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Patent No. 5970981

Mouthguard made at least partially from an edible candy

A mouthguard includes a U-shaped upper bite plate which removably fits over upper teeth of a person, with the entire upper bite plate being made from a soft, deformable and edible gummi candy.

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Assignee: Sanofi-Synthelabo


Location: Paris, FR
No. of patents: 153

1        
NumberTitleIssue Date
74276153-substituted-4-pyrimidone derivatives
A pyrimidone derivative represented by formula (I) or a salt thereof, or a solvate thereof or a hydrate thereof having inhibitory activity against tau protein kinase 1: wherein R1 represents a C1-C12 alkyl group which may be substitu...
09/23/2008
6979683Benzimidazole derivatives, preparation and therapeutic use thereof
The invention relates to benzimidazole derivatives of general formula (I) in which X represents a nitrogen atom or a carbon atom; and when X represents a nitro...
12/27/2005
6949583Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method of preparing same and compositions containing same
The invention relates to benzofuran or benzothiophene derivatives, to processes for preparing them, to pharmaceutical compositions comprising them, and to the method of use thereof in the treatment of pathological syndromes of the cardiovascular system. ...
09/27/2005
6918889Disposable injection device
A single-use injection device, includes a pre-filled syringe (1), a syringe body (5) which is integral with the said syringe, and a protective case (10), the syringe body and protective case being provided with elements (9, 14, 15, 21) fo...
07/19/2005
6916929Method for preparing 4-methylamino-4-phenylpiperidine
The invention relates to a process for preparing a 4-alkoxycarbonylamino-1-benzyl-4-phenylpiperidine of formula (I) via hydrolysis of 1-benzyl-4-cyano-4-phenylpiperidine (II) in acidic medium and treatment of the 1-ben...
07/12/2005
6908927Pyridopyranoazepine derivatives, their preparation and their therapeutic application
The invention relates to pyridopyranoazepine derivatives, to pharmaceutical compositions containing them, to process for preparing them, and to the method of use thereof in the treatment or prevention of disorders associated with a dysfunction of the nicotine recept...
06/21/2005
6908914Antipsychotic cyclic N-aralkylamines
The invention relates to benzene derivatives, to pharmaceutical compositions containing them, to processes for preparing them, and to the method of use thereof in the treatment of psychotic disorders. ...
06/21/2005
D505320Packaging for a drug blister-pack for clinical trial
05/24/2005
6894186Hydroxyacetic ester derivatives, preparation method and use as synthesis intermediates
Methyl (R)-2-(R1OSO2)-2-(2-chlorophenyl)acetates useful as intermediates in the preparation of methyl (S)-2(2-chlorophenyl)-2-(4,5,6,7-tetrahydrothieno[3,2-c]-5-pyridyl)acetate. ...
05/17/2005
6867220Phenoxypropanolamines, method for producing them and pharmaceutical compositions containing them
The invention relates to compounds of formula (I) where R1 represents a hydrogen or halogen atom or an —S(O)z—(C1-C4)alkyl, —S(O)z—(C1
03/15/2005
68642771,3-dihydro-2H-indol-2-one derivatives, method for preparing same and pharmaceutical compositions containing them
The invention relates to compounds of formula: and to solvates and/or hydrates thereof, with affinity for and selectivity towards the Vreceptors or both the V1b and V1a receptors of arginine-vasop...
03/08/2005
6861072Pharmaceutical composition with gastric residence and controlled release
The invention concerns a pharmaceutical composition with gastric residence and controlled release, characterized in that it comprises two or three layers and contains (a) an active principle associated with a excipient modifying its release; (b) a system generating ...
03/01/2005
6858629Heteroaryloxy propanolamines, preparation method and pharmaceutical compositions containing same
Compounds of formula (I): where X is N or CH; A represents a group of formula (a) or (b) R1 represents hydrogen or an —NH2, —NR...
