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| Number | Title | Issue Date |
| 6331636 | Therapeutically useful 2-aminotetralin derivatives This invention is therapeutically useful 2-aminotetralins and pharmaceutically acceptable acid addition salts thereof of the formula ##STR1## These compounds are useful to treat central nervous system disorders, hypertension, diabetes, sexual impotency an... | 12/18/2001 |
| 6008253 | Use of 3-guanidinopropionic acid to increase endurance, stamina and exercise capacity in a mammal The present invention provides a new food product and use for a known compound. More particularly, the present invention provides a new food product containing 3-guanidinopropionic acid and a method of using 3-guanidinopropionic acid to increase endurance... | 12/28/1999 |
| 5721132 | Synthetic gene for D4 dopamine receptors A modified gene coding for the human D4 dopamine receptor has been synthesized by chemo-enzymatic methods. The nucleotide sequence of the D4 dopamine receptor gene was changed to reduce the G+C content and to eliminate intronic sequences, while maintainin... | 02/24/1998 |
| 5663305 | Somatotropin analogs The present invention provides analogs of animal somatotropins particularly with changes in the amino acids between residue 96 to 133 which are changed to reduce hydrophobicity or helical stability.... | 09/02/1997 |
| 5650427 | Centrally acting 6,7,8,9-tetrahydro-3H-benz(e) indole heterocyclics A compound of Formula I ##STR1## or pharmaceutically acceptable salts of Formula I, where R1 is H, C1 -C3 alkyl, --(CH2)n CONH2 where n is 2 to 6, (CH2)n -1-(4,4-dimethylpip... | 07/22/1997 |
| 5643895 | Phosphonoacetic esters and acids as anti-inflammatories Compounds useful in the treatment of inflammation structurally represented as Formula I ##STR1## one of X or Y is H and the other is selected from the group consisting of: ##STR2## or X and Y are taken together to form a ring selected from the g... | 07/01/1997 |
| 5643942 | Methods, composition and solutions for treating alopecia This invention relates to the method for treating the form of alopecia commonly known as "male pattern baldness" which comprises regular topical application to the affected areas of the human scalp of a composition containing as at least one of its active... | 07/01/1997 |
| 5643940 | Dioxapyrrolomycin as an antiparasitic agent and compositions useful therefor This invention concerns a method for killing internal parasites, especially nematodes, trematodes and cestodes affecting warm blooded animals such as sheep, cattle, swine, goats, dogs, cats, horses and humans as well as poultry by administering an effecti... | 07/01/1997 |
| 5635495 | Pyrimidine bisphosphonate esters and (alkoxymethylphosphinyl)alkyl phosphonic acids as anti-inflammatories Compounds useful in the treatment of inflammation structurally represented as ##STR1## wherein X,X1 and R groups are as herein defined.... | 06/03/1997 |
| 5633374 | Pyrimidine, cyanoguanidines as K-channel blockers Pyrimidine-cyanoguanidine compounds of Formula I and its pharmaceutically acceptable acid addition salts ##STR1## wherein R1 is hydrogen or methyl; R2 is C1 -C6 alkyl, C2 -C6 alkenyl, C | 05/27/1997 |
| 5631227 | Somatotropin analogs The present invention provides analogs of somatotropins wherein the asparagine residue corresponding to position 99 of a bovine somatotropin is replaced with a compound selected from the group consisting of proline, aspartic acid, glutamic acid, serine, g... | 05/20/1997 |
| 5622845 | Fermentation method for producing norleucine The present invention provides an inexpensive fermentation medium for growing microorganisms. Also provided are fermentation media and methods for producing norleucine by growing E. coli thereon, fermentation media and methods for incorporating norleucine... | 04/22/1997 |
| 5621123 | Cyclic hydrocarbons with an aminoalkyl sidechain Provided are cyclic hydrocarbons of Formula I ##STR1## with an aminoalkyl sidechain that are useful for treating phospholipase A2 mediated conditions, diabetes, and obesity.... | 04/15/1997 |
