety of diseases and conditions such as, but not limited to aging, Alzheimer's Disease, cancer, card... | 10/10/2006 |
| 7015232 | Stabilization of quinapril using magnesium oxide The present invention is directed to ACE inhibitor-containing compositions stabilized by the presence of magnesium oxide. Preferably, the ACE inhibitor, quinapril, is protected from certain forms of degradation when prepared in a pharmaceutical composition consistin... | 03/21/2006 |
| 6962928 | Tetrahydroquinoline derivatives for the inhibition of osteoporosis, estrogen dependent breast cancer, endometriosis and uterine fibrosis The current invention provides methods for inhibiting osteoporosis, estrogen dependent breast cancer, endometriosis and uterine fibrosis comprising administering to a patient in need thereof a compound of the formula: ... | 11/08/2005 |
| 6828331 | Growth hormone secretagogues What is disclosed are growth hormone secretagogues, and their uses, of the formula wherein R1 is C6H5CH2OCH2—, C6H5 (CH2... | 12/07/2004 |
| 6723739 | Glucopyranoside benzothiophenes A compound of the formula or a pharmaceutically acceptable salt or solvate thereof. Also provided by the invention are methods of use of the above compounds, and processes for the preparation thereof. ... | 04/20/2004 |
| 6258826 | Pharmaceutical formulations and applications thereof for the treatment of estrogen deprivation syndrome Formulations and applications thereof are described which are useful for the inhibition of various medical conditions associated with estrogen deprivation syndrome including osteoporosis and hyperlipidemia utilizing compounds of structure I represented by... | 07/10/2001 |
| 6197790 | Benzothiophene compounds, intermediates, compositions, and methods A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a is --H... | 03/06/2001 |
| 6077852 | Treatment of central nervous system disorders with selective estrogen receptor modulators The present invention provides a method of treating depression, mood swings, or Alzheimer's disease in a patient in need of such treatment by administering a selective estrogen receptor modulating compound of the formula ##STR1## in which R... | 06/20/2000 |
| 6030986 | Benzothiophene compounds, intermediates, compositions, and methods A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a i... | 02/29/2000 |
| 5998441 | Benzothiophene compounds, intermediates, compositions, and methods A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a i... | 12/07/1999 |
| 5985898 | Benzothiophene compounds, intermediates, compositions, and methods A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a i... | 11/16/1999 |
| 5986109 | Benzothiophene compounds, intermediates, compositions, and methods A compound of fomula XIV: ##STR1## wherein: R1a is --H or --OR7a in which R7a is a hydoxy protecting group; R2a is --H, halo, or OR8a in which R8a is a hydroxy protecting group; and R | 11/16/1999 |
| 5981765 | Benzothiophene compounds, intermediates, compositions, and methods The present invention provides a compound of formula ##STR1## wherein R1a is --H or --OR7a in which R7a is a hydroxy protecting group; R2a is --H, halo, or --OR8a in which R8a is a hydroxy ... | 11/09/1999 |
| 5977093 | Benzothiophene compounds, intermediates, compositions, and methods A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I wherein R1a is --H or --OR7a in which R7a is --H or a hydroxy ... | 11/02/1999 |
| 5969142 | Benzothiophene compounds, intermediates, compositions and methods The present invention provides compounds and processes for the preparation of compounds of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a is --H or a hydroxy protecting group; R2a is --H, halo... | 10/19/1999 |
| 5919800 | Benzothiophene compounds, intermediates, compositions, and methods The present invention provides a method for inhibiting endometriosis comprising administering to a woman an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a is --H or a ... | 07/06/1999 |
| 5856339 | Benzothiophene compounds, intermediates, compositions, and methods The present invention provides intermediate compounds and processes for the preparation of compounds of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a is --H or a hydroxy protecting group; R2a... | 01/05/1999 |
| 5856340 | Method of treating estrogen dependent cancers A method for alleviating the symptoms of post-menopausal syndrome comprising administering to a woman in need thereof an effective amount of a compound of formula I ##STR1## wherein R1a is --H or --OR7a in which R7a i... | 01/05/1999 |
| 5734062 | Method of preparation of physostigmine carbamate derivatives from eseretholes This invention relates to a process for the preparation of a product of the formula ##STR1## wherein R is loweralkyl; R1 is hydrogen, loweralkyl, lowercycloalkyl, lowercycloalkylloweralkyl, lowerbicycloalkyl, aryl or arylloweralkyl; Rs ... | 03/31/1998 |