02/22/2005
6852736Phenoxypropanolamines, preparation and therapeutic use thereof
The invention concerns phenoxypropanolamines of formula (I) in which R1 represents a hydrogen, a group —S(O)z—(C1-C4)alk-R′, (R′ being H, phenyl or (C1-C
02/08/2005
68469362-butyl-3-(4-[3(dibutylamino)propoxy]benzoyl)-5-nitro-benzofuran hydrochloride and preparation thereof
The invention relates to 2-butyl-3-(4-[3-(dibutylamino)propoxy]benzoyl-5-nitrobenzofuran hydrochloride, to its preparation and to its use as synthetic intermediate, in particular in preparing 2-butyl-3-(4-[3-(dibutylamino)propoxy]benzoyl)-5-nitrobenzofuran, itself a...
01/25/2005
6844329Polysaccharides with antithrombotic activity comprising at least a covalent bond with biotin or a biotin derivative
The present invention relates to novel synthetic polysaccharides with antithrombotic activity exhibiting at least one covalent bond with biotin or a biotin derivative and to a process employing avidin or streptavidin which makes it possible to neutralize these polys...
01/18/2005
68443352-amino-3-(alkyl)-pyrimidone derivatives as GSK3.β.inhibitors
A pyrimidone derivative represented by formula (I) or a salt thereof: Wherein: R1 represents a hydrogen atom or a C1-6 alkyl group which may be substituted by a C
01/18/2005
68443371,4-diazabicyclo[3.2.2]nonane-phenylisoxazole derivatives, their preparation and their application in therapeutics
Compounds corresponding to general formula (I) in which R1, R2, R3, R4 and R5 each represent, independently of one another, a hydrogen or halogen atom or a nitro, ...
01/18/2005
68357304-heteroparyl-1,4-diazabicyclo[3.2.2]nonane, preparation and therapeutic use thereof
Compounds of the general formula (I) in which R1, R2, R3 and R4 each represent a hydrogen or halogen atom or a nitro, amino, trifluoromethyl, cyano, hydroxyl, alkyl or alkoxy...
12/28/2004
6828448Methanesulphonamido-benzofuran, preparation method and use thereof as synthesis intermediate
The invention relates to 2-butyl-5-(methanesulfonamido)benzofuran, its preparation and its use. This compound is a synthesis intermediate, in particular for the preparation of dronedarone. ...
12/07/2004
6806282Branched substituted amino derivatives of 3-amino-1-phenyl-1h-[1,2,4]triazol, methods for producing them and pharmaceutical compositions containing them
The present invention relates to novel branched substituted amino derivatives of 3-amino-1-phenyl-1H-[1,2,4]triazole, processes for their preparation and pharmaceutical compositions comprising them. ...
10/19/2004
6800761Form of irbesartan, methods for obtaining said form and pharmaceutical compositions containing same
The invention relates to a novel crystalline form of irbesartan, to pharmaceutical compositions containing it, to processes for preparing it, and to a method for treating cardiovascular diseases utilizing it. ...
10/05/2004
6794382Benzimidazole derivatives, preparation and therapeutic use thereof
The invention relates to benzimidazole derivatives of general formula in which X represents a nitrogen atom or a carbon atom; and when X represents a nitrogen atom: R3 represents a hydrogen atom or a...
09/21/2004
6767533Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress
A composition containing a peripheral benzodiazepine receptor ligand for topical use in the treatment of cutaneous stress. ...
07/27/2004
6761879Titanium derived compounds, preparation and use thereof
The invention relates to a titanium-derived compounds, and to processes for preparing the same. ...
07/13/2004
67306951,3-dihydro-2h-indol-2-one derivatives and their use as ligands for V1b and V1a arginine-vasopressin receptors
The invention relates to compounds of formula: as well as the possible salts thereof with mineral or organic acids, and the solvates and/or hydrates thereof, which have affinity for and selectivity towards the V1b
05/04/2004
6713053Use of IL-7 for treating auto-immune diseases and insulin-dependent diabetes mellitus in particular
The use of interleukin 7 or T cells pre-incubated in the presence of IL-7 for preparing a drug or pharmaceutical composition for treating an auto-immune disease, particularly an auto-immune disease induced by a defect in CD4+ T cell immunoregulation, is disclosed.