| 5616320 | Use of antibiotics 10381b to promote growth Antibiotic 10381a1, wherein R is hydrogen, is a cytosine-containing antibiotic producible by culturing the novel microorganism Streptomyces arginensis in an aqueous medium and isolation thereof. Derivatives wherein R is a C1 to C | 04/01/1997 |
| 5610158 | 4-oxo- and 4H-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents Imidazo-benzoxazines of Formula (I) and pharmaceutically acceptable salts thereof. ##STR1## where Q is selected from (A) through (H) ##STR2## or pharmaceutically acceptable salts thereof wherein the R groups are as defined herein. The imida... | 03/11/1997 |
| 5602115 | Bisphosphonic acid derivatives as anti-arthritic agents The bisphosphonates of formula (III) R2 --X--(CW)m1 --CR3 R4 --CH2 --CM[PO--(OR1)2 ]2 (III) bicyclic bisphosphonates (V), and cyclic bisphosphonates (VII... | 02/11/1997 |
| 5601974 | Method of detecting viral infection in vaccinated animals Provided are methods for determining whether a vaccinated animal is uninfected or infected with a virulent wild-type virus. Methods, vaccines and viruses are disclosed that are useful to seratologically distinguish infected from uninfected animals in popu... | 02/11/1997 |
| 5599930 | Substituted indoles as anti-AIDS pharmaceuticals Substituted indoles of formula (I) ##STR1## are useful anti-AIDS pharmaceuticals.... | 02/04/1997 |
| 5599841 | Use of 3-guanidinopropionic acid in the treatment and prevention of metabolic disorders The present invention provides a method for treating or preventing certain metabolic disorders comprising the systemic administration of 3-guanidinopropionic acid.... | 02/04/1997 |
| 5597816 | Pyrazoloazepino substituted oximes useful as anti-atherosclerosis and anti-hypercholesterolemic agents Pyrazoloazepino-substituted oximes, having the formula ##STR1## wherein R is ##STR2## where R5 is --(CH2)c -- and c is 3-6 are disclosed. These compounds are useful for the treatment of atherosclerosis and h... | 01/28/1997 |
| 5594140 | Imidazo[1,5-A]quinolines for treatment of anxiety and sleep disorders Imidazo[1,5-a]quinolines of formula (I) which are useful pharmaceutical agents for the treatment of anxiety, sleep disorders, panic states, convulsions and muscle disorders. ##STR1##... | 01/14/1997 |
| 5594144 | Tropolone derivatives and pharmaceutical composition thereof for preventing and treating ischemic diseases The present invention provides novel tropolone derivatives of the formula I ##STR1## wherein R10 is a substituted or unsubstituted piperazinyl or benzothiazolidinyl group, and pharamaceutical compositions thereof. These compounds are usefu... | 01/14/1997 |
| 5594024 | Centrally actig substituted phenylazacycloalkanes A compound or Formula I ##STR1## or a pharmaceutically acceptable salt thereof wherein n is 1 or 2; R1 and R2 are independently H (provided only one is H at the same time), --OH, CN, CH2 CN, 2- or 4-CF3, CH... | 01/14/1997 |
| 5593980 | Arylmethylphosphonates and phosphonic acids useful as anti-inflammatory agents This invention provides a new use of acids, esters, and salts of arylmethylphosphonates of Formula I, ##STR1## or a phosphonic acid of Formula II ##STR2## and derivatives as anti-inflammatory and anti-arthritic agents. Representative compou... | 01/14/1997 |
| 5583106 | Somatotropin for increasing reproductive performance in cattle This invention provides a method of using somatotropin to enhance the reproductive performance in cattle by commencing administration during the early postpartum period. Following one aspect of the invention, somatotropin (5 mg/day) is administered starti... | 12/10/1996 |
| 5578599 | Stimulation of hair growth with minoxidil and a 5-reductase inhibitor An improved method and composition for promoting hair growth in mammals for treating various forms of alopecia or male pattern baldness comprising the concomitant administration of potassium channel openers, such as minoxidil, cromakalim, pinacidil, or a ... | 11/26/1996 |
