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A method of swing on a swing is disclosed, in which a user positioned on a standard swing suspended by two chains from a substantially horizontal tree branch induces side to side motion by pulling alternately on one chain and then the other.
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| Number | Title | Issue Date |
| 5710165 | Use of polyamine antagonists for the treatment of glaucoma Polyamine antagonists are found to be effective in preventing or reducing visual field loss associated with glaucoma. Especially preferred are certain 1-phenyl-2-piperidinoalkanol derivatives, such as eliprodil and ifenprodil.... | 01/20/1998 |
| 5244901 | 4-pyrimidinecarboxamide derivatives, their preparation and their application in therapy The present invention provides a compound which is a 4-pyrimidinecarboxamide derivative of general formula (I) ##STR1## in which X represents one or more substituents independently chosen from fluorine, chlorine, methoxy and cyclopropyl, R1 | 09/14/1993 |
| 5244894 | 2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics Compounds corresponding to the general formula (I) ##STR1## in which n=2 or 3, X=H, F, Cl or OCH3, R=H or CH3, R1 =H or CH3, R2 =alkyl, hydroxyalkyl, (hydroxy)(methoxy)alkyl, dimethoxyalkyl, 2-(a... | 09/14/1993 |
| 5212181 | 1-(3,4-dihydro-2-oxo-1H-quinolin-6-yl)-2-[4-(2-phenylethyl)piperidin-1-yl]e t [4-(2-phenylethyl)piperidin-1-yl]ethanone, to their preparation and to their therapeutic application A compound which is an ethanol or ethanone derivative of general formula (I) ##STR1## in which X represents CO or CHOH, or is an addition salt thereof with an acid, and, when X represents CHOH, is in the form of a pure enantiomer or a mixture of... | 05/18/1993 |
| 5210086 | 2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapy A compound which is a 2-aminopyrimidine-4-carboxamide derivative, of the general formula (I) ##STR1## in which m is 0 or 1, p is 0 or 1, q is 1 or 2, n is 2 or 3, R1 represents a hydrogen atom or a methyl group, and X represents at least o... | 05/11/1993 |
| 5192797 | Derivatives of 2-aminoalkyl-5-arylalkyl-1,3-dioxanes, their preparation and their therapeutic application A compound which is a 2-aminoalkyl-5-arylalkyl-1,3-dioxane of general formula (I) ##STR1## in which m represents 0 or 1; n represents 1, 2, 3 or 4; R1 represents hydrogen or methyl; R2 represents hydrogen, methyl or an alkanoyl group... | 03/09/1993 |
| 5192763 | [(1-arylpyrrolidin-2-yl)methyl]piperazine derivatives, their preparation and their application in therapeutics [(1-Arylpyrrolidin-2-yl)methyl]piperazine compounds corresponding to the formula ##STR1## in which Z denotes a group of formula N-R1 in which R1 is either a hydrogen atom or a C1-3 alkyl group or a group of formula ... | 03/09/1993 |
| 5179108 | Derivatives of 4-(aminomethyl) piperidine, their preparation and their therapeutic application Compounds of general formula (I) ##STR1## in which n is 1 or 2; R represents a linear or branched C1 -C3 -alkyl group; and X represents at least one substituent chosen from hydrogen, halogen, C1 -C3 -alkyl and C... | 01/12/1993 |
| 5169779 | Process for the preparation of methyl (-)-(2R,3S)-2,3-epoxy-3-(4-methoxy-phenyl)propionate A process for the preparation of methyl (-)-(2R,3S)-2,3-epoxy-3-(4-methoxyphenyl)propionate, which comprises subjecting the dextrorotatory (2S,3R) enantiomer, present in a starting mixture containing both the levorotatory (2R,3S and dextrorotatory (2S,3R)... | 12/08/1992 |
| 5164397 | 2-Aminopyrimidine-4-carboxamide derivatives, their preparation and their application in urinary therapeutics A compound of formula (I) ##STR1## in which n denotes 2, 3, 4, or 5, p denotes 0 or 1, m denotes 0, 1, 2, 3, 4, or 5, and R1 denotes a hydrogen atom or a methyl group, each X, which may be identical or different to any other X if m is greater t... | 11/17/1992 |
| 5112621 | Sustained release pharmaceutical composition of diltiazem A sustained-release pharmaceutical composition which comprises microparticles comprising an active principle, said microparticles being coated with a coating mixture comprising ethyl cellulose and an acrylic resin which is a polymerizate of acrylic and me... | 05/12/1992 |
| 5102998 | Method for preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-5H-1,5-benzothiaze pine-4-one and chlorinated derivatives thereof 2-Aminothiophenol is reacted with methyl (-)-(2R,3S)-2,3-epoxy-3-(4-methoxyphenyl)propionate, and the intermediate methyl (2S,3S)-3-[(2-aminophenyl)thio]-2-hydroxy-3-(4-methoxyphenyl)propionate is cyclized in the presence of methanesulfonic acid, in ... | 04/07/1992 |
