Assignee: Glaxo Group Limited

Location: Middlesex, GB
No. of patents: 57

Number	Title	Issue Date
8178573	Compounds The present invention provides compounds of formula (I): pharmaceutical compositions comprising the compounds and the use of the compounds for the manufacture of a medicament, particularly for the treatment of inflammation ...	05/15/2012
8101775	Indole derivatives as S1P1 Receptor The invention relates to compounds of formula (I) wherein one of R5 and R6 is hydrogen or R2 and the other is (a) pharmace...	01/24/2012
8088133	Tongue cleaning device A tongue cleaning device comprising a tongue cleaning surface supported for tongue cleaning by running the surface across the tongue, a reservoir for a tongue cleaning fluid, means to dispense the fluid either onto the tongue cleaning surface, or directly onto the u...	01/03/2012
8003663	Pyrazolo[3,4-b]pyridine compounds, and their use as PDE4 inhibitors The invention provides N-{[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo [3,4-b]pyridin-5-yl]methyl}-4-({8-[(2-hydroxyethyl) (methyl)amino]octanoyl}amino)benzamide, whose formula is or a salt thereof, such as th...	08/23/2011
8003638	7-pyrazolylbenzazepines having affinity for D3 receptor Compounds of formula (I) or a salt thereof are disclosed: wherein R1 is pyrazolyl substituted by two or three substituents independently selected from halogen, C1-4alkyl and haloC1-4alkyl; R...	08/23/2011
7943651	Compounds The present invention provides compounds of formula (I): pharmaceutical compositions comprising the compounds and the use of the compounds for the manufacture of a medicament, particularly for the treatment of inflammation ...	05/17/2011
7909527	Fluid dispenser A dispensing container for application of a fluid film forming substance to a surface, particularly a therapeutic film to a user's skin comprising a reservoir of a fluid film forming substance, a dispensing nozzle for the film forming substance, and a pump to send t...	03/22/2011
7875643	Azabicyclo (3.1.0) hexane derivatives useful as modulators of dopamine D3 receptors The present invention relates to novel compounds of formula (I) or a pharmaceutically acceptable salt thereof: wherein G is selected from a group consisting of: phenyl, pyridyl, benzothiaz...	01/25/2011
7863299	Triazolyl derivatives of azabicyclo [3.1.0] hexane as dopamine D3 receptor modulators The present invention relates to novel compounds of formula (IC) or a salt thereof: wherein: p is an integer ranging from 0 to 4; R1 is independently selected from a group consisting of:...	01/04/2011
7858796	Chemical compounds The invention is directed to novel indole carboxamide derivatives. Specifically, the invention is directed to compounds according to formula I: where R1, R2, R3, U and V are defined below and to pharmaceutically acceptable ...	12/28/2010
7855298	Azabicyclo (3.1.0.) hexane derivatives useful as modulators of dopamine Dreceptors The present invention relates to novel compounds of formula (I) or a pharmaceutically acceptable salt thereof: 1. wherein G is selected from a group consisting of: phenyl...	12/21/2010
7838680	Process for preparing heterocyclic derivatives The present invention relates to a novel process, useful for preparing key intermediates of formula (I) in the synthesis of various compounds, among them compounds which are potent and specific antagonists of D3 receptors, ...	11/23/2010
7807698	Azabicyclo[3.1.0]hexane derivatives as modulators of the dopamine D3 receptor The present invention relates to novel compounds of formula (I) or a pharmaceutically acceptable salt thereof: wherein G is selected from a group consisting of: phenyl, pyridyl, benzothiaz...	10/05/2010
7803820	3-triazolylthiaalkyl-3-azabicyclo (3-1-O) hexanes and their use as dopamine D3 receptor ligands The present invention relates to novel compounds of formula (I) or a pharmaceutically acceptable salt thereof: wherein R1 is hydrogen or C1-4alkyl; R...	09/28/2010
7799815	Triazole derivatives as modulators of dopamine D3 receptors The present invention relates to novel compounds of formula (I) or a salt thereof: wherein: G is a 5- or 6-membered heteroaromatic group, or is a 9- or 10-membered bicyclic heteroaromatic ...	09/21/2010
7732020	Method and apparatus for the application of powder material to substrates An apparatus for electrostatically charging powder material and supplying it to an applicator for electrostatically applying the powder material to solid dosage forms includes a mixer for mixing a sump of the powder material to electrostatically charge the powder ma...	06/08/2010
D610674	Pharmaceutical tablet	02/23/2010
7652012	2-(R)-(4-fluoro-2-methyl-phenyl)-4-(S)-((8aS)-6-oxo-hexahydro-pyrrolo[1,2-]-pyrazin-2-yl)-piperidine-1-carboxylic acid [1-(R)-3,5-bis-trifluoromethyl-phenyl)-ethyl]-methylamide maleate and pharmaceutical compositions thereof The present invention relates to piperidine derivatives of formula (I) specifically 2-(R)-(4-Fluoro-2-methyl-phenyl)-4-(S)-((8aS)-6-oxo-hexahydro-pyrrolo[1,2-a]-pyrazin-2-yl)-piperidine-1-carboxylic acid [1-(R)-(3,5-bis-tri...	01/26/2010