| 5574038 | 5,6-cyclicimidazo [1,5-a] Quinoxalines The invention discloses imidazo[1,5-a]quinoxalines (I) ##STR1## which do not contain an endocyclic carbonyl group that are useful as anxiolytic and sedative/hypnotic agents.... | 11/12/1996 |
| 5567722 | Cyanoguanidines as K-channel blockers Cyanoguanidine compounds of Formula I and its pharmaceutically acceptable acid addition salts ##STR1## wherein R1 is hydrogen or methyl; R2 is C1 -C6 alkyl, C2 -C6 alkenyl, C2 ... | 10/22/1996 |
| 5566828 | Locking package for a syringe A locking package structure wherein the package will provide a convenient and safe disposable receptacle for the syringe and the needle thereon and which can then be closed so as to prevent the syringe and needle from being a hazard. The open box receives... | 10/22/1996 |
| 5565571 | Substituted aryl- and heteroaryl-phenyloxazolidinones The present invention discloses novel substituted aryl- and heteroarylphenyloxazolidinones which are useful as anti-bacterial agents. More specifically, the substituted aryl- and heteroarylphenyloxazolidinones of the invention are characterized by ox... | 10/15/1996 |
| 5565468 | Pyridino substituted oximes useful as anti-atherosclerosis and anti-hypercholesterolemic agents Imidazopyridino- and pyrazolopyridino- substituted oximes are disclosed having the formulas ##STR1## wherein R1, R2, R3, R4, R5 and a are as described in the claims. for the treatment of atherosc... | 10/15/1996 |
| 5565441 | Phosphonoacetic esters and acids as anti-inflammatories Compounds useful in the treatment of inflammation structurally represented as Formula I ##STR1## one of X or Y is H and the other is selected from the group consisting of: ##STR2## or X and Y are taken together to form a ring selected from the g... | 10/15/1996 |
| 5563142 | Diaromatic substituted compounds as anti-HIV-1 agents The present invention includes diaromatic substituted heterocyclic compounds (III) ##STR1## which are useful in treating individuals infected with the HIV virus.... | 10/08/1996 |
| 5556878 | Ɗ6,7 -taxols antineoplatic use and pharmaceutical compositions containing them This invention provides 7-deoxy-Ɗ6,7 -taxol and 7-deoxy-Ɗ6,7 -taxol analogs of Formula I: ##STR1## The compounds of Formula I are useful for the same cancers for which taxol has been shown active, including human ovarian cance... | 09/17/1996 |
| 5554617 | Method for treating cancer with 6-aryl pyrimidine compounds A method for altering the immunoregulatory system of humans and animals by administering a compound of the formula: ##STR1## wherein X3 is equal to X, X4, or X5 wherein X4 is fluoro, chloro, bromo or iodo, ... | 09/10/1996 |
| 5552152 | Taste masking of ibuprofen by fluid bed coating A chewable taste-masked ibuprofen tablet having controlled release characteristics.... | 09/03/1996 |
| 5547950 | Oxazolidinone antimicrobials containing substituted diazine moieties A compound of structural Formula I: ##STR1## or pharmaceutically acceptable salts thereof wherein: each n is independently 1 to 3; Y is chosen from a-n as defined herein; wherein each occurrence of said C.sub.1-6 alkyl may be substituted with one or ... | 08/20/1996 |
| 5545755 | Therapeutically useful 2-aminotetralin derivatives This invention is therapeutically useful 2-aminotetralins and pharmaceutically acceptable acid addition salts thereof of the formula ##STR1## R, R1 to R5 and p are as defined in the specification, these compounds are useful to t... | 08/13/1996 |
| 5541339 | CC-1065 analogs having two CPI subunits This invention concerns chemical compounds of general Formula I CPI1 -R5 -T-R'5 -CPI2 I The compounds of Formula I are useful as uv light absorbers, antibacterial agents, and are particularly useful as an... | 07/30/1996 |
| 5541324 | Imidazo[1,5-A]quinoxalines An invention relating to Imidazo[1,5-a]quinoxalines (I) ##STR1## which do not contain an endocyclic carbonyl group and which are useful as anxiolytic and sedative/hypnotic agents.... | 07/30/1996 |