| 5096900 | (4-piperidyl)methyl-2,3-dihydro-1H-isoindole and -2,3,4,5-tetrahydro-1H-benzazepine derivatives, their preparation and their application in therapy A benzazepine derivative which is a compound of formula (I): ##STR1## in which: each of m and n denotes the number 1, or each of m and n denoted the number 2, or m denotes the number 3 and n denoted the number 1; and R denotes hydrogen or a group of formula --... | 03/17/1992 |
| 5081128 | 2,3-dihydro-1H-isoindole derivatives and their application in therapy A benzazepine derivative which is a compound of formula (I): ##STR1## in which each of m and n denotes the number 1, or each of m and n denotes the number 2, or m denotes the number 3 and n denotes the number 1; and R denotes hydrogen or a group of formul... | 01/14/1992 |
| 5081277 | Process for the preparation of propionic acid derivatives Process for the preparation of compounds of the general formula (I) ##STR1## wherein R is hydrogen or (C1-4)alkyl.... | 01/14/1992 |
| 5075325 | N-aminobutyl-n-phenylarylamide derivatives, their preparation and their application in therapy A compound of formula (I) ##STR1## in which: X denotes hydrogen, a halogen, a trifluoromethyl group, a C1 -C4 alkyl group or a C1 -C4 alkoxy group; R1 denotes a linear or branched C2 -C | 12/24/1991 |
| 5064836 | Imidazopyridine for use as an anaesthetic A method of anaesthetizing a subject in need of anaesthetizing, which comprises administering to the subject an anaesthetically effective amount of N-[[2-(4-ethylphenyl)-3-imidazo[1,2-a]pyridinyl]methyl] N,3-dimethylbutanamide or a pharmaceutically accept... | 11/12/1991 |
| 5034401 | Derivatives of (1-hydroxy-2-piperidylalkyl-indol-2-ones, 2-quinolinones, 2-benzo(B)azapinones, benzimidazol-2-ones, and quinazolin-2-ones, their preparation and their application in therapeutics A compound, in the form of a pure optical isomer or a mixture thereof, of formula (I): ##STR1## in which: Z represents a group of formula --CH2 --, --C(CH3)2 --, --CH.dbd.CH--, --(CH2)2 --, ... | 07/23/1991 |
| 5023266 | Method of treatment of psychotic disorders Ifenprodil and its analogues are useful for the treatment of psychoses such as schizophrenia.... | 06/11/1991 |
| 5013835 | Method of preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)2,3-dihydro-5H-1,5-benzothiazep ine-4-one 2-Aminothiophenol is reacted with (-)-(2R,3S)-2,3-epoxy-3-(4-methoxyphenyl) methylpropionate, and the intermediate (2S,3S)-3-[(2-aminophenyl)thio]-2-hydroxy-3-(4-methoxyphenyl) methylpropionate is then cyclized in the presence of methane sulfonic aci... | 05/07/1991 |
| 5010079 | Indolone derivatives, their preparation and their application in therapy An indolone derivative is useful for the treatment of anxiety, depression and schizophrenia and is a 5HT1A agonist and 5HT2 antagonist, which is a compound of formula (I): ##STR1## in which R1 is a hydrogen or halogen... | 04/23/1991 |
| 5008434 | Process for the preparation of methyl (+)-(2S,3S)-3-[(2-aminophenyl)thio]-2-hydroxy-3-(4-methoxyphenyl)-propio nates A process for the preparation of a methyl (+)-(2S,3S)-3-[(2-aminophenyl)thio]-2-hydroxy-3-(4-methoxyphenyl)propionat e of the formula (I): ##STR1## in which X denotes hydrogen or chlorine, which process comprises reacting a 2-aminothiophenol of f... | 04/16/1991 |
| 5001159 | N-aminobutyl-n-phenylarylamide compounds and their application in therapy A compound of formula (I) ##STR1## in which: X denotes hydrogen, a halogen, a trifluoromethyl group, a C1 -C4 alkyl group or a C1 -C4 alkoxy group; R1 denotes a linear or branched C2 -C | 03/19/1991 |
| 5001132 | Phenyloxypropanolamine derivatives and their application in therapeutics Phenyloxypropanolamine derivatives in the form of racemates or enantiometers, of formula (I) ##STR1## in which R is H or CH3, and their pharmaceutically acceptable salts.... | 03/19/1991 |
| 4990506 | 3-(acylaminomethyl)imidazo[1,2-a]pyridine derivatives and their application in therapy A compound which is a 3-(acylaminomethyl)imidazo[1,2-a]pyridine derivative of formula (I) ##STR1## in which R1 denotes hydrogen; linear or branched C1 -C4 alkyl; or benzyl; R2 denotes linear or branched C | 02/05/1991 |
| 4983607 | Quinolinone derivatives and their preparation in therapy A quinolinone derivative which is a compound of formula (I): ##STR1## in which: R1 and R2 are each, independently of one another, a hydrogen or halogen atom or a (C1-4)alkyl radical; R3 is a hydrogen atom or a (... | 01/08/1991 |