| 5698523 | Acylated enol derivatives as prodrugs of elastase inhibitors This invention relates to acylated enol derivatives of known elastase inhibitors. These compounds are useful in the treatment of various inflammatory diseases, including cystic fibrosis and emphysema or as prodrugs of compounds which are useful in the tre... | 12/16/1997 |
| 5683982 | Synthetic lung surfactant having antioxidant properties Synthetic pulmonary surfactants having antioxidant properties consisting of a complex of a polypeptide, with an antioxidant moiety, having an alpha-helical structure and a lipid consisting of one or more of the lipids associated with natural pulmonary sur... | 11/04/1997 |
| 5681925 | Trifunctional antithrombin and antiplatelet peptides Novel compounds which contain a thrombin catalytic-site inhibitor coupled with an anion binding exosite associating moiety via an RGD-X bridging sequence are trifunctional anticoagulants useful in treating venous or arterial thrombotic conditions.... | 10/28/1997 |
| 5677457 | Method of preparation of physostigmine carbamate derivatives from eseroline ethers The present invention relates to a novel process for the preparation of physostigmine carbamate derivatives and to pharmaceutically acceptable salts thereof. The present invention further relates to a novel process for the preparation of eseroline derivat... | 10/14/1997 |
| 5672625 | Sulfonic stilbene derivatives in the treatment of viral diseases Sulfonic acid stilbenes block the infection of cells by HSV and CMV and these compounds can be used to treat viral infection.... | 09/30/1997 |
| 5670521 | Reversal of multi-drug resistance by triphenyl-azacycloalkane derivatives Certain triphenylpiperidines reverse drug resistance in multi-drug resistant tumors. These compounds apparently function by inhibiting a p-glycoprotein pump which becomes activated in late stage tumor development and which is inherently present in tumors ... | 09/23/1997 |
| 5665880 | Method of preparation of physostigmine carbamate derivatives from eseretholes This invention relates to a process for the preparation of a product of the formula ##STR1## wherein R is loweralkyl; R1, is hydrogen, loweralkyl, lowercycloalkyl, lowercycloalkylloweralkyl, lowerbicycloalkyl, aryl or arylloweralyl; R... | 09/09/1997 |
| 5665780 | Reversal of multi-drug resistance by tetraarylethylenes Certain tetraarylethylenes reverse drug resistance in multi-drug resistant tumors. These compounds apparently function by inhibiting a p-glycoprotein pump which becomes activated in late stage tumor development and which is inherently present in tumors fr... | 09/09/1997 |
| 5650416 | Piperidinyl thiacyclic derivatives Piperidinyl thiacyclic derivatives of the formula ##STR1## wherein X, Y, R1, R2, R3 and R4 are defined in the specification, are useful in the treatment of allergic diseases and diseases responding to antag... | 07/22/1997 |
| 5631268 | Piperidinyl thiacyclic derivatives Piperidinyl thiacyclic derivatives of the formula ##STR1## wherein X, Y, R1, R2, R3 and R4 are defined in the specification, are useful in the treatment of allergic diseases and diseases responding to antag... | 05/20/1997 |
| 5608095 | Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents This invention relates to compounds of the formula ##STR1## wherein R1 and R6 are each independently C1 -C6 alkyl; R2, R3 and R4 are each independently hydrogen or C1 ... | 03/04/1997 |
| 5602147 | Piperidinyl thiacyclic derivatives Piperidinyl thiacyclic derivatives useful in the treatment of allergic diseases and diseases responding to antagonism of 5HT2 receptors, pharmaceutical compositions and a methods of treatment using these compounds.... | 02/11/1997 |
| 5595979 | Method of treating a neoplastic disease state by conjunctive therapy with 2'-fluoromethylidene derivatives and radiation or chemotherapy The present invention relates to a method of treating a patient afflicted with a neoplastic disease state comprising the administration thereto of an effective antineoplastic amount of ionizing or nonionizing radiation, or an effective antineoplastic amou... | 01/21/1997 |
| 5596003 | Piperidinyl thiacyclic derivatives Piperidinyl thiacyclic derivatives useful in the treatment of allergic diseases and diseases responding to antagonism of 5HT2 receptors, pharmaceutical compositions and a methods of treatment using these compounds.... | 01/21/1997 |
| 5574012 | Analogs of hirudin having anti-platelet activity This invention relates to peptide derivatives which are useful anticoagulant agents.... | 11/12/1996 |
| 5563156 | Thrombin inhibitors This invention relates to novel polyfluorinated alkyl derivatives of certain tripeptides, to the methods for their preparation, the intermediates therefore, to their use in inhibiting thrombin and lung tryptase and in their end-use application as anti-coa... | 10/08/1996 |