03/30/2004
6710042Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
Compounds of formula (I) are useful as human NK3 receptor antagonists. ...
03/23/2004
6693118Use of 4-substituted tetrahydropyridines for the manufacture of medicaments acting upon TGF-댡
The invention relates to the use of a compound of formula (I): ##STR1## for the preparation of pharmaceutical compositions for increasing the circulating, cellular and extracellular levels of TGF-댡....
02/17/2004
6689797Tetrahydropyridines, preparation method and pharmaceutical compositions containing same
The present invention relates to compounds of formula (I): ##STR1## in which R1 represents a hydrogen or halogen atom, or a group CF3 ; R2 and R3 represent, independently, a hydrogen atom or a methyl group; n and n' ...
02/10/2004
6686182Alkyl esters of 3-(3,4-dihalophenyl)-2,6-dioxopiperidine-3-propionic acid of use as intermediates
The invention relates to lower-alkyl esters of 3-(3,4-dihalophenyl)-2,6-dioxopiperidine-3-propionic acid derivatives, and to processes for preparing the same....
02/03/2004
6680329N-(heterocyclyl)benzene or pyridinesulphonamides as antithrombotic agents and anticoagulants
Compounds of formula [I] ##STR1## in which: W may represent a --(CH2)2 --, --(CH2)3 --, --CH2 --C.ident.C-- or --CH2 --CH.dbd.CH-- group, R2 may in particular represent a pipe...
01/20/2004
6673790Indolin-2-one derivatives, preparation and their use as ocytocin receptor ligands
The present invention relates to novel indolin-2-one derivatives of formula: ##STR1## to the preparation and to the pharmaceutical compositions comprising them. These compounds have an affinity for oxytocin receptors....
01/06/2004
6670486Process for racemization
The invention relates to the racemisation process of the optically active [2-(2-thienyl)ethylamino](2-halogenophenyl)acetamides of general formula (VII) by using basic compounds. The resulting racemic compounds of general formula (VII) can thus be recycle...
12/30/2003
6670338Pentasaccharides processes for their preparation and pharmaceutical compositions containing them
Pentasaccharides in acidic form and their pharmaceutically acceptable salts, the anionic form thereof having the formula: ##STR1## wherein: R represents hydrogen or an --SO3-, (C1 -C3)alkyl or (C2...
12/30/2003
6649627Phenoxylpropanolamines, method for the production thereof and pharmaceutical compositions containing the same
The invention concerns compounds of formula (Ia) ##STR1## wherein R1a represents hydrogen, an --S(O)z --(C1 -C4)Alk group, a --CO(C1 -C4)Alk group, an --NHSO2 --(C1 ...
11/18/2003
66422331-Phenacyl-3-phenyl-3-(piperidylethyl)piperidine derivatives, process for the preparation thereof and pharmaceutical compositions containing them
The invention relates to the compounds of formula: ##STR1## as well as to the salts thereof with inorganic or organic acids, to solvates thereof and/or to hydrates thereof, which have strong affinity and high selectivity for the human NK1 recep...
11/04/2003
6642258Use of central cannabinoid receptor antagonist for preparing medicines
The invention relates to the use of a central cannabinoid receptor antagonist for the preparation of medicinal products that are useful in treating and preventing neuroinflammatory pathologies....
11/04/2003
6639083Method for preparing a thiopene derivative
The invention relates to a process for preparing 2-thienyl-2-ethanol, in which: a) thiophene is metallated using an alkali metal, in the presence of an electron transfer agent, b) the compound obtained is treated with ethylene oxide, c) the thienyl...
10/28/2003
66356452,5,-diazabicyclo[2.2.1]heptane derivatives, their preparation and therapeutic uses
The invention relates to 2,5-diazabicyclo[2.2.1]heptane derivatives, to pharmaceutical compositions containing them, and to methods for the treatment or prevention of disorders associated with a dysfunction of the nicotinic receptors utilizing them....
10/21/2003
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