| 4983598 | Pharmaceutical composition containing diltiazem and angiotensin-converting enzyme inhibitor Compositions of diltiazem and angiotensin-converting enzyme inhibitor useful for the treatment of hypertension, cardiac insufficiency and coronary insufficiency.... | 01/08/1991 |
| 4977159 | 2-[(4-piperidyl)methyl]-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole derivatives, and their application in treating depressive state, anxiety state or hypertension A compound which is a pyrido[3,4-b]derivative of formula (I) ##STR1## in which R is a hydrogen atom or an alkyl carbonyl, arylalkylcarbonyl or arylcarbonyl group of formula COR1 wherein R1 is a C1 -C6 alkyl... | 12/11/1990 |
| 4973330 | Surgical apparatus for modifying the curvature of the eye cornea A surgical apparatus for partially modifying the curvature of the cornea of an eye while the eye is within the patient is disclosed. The device is able to ablate a zone of corneal material in the form of a lenticular lamina. The thickness of the lamina at... | 11/27/1990 |
| 4963680 | Piperazine derivatives and their preparation process A piperazine derivative of formula (I) ##STR1## in which: R is hydrogen or a straight or branched (C1 -4) alkoxycarbonyl group; and A is a 7-methoxy-1-naphthalenyl, 6-methoxy-2,3-dihydro-1-(1H)-indenyl or 7-methoxy-1,2,3,4-tetra... | 10/16/1990 |
| 4950670 | 6-phenyl-3-(piperazinyalalkyl)-2,4(1H,3H)-pyrimidinedione derivatives, their preparation and their application in therapy A pyrimidinedione derivative which is a compound of formula (I): ##STR1## in which: R1 denotes hydrogen, a halogen, a methyl group or a methoxy group, R2 denotes hydrogen, a C1 -C4 alkyl group or a benzyl group, n denotes 2, 3 or 4, ... | 08/21/1990 |
| 4945096 | Treatment of a depressive state with 2-[(4-piperidyl)methyl]-1,2,3,4-tetrahydroisoquinoline derivates A compound of formula (I) ##STR1## in which R is (a) a hydrogen atom; (b) a linear or branched (C1 -C6) alkyl group; an allyl group; a cycloalkylmethyl group in which the cycloalkyl moiety has from 3 to 6 carbon atoms; a phenylm... | 07/31/1990 |
| 4931449 | 2-((4-piperidyl)methyl)benzofuro(2,3-C)pyridine derivatives, and their application in therapy A compound of formula (I) ##STR1## in which R is a benzyl, benzoyl, 3-chlorobenzoyl, 3-methylbenzoyl or (C1 -C6 alkoxy)carbonyl group, or a pharmacologically acceptable acid addition salt thereof.... | 06/05/1990 |
| 4929621 | 1-1[(2-pyrimidinyl)amino-alkyl]piperidines, their preparation and their application in therapy A compound which is a pyrimidinylamino derivative of piperidine of formula (I) ##STR1## in which: X is a (CH2)2, CH.dbd.CH or CH2 --CO group; Y is a CH.dbd.CH group or sulphur; n is 2, 3 or 4; R1 is hydrogen or ... | 05/29/1990 |
| 4925850 | Derivatives of 2-((4-piperidinyl)methyl)-1,2,3,4-tetrahydroisoquinoline, their preparation and their application in therapeutics A compound of formula (I): ##STR1## in which: X is hydrogen or a methyl or methoxy group; Y is a halogen or a methyl or methoxy group; and R is a group of formula --Z--R' in which: Z is a --CH2 -- group, and R' is a phenyl group unsubstituted or sub... | 05/15/1990 |
| 4925837 | Pharmaceutical compositions Pharmaceutical compositions containing, by way of active substance, a combination of an alpha-blocker and a calcium antagonist. The composition is useful in treating cardiovascular disorders, especially hypertension.... | 05/15/1990 |
| 4914092 | Benzothiazepin-4-one derivatives, their preparation and their application in therapy A compound, in the form of a pure diastereoisomer or mixture thereof, which is a benzothiazepin-4-one derivative of formula (I): ##STR1## in which: R1 is hydrogen or a C2 -C4 alkanoyl group; R2 and R3 independently each is hydrogen, ... | 04/03/1990 |
| 4912219 | 2-[4-pyrimidin-2-yl amino)piperidin-1-yl]benzimidazole compound Benzimidazole derivatives corresponding to the formula (I) ##STR1## in which X is CH or N, R1 is either a hydrogen atom, or a benzyl radical which can bear 1 to 3 substituents chosen from halogen atoms and trifluoromethyl, (C1-4... | 03/27/1990 |
| 4908214 | Pharmaceutical tablet for the treatment of uraemia A tablet constituted by (1) a core comprising a mixture of salts formed by a basic -amino acids and -keto analogues of branched-chain essential amino acids and (2) a gastroresistant or gastrosoluble coating.... | 03/13/1990 |
| 4904684 | 2-(4,5-dihydro-1H-imidazol-2-yl)-1,2,4,5-tetrahydropyrrolo[3,2,1 -hi]indole derivatives useful as antidiabetic agents 2-(4,5-Dihydro-1H-imidazol-2-yl)-1,2,4,5-tetrahydropyrrolo[3,2,1-hi]indole derivatives and their pharmaceutically acceptable salts are useful an antidiabetic agents.... | 02/27/1990 |