7622302	Process for improving the manufacture of clavams e.g. clavulanic acid New processes for improving the manufacture of clavams e.g. clavulanic acid. Novel DNA sequences and new microorganisms capable of producing increased amounts of clavulanic acid are also disclosed. ...	11/24/2009
7618969	Compounds which potentiate glutamate receptor and uses thereof in medicine Compounds of formula (I) or a pharmaceutically acceptable salt, solvate or prodrug thereof, are disclosed: wherein R1 is C1-6alkyl, haloC1-6alkyl, C2-6alkenyl, amino, monoC1-...	11/17/2009
D601689	Pharmaceutical tablet	10/06/2009
7566735	Compounds which potentiate AMPA receptor and uses thereof in medicine Compounds of formula (I) and salts are provided: along with pharmaceutical compositions, uses in medicine, e.g., treating disease or condition mediated by a reduction or imbalance in glutamate receptor function, such as sch...	07/28/2009
7534893	Imidazol-2-one compounds useful in the treatment of various disorders A compound of formula (I) wherein: R is a group selected from: A-B is a bivalent radical of formula (v), (vi) or (vii) —CH═C(R11	05/19/2009
7504392	2,3,4,5-tetrahydro-1H-3-benzazepines and their medical use The invention provides compounds of the formula or a pharmaceutically acceptable salts thereof. The compounds are useful in therapy, in particular as antipsychotic agents.	03/17/2009
7498326	Compounds Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man. The piperidine derivatives include compounds of formula (I): ...	03/03/2009
7498020	Medicaments This invention relates to aerosol formulations of use for the administration of medicaments by inhalation, in particular a pharmaceutical aerosol formulation which comprises particulate salbutamol and physiologically acceptable salts and solvates thereof and a fluor...	03/03/2009
7482374	Pyrrolidine-2-ones as Factor Xa inhibitors The invention relates to compounds of formula (I): wherein substituents are as defined. ...	01/27/2009
7482365	Piperidylcarboxamide derivatives and their use in the treatment of tachykinin-mediated diseases The present invention relates to piperidine derivatives of formula (I): wherein R, R1, R2, R3, R4, R5, R6, X, Y, m and n are as defined herein; and pharmaceu...	01/27/2009
7465743	Pyrazolo[3,4-]pyridine compounds, and their use as PDE4 inhibitors The invention relates to a compound of formula (I) or a salt thereof: wherein: R1 is Et, n-Pr, i-Pr, C2fluoroalkyl, or —CH2CH2OH; R2	12/16/2008
7381728	Piperazine derivatives useful for the treatment of gastrointestinal disorders The invention provides compounds of formula (I) or pharmaceutically acceptable salts thereof, wherein Ra, Rb, Rc, Rd, Re, Rf and Y are as defined in the specification. The compounds are partial or ful...	06/03/2008
7342028	Medical use for tachykinin antagonists The present invention relates to the use of tachykinin antagonists, including substance P antagonists and other neurokinin antagonists, in the treatment of emesis. Also described are novel tachykinin antagonists of formula (I), processes for their preparation, pharm...	03/11/2008
7329667	CRF receptor antagonists The present invention relates to tricyclic pyrimidines compounds of formula (I) including stereoisomers, prodrugs and pharmaceutically acceptable salts or solvates thereof, to processes for their preparation, to ...	02/12/2008
7288564	Indole derivatives Compounds of formula (I) or salts or solvates thereof or physiologically functional derivatives thereof are potent binders at the EP4 receptor and are of use in the treatment or prevention of conditions such as a...	10/30/2007
D552992	Cap	10/16/2007
7220403	Pharmaceutical formulation of fluticasone propionate There is provided according to the invention a pharmaceutical aerosol formulation which comprises: (i) fluticasone propionate and (ii) a hydrofluoroalkane (HFA) propellant, characterised in that the fluti...	05/22/2007
7214692	Medical use for tachykinin antagonists The present invention relates to the use of tachykinin antagonists, including substance P antagonists and other neurokinin antagonists, in the treatment of emesis. Also described are novel tachykinin antagonists of formula (I), processes for their preparation, pharm...	05/08/2007
7157479	Oxazol/thiazol-derivatives activators of the hPPAR-alpha receptor A compound of formula (I) and pharmaceutically acceptable salts, solvates and hydrolysable esters thereof Wherein X1 represents O or S; R1 and R2 are ind...	01/02/2007
D532701	Tube	11/28/2006
D532306	Container	11/21/2006
7122538	Sulfonamide derivatives as antipsychotic agents The invention provides compounds of formula (I): wherein A and B represent the groups —(CH2)m— and —(CH2)n— respectively; R1	10/17/2006

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Assignee: Glaxo Group Limited